CymitQuimica logo
GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

Show 19 more subcategories

Found 5983 products of "GPCR/G-Protein"

Sort by

Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
products per page.
  • Cinitapride Hydrogen Tartrate

    CAS:
    Cinitapride Hydrogen Tartrate is a gastroprokinetic agent that acts as an antagonist of the 5-HT2 receptors and as an agonist of the 5-HT1 and 5-HT4 receptors
    Formula:C25H36N4O10
    Purity:98%
    Color and Shape:Solid
    Molecular weight:552.581

    Ref: TM-T22294

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • EP3 antagonist 3

    CAS:
    EP3 antagonist 3, potent and selective oral, inhibited GR63799- or acetic acid-induced reduction in bladder capacity and PGE2-induced overactive bladder model.
    Formula:C21H18N2O4
    Color and Shape:Solid
    Molecular weight:362.38

    Ref: TM-T61357

    25mg
    915.00€
    50mg
    1,190.00€
    100mg
    1,848.00€
  • ONO-8713

    CAS:
    ONO-8713 is a selective prostaglandin E receptor subtype EP1 antagonist that can be used to study diseases of the biblical system and metabolism-related
    Formula:C25H24F3NO6S
    Purity:99.97%
    Color and Shape:Solid
    Molecular weight:523.52

    Ref: TM-T63667

    1mg
    358.00€
    5mg
    873.00€
    10mg
    1,063.00€
    25mg
    1,423.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • CP-226269

    CAS:

    CP-226269 is a potent dopamine D4 receptor agonist that regulates calcium flux and has an EC50 value of 32.0 nM.

    Formula:C18H19FN4
    Purity:99.08%
    Color and Shape:Solid
    Molecular weight:310.37

    Ref: TM-T27060

    1mg
    37.00€
    5mg
    88.00€
    10mg
    120.00€
    25mg
    210.00€
    50mg
    314.00€
    100mg
    452.00€
    200mg
    628.00€
  • L-740093

    CAS:
    L-740093 is a specific antagonist of CCK-B receptor.
    Formula:C26H31N5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:445.56

    Ref: TM-T27774

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • S 16924

    CAS:
    S 16924 is a 5-HT 1A agonist with potential anxiolytic effects and may be useful in the study of neurologic disorders.
    Formula:C22H24FNO4
    Purity:99.35% - 99.6%
    Color and Shape:Solid
    Molecular weight:385.43

    Ref: TM-T28638

    1mg
    264.00€
    5mg
    650.00€
    10mg
    888.00€
    25mg
    1,369.00€
    50mg
    1,783.00€
  • ESI-08

    CAS:
    ESI-08 is an effective antagonist of EPAC2 with an IC50 of 8.4 μM. ESI-08 selectively blocks cAMP-induced EPAC activation but not cAMP-mediated PKA activation.
    Formula:C20H23N3OS
    Purity:97.17%
    Color and Shape:Solid
    Molecular weight:353.48

    Ref: TM-T11234

    1mg
    52.00€
    5mg
    113.00€
    10mg
    178.00€
    25mg
    409.00€
    1mL*10mM (DMSO)
    126.00€
  • Dicarbine

    CAS:
    Double carbene blocks dopamine receptors, aiding schizophrenia and alcoholism research; it maintains defense reflexes despite mid-brain stimulation.
    Formula:C13H18N2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:202.3

    Ref: TM-T13652

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Aganepag

    CAS:
    Aganepag: Potent EP2 agonist, EC50 0.19 nM, inactive at EP4, used in wound healing and scar/wrinkle treatment research.
    Formula:C24H31NO4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:429.57

    Ref: TM-T14139

    25mg
    2,043.00€
    50mg
    2,682.00€
    100mg
    3,600.00€
  • Atrasentan hydrochloride

    CAS:
    Atrasentan hydrochloride (ABT-627 hydrochloride) is an antagonist of the endothelin receptor(IC50 = 55.1 μM for ETA).
    Formula:C29H39ClN2O6
    Purity:99.75%
    Color and Shape:Solid
    Molecular weight:547.08

    Ref: TM-TQ0270

    1mg
    47.00€
    5mg
    92.00€
    10mg
    130.00€
    25mg
    250.00€
    50mg
    356.00€
    1mL*10mM (DMSO)
    110.00€
  • A2AR-agonist-1

    CAS:
    A2AR-agonist-1 targets A2A Receptor/ENT1 for neuroprotection; potent with Ki of 4.39 (A2AR), 3.47 (ENT1).
    Formula:C20H22N6O4
    Purity:99.9%
    Color and Shape:Solid
    Molecular weight:410.43

    Ref: TM-T10212

    1mg
    90.00€
    2mg
    127.00€
    5mg
    178.00€
    10mg
    269.00€
    25mg
    427.00€
    50mg
    610.00€
    100mg
    820.00€
    500mg
    1,603.00€
    1mL*10mM (DMSO)
    207.00€
  • SB-269970

    CAS:
    SB-269970 is a antagonist of 5-HT7 receptor(pKi of 8.3).
    Formula:C18H28N2O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:352.49

    Ref: TM-T12842

    25mg
    2,178.00€
    50mg
    3,042.00€
    100mg
    4,140.00€
  • WS 009A

    CAS:
    WS 009A is an antagonist of the endothelin receptor.
    Formula:C24H25NO10S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:519.52

    Ref: TM-T24053

    25mg
    1,369.00€
  • VNA-932

    CAS:
    VNA-932 is an agonist of the vasopressin V2-receptor (IC50: 80.3 nM and 778 nM in human-V2 binding and V1a binding assay).
    Formula:C23H19ClN4O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:402.88

    Ref: TM-T17251

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • GBR 13069 dihydrochloride

    CAS:
    GBR 13069 dihydrochloride is a dopamine uptake inhibitor.
    Formula:C28H32Cl2F2N2O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:521.47

    Ref: TM-T22799

    5mg
    259.00€
    10mg
    500.00€
    25mg
    1,161.00€
  • (R)-SLV 319

    CAS:
    (R)-SLV 319: potent CB1 antagonist, K i of 894 nM, dextrorotatory isomer.
    Formula:C23H20Cl2N4O2S
    Color and Shape:Solid
    Molecular weight:487.4

    Ref: TM-T22140

    5mg
    1,018.00€
    10mg
    1,513.00€
  • DS-3801b

    CAS:
    DS-3801b is a non-macrolide GPR38 agonist with an N-methylaniline structure for the study of functional gastrointestinal disorders.
    Formula:C28H39N3O3
    Purity:99.21%
    Color and Shape:Solid
    Molecular weight:465.63

    Ref: TM-T62973

    1mg
    164.00€
    5mg
    402.00€
    10mg
    655.00€
    25mg
    1,305.00€
    50mg
    1,839.00€
    1mL*10mM (DMSO)
    412.00€
  • GSK1059865

    CAS:
    GSK1059865 is a potent antagonist of the orexin 1 receptor.
    Formula:C20H23BrFN3O2
    Color and Shape:Solid
    Molecular weight:436.32

    Ref: TM-T11477

    1mg
    69.00€
    5mg
    147.00€
    10mg
    To inquire
    1mL*10mM (DMSO)
    164.00€
  • MC-4R Agonist 1

    CAS:
    MC-4R Agonist 1 is an agonist of human melanocortin-4 receptor (MC-4R) and can be used in the research of sexual dysfunction, obesity, and diabetes.
    Formula:C30H38ClF2N3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:546.09

    Ref: TM-T10230

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • TSHR antagonist S37b

    CAS:
    S37b, a less effective enantiomer of TSHR antagonist S37a, offers minor thyrotropin receptor inhibition, useful for thyroid research.
    Formula:C25H20N2O3S2
    Color and Shape:Solid
    Molecular weight:460.57

    Ref: TM-T38226

    5mg
    429.00€
    25mg
    1,378.00€
    50mg
    1,791.00€
    100mg
    2,682.00€