GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,006 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(157 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(192 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(326 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5972 products of "GPCR/G-Protein"
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Orexin A (human, rat, mouse)
CAS:Orexin A, a 33 AA neuropeptide in humans, rats, mice, influences various processes, studied in pancreatic function and as an OX1R antagonist.Formula:C152H243N47O44S4Purity:98%Color and Shape:SolidMolecular weight:3561.1Abediterol napadisylate
CAS:Abediterol napadisylate is a novel long-acting β2-agonist in persistent asthma that is efficacy, safe, and tolerable.Formula:C60H68F4N4O14S2Purity:98%Color and Shape:SolidMolecular weight:1209.32RS 18286
CAS:RS 18286 is a LHRH antagonist.Formula:C74H101Cl2N17O14Color and Shape:SolidMolecular weight:1523.6PAR650097
PAR650097 is a humanized monoclonal antibody targeting PAR2, used in migraine research.Purity:96.67% (SEC-HPLC) - 98.83% (SEC-HPLC)Color and Shape:LiquidMolecular weight:144.1 kDaKisspeptin-54(human)
CAS:Endogenous ligand for KISS1 receptor; Ki values: rat 1.80 nM, human 1.45 nM. Inhibits tumor spread, stimulates gonadotropin release.Formula:C258H401N79O78Purity:98%Color and Shape:SolidMolecular weight:5857.49L 366811
CAS:L 366811 is a potent oxytocin antagonist.Formula:C43H56N8O6Color and Shape:SolidMolecular weight:780.95MM 54
CAS:Potent apelin receptor antagonist (Ki=82 nM, IC50=93 nM), counters [Pyr1]-Apelin-13, inhibits glioblastoma growth in mice.Formula:C70H121N29O15S4Purity:98%Color and Shape:SolidMolecular weight:1737.15EP3 antagonist 4
CAS:EP3 antagonist 4: hEP inhibitor, Ki = 2 nM, low clearance, high oral AUC, good bioavailability in rats, potential for diabetes research.Formula:C22H20Cl3FN4O3S2Purity:98%Color and Shape:SoildMolecular weight:577.91(S)-Azelastine hydrochloride
CAS:(S)-Azelastine HCl, an antihistamine, reduces H1R, M1R, M3R levels and inhibits HNEpC growth.Formula:C22H25Cl2N3OPurity:98%Color and Shape:SolidMolecular weight:418.36Cagrilintide acetate
.Cagrilintide is a long-acting amylin analog,treat diabetes and obesity by reducing appetite through activation of the AMY3R and calcitonin receptor.Formula:C196H316N54O61S2Purity:99.88%Color and Shape:SolidMolecular weight:4469.06R 50595
CAS:R 50595 is a selective non-competitive cisapride antagonist.Formula:C30H35Cl2F2N3O3Purity:98%Color and Shape:SolidMolecular weight:594.52ACT-1016-0707
CAS:ACT-1016-0707 is a selective, insurmountable LPA1 antagonist with antifibrotic and anti-inflammatory activity in lung fibrosis modelsFormula:C19H23ClN4O4SPurity:99.905%Color and Shape:SolidMolecular weight:438.93ACTH (1-14)
CAS:ACTH (1-14) is a pituitary hormone fragment that controls cortisol and androgen levels.Formula:C77H109N21O20SPurity:98%Color and Shape:SolidMolecular weight:1680.88(+)-Oxypeucedanin methanolate
CAS:(+)-Oxypeucedanin methanolate (compound 9) is a natural compound that inhibits prostaglandin E2 production [1].Formula:C17H18O6Color and Shape:SolidMolecular weight:318.32Hemokinin 1, human TFA
Hemokinin-1 is a human TFA and selective NK1 agonist; also activates NK2 & NK3 and induces opioid-independent analgesia.Formula:C56H85F3N14O16SColor and Shape:SolidMolecular weight:1299.42Yohimbic acid, ethyl ester
CAS:Yohimbic acid, ethyl ester is a biochemical with possible effects on reserpine action.Formula:C22H28N2O3Color and Shape:SolidMolecular weight:368.47GPR61 Inverse agonist 1
Compound 1, identified as a GPR61 inverse agonist, exhibits an IC50 of 11 nM, rendering it suitable for metabolism and body weight disorder research, includingColor and Shape:Odour SolidL-779976
CAS:L-779,976 is an agonist of somatostatin receptor.Formula:C33H43N7O3Color and Shape:SolidMolecular weight:585.74TLX agonist 2
TLX agonist 2 (compound 31) is a TLX agonist with an EC50 of 0.1 μM and a Kd of 0.16 μM. This compound enhances transcriptional activity by binding to TLX, thereby boosting the expression of TLX target genes. TLX agonist 2 is utilized in research on neurodegenerative diseases.Color and Shape:Odour SolidLUF6096
CAS:LUF6096 (CF-602) is a potent allosteric enhancer of the adenosine A3 receptor, exhibiting the capability to enhance agonist binding allosterically whileFormula:C22H21Cl2N3OPurity:99.5%Color and Shape:SolidMolecular weight:414.33
