
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,024 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,030 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(159 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(443 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(83 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(326 products)
- PAFR(13 products)
- PKA(52 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5968 products of "GPCR/G-Protein"
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GW627368
CAS:GW627368 (GW 627368X)X is a novel, potent and selective antagonist of prostanoid EP4 receptor.Formula:C30H28N2O6SPurity:99.75% - 99.92%Color and Shape:SolidMolecular weight:544.62N-Cbz-DL-tryptophan
CAS:N-Cbz-DL-tryptophan is a cholecystokinin receptor antagonist, abolished the response of the isolated heart to CCK-8.Formula:C19H18N2O4Purity:99.97%Color and Shape:SolidMolecular weight:338.36β-CGRP, human acetate
β-CGRP, human acetate is one of calcitonin peptides and acts via the complex of receptor-activity-modifying protein (RAMP) and calcitonin-receptor-like receptorFormula:C164H271N51O50S3Purity:99.35%Color and Shape:SolidMolecular weight:3853.46nifenalol.HCl
CAS:Nifenalol.HCl(INPEA) is a antagonist of β-adrenergic receptor.Formula:C11H17ClN2O3Purity:99.96%Color and Shape:SolidMolecular weight:260.72Deslorelin acetate(57773-65-6 free base)
Deslorelin acetate(57773-65-6 free base) is a gonadotropin releasing hormone super-agonist (GnRH agonist)Formula:C66H87N17O14Purity:99.84%Color and Shape:SolidMolecular weight:1342.5Tetracosactide acetate
CAS:Cosyntropin (acetate) stimulates the release of corticosteroids such as cortisol from the adrenal gland.Formula:C138H214N40O33SPurity:99.76%Color and Shape:SolidMolecular weight:2993.54I-191
CAS:I-191 is a potent antagonist of protease-activated receptor 2 (PAR2), inhibits multiple signaling functions in human cancer cells.Formula:C23H26FN5O2Purity:99.8%Color and Shape:SolidMolecular weight:423.48Ref: TM-T7137
1mg89.00€2mg116.00€5mg188.00€10mg284.00€25mg474.00€50mg688.00€100mg938.00€1mL*10mM (DMSO)210.00€ML 10302
CAS:ML 10302 is a potent 5-HT4 agonist with Ki of 1.07 nM, boosts bowel movement, and may aid in neurology research.Formula:C15H21ClN2O3Color and Shape:SolidMolecular weight:312.79AM211
CAS:AM211 (AM211 free acid) is a potent and orally bioavailable antagonist of prostaglandin D2 (PGD2) receptor type 2 (DP2)Formula:C27H27F3N2O4Purity:≥95%Color and Shape:SolidMolecular weight:500.51CYM-5520
CAS:CYM-5520 is a noncompetitive allosteric agonist of S1P2Formula:C21H19N3O2Purity:99.47%Color and Shape:SolidMolecular weight:345.39Ref: TM-T22703
1mg48.00€2mg64.00€5mg94.00€10mg142.00€25mg250.00€50mg374.00€100mg557.00€1mL*10mM (DMSO)103.00€GLPG2938
CAS:GLPG2938 (1-(2-Ethoxy-6-(trifluoromethyl)pyridin-4-yl)-3-((5-methyl-6-(1-methyl-3-(trifluoromethyl)-1H-pyrazol-4-yl)pyridazin-3-yl)methyl)urea) is a potent andFormula:C20H19F6N7O2Purity:98.25%Color and Shape:SolidMolecular weight:503.4Ref: TM-T9199
1mg84.00€2mgTo inquire5mg144.00€10mg250.00€25mg550.00€50mg792.00€100mg1,093.00€1mL*10mM (DMSO)160.00€Dioxopromethazine hydrochloride
CAS:Dioxopromethazine is a target-based classification of drug and available in a number of countries worldwide.Formula:C17H20N2O2S·HClPurity:99.58%Color and Shape:SolidMolecular weight:352.88ELA-11 (human) acetate(1784687-32-6 free base)
ELA-11: potent apelin receptor agonist, Ki=14 nM. Blocks cAMP, boosts β-arrestin. Part of ELA-32.Formula:C60H94N16O15S2Purity:99.53%Color and Shape:SolidMolecular weight:1343.61Prucalopride Succinate
CAS:Prucalopride Succinate is a 5-HT4 receptor agonist with Ki 2.5 nM (5-HT4a) and 8 nM (5-HT4b).Formula:C18H26ClN3O3·C4H6O4Purity:99.24%Color and Shape:SolidMolecular weight:485.96Dazoxiben
CAS:<p>Dazoxiben (UK-37248) is a potent inhibitor of thromboxane (TX) synthase</p>Formula:C12H13ClN2O3Purity:99.99%Color and Shape:SolidMolecular weight:268.7TRAP-6
CAS:<p>TRAP-6 (Thrombin Receptor Activator Peptide 6)(2TFA) is an agonist of protease-activated receptor 1 (PAR1).</p>Formula:C34H56N10O9Purity:>99.99%Color and Shape:SolidMolecular weight:748.87CAY10444
CAS:CAY10444 is an S1P3 specific antagonist.Formula:C15H29NO2SPurity:99.15% - 99.61%Color and Shape:SolidMolecular weight:287.46Ref: TM-T23860
5mg47.00€10mg74.00€25mg144.00€50mg235.00€100mg393.00€200mg532.00€500mg838.00€1mL*10mM (DMSO)50.00€Antazoline
CAS:Antazoline has antihistamine and anticholinergic effects.It used to treat a variety of arrhythmias.Formula:C17H19N3Purity:≥95%Color and Shape:White Crystalline Powder SolidMolecular weight:265.35Blarcamesine hydrochloride
CAS:Blarcamesine hydrochloride (AVex-73 hydrochloride) is a Sigma-1 Receptor agonist (IC50: 860 nM).Formula:C19H24ClNOPurity:99.57% - 99.9%Color and Shape:SolidMolecular weight:317.85Ref: TM-T4111
1mg35.00€2mg48.00€5mg70.00€10mg104.00€25mg207.00€50mg359.00€100mg588.00€200mg833.00€1mL*10mM (DMSO)78.00€Hydroxyzine
CAS:Hydroxyzine (Hydroxyzine free base) is an antagonist of histamine H1-receptor.Formula:C21H27ClN2O2Purity:99.54% - ≥95%Color and Shape:Oil SolidMolecular weight:374.9
