GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,024 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,030 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(159 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(443 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(83 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(326 products)
- PAFR(13 products)
- PKA(52 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5968 products of "GPCR/G-Protein"
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Darbufelone mesylate
CAS:Darbufelone mesylate blocks PGF2α, LTB4, PGHS-2 (IC50: 0.19 μM), and PGHS-1 (IC50: 20 μM).Formula:C19H28N2O5S2Purity:96.81% - 99.92%Color and Shape:SolidMolecular weight:428.57Ref: TM-T10960L
1mg49.00€5mg104.00€10mg170.00€25mg359.00€50mg587.00€100mg835.00€200mg1,121.00€1mL*10mM (DMSO)115.00€Reboxetine mesylate
CAS:<p>Reboxetine mesylate (FCE20124 mesylate) is a norepinephrine reuptake inhibitor (Ki: 8.2 nM).</p>Formula:C19H23NO3·CH4O3SPurity:99.18% - 99.87%Color and Shape:Tan Or Off-White Cyrstalline SolidMolecular weight:409.5Anisotropine Methylbromide
CAS:Anisotropine Methylbromide is an anticholinergic agent and has been used for relief of gastrointestinal spasm and for the suppression of gastric acid secretion.Formula:C17H32BrNO2Purity:99.73%Color and Shape:Crystals From Acetone SolidMolecular weight:362.35ABT-702 dihydrochloride
CAS:ABT-702 dihydrochloride is a potent adenosine kinase (AK) inhibitor.Formula:C22H21BrCl2N6OPurity:98.42% - 98.98%Color and Shape:SolidMolecular weight:536.25Ref: TM-T4668
1mg62.00€2mg87.00€5mg119.00€10mg187.00€25mg350.00€50mg530.00€100mg748.00€500mg1,578.00€1mL*10mM (DMSO)140.00€Cloprostenol sodium salt
CAS:Cloprostenol sodium salt (ICI 80996 sodium salt) is a synthetic prostaglandin analogue, an agonist at the PGF2α receptor, with luteolytic properties.Formula:C22H28ClNaO6Purity:97.17% - 98.47%Color and Shape:White To Almost White Hygroscopic PowderMolecular weight:446.9[D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate
Broad-spectrum neuropeptide inverse agonist/antagonist; potent at ghrelin receptor (EC50 = 5.2 nM); inhibits cancer growth, induces apoptosis.Formula:C81H113N19O14Purity:97.68%Color and Shape:SolidMolecular weight:1576.91[D-Trp8]-γ-MSH acetate(321351-81-9 free base)
[D-Trp8]-γ-MSH acetate(321351-81-9 free base) is a selective melanocortin 3 (MC3) receptor agonist (IC50 values are 6.7, 340 and 600 nM for human MC3, MC5 andFormula:C76H103N21O18SPurity:99.75%Color and Shape:SolidMolecular weight:1630.82Alprenolol benzoate
CAS:Alprenolol benzoate is the benzoate salt of Alprenolol -- a beta blocker.Formula:C22H29NO4Color and Shape:SolidMolecular weight:371.48TG4-155
CAS:<p>TG4-155: brain-penetrant EP2 inhibitor, KB 2.4 nM; >1000x weaker at EP4, KB 11.4 μM; selective over other receptors/channels.</p>Formula:C23H26N2O4Purity:97.2%Color and Shape:SolidMolecular weight:394.46Parmodulin 2
CAS:ML161 (Parmodulin 2) inhibits PAR1, blocking platelet activation and thrombin-induced activity (IC50: 0.26μM).Formula:C17H17BrN2O2Purity:97.35% - 99.95%Color and Shape:SolidMolecular weight:361.23Derenofylline
CAS:Derenofylline is a selective and potent adenosine A(1) antagonist in vitro (Ki=1 nM)Formula:C18H20N4OPurity:98.09%Color and Shape:SolidMolecular weight:308.38NNC-0640
CAS:NNC-0640 is a negative allosteric modulator of Human Glucagon Receptor with an IC50 of 69.2 nM.Formula:C29H31N7O4SPurity:97.04%Color and Shape:SolidMolecular weight:573.67Ref: TM-T7364
1mg48.00€2mg65.00€5mg96.00€10mg169.00€25mg298.00€50mg454.00€100mg655.00€1mL*10mM (DMSO)96.00€Alcaftadine
CAS:Alcaftadine (Lastacaft) is an H1 histamine receptor antagonist indicated for the prevention of itching associated with allergic conjunctivitis.Formula:C19H21N3OPurity:98% - 98.65%Color and Shape:SolidMolecular weight:307.39PRX-08066
CAS:PRX-08066 is a selective 5-hydroxytryptamine receptor 2B (5-HT2BR, IC50= 3.4 nM) antagonist that induces selective vasodilation of pulmonary arteries.Formula:C19H17ClFN5SPurity:97.79% - 98.07%Color and Shape:SolidMolecular weight:401.89Ref: TM-T16669
1mg60.00€5mg119.00€10mg170.00€25mg350.00€50mg522.00€100mg748.00€200mg1,026.00€1mL*10mM (DMSO)111.00€Diquafosol tetrasodium
CAS:Diquafosol Tetrasodium is a P2Y2 receptor agonist that stimulates the secretion of mucins from ocular tissues Diquafosol tetrasodium (INS365) improves tear filmFormula:C18H22N4Na4O23P4Purity:98.25% - 99.97%Color and Shape:SolidMolecular weight:878.23Zacopride hydrochloride
CAS:Zacopride is a highly potent 5-HT3 receptor antagonist (Kd = 0.38 nM) and 5-HT4 receptor agonist (Ki = 373 nM). It also is a selective IK1 channel agonist.Formula:C15H20ClN3O2·HClPurity:98.32%Color and Shape:SolidMolecular weight:346.26Ref: TM-T5336
1mg35.00€5mg74.00€10mg104.00€25mg224.00€50mg406.00€100mg652.00€200mg908.00€1mL*10mM (DMSO)84.00€Antalarmin
CAS:Antalarmin is a CRHR1 antagonist that blocks adrenocorticotropin-releasing hormone-induced hypertension, blocks CRF activation.Formula:C24H34N4Purity:99.99%Color and Shape:SolidMolecular weight:378.55Ref: TM-T70433
1mg86.00€5mg173.00€10mg255.00€25mg430.00€50mg582.00€100mg787.00€1mL*10mM (DMSO)183.00€Xaliproden hydrochloride
CAS:Xaliproden is a compound that mimics the effects of nerve growth factor and is also a serotonin 5-HT1A receptor agonist.Formula:C24H23ClF3NPurity:99.99%Color and Shape:SolidMolecular weight:417.89Ref: TM-T9272
1mg40.00€5mg85.00€10mg120.00€25mg235.00€50mg376.00€100mg540.00€200mg775.00€1mL*10mM (DMSO)96.00€[Lys8, Lys9]-Neurotensin (8-13) acetate
[Lys8, Lys9]-Neurotensin (8-13) acetate, a Neurotensin analog, exerts its analgesic effects through activation of the G protein-coupled receptors NTS1 and NTS2Formula:C40H68N8O10Purity:99.31%Color and Shape:SolidMolecular weight:821.02Ref: TM-T38807L
1mg87.00€2mg124.00€5mg187.00€10mg284.00€25mg452.00€50mg645.00€100mg867.00€200mg1,159.00€1mL*10mM (DMSO)To inquireVelneperit
CAS:Velneperit (S2367) is potent and selective neuropeptide Y (NPY) Y5 receptor under evaluating for treatment of obesity.Formula:C17H24F3N3O3SPurity:99.70%Color and Shape:SolidMolecular weight:407.45Ref: TM-T17222
1mg37.00€2mg52.00€5mg79.00€10mg119.00€25mg259.00€50mg439.00€100mg647.00€1mL*10mM (DMSO)87.00€
![[D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FTP1931L1.webp&w=3840&q=75)
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