GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,006 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(157 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(192 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(326 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5972 products of "GPCR/G-Protein"
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Israpafant
CAS:Israpafant: PAF receptor blocker, IC50 0.84nM, hinders platelet aggregation, eosinophil activation, boosts calcium transit, anti-nephrotoxic.Formula:C28H29ClN4SColor and Shape:SolidMolecular weight:489.07Seglitide
CAS:Peptide agonist targets sst2/sst5 receptors. IC50/Kd: sst1 >1000, sst2 = 0.2-1.5, sst3 = 27-36, sst4 >127, sst5 = 0.06-23 nM.Formula:C44H56N8O7Purity:98%Color and Shape:SolidMolecular weight:808.98Vazegepant
CAS:Vazegepant is an intranasal CGRP receptor antagonist utilized for conducting acute migraine research.Formula:C36H46N8O3Purity:98.61% - 99.98%Color and Shape:SolidMolecular weight:638.80Ref: TM-T38734
1mg96.00€5mg227.00€10mg335.00€25mg567.00€50mgTo inquire100mgTo inquire1mL*10mM (DMSO)305.00€Galanin (1-15) (porcine, rat)
CAS:N-terminal galanin fragment used to mediate central cardiovascular effectsFormula:C72H105N19O20Purity:98%Color and Shape:SolidMolecular weight:1556.72NESS 0327
CAS:NESS 0327 is a high selectivity antagonist of the cannabinoid CB1 receptor. NESS 0327 is more than 60,000-fold selective for the CB1 receptor.Formula:C24H23Cl3N4OPurity:99.78%Color and Shape:SolidMolecular weight:489.82N,N′-Diferuloylputrescine
CAS:N,N′-Diferuloylputrescine acts as a pigment inhibitor, showing a 57% reduction in pigmentation.Formula:C24H28N2O6Purity:98%Color and Shape:SolidMolecular weight:440.49Sigma-1 receptor antagonist 4
Sigma-1 receptor antagonist 4 (Compound 32) is a potent σ1R antagonist that significantly enhances morphine's analgesic effects and reverses morphine-inducedFormula:C22H26N2OColor and Shape:SolidMolecular weight:334.45Dexbrompheniramine maleate
CAS:Dexbrompheniramine is an antihistamine used for hay fever and urticaria, blocking H1 receptors in the body.Formula:C20H23BrN2O4Color and Shape:SolidMolecular weight:435.318AD186
AD186, a potent and selective S1R agonist, exhibits dissociation constants (Kis) of 2.7 nM for S1R and 27 nM for S2R.Formula:C22H28N2Purity:98%Color and Shape:SolidMolecular weight:320.47PSB 0777 ammonium hydrate
PSB 0777 ammonium hydrate is a potent and selective adenosine A2A receptor full agonist, exhibiting K i values of 44.4 nM for rat A2A receptors and 360 nM forFormula:C18H20N5O7S2·NH4·75H2OPurity:98%Color and Shape:SolidMolecular weight:532.09Galanin-Like Peptide (porcine)
CAS:Galanin-Like Peptide (porcine) is a 60 amino acid neuropeptide originally isolated from the porcine hypothalamus.Formula:C281H443N81O78Purity:98%Color and Shape:SolidMolecular weight:6204.02Dp[Tyr(methyl)2,Arg8]-Vasopressin
CAS:Dp[Tyr(Me)2,Arg8]-Vasopressin is a non-selective antagonist of the peptide arginine vasopressin V1b receptor [1].Formula:C49H70N14O12S2Purity:98%Color and Shape:SolidMolecular weight:1111.3PAR-4 Agonist Peptide, amide
CAS:PAR-4 Agonist Peptide, amide (AY-NH2) is an agonist of proteinase-activated receptor-4 (PAR-4).Formula:C34H48N8O7Purity:98%Color and Shape:SolidMolecular weight:680.79Kisspeptin-10, human
CAS:Kisspeptin-10, human is an effective vasoconstrictor and inhibitor of angiogenesis.Formula:C63H83N17O14Purity:98%Color and Shape:SolidMolecular weight:1302.46215(R)-17-phenyl trinor Prostaglandin F2α
CAS:17-phenyl trinor Prostaglandin F2α N-ethyl amide (17-phenyl trinor PGF2α) is an F-series prostaglandin analog which has been approved for use as an ocularFormula:C23H32O5Color and Shape:SolidMolecular weight:388.5hNTS1R agonist-1
Compound 10, an hNTS1R agonist-1, acts as a full agonist with a strong affinity for hNTS1R (K i: 6.9 nM), showing the ability to cross the blood-brain barrier (Formula:C37H62N10O9Purity:98%Color and Shape:SolidMolecular weight:790.95Galanin-Like Peptide (rat)
CAS:Galanin-Like Peptide (rat), a neuropeptide comprising 60 amino acids, plays a crucial role in regulating feeding, body weight, and energy metabolism [1].Formula:C288H461N87O83SPurity:98%Color and Shape:SolidMolecular weight:6502.34β-CGRP, human
CAS:β-CGRP, human ,a 37-amino acid peptide,is the beta form of Calcitonin-gene-related peptide (β-CGRP), involved extensively in regulation of the cardiovascularFormula:C162H267N51O48S3Purity:98%Color and Shape:SolidMolecular weight:3793.41(D-Arg8)-Inotocin
CAS:'(D-Arg8)-Inotocin is a potent, selective, and competitive antagonist of the vasopressin receptor (V 1a R), exhibiting a binding affinity (K i) of 1.3 nM.Formula:C39H68N14O11S2Purity:98%Color and Shape:SolidMolecular weight:973.17Sulfatroxazole
CAS:Sulfatroxazole (Isosulfafurazole) (compound 12) is a selective antagonist of the ETA receptor with an IC50 of 0.26 μM.Formula:C11H13N3O3SColor and Shape:SolidMolecular weight:267.3
![Dp[Tyr(methyl)2,Arg8]-Vasopressin](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FT80073.webp&w=3840&q=75)
