GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,017 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(194 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5983 products of "GPCR/G-Protein"
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PY-60
CAS:PY-60 can effectively activate YAP transcriptional activity against annexin A2 (ANXA2).Cost-effective and quality-assured.Formula:C16H15N3O2SPurity:99.5% - 99.67%Color and Shape:SolidMolecular weight:313.37Ref: TM-T9566
1mg54.00€5mg114.00€10mg177.00€25mg356.00€50mg512.00€100mg707.00€200mg973.00€1mL*10mM (DMSO)126.00€(+)-Cloprostenol
CAS:(+)-Cloprostenol is a analogue of prostaglandin F2α (PGF2α), and is selective prostaglandin receptor agonistic.Formula:C22H29ClO6Purity:98%Color and Shape:SolidMolecular weight:424.92Parstatin(human) TFA
Parstatin(human) TFA, a cell-penetrating PAR-1 thrombin receptor agonist peptide, effectively inhibits angiogenesis, as indicated by studies [1] [2].Formula:C193H331F3N64O55S3Color and Shape:SolidMolecular weight:4581.28TGR5 agonist 1
Compound 18 (TGR5 agonist 1) is a potent agonist of TGR5, exhibiting an EC50 value of 0.31 µM [1].Formula:C28H48NNaO6SColor and Shape:SolidMolecular weight:549.74WS 9326A
CAS:WS 9326A is an antagonist of tachykinin receptor from Streptomyces violaceusniger.Formula:C54H68N8O13Purity:98%Color and Shape:SolidMolecular weight:1037.181Kisspeptin 13
CAS:Kisspeptin 13 activates GPR54 & GnRH receptors, boosts memory, and aids in Alzheimer's research.Formula:C78H107N21O18Color and Shape:SolidMolecular weight:1626.81Losulazine
CAS:Losulazine: a new antihypertensive, requires functional sympathetic nervous system; mechanism undefined.Formula:C27H22F4N4O3SPurity:98.83%Color and Shape:SolidMolecular weight:558.55GRL018-21
GRL018-21 is a potent, highly selective inhibitor of G protein-coupled receptor kinase 5 (GRK5), exhibiting an IC50 of 10 nM [1].Color and Shape:Odour SolidLys-(Des-Arg9,Leu8)-Bradykinin
CAS:Lys-(Des-Arg9,Leu8)-Bradykinin is a selective antagonist of the bradykinin B1 receptor [1].Formula:C47H75N13O11Purity:98%Color and Shape:SolidMolecular weight:998.18α-MSH TFA
CAS:α-Melanocyte-stimulating hormone (α-MSH) is a 13-amino acid peptide hormone produced by post-translational processing of proopiomelanocortin (POMC) in theFormula:C79H110F3N21O21SColor and Shape:SolidMolecular weight:1778.93Cortistatin 14, human, rat
CAS:Cortistatin 14: a neuropeptide similar to somatostatin; induces sleep, depresses neuronal activity; found in cortex, hippocampus.Formula:C81H113N19O19S2Purity:98%Color and Shape:SolidMolecular weight:1721.01Icatibant
CAS:Icatibant is a selective and specific antagonist of the bradykinin B2 receptor (IC50 and Ki: 1.07 nM and 0.798 nM respectively).Formula:C59H89N19O13SPurity:98%Color and Shape:White SolidMolecular weight:1304.52PAR-2 (1-6) (human)
CAS:PAR-2 (1-6) (human) (SLIGKV), a peptide ligand, is a PAR-2 agonist [1] .Formula:C28H53N7O8Color and Shape:SolidMolecular weight:615.76PAMP-12 (unmodified)
CAS:PAMP-12 (unmodified), an endogenous peptide and potent MRGPRX2 (MrgX2) agonist (EC50=20-50 nM), induces hypotension by inhibiting catecholamine release fromFormula:C77H118N24O15Color and Shape:SolidMolecular weight:1619.91Biotin-NeurokininA
Biotin-NeurokininA: biotinylated peptide, NK-2 receptor agonist, key in human airway and gut function.Formula:C60H94N16O16S2Color and Shape:SolidMolecular weight:1359.61(p-Iodo-Phe7)-ACTH (4-10)
CAS:(p-Iodo-Phe7)-ACTH (4-10), an ACTH derivative and MC receptor antagonist, inhibits α-MSH-induced grooming in rats.Formula:C44H58IN13O10SColor and Shape:SolidMolecular weight:1087.98SBI-810
CAS:SBI-810 is a functional selective β-arrestin-biased allosteric modulator of the neurotensin receptor 1 (NTSR1). In the presence of the endogenous ligand neurotensin (NT), SBI-810 regulates NTSR1 signaling through a G protein-specific mechanism. It fully antagonizes NT-induced Gq activation and partially antagonizes NT-induced Gi1 activation, allowing NTSR1 to activate GoA and G12.Formula:C27H34N4O2Color and Shape:SolidMolecular weight:446.59DSP-1053
CAS:Dsp-1053 is a powerful SERT (Ki=1.02 nM) inhibitor with partial 5-HT1A receptor (Ki=5.05 nM) agonizing activity.Formula:C26H32BrNO4Purity:98%Color and Shape:SolidMolecular weight:502.44PACAP (1-27), human, ovine, rat
CAS:PACAP (1-27) (the N-terminal fragment of PACAP-38) is a novel neuropeptides originally isolated from bovine hypothalamus, also found in humans and rats.Formula:C142H224N40O39SPurity:98%Color and Shape:SolidMolecular weight:3147.66Urotensin I
CAS:Urotensin I, 41-aa neuropeptide, agonist for human/rat CRF receptors, lowers blood pressure in rats, isolated from white suckers.Formula:C210H340N62O67S2Purity:98%Color and Shape:SolidMolecular weight:4869.46
