
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,024 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(194 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5990 products of "GPCR/G-Protein"
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SKF 86466 hydrochloride
CAS:SKF 86466 hydrochloride is an α2-adrenoceptor antagonist.Formula:C11H15Cl2NPurity:98%Color and Shape:SolidMolecular weight:232.15BN 50341
CAS:BN 50341 is an inhibitor of antithrombotic platelet activating factor.Formula:C32H41ClN2O4Purity:98%Color and Shape:SolidMolecular weight:553.13Rolapitant
CAS:Rolapitant Hydrochloride is an oral NK1-receptor blocker that prevents nausea and has a fast onset and long half-life.Formula:C25H26F6N2O2Purity:99.86%Color and Shape:SolidMolecular weight:500.48Ref: TM-T3716
1mg48.00€2mg63.00€5mg88.00€1mL*10mM (DMSO)96.00€10mg117.00€25mg178.00€50mg295.00€100mg442.00€500mg982.00€Jmv 390-1
CAS:Jmv 390-1 is an inhibitor of metallopeptidase.Formula:C23H35N3O6Purity:98%Color and Shape:SolidMolecular weight:449.54Diftalone
CAS:Diftalone is an anti-Inflammatory agent.Formula:C16H12N2O2Purity:98%Color and Shape:SolidMolecular weight:264.28Mepixanox
CAS:Mepixanox is an analeptic drug. It is used for treating respiratory and cardiorespiratory insufficiency.Formula:C20H21NO3Purity:98%Color and Shape:SolidMolecular weight:323.39Dihydroalprenolol, (S)-
CAS:Dihydroalprenolol, (S)- is a hydrogenated alprenolol derivative. It acts as a beta-adrenergic blocker.Formula:C15H25NO2Purity:98%Color and Shape:SolidMolecular weight:251.36Methiothepin maleate
CAS:Methiothepin maleate (Metitepine) is a 5-HT1, 5-HT6, 5-HT7 serotonin receptor antagonist, which blocks serotonin autoreceptors.Formula:C24H28N2O4S2Purity:98%Color and Shape:SolidMolecular weight:472.62Amitifadine hydrochloride
CAS:Amitifadine hydrochloride (EB-1010 hydrochloride) is a triple reuptake inhibitor (TRI) or serotonin-norepinephrine-dopamine reuptake inhibitor (SNDRI).Formula:C11H12Cl3NPurity:98%Color and Shape:SolidMolecular weight:264.58Befunolol HCl
CAS:Befunolol is a beta blocker with intrinsic sympathomimetic activity and also acts as a β adrenoreceptor partial agonist.Formula:C16H22ClNO4Color and Shape:SolidMolecular weight:327.82MeSAMP
CAS:2MeSAMP is a P2Y(12) antagonist that works by inhibiting platelet activation through a P2Y(12)/G(i)-dependent mechanism.Formula:C11H16N5NaO7PSPurity:98%Color and Shape:SolidMolecular weight:416.3Radioprotectin-1
CAS:Radioprotectin-1 is a selective agonist of LPA2 with EC50 of 25 nM for murine LPA2 GPCR and exerts radioprotective and radiomitigative action.Formula:C23H19ClN2O6SPurity:98.63% - 99.27%Color and Shape:SolidMolecular weight:486.92Ref: TM-T12684
1mg81.00€5mg170.00€1mL*10mM (DMSO)187.00€10mg259.00€25mg425.00€50mg562.00€100mg775.00€Gyki 32887
CAS:Gyki 32887 is a dopamine agonist.Formula:C23H28N6O6SPurity:98%Color and Shape:SolidMolecular weight:516.57Carcainium chloride
CAS:Carcainium chloride (Carcainium (chloride)) is a derivative of Lidocaine and possesses an antitussive effect.Formula:C18H22ClN3O2Purity:99.89%Color and Shape:SolidMolecular weight:347.84PGD2-IN-1
CAS:PGD2-IN-1 (PGD2-inhibitor) is an effective DP receptor antagonist (IC50:0.3 nM), a compound that can inhibit prostaglandin D2 (PGD2) signaling.Formula:C23H23Cl2N3O3Purity:98.21%Color and Shape:SolidMolecular weight:460.35Ref: TM-T4624
1mg66.00€5mg150.00€1mL*10mM (DMSO)159.00€10mg245.00€25mg414.00€50mg610.00€100mg867.00€500mg1,738.00€S 12024-2
CAS:S 12024-2 (Dabelotine mesylate) is a new cognitive drug-enhancer.Formula:C16H26N2O5SPurity:98%Color and Shape:SolidMolecular weight:358.45RGH 1756
CAS:RGH 1756 is an atypical antipsychotic with high affinity to dopamine D(3) receptors that leads to c-Fos induction in a unique pattern.Formula:C26H30N4O2SPurity:98%Color and Shape:SolidMolecular weight:462.61Lergotrile mesylate
CAS:Lergotrile mesylate, an ergoline derivative, suppresses prolactin in vivo and in vitro.Formula:C18H22ClN3O3SColor and Shape:SolidMolecular weight:395.9Draflazine
CAS:Draflazine: ENT1 inhibitor, reverses hypersensitivity in CFA and carrageenan-induced hyperalgesia.Formula:C30H33Cl2F2N5O2Purity:98%Color and Shape:SolidMolecular weight:604.52RG-12915
CAS:RG-12915 is a selective antagonist of 5-HT3(IC50 value of 0.16 nM).Formula:C20H25ClN2O2Purity:98%Color and Shape:SolidMolecular weight:360.88
