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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5990 products of "GPCR/G-Protein"

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  • YM-17690

    CAS:
    YM-17690 is a non-analogous leukotriene agonist.
    Formula:C28H29NO7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:491.53

    Ref: TM-T29180

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • ABT-546

    CAS:
    ABT-546 is a potent, selective endothelin ETA receptor antagonist, Ki 0.46 nM for [125I]ET-1 binding.
    Formula:C30H48N2O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:532.71

    Ref: TM-T10225

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Seliforant

    CAS:
    Seliforant is a histamine H4 receptor antagonist.
    Formula:C12H21N5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:235.33

    Ref: TM-T28746

    25mg
    690.00€
    50mg
    897.00€
    100mg
    1,341.00€
  • ASP-4058 hydrochloride

    CAS:
    ASP-4058 hydrochloride: selective oral S1P1/S1P5 agonist, safe, mitigates mouse autoimmune encephalomyelitis.
    Formula:C19H13ClF6N4O2
    Color and Shape:Solid
    Molecular weight:478.78

    Ref: TM-T63141

    25mg
    887.00€
    50mg
    1,153.00€
    100mg
    1,791.00€
  • TP-680

    CAS:
    TP-680 is a antagonist of cholecystokininA receptor.
    Formula:C35H33N5O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:619.73

    Ref: TM-T28998

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Guanfacine

    CAS:
    Guanfacine is a selective agonist of the α2A receptor.
    Formula:C9H9Cl2N3O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:246.09

    Ref: TM-T22824

    25mg
    103.00€
    50mg
    170.00€
    100mg
    261.00€
  • GCGR antagonist 2

    CAS:
    Orally active GCGR antagonist 2, a furan-2-carbohydrazide, binds hGluR at 2.3 nM. Blocks glucagon, inhibits rat receptor at 0.43 nM.
    Formula:C28H26N4O2
    Color and Shape:Solid
    Molecular weight:450.53

    Ref: TM-T72621

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Ko-3290

    CAS:
    Ko-3290 is a cardioselective antagonist of β-adrenoceptors known for its antilipolytic effects in animals.
    Formula:C19H25N3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:343.42

    Ref: TM-T11763

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • S-5751

    CAS:
    S-5751, a prostanoid DP (DP1) antagonist, is used potentially for the treatment of bronchial asthma.
    Formula:C25H31NO4S
    Color and Shape:Solid
    Molecular weight:441.58

    Ref: TM-T28651

    500µg
    166.00€
    1mg
    299.00€
    5mg
    1,234.00€
  • Imiloxan hydrochloride

    CAS:
    Imiloxan hydrochloride is an α2-adrenoceptor antagonist.
    Formula:C14H17ClN2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:280.75

    Ref: TM-T22861

    10mg
    610.00€
    50mg
    2,268.00€
  • C-021 dihydrochloride

    CAS:
    C-021 dihydrochloride is a potent CCR4 antagonist. It potently inhibits functional chemotaxis in human and mouse with IC50s of 140 nM and 39 nM.
    Formula:C27H43Cl2N5O2
    Purity:98.67%
    Color and Shape:Solid
    Molecular weight:540.57

    Ref: TM-T10639

    1mg
    52.00€
    5mg
    97.00€
    1mL*10mM (DMSO)
    115.00€
    10mg
    154.00€
    25mg
    249.00€
    50mg
    374.00€
  • Gastrazole disodium

    CAS:
    Gastrazole, a CCK2 receptor antagonist, is used potentially for the treatment of pancreatic cancer.
    Formula:C34H34FN5Na2O7
    Color and Shape:Solid
    Molecular weight:689.652

    Ref: TM-T27403

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Methylcarbamyl PAF C-16

    CAS:
    Methylcarbamyl PAF C-16 (Carbamyl-PAF) is a PAF analog with PAF agonistic properties, activating inflammation in pregnancy tissues and promoting preterm birth.
    Formula:C26H55N2O7P
    Color and Shape:Solid
    Molecular weight:538.7

    Ref: TM-T36205

    1mg
    180.00€
    5mg
    718.00€
    10mg
    1,276.00€
    25mg
    2,443.00€
  • CCR4 antagonist 3-1

    CAS:
    CCR4 antagonist 3-1 is a weak inhibitor of [125I]TARC binding and CEM cell migration, with IC50 values of 1.7 μM and 6.4 μM, respectively.
    Formula:C14H12N2S
    Purity:99.87%
    Color and Shape:Solid
    Molecular weight:240.32

    Ref: TM-T60336

    1mg
    96.00€
    5mg
    205.00€
    10mg
    334.00€
    25mg
    655.00€
    50mg
    1,018.00€
    100mg
    1,378.00€
    500mg
    2,673.00€
  • Orexin receptor antagonist 2

    CAS:
    Compound 30, potent orexin antagonist with pKis of 7.69/9.78, potential for insomnia research.
    Formula:C25H31N5O2
    Color and Shape:Solid
    Molecular weight:433.55

    Ref: TM-T38139

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • Mosapramine

    CAS:
    Mosapramine is a dopamine D2-receptor antagonist.
    Formula:C28H35ClN4O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:479.06

    Ref: TM-T28086

    25mg
    2,160.00€
    50mg
    2,700.00€
    100mg
    3,600.00€
  • A 68930 hydrochloride

    CAS:
    A68930 hydrochloride is a dopamine D1 receptor agonist which can be used for the research of bronchiectasis [1].
    Formula:C16H18ClNO3
    Color and Shape:Off-White Solid
    Molecular weight:307.77

    Ref: TM-T21680

    10mg
    645.00€
  • PF-04781340

    CAS:
    PF-04781340 is an effective, selective, and CNS penetrant agonist of 5-HT2C receptor.
    Formula:C17H21N3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:267.37

    Ref: TM-T24616

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • AK-IN-1

    CAS:
    AK-IN-1: competitive adenosine inhibitor, not ATP; inhibits AK 86-89% at 2-10 µM; promising for ischaemia, inflammation, seizure research.
    Formula:C22H21N3O4
    Color and Shape:Solid
    Molecular weight:391.42

    Ref: TM-T73436

    25mg
    To inquire
    50mg
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    100mg
    To inquire
  • SC 51089 free base

    CAS:
    SC 51089 free base is a selective antagonist of the prostaglandin E2 EP1 receptor, demonstrating neuroprotective activity.
    Formula:C22H19ClN4O3
    Color and Shape:Solid
    Molecular weight:422.86

    Ref: TM-T72513

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire