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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 6012 products of "GPCR/G-Protein"

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  • BMS-457

    CAS:
    BMS-457 is a potent, CCR1-selective antagonist.
    Formula:C24H35ClN2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:451

    Ref: TM-T26849

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Org41841

    CAS:
    Org41841 is an agonist of luteinising hormone/chorionic gonadotropin receptor and thyroid stimulating hormone receptor and can be used to study hyperthyroidism.
    Formula:C19H22N4O2S2
    Purity:99.46% - 99.92%
    Color and Shape:Solid
    Molecular weight:402.53

    Ref: TM-T16403

    1mg
    180.00€
  • LY 171859

    CAS:
    LY 171859 is an agonist of D2-receptor.
    Formula:C17H14O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:298.29

    Ref: TM-T27881

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • KUL-7211

    CAS:
    KUL-7211 is an β2 and β3 adrenergic receptor agonist. KUL-7211 is a potent ureteral relaxant with a relatively small hypotensive effect.
    Formula:C19H23NO5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:345.39

    Ref: TM-T27754

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Embramine

    CAS:
    Embramine, used as an antihistamine and anticholinergic, is a monoethanolamine.
    Formula:C18H22BrNO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:348.28

    Ref: TM-T11180

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Indisetron Dihydrochloride

    CAS:
    Indisetron Dihydrochloride is a 5-HT(3) and 5-HT(4) receptor antagonist. Indisetron reduces 2-methyl-5-serotonin (HT)-induced bradycardia.
    Formula:C17H24ClN5O
    Color and Shape:Solid
    Molecular weight:349.86

    Ref: TM-T27607

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Nor-SCH-12679 Maleate

    CAS:
    Nor-SCH-12679 Maleate is a D1-dopamine receptor antagonist.
    Formula:C22H25NO6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:399.44

    Ref: TM-T25879

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Linadryl hydrochloride

    CAS:
    Linadryl hydrochloride may have antihistamine activity.
    Formula:C19H24ClNO2
    Color and Shape:Solid
    Molecular weight:333.85

    Ref: TM-T27836

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • TSHR antagonist S37b

    CAS:
    S37b, a less effective enantiomer of TSHR antagonist S37a, offers minor thyrotropin receptor inhibition, useful for thyroid research.
    Formula:C25H20N2O3S2
    Color and Shape:Solid
    Molecular weight:460.57

    Ref: TM-T38226

    5mg
    429.00€
    25mg
    1,378.00€
    50mg
    1,791.00€
    100mg
    2,682.00€
  • BKM-570

    CAS:
    BKM-570, a bradykinin antagonist, causes impressive growth inhibition of lung and prostate tumors.
    Formula:C34H34Cl2F5N3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:698.55

    Ref: TM-T26833

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • SB 258585 hydrochloride

    CAS:
    SB 258585 hydrochloride is a 5-HT6 receptor antagonist.
    Formula:C18H23ClIN3O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:523.82

    Ref: TM-T23318

    1mg
    105.00€
    5mg
    379.00€
    10mg
    600.00€
  • LRH-1 Inhibitor-3

    CAS:
    LRH-1 Inhibitor-3 is an antagonist that inhibits LRH-1 transcriptional activity, reducing SHP, cyclin E1 (CCNE1), and G0S2,antiproliferation anticancer.
    Formula:C23H25N3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:375.46

    Ref: TM-T25758

    1mg
    75.00€
    5mg
    164.00€
    10mg
    240.00€
    25mg
    480.00€
    50mg
    683.00€
    100mg
    888.00€
    200mg
    1,243.00€
  • VSN-16

    CAS:
    VSN-16, a cannabinoid receptor agonist, is used potentially for the treatment of spasticity in multiple sclerosis.
    Formula:C18H26N2O3
    Color and Shape:Solid
    Molecular weight:318.41

    Ref: TM-T29117

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • UR-PI376

    CAS:
    UR-PI376 is a selective histamine H4 receptor agonist with low H1/H2 activity and moderate H3 affinity.
    Formula:C17H22N6S
    Color and Shape:Solid
    Molecular weight:342.46

    Ref: TM-T35003

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • DR-4004

    CAS:
    DR-4004 is a selective serotonin 5-HT7 receptor antagonist.
    Formula:C26H30N2O
    Color and Shape:Solid
    Molecular weight:386.53

    Ref: TM-T27207

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Clothixamide

    CAS:
    Clothixamide(Clotixamide) is a thioxanthene derivative with antipsychotic activity.
    Formula:C24H28ClN3OS
    Purity:95.51%
    Color and Shape:Solid
    Molecular weight:442.02

    Ref: TM-T13620

    1mg
    77.00€
    5mg
    167.00€
  • MDL 73005EF hydrochloride

    CAS:
    5-HT1A receptor antagonist
    Formula:C20H27ClN2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:394.89

    Ref: TM-T22966

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Dopamine D2 receptor antagonist-1

    CAS:
    Dopamine D2 Receptor Antagonist-1 functions as a negative allosteric modulator (NAM) of the dopamine D2 receptor (D2R), demonstrating sub-millimolar affinity.
    Formula:C14H17N3S
    Purity:99.86%
    Color and Shape:Solid
    Molecular weight:259.37

    Ref: TM-T11077

    1mg
    57.00€
    5mg
    120.00€
    1mL*10mM (DMSO)
    133.00€
    10mg
    178.00€
    25mg
    334.00€
    50mg
    492.00€
    100mg
    692.00€
  • Esprolol hydrochloride

    CAS:
    Esprolol is a β-adrenergic receptor antagonist.
    Formula:C17H28ClNO4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:345.86

    Ref: TM-T27286

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • GSK-239512

    CAS:
    GSK-239512 is an antagonist of H3 receptor and can be used in studies about the treatment of cognitive dysfunction in neurodegenerative disorders.
    Formula:C23H27N3O2
    Purity:99.62% - 99.74%
    Color and Shape:Solid
    Molecular weight:377.48

    Ref: TM-T27462

    1mg
    44.00€
    1mL*10mM (DMSO)
    87.00€
    5mg
    90.00€
    10mg
    107.00€
    25mg
    178.00€
    50mg
    268.00€
    100mg
    404.00€