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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5968 products of "GPCR/G-Protein"

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  • RVD-Hpα acetate(1193362-76-3 free base)


    RVD-Hpα acetate is the N-terminally extended form of human hemopressin that acts as a selective CB1 receptor agonist.
    Formula:C67H109N19O19
    Purity:99.87%
    Color and Shape:Solid
    Molecular weight:1484.71

    Ref: TM-TP1939L1

    1mg
    213.00€
    5mg
    464.00€
    10mg
    677.00€
    25mg
    1,035.00€
    50mg
    1,406.00€
    100mg
    1,882.00€
    500mg
    3,771.00€
  • Secretin (33-59), rat

    CAS:
    <p>Secretin (33-59), rat (Secretin (rat)) is a classical hormone in the gastrointestinal system and a neuropeptide.</p>
    Formula:C129H216N42O42
    Purity:98.12%
    Color and Shape:Solid
    Molecular weight:3027.35

    Ref: TM-TP1039

    1mg
    81.00€
    5mg
    173.00€
    10mg
    256.00€
    25mg
    393.00€
    50mg
    547.00€
    100mg
    738.00€
    200mg
    979.00€
  • GR-73632

    CAS:
    Potent and selective tachykinin NK1 receptor agonist (EC50 = 2 nM in guinea pig vas deferens).
    Formula:C40H59N7O6S
    Purity:99.68%
    Color and Shape:Solid
    Molecular weight:766

    Ref: TM-TP1572

    1mg
    52.00€
    5mg
    111.00€
    10mg
    170.00€
    25mg
    283.00€
    50mg
    430.00€
    100mg
    620.00€
    200mg
    870.00€
  • Nomifensine maleate

    CAS:
    <p>Nomifensine maleate (Nomifensine (maleate)) is a selective inhibitor of dopamine uptake. Nomifensine maleate is used in adult attention deficit disorder.</p>
    Formula:C20H22N2O4
    Purity:98.46%
    Color and Shape:Solid
    Molecular weight:354.4

    Ref: TM-T7070

    10mg
    35.00€
    25mg
    49.00€
    50mg
    70.00€
    100mg
    104.00€
  • [Des-Arg9]-Bradykinin TFA

    CAS:
    [Des-Arg9]-Bradykinin is an agonist of Bradykinin (B1) receptor that displays selectivity for B1 over B2 receptors.
    Formula:C46H62F3N11O12
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:1018.05

    Ref: TM-T8809

    2mg
    35.00€
    5mg
    39.00€
    10mg
    52.00€
    25mg
    88.00€
    50mg
    133.00€
    100mg
    192.00€
    200mg
    279.00€
  • AdipoRon hydrochloride

    CAS:
    AdipoRon hydrochloride is a specific, orally active AdipoR agonist, capable of binding AdipoR1 (Kd: 1.8 μM) and AdipoR2 (Kd: 3.1 μM).
    Formula:C27H29ClN2O3
    Color and Shape:Solid
    Molecular weight:464.99

    Ref: TM-T62964

    10mg
    948.00€
  • Empagliflozin

    CAS:
    Empagliflozin (BI 10773) is an SGLT-2 inhibitor (IC50=3.1 nM) that is potent and selective, with more than 300-fold selectivity for SGLT-1/4/5/6.
    Formula:C23H27ClO7
    Purity:98% - 99.98%
    Color and Shape:Solid
    Molecular weight:450.91

    Ref: TM-T1766

    1g
    278.00€
    5mg
    47.00€
    10mg
    60.00€
    50mg
    79.00€
    100mg
    96.00€
    200mg
    144.00€
    500mg
    188.00€
    1mL*10mM (DMSO)
    50.00€
  • JNJ-5207852

    CAS:
    JNJ-5207852 is a novel, non-imidazole histamine H3 receptor antagonist, with high affinity at the rat (pKi=8.9) and human (pKi=9.24) H3 receptor.
    Formula:C20H32N2O
    Purity:97.19%
    Color and Shape:Solid
    Molecular weight:316.48

    Ref: TM-T7413

    5mg
    35.00€
    10mg
    52.00€
    25mg
    99.00€
    50mg
    188.00€
    100mg
    276.00€
    200mg
    393.00€
    1mL*10mM (DMSO)
    39.00€
  • N-ACETYLTRYPTAMINE

    CAS:
    <p>N-ACETYLTRYPTAMINE is a partial agonist for melatonin receptors in the retina. Also used for determination of serotonin N-acetyl transferase.</p>
    Formula:C12H14N2O
    Purity:98.79%
    Color and Shape:Powder
    Molecular weight:202.25

    Ref: TM-T8600

    10mg
    44.00€
    25mg
    77.00€
    50mg
    111.00€
    100mg
    170.00€
    200mg
    244.00€
  • Epinastine hydrochloride

    CAS:
    Epinastine hydrochloride (WAL-801CL HCl) is an antihistamine and mast cell stabilizer that is used in eye drops to treat allergic conjunctivitis.
    Formula:C16H15N3·HCl
    Purity:99.26% - 99.62%
    Color and Shape:White Solid
    Molecular weight:285.77

    Ref: TM-T6488

    10mg
    39.00€
    25mg
    55.00€
    50mg
    71.00€
    100mg
    96.00€
    200mg
    173.00€
    500mg
    323.00€
    1mL*10mM (DMSO)
    47.00€
  • Ipragliflozin

    CAS:
    <p>Ipragliflozin (ASP1941) is under investigation in Type 2 Diabetes and Diabetes Mellitus, Type 2.</p>
    Formula:C21H21FO5S
    Purity:99.38% - 99.70%
    Color and Shape:Solid
    Molecular weight:404.45

    Ref: TM-T2385

    25mg
    57.00€
    50mg
    92.00€
    100mg
    135.00€
    200mg
    207.00€
    500mg
    439.00€
  • Exenatide

    CAS:
    Exenatide (Extendin-4) is a glucagon-like protein-1 (GLP-1) receptor agonist.
    Formula:C186H286N50O62S
    Purity:99.42%
    Color and Shape:Solid
    Molecular weight:4247

    Ref: TM-T8355

    1mg
    63.00€
    2mg
    90.00€
    5mg
    135.00€
    10mg
    187.00€
    25mg
    283.00€
    50mg
    420.00€
    100mg
    607.00€
  • CYM 50358 hydrochloride (1314212-39-9 free base)

    CAS:
    CYM50358 HCl is an S1P4 antagonist.
    Formula:C20H19Cl3N2O2
    Purity:99.57%
    Color and Shape:Solid
    Molecular weight:425.73

    Ref: TM-T25282

    1mg
    88.00€
    5mg
    177.00€
    10mg
    248.00€
    25mg
    393.00€
    50mg
    532.00€
    100mg
    712.00€
    200mg
    950.00€
  • Ciproxifan maleate

    CAS:
    <p>Ciproxifan maleate (FUB 359)(FUB-359 maleate) is a highly potent and selective histamin H3-receptor antagonist with IC50 of 9.2 nM, with low apparent affinity</p>
    Formula:C20H22N2O6
    Purity:99.39%
    Color and Shape:Solid
    Molecular weight:386.4

    Ref: TM-T2004

    1mg
    43.00€
    2mg
    55.00€
    5mg
    80.00€
    10mg
    106.00€
    25mg
    215.00€
    50mg
    401.00€
    100mg
    595.00€
  • Exo-1

    CAS:
    Exo-1 (Methyl 3-(4-fluorobenzoyl)-6-methyl-2-pyridinecarboxylate) is a synthetic compound that has been shown to affect the metabolism of various nutrients, as
    Formula:C15H12FNO3
    Purity:99.45%
    Color and Shape:Solid
    Molecular weight:273.26

    Ref: TM-T9200

    5mg
    55.00€
    10mg
    82.00€
    25mg
    126.00€
    50mg
    182.00€
    100mg
    273.00€
    200mg
    409.00€
    500mg
    677.00€
    1mL*10mM (DMSO)
    69.00€
  • AF38469

    CAS:
    AF38469 is a new, specific and orally bioavailable Sortilin inhibitor (IC50: 330 nM).
    Formula:C15H11F3N2O3
    Purity:99.18%
    Color and Shape:Solid
    Molecular weight:324.25

    Ref: TM-TQ0086

    1mg
    87.00€
    2mg
    120.00€
    5mg
    180.00€
    10mg
    283.00€
    25mg
    550.00€
    50mg
    847.00€
    100mg
    1,159.00€
    200mg
    1,549.00€
    1mL*10mM (DMSO)
    188.00€
  • Neurotensin

    CAS:
    Neurotensin, a 13 amino acid peptide, regulates LH and prolactin, interacts with dopamine system.
    Formula:C78H121N21O20
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:1672.92

    Ref: TM-TP1310

    1mg
    57.00€
    2mg
    88.00€
    5mg
    159.00€
    10mg
    216.00€
    25mg
    435.00€
    50mg
    627.00€
    100mg
    878.00€
  • TCS-OX2-29

    CAS:
    TCS-OX2-29 is a potent and selective OX2 receptor antagonist (IC50: 40 nM). It displays >250-fold selectivity for OX2 over OX1.
    Formula:C23H31N3O3
    Purity:99.81%
    Color and Shape:Solid
    Molecular weight:397.51

    Ref: TM-T4965

    1mg
    35.00€
    5mg
    70.00€
    10mg
    96.00€
    25mg
    156.00€
    50mg
    215.00€
    100mg
    303.00€
    200mg
    449.00€
    1mL*10mM (DMSO)
    77.00€
  • Xanthotoxol

    CAS:
    Xanthotoxol (Psoralen) is a bioactive furocoumarin with anti-inflammatory, antioxidant, 5-HT antagonist, and neuroprotective properties.
    Formula:C11H6O4
    Purity:99.97%
    Color and Shape:Solid
    Molecular weight:202.16

    Ref: TM-T4S1659

    5mg
    38.00€
    10mg
    57.00€
    25mg
    86.00€
    50mg
    106.00€
    1mL*10mM (DMSO)
    44.00€
  • Emedastine

    CAS:
    Emedastine (LY188695) is a second generation, selective histamine H1 receptor antagonist with anti-allergic activity.
    Formula:C17H26N4O
    Purity:97.1% - 97.76%
    Color and Shape:Oil
    Molecular weight:302.41

    Ref: TM-T3979

    1mg
    37.00€
    5mg
    79.00€
    10mg
    115.00€
    25mg
    187.00€
    50mg
    279.00€
    100mg
    415.00€
    500mg
    933.00€
    1mL*10mM (DMSO)
    87.00€