
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,024 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,030 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(159 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(443 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(83 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(326 products)
- PAFR(13 products)
- PKA(52 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5968 products of "GPCR/G-Protein"
Sort by
Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
RVD-Hpα acetate(1193362-76-3 free base)
RVD-Hpα acetate is the N-terminally extended form of human hemopressin that acts as a selective CB1 receptor agonist.Formula:C67H109N19O19Purity:99.87%Color and Shape:SolidMolecular weight:1484.71Ref: TM-TP1939L1
1mg213.00€5mg464.00€10mg677.00€25mg1,035.00€50mg1,406.00€100mg1,882.00€500mg3,771.00€Secretin (33-59), rat
CAS:<p>Secretin (33-59), rat (Secretin (rat)) is a classical hormone in the gastrointestinal system and a neuropeptide.</p>Formula:C129H216N42O42Purity:98.12%Color and Shape:SolidMolecular weight:3027.35GR-73632
CAS:Potent and selective tachykinin NK1 receptor agonist (EC50 = 2 nM in guinea pig vas deferens).Formula:C40H59N7O6SPurity:99.68%Color and Shape:SolidMolecular weight:766Nomifensine maleate
CAS:<p>Nomifensine maleate (Nomifensine (maleate)) is a selective inhibitor of dopamine uptake. Nomifensine maleate is used in adult attention deficit disorder.</p>Formula:C20H22N2O4Purity:98.46%Color and Shape:SolidMolecular weight:354.4[Des-Arg9]-Bradykinin TFA
CAS:[Des-Arg9]-Bradykinin is an agonist of Bradykinin (B1) receptor that displays selectivity for B1 over B2 receptors.Formula:C46H62F3N11O12Purity:>99.99%Color and Shape:SolidMolecular weight:1018.05AdipoRon hydrochloride
CAS:AdipoRon hydrochloride is a specific, orally active AdipoR agonist, capable of binding AdipoR1 (Kd: 1.8 μM) and AdipoR2 (Kd: 3.1 μM).Formula:C27H29ClN2O3Color and Shape:SolidMolecular weight:464.99Empagliflozin
CAS:Empagliflozin (BI 10773) is an SGLT-2 inhibitor (IC50=3.1 nM) that is potent and selective, with more than 300-fold selectivity for SGLT-1/4/5/6.Formula:C23H27ClO7Purity:98% - 99.98%Color and Shape:SolidMolecular weight:450.91Ref: TM-T1766
1g278.00€5mg47.00€10mg60.00€50mg79.00€100mg96.00€200mg144.00€500mg188.00€1mL*10mM (DMSO)50.00€JNJ-5207852
CAS:JNJ-5207852 is a novel, non-imidazole histamine H3 receptor antagonist, with high affinity at the rat (pKi=8.9) and human (pKi=9.24) H3 receptor.Formula:C20H32N2OPurity:97.19%Color and Shape:SolidMolecular weight:316.48N-ACETYLTRYPTAMINE
CAS:<p>N-ACETYLTRYPTAMINE is a partial agonist for melatonin receptors in the retina. Also used for determination of serotonin N-acetyl transferase.</p>Formula:C12H14N2OPurity:98.79%Color and Shape:PowderMolecular weight:202.25Epinastine hydrochloride
CAS:Epinastine hydrochloride (WAL-801CL HCl) is an antihistamine and mast cell stabilizer that is used in eye drops to treat allergic conjunctivitis.Formula:C16H15N3·HClPurity:99.26% - 99.62%Color and Shape:White SolidMolecular weight:285.77Ipragliflozin
CAS:<p>Ipragliflozin (ASP1941) is under investigation in Type 2 Diabetes and Diabetes Mellitus, Type 2.</p>Formula:C21H21FO5SPurity:99.38% - 99.70%Color and Shape:SolidMolecular weight:404.45Exenatide
CAS:Exenatide (Extendin-4) is a glucagon-like protein-1 (GLP-1) receptor agonist.Formula:C186H286N50O62SPurity:99.42%Color and Shape:SolidMolecular weight:4247CYM 50358 hydrochloride (1314212-39-9 free base)
CAS:CYM50358 HCl is an S1P4 antagonist.Formula:C20H19Cl3N2O2Purity:99.57%Color and Shape:SolidMolecular weight:425.73Ciproxifan maleate
CAS:<p>Ciproxifan maleate (FUB 359)(FUB-359 maleate) is a highly potent and selective histamin H3-receptor antagonist with IC50 of 9.2 nM, with low apparent affinity</p>Formula:C20H22N2O6Purity:99.39%Color and Shape:SolidMolecular weight:386.4Exo-1
CAS:Exo-1 (Methyl 3-(4-fluorobenzoyl)-6-methyl-2-pyridinecarboxylate) is a synthetic compound that has been shown to affect the metabolism of various nutrients, asFormula:C15H12FNO3Purity:99.45%Color and Shape:SolidMolecular weight:273.26Ref: TM-T9200
5mg55.00€10mg82.00€25mg126.00€50mg182.00€100mg273.00€200mg409.00€500mg677.00€1mL*10mM (DMSO)69.00€AF38469
CAS:AF38469 is a new, specific and orally bioavailable Sortilin inhibitor (IC50: 330 nM).Formula:C15H11F3N2O3Purity:99.18%Color and Shape:SolidMolecular weight:324.25Ref: TM-TQ0086
1mg87.00€2mg120.00€5mg180.00€10mg283.00€25mg550.00€50mg847.00€100mg1,159.00€200mg1,549.00€1mL*10mM (DMSO)188.00€Neurotensin
CAS:Neurotensin, a 13 amino acid peptide, regulates LH and prolactin, interacts with dopamine system.Formula:C78H121N21O20Purity:>99.99%Color and Shape:SolidMolecular weight:1672.92TCS-OX2-29
CAS:TCS-OX2-29 is a potent and selective OX2 receptor antagonist (IC50: 40 nM). It displays >250-fold selectivity for OX2 over OX1.Formula:C23H31N3O3Purity:99.81%Color and Shape:SolidMolecular weight:397.51Ref: TM-T4965
1mg35.00€5mg70.00€10mg96.00€25mg156.00€50mg215.00€100mg303.00€200mg449.00€1mL*10mM (DMSO)77.00€Xanthotoxol
CAS:Xanthotoxol (Psoralen) is a bioactive furocoumarin with anti-inflammatory, antioxidant, 5-HT antagonist, and neuroprotective properties.Formula:C11H6O4Purity:99.97%Color and Shape:SolidMolecular weight:202.16Emedastine
CAS:Emedastine (LY188695) is a second generation, selective histamine H1 receptor antagonist with anti-allergic activity.Formula:C17H26N4OPurity:97.1% - 97.76%Color and Shape:OilMolecular weight:302.41Ref: TM-T3979
1mg37.00€5mg79.00€10mg115.00€25mg187.00€50mg279.00€100mg415.00€500mg933.00€1mL*10mM (DMSO)87.00€

