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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5968 products of "GPCR/G-Protein"

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  • GW627368

    CAS:
    GW627368 (GW 627368X)X is a novel, potent and selective antagonist of prostanoid EP4 receptor.
    Formula:C30H28N2O6S
    Purity:99.75% - 99.92%
    Color and Shape:Solid
    Molecular weight:544.62

    Ref: TM-T1978

    2mg
    35.00€
    5mg
    52.00€
    10mg
    87.00€
    25mg
    131.00€
    50mg
    215.00€
    100mg
    378.00€
    1mL*10mM (DMSO)
    64.00€
  • N-Cbz-DL-tryptophan

    CAS:
    N-Cbz-DL-tryptophan is a cholecystokinin receptor antagonist, abolished the response of the isolated heart to CCK-8.
    Formula:C19H18N2O4
    Purity:99.97%
    Color and Shape:Solid
    Molecular weight:338.36

    Ref: TM-T9343

    25mg
    48.00€
    50mg
    67.00€
    100mg
    88.00€
    500mg
    212.00€
    1mL*10mM (DMSO)
    34.00€
  • β-CGRP, human acetate


    β-CGRP, human acetate is one of calcitonin peptides and acts via the complex of receptor-activity-modifying protein (RAMP) and calcitonin-receptor-like receptor
    Formula:C164H271N51O50S3
    Purity:99.35%
    Color and Shape:Solid
    Molecular weight:3853.46

    Ref: TM-TP2167

    1mg
    363.00€
    5mg
    817.00€
    10mg
    1,121.00€
    25mg
    1,673.00€
    50mg
    2,252.00€
    100mg
    3,022.00€
  • nifenalol.HCl

    CAS:
    Nifenalol.HCl(INPEA) is a antagonist of β-adrenergic receptor.
    Formula:C11H17ClN2O3
    Purity:99.96%
    Color and Shape:Solid
    Molecular weight:260.72

    Ref: TM-T8663

    25mg
    44.00€
    50mg
    66.00€
    1mL*10mM (DMSO)
    34.00€
  • Deslorelin acetate(57773-65-6 free base)


    Deslorelin acetate(57773-65-6 free base) is a gonadotropin releasing hormone super-agonist (GnRH agonist)
    Formula:C66H87N17O14
    Purity:99.84%
    Color and Shape:Solid
    Molecular weight:1342.5

    Ref: TM-TP2323L

    1mg
    93.00€
    2mg
    119.00€
    5mg
    168.00€
    10mg
    227.00€
    25mg
    409.00€
    50mg
    605.00€
    100mg
    842.00€
  • Tetracosactide acetate

    CAS:
    Cosyntropin (acetate) stimulates the release of corticosteroids such as cortisol from the adrenal gland.
    Formula:C138H214N40O33S
    Purity:99.76%
    Color and Shape:Solid
    Molecular weight:2993.54

    Ref: TM-T35664

    1mg
    55.00€
    5mg
    116.00€
    10mg
    183.00€
    25mg
    311.00€
    50mg
    449.00€
    100mg
    615.00€
    200mg
    830.00€
  • I-191

    CAS:
    I-191 is a potent antagonist of protease-activated receptor 2 (PAR2), inhibits multiple signaling functions in human cancer cells.
    Formula:C23H26FN5O2
    Purity:99.8%
    Color and Shape:Solid
    Molecular weight:423.48

    Ref: TM-T7137

    1mg
    89.00€
    2mg
    116.00€
    5mg
    188.00€
    10mg
    284.00€
    25mg
    474.00€
    50mg
    688.00€
    100mg
    938.00€
    1mL*10mM (DMSO)
    210.00€
  • ML 10302

    CAS:
    ML 10302 is a potent 5-HT4 agonist with Ki of 1.07 nM, boosts bowel movement, and may aid in neurology research.
    Formula:C15H21ClN2O3
    Color and Shape:Solid
    Molecular weight:312.79

    Ref: TM-T60787

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • AM211

    CAS:
    AM211 (AM211 free acid) is a potent and orally bioavailable antagonist of prostaglandin D2 (PGD2) receptor type 2 (DP2)
    Formula:C27H27F3N2O4
    Purity:≥95%
    Color and Shape:Solid
    Molecular weight:500.51

    Ref: TM-T7652

    1mg
    37.00€
    5mg
    79.00€
    10mg
    119.00€
    25mg
    235.00€
    50mg
    359.00€
    100mg
    532.00€
    1mL*10mM (DMSO)
    87.00€
  • CYM-5520

    CAS:
    CYM-5520 is a noncompetitive allosteric agonist of S1P2
    Formula:C21H19N3O2
    Purity:99.47%
    Color and Shape:Solid
    Molecular weight:345.39

    Ref: TM-T22703

    1mg
    48.00€
    2mg
    64.00€
    5mg
    94.00€
    10mg
    142.00€
    25mg
    250.00€
    50mg
    374.00€
    100mg
    557.00€
    1mL*10mM (DMSO)
    103.00€
  • GLPG2938

    CAS:
    GLPG2938 (1-(2-Ethoxy-6-(trifluoromethyl)pyridin-4-yl)-3-((5-methyl-6-(1-methyl-3-(trifluoromethyl)-1H-pyrazol-4-yl)pyridazin-3-yl)methyl)urea) is a potent and
    Formula:C20H19F6N7O2
    Purity:98.25%
    Color and Shape:Solid
    Molecular weight:503.4

    Ref: TM-T9199

    1mg
    84.00€
    2mg
    To inquire
    5mg
    144.00€
    10mg
    250.00€
    25mg
    550.00€
    50mg
    792.00€
    100mg
    1,093.00€
    1mL*10mM (DMSO)
    160.00€
  • Dioxopromethazine hydrochloride

    CAS:
    Dioxopromethazine is a target-based classification of drug and available in a number of countries worldwide.
    Formula:C17H20N2O2S·HCl
    Purity:99.58%
    Color and Shape:Solid
    Molecular weight:352.88

    Ref: TM-T3723

    25mg
    35.00€
    50mg
    52.00€
    100mg
    88.00€
    500mg
    233.00€
    1mL*10mM (DMSO)
    34.00€
  • ELA-11 (human) acetate(1784687-32-6 free base)


    ELA-11: potent apelin receptor agonist, Ki=14 nM. Blocks cAMP, boosts β-arrestin. Part of ELA-32.
    Formula:C60H94N16O15S2
    Purity:99.53%
    Color and Shape:Solid
    Molecular weight:1343.61

    Ref: TM-TP1922L1

    1mg
    131.00€
    5mg
    286.00€
    10mg
    430.00€
    25mg
    710.00€
    50mg
    998.00€
    100mg
    1,349.00€
  • Prucalopride Succinate

    CAS:
    Prucalopride Succinate is a 5-HT4 receptor agonist with Ki 2.5 nM (5-HT4a) and 8 nM (5-HT4b).
    Formula:C18H26ClN3O3·C4H6O4
    Purity:99.24%
    Color and Shape:Solid
    Molecular weight:485.96

    Ref: TM-T6958

    10mg
    46.00€
    25mg
    55.00€
    50mg
    74.00€
    100mg
    111.00€
    1mL*10mM (DMSO)
    35.00€
  • Dazoxiben

    CAS:
    <p>Dazoxiben (UK-37248) is a potent inhibitor of thromboxane (TX) synthase</p>
    Formula:C12H13ClN2O3
    Purity:99.99%
    Color and Shape:Solid
    Molecular weight:268.7

    Ref: TM-T7968

    1mg
    38.00€
    2mg
    49.00€
    5mg
    80.00€
    10mg
    127.00€
    25mg
    250.00€
    50mg
    369.00€
    100mg
    512.00€
    500mg
    1,093.00€
  • TRAP-6

    CAS:
    <p>TRAP-6 (Thrombin Receptor Activator Peptide 6)(2TFA) is an agonist of protease-activated receptor 1 (PAR1).</p>
    Formula:C34H56N10O9
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:748.87

    Ref: TM-T7625

    1mg
    40.00€
    2mg
    52.00€
    5mg
    88.00€
    10mg
    126.00€
    25mg
    274.00€
    50mg
    411.00€
    100mg
    597.00€
  • CAY10444

    CAS:
    CAY10444 is an S1P3 specific antagonist.
    Formula:C15H29NO2S
    Purity:99.15% - 99.61%
    Color and Shape:Solid
    Molecular weight:287.46

    Ref: TM-T23860

    5mg
    47.00€
    10mg
    74.00€
    25mg
    144.00€
    50mg
    235.00€
    100mg
    393.00€
    200mg
    532.00€
    500mg
    838.00€
    1mL*10mM (DMSO)
    50.00€
  • Antazoline

    CAS:
    Antazoline has antihistamine and anticholinergic effects.It used to treat a variety of arrhythmias.
    Formula:C17H19N3
    Purity:≥95%
    Color and Shape:White Crystalline Powder Solid
    Molecular weight:265.35

    Ref: TM-T7477

    10mg
    47.00€
    25mg
    67.00€
    50mg
    89.00€
    100mg
    131.00€
    1mL*10mM (DMSO)
    47.00€
  • Blarcamesine hydrochloride

    CAS:
    Blarcamesine hydrochloride (AVex-73 hydrochloride) is a Sigma-1 Receptor agonist (IC50: 860 nM).
    Formula:C19H24ClNO
    Purity:99.57% - 99.9%
    Color and Shape:Solid
    Molecular weight:317.85

    Ref: TM-T4111

    1mg
    35.00€
    2mg
    48.00€
    5mg
    70.00€
    10mg
    104.00€
    25mg
    207.00€
    50mg
    359.00€
    100mg
    588.00€
    200mg
    833.00€
    1mL*10mM (DMSO)
    78.00€
  • Hydroxyzine

    CAS:
    Hydroxyzine (Hydroxyzine free base) is an antagonist of histamine H1-receptor.
    Formula:C21H27ClN2O2
    Purity:99.54% - ≥95%
    Color and Shape:Oil Solid
    Molecular weight:374.9

    Ref: TM-T20884

    50mg
    43.00€
    1mL*10mM (DMSO)
    47.00€