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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 6011 products of "GPCR/G-Protein"

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  • VUF-10497

    CAS:
    VUF-10497: H4 receptor inverse agonist, anti-inflammatory in rats, binds human H1 receptor (pKi=7.57).
    Formula:C18H20ClN5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:373.9

    Ref: TM-T24951

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • (R)-V-0219


    (R)-V-0219: GLP-1R PAM, orally active, triggers Ca++ flux in HEK-hGLP-1R cells.
    Formula:C20H25F3N4O2
    Color and Shape:Solid
    Molecular weight:410.43

    Ref: TM-T73080

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Argtide

    CAS:
    Argtide is an luteinizing hormone releasing hormone (LHRH) antagonist.
    Formula:C80H104ClN21O14
    Color and Shape:Solid
    Molecular weight:1619.27

    Ref: TM-T70819

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • DOV-216,303 Free Base

    CAS:
    DOV-216,303 inhibits serotonin, norepinephrine, dopamine reuptake (IC50s: 14, 20, 78 nM) with antidepressant properties.
    Formula:C11H11Cl2N
    Purity:96.7%
    Color and Shape:Solid
    Molecular weight:228.12

    Ref: TM-T11087

    2mg
    43.00€
    5mg
    63.00€
    1mL*10mM (DMSO)
    64.00€
    10mg
    92.00€
    25mg
    150.00€
    50mg
    215.00€
    100mg
    321.00€
  • L-692585

    CAS:
    ghrelin receptor (GHS-R1a) agonist
    Formula:C32H37N7O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:567.68

    Ref: TM-T22898

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • Belaperidone

    CAS:
    Belaperidone, an antipsychotic, resembles clozapine, binds D(4) and 5-HT(2A) receptors, minimally extends Q-T without causing arrhythmias.
    Formula:C22H22FN3O2
    Color and Shape:Solid
    Molecular weight:379.43

    Ref: TM-T26763

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Chlorazanil

    CAS:
    Chlorazanil is a triazine-based, orally active diuretic that blocks Na+ and Cl– reabsorption in distal tubules, increases renal prostaglandin.
    Formula:C9H8ClN5
    Purity:98.89%
    Color and Shape:Solid
    Molecular weight:221.65

    Ref: TM-T13609L

    50mg
    To inquire
    10mg
    33.00€
    25mg
    33.00€
    1mL*10mM (DMSO)
    44.00€
  • UNC9995

    CAS:
    UNC9995 is a β-Arrestin-Biased Dopamine D2 Receptor agonist (β-Arrestin, EC50 = 120 nM; Emax = 88%).
    Formula:C20H21Cl2N3OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:422.37

    Ref: TM-T29066

    25mg
    887.00€
    50mg
    1,153.00€
    100mg
    1,746.00€
  • Pirolate

    CAS:
    Pirolate is a receptor of histamine H1.
    Formula:C16H15N3O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:329.31

    Ref: TM-T16541

    25mg
    1,369.00€
  • Nedocromil

    CAS:
    Nedocromil (FPL 59002) inhibits the action or formation of multiple mediators. Which including histamine, leukotriene C4 (LTC4), and prostaglandin D2 (PGD2).
    Formula:C19H17NO7
    Purity:95% - 97.34%
    Color and Shape:Solid
    Molecular weight:371.34

    Ref: TM-T16280

    5mg
    66.00€
    10mg
    90.00€
    25mg
    192.00€
    50mg
    313.00€
    100mg
    492.00€
  • RP101988


    RP101988, a potent Ozanimod metabolite, selectively targets S1PR1 with EC50 of 0.19 nM and S1PR5 at 32.8 nM.
    Formula:C23H22N4O4
    Color and Shape:Solid
    Molecular weight:418.45

    Ref: TM-T73361

    25mg
    1,260.00€
    50mg
    1,639.00€
    100mg
    2,250.00€
  • AS604872

    CAS:
    AS604872: Selective FP receptor antagonist, expedites cerebral/aorta degeneration, aids vascular disease models, inhibits uterine contraction.
    Formula:C28H25N3O3S2
    Color and Shape:Solid
    Molecular weight:515.65

    Ref: TM-T26665

    25mg
    1,369.00€
  • H3R-IN-1 Hydrochloride

    CAS:
    H3R-IN-1 Hydrochloride is an inverse agonist of histamine receptor 3( H3R ) .
    Formula:C19H24ClN3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:377.86

    Ref: TM-T11531

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Piclozotan

    CAS:
    Piclozotan (anhydrous), a 5-HT1A receptor agonist, demonstrated significant neuroprotective activity in a transient middle cerebral artery occlusion (t-MCAO)
    Formula:C23H24ClN3O2
    Purity:98.59%
    Color and Shape:Solid
    Molecular weight:409.91

    Ref: TM-T28414

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • TAS 205

    CAS:
    TAS 205 blocks H-PGDS (IC50= 55.8 nM), beats L-PGDS at 100 μM. Reduces PGD2 in human/rat basophils, dampens allergy in guinea pigs (30 mg/kg).
    Formula:C27H38N6O5
    Color and Shape:Solid
    Molecular weight:526.638

    Ref: TM-T38350

    1mg
    268.00€
    5mg
    1,161.00€
  • 2-CMDO

    CAS:
    2-CMDO is a Dopamine D2-like receptor antagonist.
    Formula:C23H23ClN2O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:442.89

    Ref: TM-T22493

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • ASP1126

    CAS:
    ASP1126 is a selective and orally active sphingosine-1-phosphate (S1P) agonist (EC50s: 7.12 nM, 517 nM for hS1P1 and hS1P3).
    Formula:C26H26ClF6NO5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:581.93

    Ref: TM-T10387

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • YM-264

    CAS:
    YM-264 is a selective and orally active antagonist of platelet-activating factor (PAF) (pKi value of 8.85 for rabbit platelet membranes).
    Formula:C28H36N4O5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:540.67

    Ref: TM-T13369

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • MS47134


    MS47134: potent MRGPRX4 agonist, EC50 = 149 nM, for pain/itch/hypersensitivity research.
    Formula:C22H29NO3
    Color and Shape:Solid
    Molecular weight:355.47

    Ref: TM-T73433

    25mg
    812.00€
    50mg
    1,054.00€
    100mg
    1,691.00€
  • S-14671

    CAS:
    S-14671: 5-HT1A agonist (pKi 9.3), potent in vivo; 5-HT2A/2C antagonist (pKi 7.8).
    Formula:C22H25N3O2S
    Color and Shape:Solid
    Molecular weight:395.52

    Ref: TM-T28641

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€