GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,024 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,029 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(159 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(443 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(83 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(42 products)
- Opioid Receptor(326 products)
- PAFR(14 products)
- PKA(52 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5972 products of "GPCR/G-Protein"
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Quinelorane
CAS:Quinelorane is dextrorotary isomer.Formula:C14H22N4Color and Shape:SolidMolecular weight:246.3516-phenoxy tetranor Prostaglandin F2α isopropyl ester
CAS:Prostaglandin F2α (PGF2α) drives luteolysis and smooth muscle contraction by activating the FP receptor.Formula:C25H36O6Color and Shape:SolidMolecular weight:432.557Calcitonin Gene Related Peptide (CGRP) II, rat TFA
<p>Rat CGRP II TFA: potent vasodilator and CGRP receptor activator for cardiovascular research.</p>Formula:C165H268F3N51O52S2Color and Shape:SolidMolecular weight:3919.33PG 931 acetate
<p>PG 931 acetate is a potent agonist of melanocortin 4 (MC4) receptors.</p>Formula:C61H89N15O13Purity:98.74%Color and Shape:SolidMolecular weight:1240.45CCR4 antagonist 3
CAS:Orally active CCR4 antagonist with piperidinyl-azetidine; IC50: 22 nM (calcium flux), 50 nM (CTX); antitumor effects.Formula:C24H27Cl2N7OColor and Shape:SolidMolecular weight:500.43LH-RH (4-10)
CAS:LH-RH (4-10), a heptapeptide from LHRH degradation, is made in macrophages and type II pneumocytes.Formula:C33H53N11O9Molecular weight:747.84ORG 2766
CAS:ORG 2766 is an ACTH 4-9 (H-Met(O)-Glu-His-Phe-D-Lys-Phe-OH) analog and neurotrophic peptide.Formula:C40H55N9O11SColor and Shape:SolidMolecular weight:869.99Anti-GLP-1R Antibody
Anti-GLP-1R Antibody is an anti-GLP-1R antibody that can be used for immunohistochemistry of paraffin sections.Purity:98.3% (SDS-PAGE); 97.2% (SEC-HPLC) - 98.3% (SDS-PAGE); 97.2% (SEC-HPLC)Color and Shape:Odour Liquid17-TFM-PGF1α
CAS:17-TFM-PGF1α (Compound 8) is a saturated prostaglandin analog. It exhibits a high affinity and receptor selectivity for the human prostaglandin F receptor (hFP receptor), with an EC50 of 85 nM.Formula:C24H35F3O5Color and Shape:SolidMolecular weight:460.53P2Y14R antagonist 3
<p>P2Y14R antagonist 3 (compound A) is an orally active P2Y14R antagonist with an IC50 of 23.60 nM and a Kd of 7.26 μM. It mitigates lung injury in mice induced by Lipopolysaccharides (LPS) and can be utilized in the study of inflammatory diseases.</p>Formula:C26H25N5O5Color and Shape:SolidMolecular weight:487.514-Hydroxy MPT
CAS:4-Hydroxy MPT (4-OH-MPT) is a serotonin-active compound that acts as an agonist for 5-HT2A and 5-HT2B receptors, with EC50 values of 3.82 nM and 3.4 nM, respectively.Formula:C14H20N2OColor and Shape:SolidMolecular weight:232.32Vapitadine
CAS:Vapitadine is a non-sedative antihistamine compound that relieves itching caused by atopic dermatitis.Formula:C17H20N4OPurity:99.77% - 99.86%Color and Shape:SoildMolecular weight:296.37Prostaglandin K1
CAS:Prostaglandin K1 (compound 46) is a structurally modified prostanoid analog with an EC50 and Ki of 2800 nM for the EP1 receptor.Formula:C20H32O5Color and Shape:SolidMolecular weight:352.47dCNP
<p>dCNP binds to NPR-B/C receptors (NPR-B/C receptor), initiating the cGMP signaling pathway and regulating vascular function. It exhibits anti-hypoxic effects by downregulating hypoxia-related genes such as HIF1α and HIF2α. Additionally, dCNP inhibits tumor stroma induction, demonstrating antifibrotic properties. It also enhances immune response by upregulating CTL, NK cells, and conventional type 1 dendritic cells in tumors.</p>Formula:C141H248N38O36S3Color and Shape:SolidMolecular weight:3147.911-39-Corticotropin (human)(TFA)
ACTH (1-39) human (TFA) is a melanocortin agonist that boosts adrenal CS production and affects the CNS and immune system.Formula:C207H308N56O58S·C2HF3O2Purity:98%Color and Shape:SolidMolecular weight:4655.16Galanin-Like Peptide (rat)
CAS:Galanin-Like Peptide (rat), a neuropeptide comprising 60 amino acids, plays a crucial role in regulating feeding, body weight, and energy metabolism [1].Formula:C288H461N87O83SPurity:98%Color and Shape:SolidMolecular weight:6502.34BQ-3020 ammonium
BQ-3020 ammonium, a selective endothelin receptor (ET B receptor) agonist, demonstrates inhibition of [125 I] ET-1 binding to ET B receptors with an IC50 of 0.2Formula:C96H140N20O25S·xNH3Purity:98%Color and Shape:SolidMolecular weight:2006.32 (free base)CB2 PET Radioligand 1
CB2 PET Radioligand 1 (compound [18F]9) is a positron emission tomography (PET) radioligand with high affinity for the human cannabinoid receptor 2 (hCB2, Ki=7.Formula:C20H19F3N4OPurity:98%Color and Shape:SolidMolecular weight:388.39Danshenol B
Danshenol B is a natural product that can be used as a reference standard.Formula:C22H26O4Color and Shape:SolidMolecular weight:354.446Cortistatin 29
Cortistatin 29: neuropeptide, relieves neuropathic pain, binds SS receptors (IC50: 2.8-13.7 nM), anti-fibrotic.Formula:C161H242N46O41S2Color and Shape:SolidMolecular weight:3539.77
