
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(251 products)
- Adrenergic Receptor(3,028 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(218 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(36 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(42 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(61 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 6012 products of "GPCR/G-Protein"
Sort by
Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
BMS-457
CAS:BMS-457 is a potent, CCR1-selective antagonist.Formula:C24H35ClN2O4Purity:98%Color and Shape:SolidMolecular weight:451Org41841
CAS:Org41841 is an agonist of luteinising hormone/chorionic gonadotropin receptor and thyroid stimulating hormone receptor and can be used to study hyperthyroidism.Formula:C19H22N4O2S2Purity:99.46% - 99.92%Color and Shape:SolidMolecular weight:402.53LY 171859
CAS:LY 171859 is an agonist of D2-receptor.Formula:C17H14O5Purity:98%Color and Shape:SolidMolecular weight:298.29KUL-7211
CAS:KUL-7211 is an β2 and β3 adrenergic receptor agonist. KUL-7211 is a potent ureteral relaxant with a relatively small hypotensive effect.Formula:C19H23NO5Purity:98%Color and Shape:SolidMolecular weight:345.39Embramine
CAS:Embramine, used as an antihistamine and anticholinergic, is a monoethanolamine.Formula:C18H22BrNOPurity:98%Color and Shape:SolidMolecular weight:348.28Indisetron Dihydrochloride
CAS:Indisetron Dihydrochloride is a 5-HT(3) and 5-HT(4) receptor antagonist. Indisetron reduces 2-methyl-5-serotonin (HT)-induced bradycardia.Formula:C17H24ClN5OColor and Shape:SolidMolecular weight:349.86Nor-SCH-12679 Maleate
CAS:Nor-SCH-12679 Maleate is a D1-dopamine receptor antagonist.Formula:C22H25NO6Purity:98%Color and Shape:SolidMolecular weight:399.44Linadryl hydrochloride
CAS:Linadryl hydrochloride may have antihistamine activity.Formula:C19H24ClNO2Color and Shape:SolidMolecular weight:333.85TSHR antagonist S37b
CAS:S37b, a less effective enantiomer of TSHR antagonist S37a, offers minor thyrotropin receptor inhibition, useful for thyroid research.Formula:C25H20N2O3S2Color and Shape:SolidMolecular weight:460.57BKM-570
CAS:BKM-570, a bradykinin antagonist, causes impressive growth inhibition of lung and prostate tumors.Formula:C34H34Cl2F5N3O3Purity:98%Color and Shape:SolidMolecular weight:698.55SB 258585 hydrochloride
CAS:SB 258585 hydrochloride is a 5-HT6 receptor antagonist.Formula:C18H23ClIN3O3SPurity:98%Color and Shape:SolidMolecular weight:523.82LRH-1 Inhibitor-3
CAS:LRH-1 Inhibitor-3 is an antagonist that inhibits LRH-1 transcriptional activity, reducing SHP, cyclin E1 (CCNE1), and G0S2,antiproliferation anticancer.Formula:C23H25N3O2Purity:98%Color and Shape:SolidMolecular weight:375.46VSN-16
CAS:VSN-16, a cannabinoid receptor agonist, is used potentially for the treatment of spasticity in multiple sclerosis.Formula:C18H26N2O3Color and Shape:SolidMolecular weight:318.41UR-PI376
CAS:UR-PI376 is a selective histamine H4 receptor agonist with low H1/H2 activity and moderate H3 affinity.Formula:C17H22N6SColor and Shape:SolidMolecular weight:342.46DR-4004
CAS:DR-4004 is a selective serotonin 5-HT7 receptor antagonist.Formula:C26H30N2OColor and Shape:SolidMolecular weight:386.53Clothixamide
CAS:Clothixamide(Clotixamide) is a thioxanthene derivative with antipsychotic activity.Formula:C24H28ClN3OSPurity:95.51%Color and Shape:SolidMolecular weight:442.02MDL 73005EF hydrochloride
CAS:5-HT1A receptor antagonistFormula:C20H27ClN2O4Purity:98%Color and Shape:SolidMolecular weight:394.89Dopamine D2 receptor antagonist-1
CAS:Dopamine D2 Receptor Antagonist-1 functions as a negative allosteric modulator (NAM) of the dopamine D2 receptor (D2R), demonstrating sub-millimolar affinity.Formula:C14H17N3SPurity:99.86%Color and Shape:SolidMolecular weight:259.37Ref: TM-T11077
1mg57.00€5mg120.00€1mL*10mM (DMSO)133.00€10mg178.00€25mg334.00€50mg492.00€100mg692.00€Esprolol hydrochloride
CAS:Esprolol is a β-adrenergic receptor antagonist.Formula:C17H28ClNO4Purity:98%Color and Shape:SolidMolecular weight:345.86GSK-239512
CAS:GSK-239512 is an antagonist of H3 receptor and can be used in studies about the treatment of cognitive dysfunction in neurodegenerative disorders.Formula:C23H27N3O2Purity:99.62% - 99.74%Color and Shape:SolidMolecular weight:377.48
