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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 6011 products of "GPCR/G-Protein"

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  • AP521

    CAS:
    AP521 is an agonist of the human 5-HT1A receptor (IC50: 94 nM).
    Formula:C20H19ClN2O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:402.89

    Ref: TM-T10344

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • 5-HT7 agonist 2

    CAS:
    Potent 5-HT7 agonist with 28.7 nM IC50; promising for CNS disorder research.
    Formula:C23H29N3O
    Color and Shape:Solid
    Molecular weight:363.5

    Ref: TM-T61375

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Hedgehog Antagonist VIII

    CAS:
    Hh antagonist VIII is a quinazolinyl-urea that inhibits Gli transcription in the Hh pathway, linked to cancer, with an IC50 of 70 nM.
    Formula:C23H15ClF4N4O2
    Color and Shape:Solid
    Molecular weight:490.84

    Ref: TM-T35537

    500µg
    170.00€
    1mg
    266.00€
    5mg
    489.00€
  • PD 118717

    CAS:
    PD 118717: a piperazinyl benzopyranone dopamine agonist with potential antipsychotic properties and no neurological side effects in tests.
    Formula:C20H22N4O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:366.41

    Ref: TM-T28316

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Zenidolol

    CAS:
    Zenidolol (ICI-118551) is a β2 adrenoceptor blocker with K i values: β2 (0.7 nM), β1 (49.5 nM), β3 (611 nM); used in eye disease research.
    Formula:C17H27NO2
    Color and Shape:Solid
    Molecular weight:277.4

    Ref: TM-T68385

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • NR2F1 agonist 1

    CAS:
    NR2F1 agonist 1 activates cancer cell dormancy, suppresses growth in HNSCC, and inhibits tumor growth in mice.
    Formula:C28H30N4OS
    Color and Shape:Solid
    Molecular weight:470.63

    Ref: TM-T72776

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • GBR-12935 maleate

    CAS:
    GBR-12935: dopamine reuptake inhibitor, used in research for Parkinson's and brain's dopamine pathways.
    Formula:C32H38N2O5
    Color and Shape:Solid
    Molecular weight:530.665

    Ref: TM-T70914

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Butaclamol HCl

    CAS:
    Butaclamol (AY-23,028), an unmarketed typical antipsychotic, is a research chemical that inhibits dopamine receptors.
    Formula:C25H32ClNO
    Color and Shape:Solid
    Molecular weight:397.98

    Ref: TM-T69355

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Ambucetamide

    CAS:
    Ambucetamide is an antispasmodic, it may inhibit or diminish the spontaneous rhythmical activity of the human myometrium.
    Formula:C17H28N2O2
    Color and Shape:Solid
    Molecular weight:292.42

    Ref: TM-T26614

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • (S)-Viloxazine Hydrochloride

    CAS:
    (S)-Viloxazine Hydrochloride is an S-isomer and NRI used as an antidepressant.
    Formula:C13H20ClNO3
    Purity:99.95%
    Color and Shape:Solid
    Molecular weight:273.76

    Ref: TM-T22420

    1mg
    34.00€
    5mg
    63.00€
    1mL*10mM (DMSO)
    65.00€
    10mg
    85.00€
    25mg
    117.00€
    50mg
    168.00€
    100mg
    239.00€
    500mg
    592.00€
  • Octahydroisoindole

    CAS:
    Octahydroisoindole is a natural product and a reference standard.
    Formula:C8H15N
    Purity:≥98%
    Color and Shape:Solid
    Molecular weight:125.21

    Ref: TM-TMA0432

    1g
    33.00€
    1mL*10mM (DMSO)
    33.00€
  • Lidanserin

    CAS:
    Lidanserin is an antagonist of the 5-HT2A and α1-adrenergic receptor.
    Formula:C26H31FN2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:454.53

    Ref: TM-T15754

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • Atigliflozin

    CAS:
    Atigliflozin is an antihyperglycaemic drug candidate.
    Formula:C18H22O7S
    Color and Shape:Solid
    Molecular weight:382.43

    Ref: TM-T30198

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Ro 363 hydrochloride

    CAS:
    Ro 363 hydrochloride: selective β1-adrenoceptor agonist, boosts heart contraction, lowers diastolic pressure.
    Formula:C19H26ClNO6
    Color and Shape:Solid
    Molecular weight:399.87

    Ref: TM-T61918

    100mg
    897.00€
  • Isoproterenol-d7 HCl

    CAS:
    Isoproterenol-d7: internal standard for GC/LC-MS. β1-/β2-AR agonist, not for β3. Lowers blood pressure, tackles bradydysrhythmias, asthma.
    Formula:C11H18ClNO3
    Color and Shape:Solid
    Molecular weight:254.76

    Ref: TM-T69598

    1mg
    359.00€
  • Ampreloxetine

    CAS:
    Ampreloxetine (TD-9855) is a norepinephrine reuptake inhibitor used to study neurological diseases.
    Formula:C18H18F3NO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:321.34

    Ref: TM-T26622

    25mg
    1,369.00€
  • Levobunolol hydrochloride

    CAS:
    Levobunolol hydrochloride 是一种非选择性的 β-肾上腺素受体阻滞剂,可用于治疗青光眼和上斜肌肌障碍的研究。
    Formula:C17H26ClNO3
    Purity:98.49% - >99.99%
    Color and Shape:Solid
    Molecular weight:327.85

    Ref: TM-T15742

    10mg
    62.00€
    1mL*10mM (DMSO)
    66.00€
    25mg
    92.00€
  • OPC-14523 hydrochloride

    CAS:
    OPC-14523 hydrochloride, an oral sigma/5-HT1A agonist, shows potent antidepressant activity with strong receptor affinity.
    Formula:C23H29Cl2N3O2
    Purity:99.60%
    Color and Shape:Solid
    Molecular weight:450.4

    Ref: TM-T62711

    5mg
    873.00€
    1mL*10mM (DMSO)
    925.00€
    10mg
    1,160.00€
    25mg
    1,458.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • L748337

    CAS:
    L748337 is a β3-adrenoceptor antagonist that inhibits β3-, β2-, and β1-adrenoceptors and inhibits the protective effects of CL316243.
    Formula:C26H31N3O5S
    Purity:99.67% - >99.99%
    Color and Shape:Solid
    Molecular weight:497.61

    Ref: TM-T22905

    1mg
    65.00€
  • FG-5893

    CAS:
    FG-5893 is a 5-HT1A agonist and 5-HT2 antagonist with potential anxiolytic activity.
    Formula:C27H29F2N3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:465.53

    Ref: TM-T27317

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€