
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(251 products)
- Adrenergic Receptor(3,025 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(218 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(36 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 6011 products of "GPCR/G-Protein"
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AP521
CAS:AP521 is an agonist of the human 5-HT1A receptor (IC50: 94 nM).Formula:C20H19ClN2O3SPurity:98%Color and Shape:SolidMolecular weight:402.895-HT7 agonist 2
CAS:Potent 5-HT7 agonist with 28.7 nM IC50; promising for CNS disorder research.Formula:C23H29N3OColor and Shape:SolidMolecular weight:363.5Hedgehog Antagonist VIII
CAS:Hh antagonist VIII is a quinazolinyl-urea that inhibits Gli transcription in the Hh pathway, linked to cancer, with an IC50 of 70 nM.Formula:C23H15ClF4N4O2Color and Shape:SolidMolecular weight:490.84PD 118717
CAS:PD 118717: a piperazinyl benzopyranone dopamine agonist with potential antipsychotic properties and no neurological side effects in tests.Formula:C20H22N4O3Purity:98%Color and Shape:SolidMolecular weight:366.41Zenidolol
CAS:Zenidolol (ICI-118551) is a β2 adrenoceptor blocker with K i values: β2 (0.7 nM), β1 (49.5 nM), β3 (611 nM); used in eye disease research.Formula:C17H27NO2Color and Shape:SolidMolecular weight:277.4NR2F1 agonist 1
CAS:NR2F1 agonist 1 activates cancer cell dormancy, suppresses growth in HNSCC, and inhibits tumor growth in mice.Formula:C28H30N4OSColor and Shape:SolidMolecular weight:470.63GBR-12935 maleate
CAS:GBR-12935: dopamine reuptake inhibitor, used in research for Parkinson's and brain's dopamine pathways.Formula:C32H38N2O5Color and Shape:SolidMolecular weight:530.665Butaclamol HCl
CAS:Butaclamol (AY-23,028), an unmarketed typical antipsychotic, is a research chemical that inhibits dopamine receptors.Formula:C25H32ClNOColor and Shape:SolidMolecular weight:397.98Ambucetamide
CAS:Ambucetamide is an antispasmodic, it may inhibit or diminish the spontaneous rhythmical activity of the human myometrium.Formula:C17H28N2O2Color and Shape:SolidMolecular weight:292.42(S)-Viloxazine Hydrochloride
CAS:(S)-Viloxazine Hydrochloride is an S-isomer and NRI used as an antidepressant.Formula:C13H20ClNO3Purity:99.95%Color and Shape:SolidMolecular weight:273.76Ref: TM-T22420
1mg34.00€5mg63.00€1mL*10mM (DMSO)65.00€10mg85.00€25mg117.00€50mg168.00€100mg239.00€500mg592.00€Octahydroisoindole
CAS:Octahydroisoindole is a natural product and a reference standard.Formula:C8H15NPurity:≥98%Color and Shape:SolidMolecular weight:125.21Lidanserin
CAS:Lidanserin is an antagonist of the 5-HT2A and α1-adrenergic receptor.Formula:C26H31FN2O4Purity:98%Color and Shape:SolidMolecular weight:454.53Atigliflozin
CAS:Atigliflozin is an antihyperglycaemic drug candidate.Formula:C18H22O7SColor and Shape:SolidMolecular weight:382.43Ro 363 hydrochloride
CAS:Ro 363 hydrochloride: selective β1-adrenoceptor agonist, boosts heart contraction, lowers diastolic pressure.Formula:C19H26ClNO6Color and Shape:SolidMolecular weight:399.87Isoproterenol-d7 HCl
CAS:Isoproterenol-d7: internal standard for GC/LC-MS. β1-/β2-AR agonist, not for β3. Lowers blood pressure, tackles bradydysrhythmias, asthma.Formula:C11H18ClNO3Color and Shape:SolidMolecular weight:254.76Ampreloxetine
CAS:Ampreloxetine (TD-9855) is a norepinephrine reuptake inhibitor used to study neurological diseases.Formula:C18H18F3NOPurity:98%Color and Shape:SolidMolecular weight:321.34Levobunolol hydrochloride
CAS:Levobunolol hydrochloride 是一种非选择性的 β-肾上腺素受体阻滞剂,可用于治疗青光眼和上斜肌肌障碍的研究。Formula:C17H26ClNO3Purity:98.49% - >99.99%Color and Shape:SolidMolecular weight:327.85OPC-14523 hydrochloride
CAS:OPC-14523 hydrochloride, an oral sigma/5-HT1A agonist, shows potent antidepressant activity with strong receptor affinity.Formula:C23H29Cl2N3O2Purity:99.60%Color and Shape:SolidMolecular weight:450.4L748337
CAS:L748337 is a β3-adrenoceptor antagonist that inhibits β3-, β2-, and β1-adrenoceptors and inhibits the protective effects of CL316243.Formula:C26H31N3O5SPurity:99.67% - >99.99%Color and Shape:SolidMolecular weight:497.61FG-5893
CAS:FG-5893 is a 5-HT1A agonist and 5-HT2 antagonist with potential anxiolytic activity.Formula:C27H29F2N3O2Purity:98%Color and Shape:SolidMolecular weight:465.53
