
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(251 products)
- Adrenergic Receptor(3,027 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(218 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(36 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 6011 products of "GPCR/G-Protein"
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Azatadine
CAS:Azatadine is histamine and cholinergic inhibitor (IC50: 6.5 nM and 10 nM, respectively).Formula:C20H22N2Purity:98%Color and Shape:SolidMolecular weight:290.4SN 003
CAS:SN 003 is a CRF1 antagonist.Formula:C19H25N5O2Purity:98%Color and Shape:SolidMolecular weight:355.43YQA14
CAS:YQA14 is a selective, high-affinity dopamine D3 receptor antagonist that inhibits cocaine self-administration in rats and mice, opioid addiction research.Formula:C23H27ClN4O3Purity:99.52%Color and Shape:SolidMolecular weight:442.94EPAC 5376753
CAS:EPAC 5376753 is an allosteric inhibitor of EPAC1 with an IC50 of 4 µM in Swiss 3T3 cells.Formula:C15H8Cl2N2O3SPurity:97.48%Color and Shape:SolidMolecular weight:367.21Amibegron hydrochloride
CAS:Amibegron hydrochloride is a selective β3-adrenoceptor agonist (EC50: 3.5 nM for β-adrenoceptor in rat colon). It has anxiolytic and antidepressant activity.Formula:C22H27Cl2NO4Color and Shape:SolidMolecular weight:440.36Sograzepide
CAS:Sograzepide (Netazepide) is a gastrin/CCK-B antagonist, inhibits gastrin/CCK-A activity, and can induce regression of type 1 gastric neuroendocrine tumorsFormula:C28H30N6O3Purity:98%Color and Shape:SolidMolecular weight:498.58AChE-IN-14
CAS:AChE-IN-14 inhibits eeAChE, hAChE, eqBuChE (IC50: 0.46-0.48 μM) and binds to H3R (Ki: 159.8 nM), useful for Alzheimer's research.Formula:C28H35NO3Color and Shape:SolidMolecular weight:433.58Dopamine D4 receptor antagonist-1
CAS:Dopamine D4 receptor antagonist-1 can be used in schizophrenia study.Formula:C18H19ClN4Color and Shape:SolidMolecular weight:326.82Org37684
CAS:5-HT2 receptors agonistFormula:C14H20ClNO2Purity:98%Color and Shape:SolidMolecular weight:269.77OX2R-IN-1
CAS:OX2R-IN-1: OX2R antagonist, low cytotoxicity, blood-brain barrier permeable, short half-life.Formula:C20H28ClN3O5SColor and Shape:SolidMolecular weight:457.97Prasugrel (Maleic acid)
CAS:Prasugrel Maleic acid: oral P2Y12 antagonist, thienopyridine prodrug, inhibits ADP-induced platelet aggregation.Formula:C24H24FNO7SPurity:98%Color and Shape:SolidMolecular weight:489.51GSK 894281
CAS:GSK 894281 is a ghrelin receptor agonist. It may produces myocardial degeneration/necrosis in rats.Formula:C24H28FN3O4SPurity:98%Color and Shape:SolidMolecular weight:473.56CB1R Allosteric modulator 4
CAS:Modulates CB1R positively; inhibits cAMP production; strong β-arrestin-2 recruitment.Formula:C20H17N3O2SColor and Shape:SolidMolecular weight:363.43SB357134
CAS:SB357134 is a potent, selective and orally active antagonist of 5-HT6 receptor and shows nootropic effects in animal studies.Formula:C17H18Br2FN3O3SPurity:98%Color and Shape:SolidMolecular weight:523.21CGS-12066 maleate salt
CAS:CGS-12066 maleate salt is an agonist of 5-HT1B serotonin receptor.Formula:C21H21F3N4O4Color and Shape:SolidMolecular weight:450.41(4-Acetamidocyclohexyl) nitrate
CAS:(4-Acetamidocyclohexyl) nitrate (BM121307) is an activator of guanylate cyclase.Formula:C8H14N2O4Purity:98%Color and Shape:SolidMolecular weight:202.21A412997
CAS:A412997 is a selective agonist of dopamine D4 receptor.Formula:C19H23N3OPurity:98%Color and Shape:SolidMolecular weight:309.41GP531
CAS:GP531, a second-gen adenosine regulator, is inactive at rest but boosts adenosine in ischemia.Formula:C16H21N5O4Color and Shape:SolidMolecular weight:347.37LG 82-4-01
CAS:LG 82-4-01 is an inhibitor of thromboxane (TX) synthetase.Formula:C10H10Cl2N2O3SPurity:98%Color and Shape:SolidMolecular weight:309.17EMD 386088 hydrochloride
CAS:EMD 386088 hydrochloride is a 5-HT6 receptor agonist.Formula:C14H16Cl2N2Purity:98%Color and Shape:SolidMolecular weight:283.2
