GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(248 products)
- Adrenergic Receptor(2,997 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(154 products)
- CaSR(34 products)
- Cannabinoid Receptor(216 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(191 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(40 products)
- Opioid Receptor(325 products)
- PAFR(14 products)
- PKA(59 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5957 products of "GPCR/G-Protein"
Sort by
Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
Cortistatin-14 acetate
Cortistatin-14 acetate, a neuropeptide have structural similarity to somatostatin-14, binds and exerts its function via the somatostatin receptors (sst1-sst5).
Formula:C83H118N20O20S2Purity:98.24% - 99.63%Color and Shape:SoildMolecular weight:1780.08Vapreotide
CAS:Vapreotide is an antagonist of the neurokinin-1 (NK1) receptor (IC50: 330 nM).Formula:C57H70N12O9S2Purity:98%Color and Shape:SolidMolecular weight:1131.38MK-0493 HCl
CAS:MK-0493 is a novel, potent, and selective agonist for melanocortin receptor 4 (MC4R).Formula:C30H39Cl2F2N3O2Color and Shape:SolidMolecular weight:582.55Metaterol
CAS:Metaterol is a bioactive chemical.Formula:C11H17NO2Color and Shape:SolidMolecular weight:195.2582ACTH (1-17)
CAS:ACTH (1-17), a potent MC1 receptor agonist with a Ki of 0.21 nM, is a variant of corticotropin from the pituitary gland.Formula:C95H145N29O23SPurity:98%Color and Shape:SolidMolecular weight:2093.41Urocortin II, human TFA
hUcn II, a CRF family member, targets CRF2 receptor, has time-linked stress regulation effects, showing mild motor suppression and delayed anxiolytic action.Formula:C196H340F3N63O56SPurity:98%Color and Shape:SolidMolecular weight:4564.3Methionyl-Lysyl-Bradykinin
CAS:Methionyl-Lysyl-Bradykinin (Met-Lys-Bradykinin), a Bradykinin analogue, is a kinin [1] [2] .Formula:C61H94N18O13SColor and Shape:SolidMolecular weight:1319.58Neuropeptide Y (22-36)
CAS:Neuropeptide Y (22-36) is a 15-amino acid fragment of NPY, which is abundant in the mammalian brain and involved in multiple physiological functions.Formula:C85H139N29O21Purity:98%Color and Shape:SolidMolecular weight:1903.19Antidepressant agent 4
Antidepressant agent 4: orally active, has antidepressant, anxiolytic, and nootropic effects.Formula:C19H38ClN5O2SColor and Shape:SolidMolecular weight:436.06Satavaptan
CAS:Satavaptan is a vasopressin V2 receptor antagonist. Satavaptan improves the control of ascites in cirrhosis.Formula:C33H45N3O8SColor and Shape:SolidMolecular weight:643.79FLLRN
CAS:FLLRN is a biologically active peptide serving as a PAR1-specific antagonist.Formula:C31H51N9O7Color and Shape:SolidMolecular weight:661.79Kisspeptin-10, rat
CAS:Kisspeptin-10, rat is an Endogenous ligand for the rodent kisspeptin receptor (KISS1, GPR54).
Formula:C63H83N17O15Purity:98%Color and Shape:SolidMolecular weight:1318.44Secretin, porcine
CAS:Porcine secretin: 27-amino acid peptide for diagnosing pancreatic dysfunction and gastrinoma, stimulates bicarbonate fluid.Formula:C130H220N44O41·xC2H4O2Purity:98%Color and Shape:SolidMolecular weight:N/ACAY10580
CAS:CAY10580 is a potent and selective prostaglandin EP 4 receptor agonist ( K i =35 nM).Formula:C19H35NO4Color and Shape:SolidMolecular weight:341.49tetranor-PGJM
CAS:Tetranor-PGJM is a metabolite of prostaglandin D2 and is associated with the anti-inflammatory effects of curcumin.
Formula:C16H22O6Color and Shape:SolidMolecular weight:310.346Sarafotoxin S6b
CAS:non-selective endothelin receptor agonistFormula:C110H163N27O34S5Purity:98%Color and Shape:SolidMolecular weight:2567.96Adrenomedullin (AM) (22-52), human
CAS:Adrenomedullin (ADM) is a 52-aa hypotensive peptide. Adrenomedullin (ADM) has structural similarity with amylin.Formula:C159H252N46O48Purity:98%Color and Shape:SolidMolecular weight:3576.04MrgprX2 antagonist-2
CAS:MrgprX2 antagonist-2, from patent WO2021092262A1 E163, is potent for skin inflammation studies.Formula:C17H16F5N3O3Color and Shape:SolidMolecular weight:405.325YFLLRNP
CAS:YFLLRNP is a biologically active peptide functioning as a partial agonist of PAR-1, selectively activating the G12/13 signaling pathway.Formula:C45H67N11O10Color and Shape:SolidMolecular weight:922.08[Pro34]Neuropeptide Y, porcine
CAS:[Pro34]Neuropeptide Y, porcine functions as a selective agonist for the NPY (Y1) receptor and induces vasoconstriction in the guinea pig's caval vein [1].Formula:C190H286N54O56Color and Shape:SolidMolecular weight:4222.63
