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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5983 products of "GPCR/G-Protein"

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  • Bucumarol (HCl)

    CAS:
    Bucumarol is a beta-adrenergic blocking agent.
    Formula:C17H24ClNO4
    Color and Shape:Solid
    Molecular weight:341.83

    Ref: TM-T30606

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • APC-3316 tosylate

    CAS:
    APC-3316 tosylate is a vinyl sulfone cysteine protease inhibitor and selective CCR4 antagonist.
    Formula:C39H46N4O7S2
    Color and Shape:Solid
    Molecular weight:746.94

    Ref: TM-T69183

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Benzoctamine

    CAS:
    Benzoctamine: oral psychoactive with tranquillizing effects; boosts catecholamine turnover; enhances rat heart [3H]noradrenaline uptake.
    Formula:C18H19N
    Color and Shape:Solid
    Molecular weight:249.35

    Ref: TM-T60368

    25mg
    1,927.00€
    50mg
    2,507.00€
    100mg
    3,168.00€
  • CCK-B Receptor Antagonist 1

    CAS:
    CCK-B Receptor Antagonist 1 is a cholecystokinin B (CCK-B) receptor agonist and has the potential of reducing the secretion of gastric acid.
    Formula:C28H30N6O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:498.58

    Ref: TM-T13261

    2mg
    50.00€
  • Efpeglenatide

    CAS:
    Efpeglenatide is a long-acting GLP-1 receptor agonist that improves insulin sensitivity, lowers blood glucose, delays weight gain, and supports metabolic disease research.
    Purity:100% - 100%
    Color and Shape:Solid

    Ref: TM-T64252

    1mg
    285.00€
    5mg
    692.00€
    10mg
    947.00€
    25mg
    1,458.00€
    50mg
    1,839.00€
    100mg
    2,322.00€
  • GB83

    CAS:
    GB83 is a selective human protease activated receptor 2 (PAR2) antagonist.
    Formula:C32H44N4O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:548.72

    Ref: TM-T27406

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • VPC12249

    CAS:
    VPC12249, a lysophosphatidic acid receptor type 1 (LPA1) antagonist, plays a functional role in osteoclast differentiation and bone resorption activity.
    Formula:C34H52NO6P
    Color and Shape:Solid
    Molecular weight:601.75

    Ref: TM-T29109

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • ABT-239

    CAS:
    ABT-239 is a novel, highly efficacious antagonist belonging to the non-imidazole class of histamine H3 receptor (H3R) antagonists.
    Formula:C22H22N2O
    Purity:99.94%
    Color and Shape:Solid
    Molecular weight:330.42

    Ref: TM-T14087

    1mg
    44.00€
    5mg
    93.00€
    10mg
    133.00€
    25mg
    270.00€
    50mg
    409.00€
    100mg
    595.00€
    200mg
    833.00€
    1mL*10mM (DMSO)
    90.00€
  • Zolantidine dimaleate

    CAS:
    H2 receptor antagonist
    Formula:C26H31N3O5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:497.61

    Ref: TM-T23565

    10mg
    705.00€
    50mg
    2,907.00€
  • GSK-894490A

    CAS:
    GSK-894490A is an agonist of ghrelin receptor. GSK-894490A crosses the blood/brain barrier and elicit pro-cognitive effects.
    Formula:C24H30ClN3O4S
    Color and Shape:Solid
    Molecular weight:492.03

    Ref: TM-T27493

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • A2AAR antagonist 1

    CAS:
    Compound 21a, A2AAR antagonist with 20 nM Ki, useful in neurodegenerative disease study.
    Formula:C12H8BrN3O
    Color and Shape:Solid
    Molecular weight:290.12

    Ref: TM-T60591

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Alprenolol hydrochloride, (S)-

    CAS:
    Alprenolol hydrochloride, (S)- is a nonselective β-blocker. It is also a serotonin 5HT1A receptor antagonist.
    Formula:C15H24ClNO2
    Color and Shape:Solid
    Molecular weight:285.81

    Ref: TM-T4560L1

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • LEI-101

    CAS:
    LEI-101: potent CB2 agonist, pEC50=8, bioavailable, >100x selective over CB1, potential for inflammatory diseases.
    Formula:C23H25FN4O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:472.53

    Ref: TM-T27809

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • RS 64459-193

    CAS:
    RS 64459-193 has a high affinity for the 5-HT1A binding site.
    Formula:C26H36Cl2N2O2
    Color and Shape:Solid
    Molecular weight:479.48

    Ref: TM-T34415

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • TC-C 14G

    CAS:
    CB1 receptor inverse agonist
    Formula:C24H17Cl2F2NO4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:492.3

    Ref: TM-T23427

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Aminopotentidine

    CAS:
    H2 antagonist
    Formula:C26H35N7O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:477.6

    Ref: TM-T22566

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • NGB 2904 hydrochloride

    CAS:
    dopamine D3 receptor antagonist
    Formula:C28H30Cl3N3O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:530.92

    Ref: TM-T23065

    1mg
    132.00€
    5mg
    375.00€
  • Alimemazine

    CAS:
    Alimemazine, an antipruritic and HA-receptor antagonist, also partially activates H1R and other GPCRs.
    Formula:C18H22N2S
    Purity:98%
    Color and Shape:Crystals Solid
    Molecular weight:298.45

    Ref: TM-T10281

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • JNJ-10191584

    CAS:
    JNJ-10191584, a potent and selective antagonist at the histamine H4 receptor, has antiinflammatory and analgesic effects in animal studies of acute inflammation
    Formula:C13H15ClN4O
    Color and Shape:Solid
    Molecular weight:278.74

    Ref: TM-T27658

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Glucagon receptor antagonists-2

    CAS:
    Glucagon receptor antagonist -2 is a highly effective glucagon receptor antagonist.
    Formula:C22H30FNO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:359.48

    Ref: TM-T11414

    25mg
    680.00€
    50mg
    884.00€