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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5990 products of "GPCR/G-Protein"

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  • SKF 86466 hydrochloride

    CAS:
    SKF 86466 hydrochloride is an α2-adrenoceptor antagonist.
    Formula:C11H15Cl2N
    Purity:98%
    Color and Shape:Solid
    Molecular weight:232.15

    Ref: TM-T23366

    1mg
    105.00€
    5mg
    355.00€
    10mg
    500.00€
  • BN 50341

    CAS:
    BN 50341 is an inhibitor of antithrombotic platelet activating factor.
    Formula:C32H41ClN2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:553.13

    Ref: TM-T26874

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • Rolapitant

    CAS:
    Rolapitant Hydrochloride is an oral NK1-receptor blocker that prevents nausea and has a fast onset and long half-life.
    Formula:C25H26F6N2O2
    Purity:99.86%
    Color and Shape:Solid
    Molecular weight:500.48

    Ref: TM-T3716

    1mg
    48.00€
    2mg
    63.00€
    5mg
    88.00€
    1mL*10mM (DMSO)
    96.00€
    10mg
    117.00€
    25mg
    178.00€
    50mg
    295.00€
    100mg
    442.00€
    500mg
    982.00€
  • Jmv 390-1

    CAS:
    Jmv 390-1 is an inhibitor of metallopeptidase.
    Formula:C23H35N3O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:449.54

    Ref: TM-T25554

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Diftalone

    CAS:
    Diftalone is an anti-Inflammatory agent.
    Formula:C16H12N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:264.28

    Ref: TM-T23997

    25mg
    1,369.00€
  • Mepixanox

    CAS:
    Mepixanox is an analeptic drug. It is used for treating respiratory and cardiorespiratory insufficiency.
    Formula:C20H21NO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:323.39

    Ref: TM-T16041

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • Dihydroalprenolol, (S)-

    CAS:
    Dihydroalprenolol, (S)- is a hydrogenated alprenolol derivative. It acts as a beta-adrenergic blocker.
    Formula:C15H25NO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:251.36

    Ref: TM-T23999

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Methiothepin maleate

    CAS:
    Methiothepin maleate (Metitepine) is a 5-HT1, 5-HT6, 5-HT7 serotonin receptor antagonist, which blocks serotonin autoreceptors.
    Formula:C24H28N2O4S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:472.62

    Ref: TM-T4375

    10mg
    155.00€
    25mg
    324.00€
    50mg
    439.00€
    100mg
    780.00€
  • Amitifadine hydrochloride

    CAS:
    Amitifadine hydrochloride (EB-1010 hydrochloride) is a triple reuptake inhibitor (TRI) or serotonin-norepinephrine-dopamine reuptake inhibitor (SNDRI).
    Formula:C11H12Cl3N
    Purity:98%
    Color and Shape:Solid
    Molecular weight:264.58

    Ref: TM-T2092

    1mg
    90.00€
    5mg
    215.00€
    1mL*10mM (DMSO)
    236.00€
    10mg
    356.00€
  • Befunolol HCl

    CAS:
    Befunolol is a beta blocker with intrinsic sympathomimetic activity and also acts as a β adrenoreceptor partial agonist.
    Formula:C16H22ClNO4
    Color and Shape:Solid
    Molecular weight:327.8

    Ref: TM-T26762

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • 2MeSAMP

    CAS:
    2MeSAMP is a P2Y(12) antagonist that works by inhibiting platelet activation through a P2Y(12)/G(i)-dependent mechanism.
    Formula:C11H16N5NaO7PS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:416.3

    Ref: TM-T24975

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Radioprotectin-1

    CAS:
    Radioprotectin-1 is a selective agonist of LPA2 with EC50 of 25 nM for murine LPA2 GPCR and exerts radioprotective and radiomitigative action.
    Formula:C23H19ClN2O6S
    Purity:98.63% - 99.27%
    Color and Shape:Solid
    Molecular weight:486.92

    Ref: TM-T12684

    1mg
    81.00€
    5mg
    170.00€
    1mL*10mM (DMSO)
    187.00€
    10mg
    259.00€
    25mg
    425.00€
    50mg
    562.00€
    100mg
    775.00€
  • Gyki 32887

    CAS:
    Gyki 32887 is a dopamine agonist.
    Formula:C23H28N6O6S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:516.57

    Ref: TM-T25475

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • Carcainium chloride

    CAS:
    Carcainium chloride (Carcainium (chloride)) is a derivative of Lidocaine and possesses an antitussive effect.
    Formula:C18H22ClN3O2
    Purity:99.89%
    Color and Shape:Solid
    Molecular weight:347.84

    Ref: TM-T10679

    25mg
    To inquire
    50mg
    To inquire
    10mg
    34.00€
  • PGD2-IN-1

    CAS:
    PGD2-IN-1 (PGD2-inhibitor) is an effective DP receptor antagonist (IC50:0.3 nM), a compound that can inhibit prostaglandin D2 (PGD2) signaling.
    Formula:C23H23Cl2N3O3
    Purity:98.21%
    Color and Shape:Solid
    Molecular weight:460.35

    Ref: TM-T4624

    1mg
    66.00€
    5mg
    150.00€
    1mL*10mM (DMSO)
    159.00€
    10mg
    245.00€
    25mg
    414.00€
    50mg
    610.00€
    100mg
    867.00€
    500mg
    1,738.00€
  • S 12024-2

    CAS:
    S 12024-2 (Dabelotine mesylate) is a new cognitive drug-enhancer.
    Formula:C16H26N2O5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:358.45

    Ref: TM-T24748

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • RGH 1756

    CAS:
    RGH 1756 is an atypical antipsychotic with high affinity to dopamine D(3) receptors that leads to c-Fos induction in a unique pattern.
    Formula:C26H30N4O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:462.61

    Ref: TM-T26069

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Lergotrile mesylate

    CAS:
    Lergotrile mesylate, an ergoline derivative, suppresses prolactin in vivo and in vitro.
    Formula:C18H22ClN3O3S
    Color and Shape:Solid
    Molecular weight:395.9

    Ref: TM-T25671L

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Draflazine

    CAS:
    Draflazine: ENT1 inhibitor, reverses hypersensitivity in CFA and carrageenan-induced hyperalgesia.
    Formula:C30H33Cl2F2N5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:604.52

    Ref: TM-T15167

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • RG-12915

    CAS:
    RG-12915 is a selective antagonist of 5-HT3(IC50 value of 0.16 nM).
    Formula:C20H25ClN2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:360.88

    Ref: TM-T12716

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€