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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5965 products of "GPCR/G-Protein"

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  • Conivaptan hydrochloride
    Targetmol
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    Conivaptan hydrochloride

    CAS:
    <p>Conivaptan hydrochloride (Vaprisol) is an orally active vasopressin V2 and V1A receptor antagonist, used in the therapy of hypervolemic hyponatremia and</p>
    Formula:C32H26N4O2·HCl
    Purity:98.33% - 99.86%
    Color and Shape:Solid
    Molecular weight:535.04

    Ref: TM-T6453

  • 1-[(5-methylisoxazol-3-yl)methyl]piperazine
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    1-[(5-methylisoxazol-3-yl)methyl]piperazine

    CAS:
    <p>1-[(5-methylisoxazol-3-yl)methyl]piperazine (Piperazine, 1-[(5-methyl-3-isoxazolyl)methyl]- (9CI)) is a P2Y12 inhibitor.</p>
    Formula:C9H15N3O
    Purity:95%
    Color and Shape:Solid
    Molecular weight:181.23

    Ref: TM-T8582

  • DAPTA
    Targetmol
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    DAPTA

    CAS:
    DAPTA (Adaptavir) is an inhibitor of CCR5, shows potent anti-HIV activities.
    Formula:C35H56N10O15
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:856.88

    Ref: TM-T7624

  • Sertindole
    Targetmol
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    Sertindole

    CAS:
    <p>Sertindole, atypical antipsychotic, targets D2, 5-HT1D, 5-HT2A, 5-HT2C receptors (Kds: 2.7, 20, 0.14, 6 nM).</p>
    Formula:C24H26ClFN4O
    Purity:99.87% - 99.92%
    Color and Shape:Off-White To Pale Yellow Solid
    Molecular weight:440.94

    Ref: TM-T5858

  • Midodrine
    Targetmol
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    Midodrine

    CAS:
    Midodrine ((±)-Midodrin), an adrenergic alpha-1 agonist, belongs to the class of medications known as vasopressors.
    Formula:C12H18N2O4
    Purity:99.89%
    Color and Shape:Solid
    Molecular weight:254.28

    Ref: TM-T22369

  • Perospirone
    Targetmol
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    Perospirone

    CAS:
    Perospirone (Lullan) is an antagonist of serotonin 5HT2A receptors and dopamine D2 receptors.
    Formula:C23H30N4O2S
    Purity:99.23%
    Color and Shape:White Powder
    Molecular weight:426.57

    Ref: TM-T4576

  • RU 24969 succinate
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    RU 24969 succinate

    CAS:
    <p>RU 24969 succinate, a 5-HT receptor agonist, exhibits K i values of 0.38 nM for 5-HT 1B and 2.5 nM for 5-HT 1A, indicating its affinity towards these receptors. It reduces fluid consumption and enhances forward locomotion. This compound is utilized in neurological disease research.</p>
    Formula:C18H22N2O5
    Color and Shape:Solid
    Molecular weight:346.38

    Ref: TM-T71502

  • Ro 46-2005
    Targetmol
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    Ro 46-2005

    CAS:
    Ro 46-2005: Synthetic non-peptide, blocks 125I-ET-1 at ETA receptors on human vascular cells (IC50: 220 nM).
    Formula:C23H27N3O6S
    Purity:98.02% - 98.8%
    Color and Shape:Solid
    Molecular weight:473.54

    Ref: TM-T3194

  • Tetradecyl Phosphonate
    Targetmol
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    Tetradecyl Phosphonate

    CAS:
    Tetradecyl Phosphonate 是溶血磷脂酸 1 (LPA1)、LPA2 和 LPA3 受体的泛拮抗剂。
    Formula:C14H31O3P
    Purity:99.95%
    Color and Shape:White To Off-White Powder
    Molecular weight:278.37

    Ref: TM-T7689

  • CGP71683 hydrochloride
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    CGP71683 hydrochloride

    CAS:
    CGP71683 hydrochloride: NPY5 receptor antagonist, Ki=1.3 nM; inactive at Y1 (Ki >4000 nM) and Y2 (Ki=200 nM).
    Formula:C26H30ClN5O2S
    Purity:99.92%
    Color and Shape:Solid
    Molecular weight:512.07

    Ref: TM-T5587

  • GLPG2938
    Targetmol
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    GLPG2938

    CAS:
    GLPG2938 (1-(2-Ethoxy-6-(trifluoromethyl)pyridin-4-yl)-3-((5-methyl-6-(1-methyl-3-(trifluoromethyl)-1H-pyrazol-4-yl)pyridazin-3-yl)methyl)urea) is a potent and
    Formula:C20H19F6N7O2
    Purity:98.25%
    Color and Shape:Solid
    Molecular weight:503.4

    Ref: TM-T9199

  • SORT-PGRN interaction inhibitor 1
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    SORT-PGRN interaction inhibitor 1

    CAS:
    SORT-PGRN interaction inhibitor 1 is a potent sortilin-progranulin interaction inhibitor(IC50 of 2 μM).
    Formula:C15H18N2O2
    Purity:98.72%
    Color and Shape:Solid
    Molecular weight:258.32

    Ref: TM-T9044

  • 4i
    Targetmol
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    4i

    CAS:
    4i (CHEMBL1269981) is a 5-HT3 receptor antagonist,It modulates the serotonergic system.
    Formula:C16H12ClN3O
    Purity:99.49%
    Color and Shape:Solid
    Molecular weight:297.74

    Ref: TM-T8438

  • MK-0557
    Targetmol
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    MK-0557

    CAS:
    MK-0557 is a selective and orally available antagonist of the neuropeptide Y5 receptor (Ki: 1.6 nM).
    Formula:C22H19FN4O3
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:406.41

    Ref: TM-TQ0286

  • JNJ-7777120
    Targetmol
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    JNJ-7777120

    CAS:
    JNJ-7777120 is the first potent and selective non-imidazole histamine H4 receptor antagonist, exhibits >1000-fold selectivity over the other histamin receptors.
    Formula:C14H16ClN3O
    Purity:99.83% - 99.96%
    Color and Shape:Solid
    Molecular weight:277.75

    Ref: TM-T2232

  • OXA (17-33) acetate
    Targetmol
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    OXA (17-33) acetate

    OXA (17-33) acetate is a more potent agonist of orexin-1 receptor (OX1, EC50 = 8.29 nM)) over OX2 (EC50 = 187 nM).
    Formula:C79H125N23O22
    Purity:98.52%
    Color and Shape:Solid
    Molecular weight:1748.98

    Ref: TM-TP1973L

  • Dobutamine
    Targetmol
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    Dobutamine

    CAS:
    Dobutamine, a synthetic catecholamine, boosts cardiac output and improves blood flow, mainly targeting β1-AR.
    Formula:C18H23NO3
    Color and Shape:Solid
    Molecular weight:301.38

    Ref: TM-T60677

  • Dioxopromethazine hydrochloride
    Targetmol
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    Dioxopromethazine hydrochloride

    CAS:
    Dioxopromethazine is a target-based classification of drug and available in a number of countries worldwide.
    Formula:C17H20N2O2S·HCl
    Purity:99.58%
    Color and Shape:Solid
    Molecular weight:352.88

    Ref: TM-T3723

  • L-745870 trihydrochloride
    Targetmol
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    L-745870 trihydrochloride

    CAS:
    <p>L-745870 trihydrochloride is a highly potent and selective D4 dopamine receptor antagonist.</p>
    Formula:C18H22Cl4N4
    Purity:97.52%
    Color and Shape:Solid
    Molecular weight:436.21

    Ref: TM-T22904

  • SCH 58261
    Targetmol
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    SCH 58261

    CAS:
    SCH 58261 is a potent and selective A2a adenosine receptor antagonist.The Ki =2.3 nM for rat A2a and 2 nM is for bovine A2a.
    Formula:C18H15N7O
    Purity:99.07% - 99.75%
    Color and Shape:Solid
    Molecular weight:345.36

    Ref: TM-T6979