GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,017 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(194 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5983 products of "GPCR/G-Protein"
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Eptinezumab
CAS:Eptinezumab is a humanised monoclonal antibody targeting CGRP (calcitonin gene-related peptide), which prevents CGRP binding to its receptor, migraine.
Purity:95% - 95%Color and Shape:LiquidEscitalopram
CAS:Escitalopram (Seroplex), a serotonin inhibitor for depression, curbs alcohol intake and is favored over tricyclics for tardive dyskinesia.Formula:C20H21FN2OPurity:99.82%Color and Shape:White Or White Crystalline PowderMolecular weight:324.39Carlumab
CAS:Carlumab is a high-affinity human monoclonal antibody that targets CCL2, suppressing the recruitment of monocytes/macrophages in the tumour microenvironment.Purity:95%Color and Shape:LiquidMolecular weight:144.87 kDa17-phenyl trinor Prostaglandin F2α isopropyl ester
CAS:17-phenyl trinor PGF2α N-ethyl amide is an F-series prostaglandin analog which has been approved for use as an ocular hypotensive drug, sold under the AllerganFormula:C26H38O5Color and Shape:SolidMolecular weight:430.58Buflomedil
CAS:Buflomedil is a vasoactive compound. Buflomedil has been used for peripheral arterial diseases.Formula:C17H25NO4Purity:98%Color and Shape:SolidMolecular weight:307.38Rocatinlimab
CAS:Rocatinlimab (AMG 451) (KHK4083) is a fully human, non-fucosylated IgG1 anti-OX40 monoclonal antibody indicated for atopic dermatitis (AD) research [1].Color and Shape:LiquidBlontuvetmab
CAS:Blontuvetmab (AT 004), a caninized CD20 monoclonal antibody, is utilized in the study of Canine B-cell lymphoma [1].Color and Shape:Liquid15-keto Prostaglandin F2α
CAS:15-keto Prostaglandin F2α is a metabolite of Prostaglandin F2α that lowers intraocular pressure in rabbits.Formula:C20H32O5Purity:98%Color and Shape:SolidMolecular weight:352.47Brexpiprazole-d8
CAS:Brexpiprazole D8 is a deuterium-modified partial agonist of 5-HT1A and dopamine receptors, with Ki values of 0.12 nM and 0.3 nM respectively.Formula:C25H27N3O2SPurity:98%Color and Shape:SolidMolecular weight:441.62Dapagliflozin-d5
CAS:Dapagliflozin D5 (BMS-512148 D5) is deuterated Dapagliflozin. Dapagliflozin is a competitive SGLT2 inhibitor.Formula:C21H25ClO6Purity:98%Color and Shape:SolidMolecular weight:413.9Cinnarizine D8
CAS:Cinnarizine D8 is a deuterium-labeled Cinnarizine which is an antihistamine and a calcium channel blocker.Formula:C26H28N2Purity:98%Color and Shape:SolidMolecular weight:376.573Mirtazapine D3
CAS:Mirtazapine D3 is a deuterium labeled Mirtazapine. Mirtazapine is an inhibitor of 5-HT receptor .Formula:C17H19N3Purity:98%Color and Shape:SolidMolecular weight:268.37Mianserin-d3
CAS:Mianserin-d3 is a deuterated compound of Mianserin. Mianserin has a CAS number of 24219-97-4. Mianserin, an H1 receptor reverse agonist, is a psychoactive compound in the tetracyclic antidepressant (TeCA) treatment family. Mianserin has antidepressant, antianxiety, antiemetic, hypotrophic, hypnotic and antihistamine effects, and can be used as a combination of norepinephrine and specific serotonin to treat depression.Formula:C18H17D3N2Color and Shape:SolidMolecular weight:267.38Amitriptyline-d6 Hydrochloride
CAS:Amitriptyline-d6 Hydrochloride is a deuterated compound of Amitriptyline Hydrochloride. Amitriptyline Hydrochloride has a CAS number of 549-18-8. Amitriptyline Hydrochloride is the hydrochloride salt of the tricyclic dibenzocycloheptadiene amitriptyline with antidepressant and antinociceptive activities.Formula:C20H18D6ClNColor and Shape:SolidMolecular weight:319.907-Desmethyl-3-hydroxyagomelatine
CAS:7-Desmethyl-3-hydroxyagomelatine, less active than parent drug Agomelatine, is a melatonergic agonist and 5-HT2C antagonist.Formula:C14H15NO3Purity:98%Color and Shape:SolidMolecular weight:245.27SB 271046 hydrochloride
CAS:SB 271046 hydrochloride (SB 271046A) is selective, orally active 5-HT6 antagonist and is > 200-fold selective over 55 other receptors, enzymes and ion channels.Formula:C20H22ClN3O3S2·HClPurity:99.77%Color and Shape:SolidMolecular weight:488.45Proxyfan Oxalate
CAS:Proxyfan Oxalate is a potent antagonist of the histamine H3 receptor (histamine H3 receptor), with Ki values of 2.9 nM for rats and 2.7 nM for humans. Its inhibitory effect on H3 receptors is over 1000 times stronger than its effect on other histamine receptors.Formula:C15H18N2O5Color and Shape:SolidMolecular weight:306.31R-138727
CAS:R-138727 is a novel P2Y12 receptor inhibitor.Formula:C18H20FNO3SPurity:98%Color and Shape:SolidMolecular weight:349.42Litorin
CAS:Litorin suppresses appetite and stimulates smooth muscle, gastrin, gastric acid, and pancreatic secretion.Formula:C51H68N14O11SColor and Shape:White PowderMolecular weight:1085.24Isoproterenol sulfate anhydrous
CAS:Isoproterenol sulfate anhydrous is a useful alkaloid. It is used for biological research.Formula:C22H36N2O10SPurity:98%Color and Shape:CoaMolecular weight:520.59
