GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,024 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,030 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(159 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(443 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(83 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(326 products)
- PAFR(13 products)
- PKA(52 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5968 products of "GPCR/G-Protein"
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Alimemazine hemitartrate
CAS:Alimemazine hemitartrate (Trimeprazine hemitartrate) is aphenothiazine derivative that is used as an antipruritic.Formula:C18H22N2SC4H6O6Purity:98.16% - 99.69%Color and Shape:SolidMolecular weight:448.53BP 897
CAS:BP 897: potent selective dopamine D3 agonist, weak D2 antagonist. Ki: 0.92 nM (D3), 61 nM (D2), low affinity at D1/D4.Formula:C26H31N3O2Purity:99.44%Color and Shape:SolidMolecular weight:417.54Ref: TM-T9100
1mg80.00€5mg162.00€10mg227.00€25mg379.00€50mg540.00€100mg730.00€200mg938.00€1mL*10mM (DMSO)177.00€Substance P (7-11)
CAS:<p>Substance P (7-11) (Substance P 7-11(TFA)) is a C-terminal fragment of Substance P .</p>Formula:C31H44N6O5SPurity:98.39%Color and Shape:SolidMolecular weight:612.78MRT-10
CAS:<p>MRT-10 is a Smoothened (Smo) receptor antagonist.</p>Formula:C24H23N3O5SPurity:99.73%Color and Shape:SolidMolecular weight:465.52Dexmedetomidine hydrochloride
CAS:Dexmedetomidine hydrochloride (Precedex) is a potent, selective, orally active α2-adrenoceptor agonist.Cost-effective and quality-assured.Formula:C13H16N2·HClPurity:99.94% - 99.94%Color and Shape:White Or Almost White Crystalline PowderMolecular weight:236.74Ref: TM-T6466
5mg42.00€10mg55.00€25mg88.00€50mg159.00€100mg226.00€200mg340.00€500mg563.00€1mL*10mM (DMSO)50.00€Alloxazine
CAS:Alloxazine (Isoalloxazine) is an A2 receptor antagonist, which is approximately 10-fold more selective for the A2B receptor than for the A2A receptor.Formula:C10H6N4O2Purity:99.75%Color and Shape:SolidMolecular weight:214.18Cenicriviroc
CAS:Cenicriviroc (TAK-652), oral CCR2/CCR5 blocker, inhibits HIV-1/HIV-2, with strong anti-infective/anti-inflammatory effects.Formula:C41H52N4O4SPurity:97.87%Color and Shape:SolidMolecular weight:696.94Ref: TM-TQ0297
1mg66.00€2mg95.00€5mg140.00€10mg224.00€25mg445.00€50mg582.00€100mg755.00€200mg1,017.00€1mL*10mM (DMSO)210.00€SB-200646
CAS:SB-200646 is a selective and potent antagonist of 5-HT2B/5-HT2C receptorFormula:C15H14N4OPurity:99.61%Color and Shape:SolidMolecular weight:266.3Naratriptan hydrochloride
CAS:Naratriptan Hydrochloride, a selective 5-HT1 receptor agonist with anti-migraine effect, induces vasoconstriction and reduces inflammation in migraines.Formula:C17H25N3O2S·HClPurity:99.17% - 99.93%Color and Shape:Beige SolidMolecular weight:371.93Ref: TM-T6602
10mg50.00€25mg88.00€50mg133.00€100mg188.00€200mg283.00€500mg467.00€1mL*10mM (DMSO)52.00€EST64454 free base
CAS:EST64454: σ1R antagonist for pain, high solubility, permeable, BCS class I, metabolically stable.Formula:C18H22F2N4O2Color and Shape:SolidMolecular weight:364.39Lofexidine
CAS:<p>Lofexidine is a selective α2-receptor agonist, Lofexidine reduces narcotic withdrawal symptoms.</p>Formula:C11H12Cl2N2OPurity:98.78%Color and Shape:SolidMolecular weight:259.13[Lys8, Lys9]-Neurotensin (8-13) acetate
[Lys8, Lys9]-Neurotensin (8-13) acetate, a Neurotensin analog, exerts its analgesic effects through activation of the G protein-coupled receptors NTS1 and NTS2Formula:C40H68N8O10Purity:99.31%Color and Shape:SolidMolecular weight:821.02Ref: TM-T38807L
1mg87.00€2mg124.00€5mg187.00€10mg284.00€25mg452.00€50mg645.00€100mg867.00€200mg1,159.00€1mL*10mM (DMSO)To inquireBupranolol HCl
CAS:Bupranolol: non-selective beta blocker, no ISA, strong membrane stabilizer, fast gut absorption, high first-pass metabolism, 2-4hr half-life.Formula:C14H23Cl2NO2Color and Shape:SolidMolecular weight:308.243Sarpogrelate
CAS:Sarpogrelate (MCI-9042), an oral 5-HT2 antagonist, boosts platelet aggregation and aids in studying Buerger's disease.Formula:C24H31NO6Color and Shape:SolidMolecular weight:429.51Maraviroc
CAS:Maraviroc: a CCR5 antagonist blocking HIV-1 entry; IC50s—MIP-1α: 3.3nM, MIP-1β: 7.2nM, RANTES: 5.2nM.Formula:C29H41F2N5OPurity:97.13% - 99.59%Color and Shape:Brown SolidMolecular weight:513.67Ref: TM-T6016
5mg51.00€10mg95.00€25mg160.00€50mg273.00€100mg492.00€200mg633.00€500mg998.00€1mL*10mM (DMSO)59.00€S 38093
CAS:S 38093 is a brain-penetrant antagonist of the H3 receptor (Ki: 8.8/1.44/1.2 μM, for rat/mouse/human).Formula:C17H24N2O2Purity:99.95%Color and Shape:SolidMolecular weight:288.38Ref: TM-T4099
2mg38.00€5mg52.00€10mg80.00€25mg131.00€50mg210.00€100mg334.00€200mg467.00€1mL*10mM (DMSO)52.00€Bepotastine Besilate
CAS:Bepotastine Besilate (TAU 284) is a non-sedating and selective H1 receptor antagonist (pIC50: 5.7).Formula:C21H25ClN2O3·C6H6O3SPurity:99.83% - 99.9%Color and Shape:Brown Viscous LiquidMolecular weight:547.06CYM5442
CAS:CYM5442 is an S1P agonist, targeting to Sphingosine.Formula:C23H27N3O4Purity:98.02% - 99.48%Color and Shape:SolidMolecular weight:409.48L-DOPA methyl ester (hydrochloride)
CAS:<p>L-DOPA methyl ester (LDME) is an agonist of dopamine D1 receptor.</p>Formula:C10H14ClNO4Purity:98.69% - 99.81%Color and Shape:White SolidMolecular weight:247.675SBI-553
CAS:SBI-553 is an effective and brain penetrant NTR1 allosteric modulator (EC50: 0.34 μM).Formula:C26H31FN4O2Purity:99.33%Color and Shape:SolidMolecular weight:450.55
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