GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(248 products)
- Adrenergic Receptor(2,995 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(154 products)
- CaSR(34 products)
- Cannabinoid Receptor(216 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(191 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(40 products)
- Opioid Receptor(325 products)
- PAFR(14 products)
- PKA(59 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5957 products of "GPCR/G-Protein"
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TT-OAD2 free base
CAS:TT-OAD2 free base, a non-peptide GLP-1 receptor agonist, can treat diabetes; has an EC50 of 5 nM.Formula:C50H47Cl2N3O6Purity:98%Color and Shape:SolidMolecular weight:856.83Tocrifluor T1117
CAS:Fluorescent form of AM 251, CB1 receptor antagonistFormula:C56H53Cl2N7O5Purity:98%Color and Shape:SolidMolecular weight:974.97Peptide YY (pig)
CAS:Peptide YY (pig), a 36 amino acid gut peptide from porcine duodenum, reduces appetite via Y2 receptor, affecting digestion and the heart.Formula:C190H288N54O57Color and Shape:SolidMolecular weight:4240.72VU0453379 hydrochloride
VU0453379 hydrochloride: selective CNS-penetrant GLP-1R PAM, EC50 1.3 μM.Formula:C26H35ClN4O2Color and Shape:SolidMolecular weight:471.03TT 232
CAS:sst1/sst4 somatostatin receptors agonistFormula:C45H58N10O9S2Purity:98%Color and Shape:SolidMolecular weight:947.1315(S)-HpEPE
CAS:15(S)-HpEPE, a monohydroperoxy fatty acid, forms when 15-lipoxygenase acts on EPA, with expected biological activities akin to 15(S)-HpETE.Formula:C20H30O4Color and Shape:SolidMolecular weight:334.456Clomipramine D3
CAS:Clomipramine D3 is deuterium-labeled Clomipramine, blocking serotonin, norepinephrine, dopamine transporters (Ki: 0.14, 54, 3 nM).Formula:C19H23ClN2Purity:98%Color and Shape:SolidMolecular weight:317.87Cholic Acid 7-sulfate
CAS:Cholic acid 7-sulfate: a cholic acid metabolite with added sulfate at position 7, increased in feces of male mice with specific diets.Formula:C24H40O8SColor and Shape:SolidMolecular weight:488.64ACTH (1-17)
CAS:ACTH (1-17), a potent MC1 receptor agonist with a Ki of 0.21 nM, is a variant of corticotropin from the pituitary gland.Formula:C95H145N29O23SPurity:98%Color and Shape:SolidMolecular weight:2093.41Bim 21009
CAS:Bim 21009 is an inhibitor of gonadorelin.Formula:C74H92ClN17O13Purity:98%Color and Shape:SolidMolecular weight:1463.08Antisauvagine-30 TFA
aSvg-30 TFA: potent CRF2 receptor antagonist, Kd 1.4 nM (mCRFR2β), 150 nM (CRFR1).Formula:C163H275N48F3O49SColor and Shape:SolidMolecular weight:3764.28Adrogolide HCl
CAS:Adrogolide Hydrochloride is a selective dopamine receptor D1 agonist.Formula:C22H26ClNO4SColor and Shape:SolidMolecular weight:435.96Glucagon-like peptide 1 (1-37), human TFA
Human Glucagon-like peptide 1 (1-37) TFA is a potent GLP-1 receptor agonist derived from proglucagon.Formula:C188H276N51F3O61Purity:98%Color and Shape:SolidMolecular weight:4283.5α-Helical CRF(9-41)
CAS:Corticotropin-releasing factor receptor antagonist (Ki values are 17, 5 and 0.97 at human CRF1, rat CRF2α and mouse CRF2β receptors respectively).Formula:C166H274N46O53S2Purity:98%Color and Shape:SolidMolecular weight:3827Piperulin A
CAS:Piperulin A effectively inhibits platelet-activating factor receptor (PAFR) by specifically blocking its binding to isolated rabbit platelet plasma membranes,Formula:C23H28O6Color and Shape:SolidMolecular weight:400.46CAY10580
CAS:CAY10580 is a potent and selective prostaglandin EP 4 receptor agonist ( K i =35 nM).Formula:C19H35NO4Color and Shape:SolidMolecular weight:341.49Neuromedin N
CAS:Neuromedin N is a neuropeptide derived from the same precursor polypeptide as neurotensin, and with similar but subtly distinct expression and effects.Formula:C38H63N7O8Purity:98%Color and Shape:SolidMolecular weight:745.95(D-Phe6,Leu-NHEt13,des-Met14)-Bombesin (6-14)
CAS:(D-Phe6,Leu-NHEt13,des-Met14)-Bombesin (6-14), a bombesin (BBN) antagonist, holds potential for cancer research applications [1].Formula:C49H69N13O9Color and Shape:SolidMolecular weight:984.15PAMP-12 (unmodified)
CAS:PAMP-12 (unmodified), an endogenous peptide and potent MRGPRX2 (MrgX2) agonist (EC50=20-50 nM), induces hypotension by inhibiting catecholamine release fromFormula:C77H118N24O15Color and Shape:SolidMolecular weight:1619.91Relaxin H3 (human)
CAS:Relaxin H3 (human) is a relaxin peptide that exhibits antifibrotic effects through activation of RXFP1 [1].Color and Shape:Solid
