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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5983 products of "GPCR/G-Protein"

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  • Irindalone

    CAS:
    IrindaloneIrindalone is a potent serotonin (5-HT2) antagonist.
    Formula:C24H29FN4O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:408.51

    Ref: TM-T11677

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • PNU-96391

    CAS:
    PNU-96391 (OSU-6162) is an antagonist of dopamine D2 and a partial agonist of 5-HT2A. PNU-96391 can be used in research on the treatment of chronic diseases.
    Formula:C15H23NO2S
    Purity:99.53%
    Color and Shape:Solid
    Molecular weight:281.41

    Ref: TM-T28435

    1mg
    73.00€
    1mL*10mM (DMSO)
    138.00€
    5mg
    146.00€
    10mg
    210.00€
    25mg
    319.00€
    50mg
    447.00€
    100mg
    600.00€
    200mg
    800.00€
  • Levobunolol

    CAS:
    Levobunolol is a nonselective beta-blocker. It is used topically to treat glaucoma.
    Formula:C17H25NO3
    Color and Shape:White To Pink Powder
    Molecular weight:291.39

    Ref: TM-T32699

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • EA-230

    CAS:
    Ea-230 is an immunomodulator that may be used in the treatment of renal failure.
    Formula:C15H27N5O6
    Color and Shape:Solid
    Molecular weight:373.4

    Ref: TM-T31594

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Amosulalol, (-)-

    CAS:
    Amosulalol, (-)-, is an adrenergic agent.
    Formula:C18H24N2O5S
    Color and Shape:Solid
    Molecular weight:380.46

    Ref: TM-T30028

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • NPEC-caged-dopamine

    CAS:
    Dopamine receptor agonist
    Formula:C17H18N2O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:346.33

    Ref: TM-T23082

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Afurolol Hydrochloride

    CAS:
    Afurolol Hydrochloride (DL 071-IT) is a non-selective β-adrenergic receptor antagonist. DL 071 IT exhibits intrinsic sympathomimetic activity.
    Formula:C15H22ClNO4
    Purity:98.86%
    Color and Shape:Solid
    Molecular weight:315.79

    Ref: TM-T5450

    1mg
    95.00€
    5mg
    195.00€
    10mg
    293.00€
    25mg
    519.00€
    50mg
    750.00€
    100mg
    1,046.00€
    200mg
    1,410.00€
  • 5-HT3 antagonist 2

    CAS:
    5-HT3 antagonist 2 is an antagonist of 5-HT3 receptor.
    Formula:C18H21N3O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:295.38

    Ref: TM-T12988

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Amitifadine hydrochloride

    CAS:
    Amitifadine hydrochloride (EB-1010 hydrochloride) is a triple reuptake inhibitor (TRI) or serotonin-norepinephrine-dopamine reuptake inhibitor (SNDRI).
    Formula:C11H12Cl3N
    Purity:98%
    Color and Shape:Solid
    Molecular weight:264.58

    Ref: TM-T2092

    1mg
    90.00€
    5mg
    215.00€
    1mL*10mM (DMSO)
    236.00€
    10mg
    356.00€
  • Prucalopride hydrochloride

    CAS:
    Prucalopride hydrochloride is a selective agonist of the 5-HT4.
    Formula:C18H27Cl2N3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:404.33

    Ref: TM-T2542L

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Methiothepin maleate

    CAS:
    Methiothepin maleate (Metitepine) is a 5-HT1, 5-HT6, 5-HT7 serotonin receptor antagonist, which blocks serotonin autoreceptors.
    Formula:C24H28N2O4S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:472.62

    Ref: TM-T4375

    10mg
    155.00€
    25mg
    324.00€
    50mg
    439.00€
    100mg
    780.00€
  • SGS518 oxalate

    CAS:
    SGS518 oxalate is a 5-HT6 antagonist.
    Formula:C23H24F2N2O7S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:510.51

    Ref: TM-T23350

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • LY 163443

    CAS:
    LY 163443 is an dual receptor antagonist of LTD4 and LTE4.
    Formula:C20H22N4O3
    Color and Shape:Solid
    Molecular weight:366.41

    Ref: TM-T27877

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • ST1936

    CAS:
    ST1936 (ST 1936 oxalate) is a 5-HT6 receptor agonist that stimulates cAMP, Ca2+, ERK1/2, and Fyn kinases by fully activating cloned human 5-HT6 receptors.
    Formula:C13H17ClN2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:236.74

    Ref: TM-T23396

    1mg
    44.00€
    5mg
    111.00€
    1mL*10mM (DMSO)
    123.00€
    10mg
    178.00€
    25mg
    316.00€
    50mg
    470.00€
    100mg
    682.00€
    200mg
    954.00€
  • BGC201531

    CAS:
    BGC201531 (AP-1531) is a EP4 antagonist for the treatment of acute migraine.
    Formula:C26H28N2O6S
    Purity:98.51% - 99.33%
    Color and Shape:Solid
    Molecular weight:496.58

    Ref: TM-T8993

    1mg
    129.00€
    5mg
    304.00€
    10mg
    442.00€
    25mg
    735.00€
    50mg
    1,018.00€
    100mg
    1,378.00€
  • SCH-23390 maleate

    CAS:
    SCH-23390 maleate (R-(+)-SCH-23390 maleate) is a potent and selective antagonist of dopamine D1-like receptor (1 and D5 receptor with Kis of 0.2 nM and 0.3 nM,
    Formula:C21H22ClNO5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:403.86

    Ref: TM-T12865

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • 2-Methylthioadenosine diphosphate trisodium

    CAS:
    2-Methylthioadenosine diphosphate trisodium(2-MeS-ADP) is a purinergic P2Y receptor agonist that agonizes P2Y13 and P2Y12, induces platelet aggregation.
    Formula:C11H14N5Na3O10P2S
    Color and Shape:Solid
    Molecular weight:539.24

    Ref: TM-T23581

    1mg
    133.00€
    5mg
    570.00€
    10mg
    875.00€
  • PNU-282987 S enantiomer hydrochloride

    CAS:
    (S)-PNU-282987, selective α7 nAChR agonist; Ki=26 nM (rat), weak on other receptors except 5-HT3; Ki=930 nM.
    Formula:C14H18Cl2N2O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:301.21

    Ref: TM-T22401

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • TC-G 1004

    CAS:
    adenosine A2A receptors antagonist
    Formula:C22H27N7O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:421.5

    Ref: TM-T23435

    50mg
    2,970.00€
  • Indisetron Dihydrochloride

    CAS:
    Indisetron Dihydrochloride is a 5-HT(3) and 5-HT(4) receptor antagonist. Indisetron reduces 2-methyl-5-serotonin (HT)-induced bradycardia.
    Formula:C17H24ClN5O
    Color and Shape:Solid
    Molecular weight:349.86

    Ref: TM-T27607

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€