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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 6011 products of "GPCR/G-Protein"

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  • Azatadine

    CAS:
    Azatadine is histamine and cholinergic inhibitor (IC50: 6.5 nM and 10 nM, respectively).
    Formula:C20H22N2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:290.4

    Ref: TM-T22593

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • SN 003

    CAS:
    SN 003 is a CRF1 antagonist.
    Formula:C19H25N5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:355.43

    Ref: TM-T23373

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • YQA14

    CAS:
    YQA14 is a selective, high-affinity dopamine D3 receptor antagonist that inhibits cocaine self-administration in rats and mice, opioid addiction research.
    Formula:C23H27ClN4O3
    Purity:99.52%
    Color and Shape:Solid
    Molecular weight:442.94

    Ref: TM-T29195

    1mg
    77.00€
    5mg
    170.00€
    10mg
    262.00€
    25mg
    546.00€
    50mg
    855.00€
    100mg
    1,170.00€
  • EPAC 5376753

    CAS:
    EPAC 5376753 is an allosteric inhibitor of EPAC1 with an IC50 of 4 µM in Swiss 3T3 cells.
    Formula:C15H8Cl2N2O3S
    Purity:97.48%
    Color and Shape:Solid
    Molecular weight:367.21

    Ref: TM-T11212

    1mg
    49.00€
    5mg
    92.00€
    1mL*10mM (DMSO)
    105.00€
    10mg
    147.00€
    25mg
    286.00€
  • Amibegron hydrochloride

    CAS:
    Amibegron hydrochloride is a selective β3-adrenoceptor agonist (EC50: 3.5 nM for β-adrenoceptor in rat colon). It has anxiolytic and antidepressant activity.
    Formula:C22H27Cl2NO4
    Color and Shape:Solid
    Molecular weight:440.36

    Ref: TM-T10302

    25mg
    837.00€
    50mg
    1,089.00€
    100mg
    1,648.00€
  • Sograzepide

    CAS:
    Sograzepide (Netazepide) is a gastrin/CCK-B antagonist, inhibits gastrin/CCK-A activity, and can induce regression of type 1 gastric neuroendocrine tumors
    Formula:C28H30N6O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:498.58

    Ref: TM-T16906

    1mL*10mM (DMSO)
    To inquire
    1mg
    224.00€
    5mg
    623.00€
  • AChE-IN-14

    CAS:
    AChE-IN-14 inhibits eeAChE, hAChE, eqBuChE (IC50: 0.46-0.48 μM) and binds to H3R (Ki: 159.8 nM), useful for Alzheimer's research.
    Formula:C28H35NO3
    Color and Shape:Solid
    Molecular weight:433.58

    Ref: TM-T62441

    25mg
    1,927.00€
    50mg
    2,507.00€
    100mg
    3,168.00€
  • Dopamine D4 receptor antagonist-1

    CAS:
    Dopamine D4 receptor antagonist-1 can be used in schizophrenia study.
    Formula:C18H19ClN4
    Color and Shape:Solid
    Molecular weight:326.82

    Ref: TM-T60917

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Org37684

    CAS:
    5-HT2 receptors agonist
    Formula:C14H20ClNO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:269.77

    Ref: TM-T23112

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • OX2R-IN-1

    CAS:
    OX2R-IN-1: OX2R antagonist, low cytotoxicity, blood-brain barrier permeable, short half-life.
    Formula:C20H28ClN3O5S
    Color and Shape:Solid
    Molecular weight:457.97

    Ref: TM-T62855

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Prasugrel (Maleic acid)

    CAS:
    Prasugrel Maleic acid: oral P2Y12 antagonist, thienopyridine prodrug, inhibits ADP-induced platelet aggregation.
    Formula:C24H24FNO7S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:489.51

    Ref: TM-T16572

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • GSK 894281

    CAS:
    GSK 894281 is a ghrelin receptor agonist. It may produces myocardial degeneration/necrosis in rats.
    Formula:C24H28FN3O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:473.56

    Ref: TM-T27443

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • CB1R Allosteric modulator 4

    CAS:
    Modulates CB1R positively; inhibits cAMP production; strong β-arrestin-2 recruitment.
    Formula:C20H17N3O2S
    Color and Shape:Solid
    Molecular weight:363.43

    Ref: TM-T61371

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • SB357134

    CAS:
    SB357134 is a potent, selective and orally active antagonist of 5-HT6 receptor and shows nootropic effects in animal studies.
    Formula:C17H18Br2FN3O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:523.21

    Ref: TM-T28689

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • CGS-12066 maleate salt

    CAS:
    CGS-12066 maleate salt is an agonist of 5-HT1B serotonin receptor.
    Formula:C21H21F3N4O4
    Color and Shape:Solid
    Molecular weight:450.41

    Ref: TM-T27000

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • (4-Acetamidocyclohexyl) nitrate

    CAS:
    (4-Acetamidocyclohexyl) nitrate (BM121307) is an activator of guanylate cyclase.
    Formula:C8H14N2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:202.21

    Ref: TM-T10562

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • A412997

    CAS:
    A412997 is a selective agonist of dopamine D4 receptor.
    Formula:C19H23N3O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:309.41

    Ref: TM-T19691

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • GP531

    CAS:
    GP531, a second-gen adenosine regulator, is inactive at rest but boosts adenosine in ischemia.
    Formula:C16H21N5O4
    Color and Shape:Solid
    Molecular weight:347.37

    Ref: TM-T13713

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • LG 82-4-01

    CAS:
    LG 82-4-01 is an inhibitor of thromboxane (TX) synthetase.
    Formula:C10H10Cl2N2O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:309.17

    Ref: TM-T25710

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • EMD 386088 hydrochloride

    CAS:
    EMD 386088 hydrochloride is a 5-HT6 receptor agonist.
    Formula:C14H16Cl2N2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:283.2

    Ref: TM-T22763

    10mg
    677.00€