GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,024 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,029 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(159 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(443 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(83 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(42 products)
- Opioid Receptor(326 products)
- PAFR(14 products)
- PKA(52 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5972 products of "GPCR/G-Protein"
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RE-640
CAS:NSC-5844 (RE-640) (RE640) is a bisquinoline compound with C-C chemokine receptor type 1 (CCR1)-agonistic activities.Formula:C20H16Cl2N4Purity:99.60% - 99.87%Color and Shape:SolidMolecular weight:383.27Hydroxyzine
CAS:Hydroxyzine (Hydroxyzine free base) is an antagonist of histamine H1-receptor.Formula:C21H27ClN2O2Purity:99.54% - ≥95%Color and Shape:Oil SolidMolecular weight:374.9GUANABENZ
CAS:GUANABENZ is a Central alpha-2 Adrenergic Agonist. The mechanism of action of guanabenz is as an Adrenergic alpha2-Agonist.Formula:C8H8Cl2N4Purity:98.31%Color and Shape:White Solid From Acetonitrile SolidMolecular weight:231.08Zuclopenthixol
CAS:<p>Zuclopenthixol (cis-Clopenthixol) is a thioxanthene with therapeutic actions similar to the phenothiazine antipsychotics.</p>Formula:C22H25ClN2OSPurity:98.9% - 99.82%Color and Shape:SolidMolecular weight:400.96HS 014 acetate(207678-81-7 free base)
HS 014 acetate is a potent MC4R antagonist with Ki: 3.16 nM (MC4), and boosts food intake and nociception in animals.Formula:C73H98N20O19S2Purity:>99.99%Color and Shape:SolidMolecular weight:1623.83BQ-788 sodium salt
CAS:BQ-788 sodium salt is a potent and selective antagonist of ETB receptor(ETB receptors with an IC50 of 1.2 nM in human Girrardi heart cells).Formula:C34H51N5NaO7Color and Shape:SolidMolecular weight:664.8Takeda103A
CAS:Takeda103A (CMPD103A) is the GRK2-dependent bovine tubulin oxidation effective inhibitor.Formula:C24H23F2N7OPurity:97.17%Color and Shape:SolidMolecular weight:463.48Ref: TM-T24850
1mg85.00€2mg105.00€5mg164.00€10mg258.00€25mg424.00€50mg562.00€100mg787.00€200mg1,035.00€1mL*10mM (DMSO)187.00€CS 2100
CAS:<p>CS 2100 (1-[[4-Ethyl-5-[5-(4-phenoxyphenyl)-1,2,4-oxadiazol-3-yl]-2-thienyl]methyl]-3-azetidinecarboxylic acid) is an S1P1 agonist.</p>Formula:C25H23N3O4SPurity:99.19%Color and Shape:SolidMolecular weight:461.53SB 242084
CAS:SB 242084 dihydrochloride hydrate is a psychoactive drug and research chemical which acts as a selective antagonist for the 5HT2C receptor.Formula:C21H19ClN4O2Purity:99.75% - ≥98%Color and Shape:SolidMolecular weight:394.85Diphenhydramine
CAS:Diphenhydramine (Syntedril): first-gen antihistamine for allergies, antiemetic, antitussive, anticholinergic, sedative, treats drug-induced parkinsonism.Formula:C17H21NOPurity:98.07%Color and Shape:SolidMolecular weight:255.35Alimemazine hemitartrate
CAS:Alimemazine hemitartrate (Trimeprazine hemitartrate) is aphenothiazine derivative that is used as an antipruritic.Formula:C18H22N2SC4H6O6Purity:98.16% - 99.69%Color and Shape:SolidMolecular weight:448.536-fluoro-DL-Tryptophan
CAS:6-fluoro-DL-Tryptophan is an inhibitor of serotonin (5-HT) synthesis.Formula:C11H11FN2O2Purity:99.25%Color and Shape:Off-White PowderMolecular weight:222.22Pemirolast
CAS:Pemirolast: oral antiallergic, reduces paclitaxel reactions, inhibits neuropeptides, for asthma and conjunctivitis study.Formula:C10H8N6OColor and Shape:SolidMolecular weight:228.21AnaMorelin hydrochloride
CAS:AnaMorelin hydrochloride (RC-1291 hydrochloride) is a novel ghrelin receptor agonist(EC50 : 0.74 nM, in the FLIPR assay).Formula:C31H43ClN6O3Purity:99.18% - ≥98%Color and Shape:SolidMolecular weight:583.16Ref: TM-T7225
1mg35.00€2mg50.00€5mg73.00€10mg96.00€25mg145.00€50mg177.00€100mg235.00€1mL*10mM (DMSO)95.00€Atrasentan sodium
CAS:Atrasentan (ABT-627) is an oral ETA receptor blocker with potential cancer-fighting properties, inhibiting angiogenesis and tumor growth.Formula:C29H37N2NaO6Color and Shape:SolidMolecular weight:532.61Exo1
CAS:Exo1 is an inhibitor of the exocytic pathwayFormula:C15H12FNO3Purity:98.75%Color and Shape:SolidMolecular weight:273.26Neurokinin A
CAS:Neurokinin A (NKA), formerly known as Substance K, is a neurologically active peptide translated from the pre-protachykinin gene.Formula:C50H80N14O14SPurity:>99.99%Color and Shape:White To Off-White Lyophilized SolidMolecular weight:1133.32Dexmedetomidine
CAS:Dexmedetomidine: a central alpha-2 adrenergic agonist for general anesthesia.Formula:C13H16N2Purity:99% - >99.99%Color and Shape:SolidMolecular weight:200.28Nafarelin acetate(76932-56-4 free base)
CAS:Nafarelin acetate (76932-56-4) is a GnRH analog that reduces LH and FSH release, used for estrogen-related treatments.Formula:C68H87N17O15Purity:99.98%Color and Shape:SolidMolecular weight:1382.55HAEGTFTSDVSSYLE
<p>HAEGTFTSDVSSYLE is a peptide. GLP-I analog contains the sequence.</p>Formula:C71H103N17O28Purity:>99.99%Color and Shape:SolidMolecular weight:1642.71
