GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,017 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(194 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5983 products of "GPCR/G-Protein"
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Hydroxy ziprasidone
CAS:Hydroxy ziprasidone is an impurity of Ziprasidone. Ziprasidone, an antipsychotic agent, is a 5-HT and dopamine receptor antagonist.Formula:C21H21ClN4O2SPurity:98%Color and Shape:SolidMolecular weight:428.947-Desmethyl-3-hydroxyagomelatine
CAS:7-Desmethyl-3-hydroxyagomelatine, less active than parent drug Agomelatine, is a melatonergic agonist and 5-HT2C antagonist.Formula:C14H15NO3Purity:98%Color and Shape:SolidMolecular weight:245.27SB 271046 hydrochloride
CAS:SB 271046 hydrochloride (SB 271046A) is selective, orally active 5-HT6 antagonist and is > 200-fold selective over 55 other receptors, enzymes and ion channels.Formula:C20H22ClN3O3S2·HClPurity:99.77%Color and Shape:SolidMolecular weight:488.45Amthamine
CAS:Compound AMTHAMINE DIHYDROBROMIDE is a useful organic compound for research related to life sciences.Formula:C6H11N3SColor and Shape:SoildMolecular weight:157.24Roxatidine acetate
CAS:Roxatidine acetate: anti-ulcer, blocks histamine, reduces acid. Safer at lower doses.Formula:C19H28N2O4Purity:98%Color and Shape:White Or Off-White PowderMolecular weight:348.44Ridazolol HCl
CAS:Ridazolol HCl (CAS 413) is a novel β-adrenoceptor (β-AR) blocker with α-adrenerolytic activity.Formula:C15H19Cl3N4O3Purity:99.48%Color and Shape:SoildMolecular weight:409.7Isoproterenol sulfate anhydrous
CAS:Isoproterenol sulfate anhydrous is a useful alkaloid. It is used for biological research.Formula:C22H36N2O10SPurity:98%Color and Shape:CoaMolecular weight:520.59Ketanserinol
CAS:Ketanserinol is a metabolite of the antihypertensive drug ketanserin, which blocks 5-HT2 receptors to treat protamine-induced pulmonary hypertension.Formula:C22H24FN3O3Color and Shape:SolidMolecular weight:397.44S 25585
CAS:S 25585 is a neuropeptide Y (NPY) Y5 receptor antagonist.Formula:C22H23F3N4O6SPurity:98%Color and Shape:SolidMolecular weight:528.5Dopamine D4 receptor ligand 2
CAS:Compound 17, a dopamine D4 receptor ligand, exhibits high potency and selectivity with IC 50 values of 0.057 nM for D4, and >1000, 220, and 270 nM for D2, 5-HT1A, and α1 receptors, respectively [1].Formula:C20H24ClN3O2Color and Shape:SolidMolecular weight:373.88Dolasetron Mesylate
CAS:Dolasetron Mesylate (MDL-73147EF) is an antagonist of the 5-HT3 receptor and can be used in research on the treatment of vomiting and nausea followingFormula:C20H24N2O6SPurity:99.05%Color and Shape:White PowderMolecular weight:420.48Lodoxamide tromethamine
CAS:Lodoxamide tromethamine is a mast cell stabilizer with anti-allergic properties and can be used in studies about the treatment of asthma and allergicFormula:C19H28ClN5O12Purity:98.8%Color and Shape:SolidMolecular weight:553.91MK-5046
CAS:MK-5046 is a novel BRS-3 agonist, binding to BRS-3 with high affinity (mouse Ki = 1.6 nM, human Ki = 25 nM).Formula:C20H18F6N4OPurity:98.56%Color and Shape:SolidMolecular weight:444.37LY 344864
CAS:LY 344864, a specifc receptor agonist, is an affinity of 6 nM (Ki) at the recently cloned 5-HT1F receptor.Formula:C21H22FN3OPurity:98%Color and Shape:SolidMolecular weight:351.42Paroxetine hydrochloride hemihydrate
CAS:Paroxetine hydrochloride hemihydrate (Paxil) is an effective and selective serotonin reuptake inhibitor (SSRI).Formula:C38H44Cl2F2N2O7Purity:99.949%Color and Shape:SolidMolecular weight:749.67Guacetisal
CAS:Guacetisal, from acetylsalicylic acid and guaiacol, may treat chronic bronchitis.
Formula:C16H14O5Purity:99.18%Color and Shape:SolidMolecular weight:286.28Photoregulin1
CAS:Photoregulin1 modulates Nr2e3, slows photoreceptor degeneration in RhoP23H, Pde6brd1 mouse RP models.Formula:C21H23N3O2SColor and Shape:SolidMolecular weight:381.49HSK0935
CAS:HSK0935 is a highly selective and orally available SGLT2 inhibitor (IC50: 1.3 nM). It has antihyperglycemic activities.Formula:C22H25ClO7Purity:98%Color and Shape:SolidMolecular weight:436.88Ipsapirone
CAS:Ipsapirone is a partial agonist of 5-HT1A receptor and produces an inhibitory effect on 5-HT2 and the α1-adrenergic function at high doses.
Formula:C19H23N5O3SPurity:99.51%Color and Shape:SolidMolecular weight:401.48N,N-Dimethylsphingosine
CAS:N,N-Dimethylsphingosine,is a potent competitive SphK phosphorylation inhibitor.DMS is elevated in models of neuropathic pain by increasing IL-1β and MCP-1.Formula:C20H41NO2Purity:98%Color and Shape:Clear Colorless To Faint Yellow Liquid/White To Off-White PowderMolecular weight:327.55
