GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,024 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,030 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(159 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(443 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(83 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(326 products)
- PAFR(13 products)
- PKA(52 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5968 products of "GPCR/G-Protein"
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BD-1047 dihydrobromide
CAS:BD-1047 dihydrobromide (BD1047.2HBr) , a selective functional antagonist of sigma receptors, has antipsychotic activity in animal models predictive of efficacyFormula:C13H22Br2Cl2N2Purity:98.13% - 99.39%Color and Shape:SolidMolecular weight:437.04Ref: TM-T1740
1mg37.00€2mg48.00€5mg73.00€10mg95.00€25mg168.00€50mg290.00€100mg490.00€1mL*10mM (DMSO)74.00€Sigma-LIGAND-1 hydrochloride
CAS:Sigma-LIGAND-1 HCl: selective sigma receptor ligand; DTG IC50: 16 nM, PPP IC50: 19 nM; weak D2 receptor affinity, Ki: 4000 nM.Formula:C27H34ClNO4Color and Shape:SolidMolecular weight:472.02Hemopressin (rat) acetate(568588-77-2 free base)
Hemopressin is a nonapeptide, CB2 agonist, derived from rat hemoglobin, with antinociceptive properties.Formula:C5H81N13O14Purity:99.37%Color and Shape:SolidMolecular weight:1148.31Phenylbiguanide
CAS:<p>Phenylbiguanide (N-Phenylbiguanide) is a 5-HT3 receptor selective agonist(EC50 : 3.0±0.1 μM)</p>Formula:C8H11N5Purity:99.54%Color and Shape:SolidMolecular weight:177.21Volinanserin
CAS:Volinanserin (MDL100907) is a potent 5-HT2 receptor antagonist with a Ki of 0.36 nM, 300x selective over 5-HT1c, alpha-1, and sigma receptors.Formula:C22H28FNO3Purity:98.94% - 99.95%Color and Shape:SolidMolecular weight:373.46Ref: TM-T5389
1mg42.00€5mg88.00€10mg124.00€25mg233.00€50mg301.00€100mg393.00€200mg560.00€1mL*10mM (DMSO)96.00€Lixisenatide acetate (320367-13-3 free base)
CAS:<p>Lixisenatide acetate is a receptor agonist similar to glucagon-like peptide-1 (glp-1) for the treatment of type 2 diabetes mellitus (T2DM).</p>Formula:C215H347N61O65S·6C2H4O2Purity:98% - 99.9%Color and Shape:SolidMolecular weight:5218.88Enprofylline
CAS:Enprofylline (Enprofilina), a bronchodilator, acts primarily as a competitive nonselective phosphodiesterase inhibitor.Formula:C8H10N4O2Purity:98.37%Color and Shape:SolidMolecular weight:194.19Ref: TM-T21389
2mg44.00€5mg65.00€10mg93.00€25mg149.00€50mg226.00€100mg335.00€200mg465.00€1mL*10mM (DMSO)63.00€Emedastine
CAS:Emedastine (LY188695) is a second generation, selective histamine H1 receptor antagonist with anti-allergic activity.Formula:C17H26N4OPurity:97.1% - 97.76%Color and Shape:OilMolecular weight:302.41Ref: TM-T3979
1mg37.00€5mg79.00€10mg115.00€25mg187.00€50mg279.00€100mg415.00€500mg933.00€1mL*10mM (DMSO)87.00€Naftopidil hydrochloride
CAS:Naftopidil HCl (BM-15275) is a selective alpha1 blocker with Ki: α1a-3.7 nM, α1b-20 nM, α1d-1.2 nM; it also inhibits cell growth.Formula:C24H29ClN2O3Purity:99.5%Color and Shape:SolidMolecular weight:428.95Ref: TM-T9220
1mg44.00€5mg87.00€10mg117.00€25mg202.00€50mg304.00€100mg437.00€200mg612.00€1mL*10mM (DMSO)97.00€Sarpogrelate
CAS:Sarpogrelate (MCI-9042), an oral 5-HT2 antagonist, boosts platelet aggregation and aids in studying Buerger's disease.Formula:C24H31NO6Color and Shape:SolidMolecular weight:429.51Niaprazine
CAS:<p>Niaprazine is a histamine H1-receptor antagonist with marked sedative properties.</p>Formula:C20H25FN4OPurity:99.56%Color and Shape:SolidMolecular weight:356.44Neurokinin A
CAS:Neurokinin A (NKA), formerly known as Substance K, is a neurologically active peptide translated from the pre-protachykinin gene.Formula:C50H80N14O14SPurity:>99.99%Color and Shape:White To Off-White Lyophilized SolidMolecular weight:1133.32Exendin-4
CAS:<p>Exenatide: GLP-1 receptor agonist, 39-amino acid, longer half-life (2.4 hrs), IC50 of 3.22 nM.</p>Formula:C184H282N50O60SPurity:97.71% - 99.78%Color and Shape:SolidMolecular weight:4186.57Nelociguat
CAS:<p>Nelociguat (BAY60-4552) is an sGC stimulator, crucial in NO signal pathways.</p>Formula:C19H17FN8O2Purity:99.19%Color and Shape:SolidMolecular weight:408.39Nefazodone hydrochloride
CAS:Nefazodone hydrochloride (Serzone) is a serotoninergic modulating antidepressant that is used in therapy of depression, aggressive behavior and panic disorder.Formula:C25H33Cl2N5O2Purity:99% - 99.86%Color and Shape:White SolidMolecular weight:506.47Ref: TM-T3275
5mg47.00€10mg70.00€25mg120.00€50mg216.00€100mg325.00€200mg472.00€500mg775.00€1mL*10mM (DMSO)77.00€TY-52156
CAS:TY-52156 is an effective and selective S1P3 receptor antagonist (Ki: 110 nM).Formula:C18H19Cl2N3OPurity:99.91% - 99.91%Color and Shape:SolidMolecular weight:364.27Ref: TM-T17183
2mg40.00€5mg60.00€10mg87.00€25mg166.00€50mg298.00€100mg510.00€200mg683.00€1mL*10mM (DMSO)66.00€Metoclopramide hydrochloride hydrate
CAS:Metoclopramide hydrochloride hydrate (Metoclopramide monohydrochloride monohydrate) is a dopamine D2 antagonist that is a drug used for digestive dysfunction.Formula:C14H25Cl2N3O3Purity:99.33%Color and Shape:SolidMolecular weight:354.27Darusentan
CAS:Darusentan (Lu-135252) is a potent inhibitor of endothelin signaling and function in both large and small arteriesFormula:C22H22N2O6Purity:98.72%Color and Shape:SolidMolecular weight:410.43Ref: TM-T5458
2mg46.00€5mg69.00€10mg105.00€25mg183.00€50mg304.00€100mg437.00€200mg615.00€1mL*10mM (DMSO)71.00€Rizatriptan benzoate
CAS:Rizatriptan benzoate (MK-462 Benzoate) selectively binds to and activates serotonin (5-HT) 1B receptors and 5-HT 1D receptors providing relief of migraineFormula:C22H25N5O2Purity:99% - 99.79%Color and Shape:White To Off-White Crystalline PowderMolecular weight:391.47Ref: TM-T1512
10mg47.00€25mg79.00€50mg126.00€100mg183.00€200mg273.00€500mg462.00€1mL*10mM (DMSO)50.00€CGP 71683 (free base)
CAS:CGP 71683 (free base) is a potent and highly selective non-peptide antagonist of the NPY Y(5) receptor in the study of obesity.Formula:C26H29N5O2SColor and Shape:SolidMolecular weight:475.61
