
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,023 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(194 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5990 products of "GPCR/G-Protein"
Sort by
Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
YM-17690
CAS:YM-17690 is a non-analogous leukotriene agonist.Formula:C28H29NO7Purity:98%Color and Shape:SolidMolecular weight:491.53ABT-546
CAS:ABT-546 is a potent, selective endothelin ETA receptor antagonist, Ki 0.46 nM for [125I]ET-1 binding.Formula:C30H48N2O6Purity:98%Color and Shape:SolidMolecular weight:532.71Seliforant
CAS:Seliforant is a histamine H4 receptor antagonist.Formula:C12H21N5Purity:98%Color and Shape:SolidMolecular weight:235.33ASP-4058 hydrochloride
CAS:ASP-4058 hydrochloride: selective oral S1P1/S1P5 agonist, safe, mitigates mouse autoimmune encephalomyelitis.Formula:C19H13ClF6N4O2Color and Shape:SolidMolecular weight:478.78TP-680
CAS:TP-680 is a antagonist of cholecystokininA receptor.Formula:C35H33N5O4SPurity:98%Color and Shape:SolidMolecular weight:619.73Guanfacine
CAS:Guanfacine is a selective agonist of the α2A receptor.Formula:C9H9Cl2N3OPurity:98%Color and Shape:SolidMolecular weight:246.09GCGR antagonist 2
CAS:Orally active GCGR antagonist 2, a furan-2-carbohydrazide, binds hGluR at 2.3 nM. Blocks glucagon, inhibits rat receptor at 0.43 nM.Formula:C28H26N4O2Color and Shape:SolidMolecular weight:450.53Ko-3290
CAS:Ko-3290 is a cardioselective antagonist of β-adrenoceptors known for its antilipolytic effects in animals.Formula:C19H25N3O3Purity:98%Color and Shape:SolidMolecular weight:343.42S-5751
CAS:S-5751, a prostanoid DP (DP1) antagonist, is used potentially for the treatment of bronchial asthma.Formula:C25H31NO4SColor and Shape:SolidMolecular weight:441.58Imiloxan hydrochloride
CAS:Imiloxan hydrochloride is an α2-adrenoceptor antagonist.Formula:C14H17ClN2O2Purity:98%Color and Shape:SolidMolecular weight:280.75C-021 dihydrochloride
CAS:C-021 dihydrochloride is a potent CCR4 antagonist. It potently inhibits functional chemotaxis in human and mouse with IC50s of 140 nM and 39 nM.Formula:C27H43Cl2N5O2Purity:98.67%Color and Shape:SolidMolecular weight:540.57Gastrazole disodium
CAS:Gastrazole, a CCK2 receptor antagonist, is used potentially for the treatment of pancreatic cancer.Formula:C34H34FN5Na2O7Color and Shape:SolidMolecular weight:689.652Methylcarbamyl PAF C-16
CAS:Methylcarbamyl PAF C-16 (Carbamyl-PAF) is a PAF analog with PAF agonistic properties, activating inflammation in pregnancy tissues and promoting preterm birth.Formula:C26H55N2O7PColor and Shape:SolidMolecular weight:538.7CCR4 antagonist 3-1
CAS:CCR4 antagonist 3-1 is a weak inhibitor of [125I]TARC binding and CEM cell migration, with IC50 values of 1.7 μM and 6.4 μM, respectively.Formula:C14H12N2SPurity:99.87%Color and Shape:SolidMolecular weight:240.32Orexin receptor antagonist 2
CAS:Compound 30, potent orexin antagonist with pKis of 7.69/9.78, potential for insomnia research.Formula:C25H31N5O2Color and Shape:SolidMolecular weight:433.55Mosapramine
CAS:Mosapramine is a dopamine D2-receptor antagonist.Formula:C28H35ClN4OPurity:98%Color and Shape:SolidMolecular weight:479.06A 68930 hydrochloride
CAS:A68930 hydrochloride is a dopamine D1 receptor agonist which can be used for the research of bronchiectasis [1].Formula:C16H18ClNO3Color and Shape:Off-White SolidMolecular weight:307.77PF-04781340
CAS:PF-04781340 is an effective, selective, and CNS penetrant agonist of 5-HT2C receptor.Formula:C17H21N3Purity:98%Color and Shape:SolidMolecular weight:267.37AK-IN-1
CAS:AK-IN-1: competitive adenosine inhibitor, not ATP; inhibits AK 86-89% at 2-10 µM; promising for ischaemia, inflammation, seizure research.Formula:C22H21N3O4Color and Shape:SolidMolecular weight:391.42SC 51089 free base
CAS:SC 51089 free base is a selective antagonist of the prostaglandin E2 EP1 receptor, demonstrating neuroprotective activity.Formula:C22H19ClN4O3Color and Shape:SolidMolecular weight:422.86
