
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,022 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(194 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5983 products of "GPCR/G-Protein"
Sort by
Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
Cinitapride Hydrogen Tartrate
CAS:Cinitapride Hydrogen Tartrate is a gastroprokinetic agent that acts as an antagonist of the 5-HT2 receptors and as an agonist of the 5-HT1 and 5-HT4 receptorsFormula:C25H36N4O10Purity:98%Color and Shape:SolidMolecular weight:552.581EP3 antagonist 3
CAS:EP3 antagonist 3, potent and selective oral, inhibited GR63799- or acetic acid-induced reduction in bladder capacity and PGE2-induced overactive bladder model.Formula:C21H18N2O4Color and Shape:SolidMolecular weight:362.38ONO-8713
CAS:ONO-8713 is a selective prostaglandin E receptor subtype EP1 antagonist that can be used to study diseases of the biblical system and metabolism-relatedFormula:C25H24F3NO6SPurity:99.97%Color and Shape:SolidMolecular weight:523.52CP-226269
CAS:CP-226269 is a potent dopamine D4 receptor agonist that regulates calcium flux and has an EC50 value of 32.0 nM.
Formula:C18H19FN4Purity:99.08%Color and Shape:SolidMolecular weight:310.37L-740093
CAS:L-740093 is a specific antagonist of CCK-B receptor.Formula:C26H31N5O2Purity:98%Color and Shape:SolidMolecular weight:445.56S 16924
CAS:S 16924 is a 5-HT 1A agonist with potential anxiolytic effects and may be useful in the study of neurologic disorders.Formula:C22H24FNO4Purity:99.35% - 99.6%Color and Shape:SolidMolecular weight:385.43ESI-08
CAS:ESI-08 is an effective antagonist of EPAC2 with an IC50 of 8.4 μM. ESI-08 selectively blocks cAMP-induced EPAC activation but not cAMP-mediated PKA activation.Formula:C20H23N3OSPurity:97.17%Color and Shape:SolidMolecular weight:353.48Dicarbine
CAS:Double carbene blocks dopamine receptors, aiding schizophrenia and alcoholism research; it maintains defense reflexes despite mid-brain stimulation.Formula:C13H18N2Purity:98%Color and Shape:SolidMolecular weight:202.3Aganepag
CAS:Aganepag: Potent EP2 agonist, EC50 0.19 nM, inactive at EP4, used in wound healing and scar/wrinkle treatment research.Formula:C24H31NO4SPurity:98%Color and Shape:SolidMolecular weight:429.57Atrasentan hydrochloride
CAS:Atrasentan hydrochloride (ABT-627 hydrochloride) is an antagonist of the endothelin receptor(IC50 = 55.1 μM for ETA).Formula:C29H39ClN2O6Purity:99.75%Color and Shape:SolidMolecular weight:547.08A2AR-agonist-1
CAS:A2AR-agonist-1 targets A2A Receptor/ENT1 for neuroprotection; potent with Ki of 4.39 (A2AR), 3.47 (ENT1).Formula:C20H22N6O4Purity:99.9%Color and Shape:SolidMolecular weight:410.43Ref: TM-T10212
1mg90.00€2mg127.00€5mg178.00€10mg269.00€25mg427.00€50mg610.00€100mg820.00€500mg1,603.00€1mL*10mM (DMSO)207.00€SB-269970
CAS:SB-269970 is a antagonist of 5-HT7 receptor(pKi of 8.3).Formula:C18H28N2O3SPurity:98%Color and Shape:SolidMolecular weight:352.49WS 009A
CAS:WS 009A is an antagonist of the endothelin receptor.Formula:C24H25NO10SPurity:98%Color and Shape:SolidMolecular weight:519.52VNA-932
CAS:VNA-932 is an agonist of the vasopressin V2-receptor (IC50: 80.3 nM and 778 nM in human-V2 binding and V1a binding assay).Formula:C23H19ClN4OPurity:98%Color and Shape:SolidMolecular weight:402.88GBR 13069 dihydrochloride
CAS:GBR 13069 dihydrochloride is a dopamine uptake inhibitor.Formula:C28H32Cl2F2N2OPurity:98%Color and Shape:SolidMolecular weight:521.47(R)-SLV 319
CAS:(R)-SLV 319: potent CB1 antagonist, K i of 894 nM, dextrorotatory isomer.Formula:C23H20Cl2N4O2SColor and Shape:SolidMolecular weight:487.4DS-3801b
CAS:DS-3801b is a non-macrolide GPR38 agonist with an N-methylaniline structure for the study of functional gastrointestinal disorders.Formula:C28H39N3O3Purity:99.21%Color and Shape:SolidMolecular weight:465.63GSK1059865
CAS:GSK1059865 is a potent antagonist of the orexin 1 receptor.Formula:C20H23BrFN3O2Color and Shape:SolidMolecular weight:436.32MC-4R Agonist 1
CAS:MC-4R Agonist 1 is an agonist of human melanocortin-4 receptor (MC-4R) and can be used in the research of sexual dysfunction, obesity, and diabetes.Formula:C30H38ClF2N3O2Purity:98%Color and Shape:SolidMolecular weight:546.09TSHR antagonist S37b
CAS:S37b, a less effective enantiomer of TSHR antagonist S37a, offers minor thyrotropin receptor inhibition, useful for thyroid research.Formula:C25H20N2O3S2Color and Shape:SolidMolecular weight:460.57
