GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,017 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(194 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5983 products of "GPCR/G-Protein"
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Alosetron
CAS:Alosetron, a 5-HT3 antagonist, is used for the management of severe diarrhea-predominant irritable bowel syndrome (IBS) in women only.Formula:C17H18N4OPurity:98%Color and Shape:Crystalline PowderMolecular weight:294.36ARC 239 dihydrochloride
CAS:ARC 239 dihydrochloride is a selective α2B adrenoceptor antagonist (pKD values are 8.8, 6.7 and 6.4 at α2B, α2A, and α2D receptors respectively).Formula:C24H31Cl2N3O3Purity:99.72%Color and Shape:SolidMolecular weight:480.43Maridebart
CAS:Maridebart is a humanized IgG1-kappa monoclonal antibody that targets the GIPR (gastric inhibitory polypeptide receptor) [1].Color and Shape:LiquidVixticibart
Vixticibart is a humanized IgG4κ antibody targeting NPR1, with HumanIgG4(S228P) kappa serving as its corresponding isotype control.Color and Shape:Odour LiquidOsanetant
CAS:Osanetant produces anxiolytic- and antidepressant-like effects. Osanetant is a selective NK3 receptor antagonist. It is researched for schizophrenia.Formula:C35H41Cl2N3O2Purity:98%Color and Shape:SolidMolecular weight:606.62PSB 0777 ammonium salt
CAS:adenosine A2A receptor full agonistFormula:C18H24N6O7S2Purity:98%Color and Shape:SolidMolecular weight:500.55Xenin-8
CAS:neurotensin-like peptide that modulate pancreatic insulin and glucagon secretion/effectsFormula:C51H79N15O9Purity:98%Color and Shape:SolidMolecular weight:1046.27[D-Trp34]-Neuropeptide Y
CAS:Potent NPY Y5 receptor agonist (pEC50 = 7.82); highly selective; induces hyperphagia, body weight gain; orally active.Formula:C196H289N55O56Purity:98%Color and Shape:SolidMolecular weight:4311.77Cholecystokinin (26-33) free acid
CAS:Cholecystokinin (26-33) free acid is part of CCK and induces mild taste aversion conditioning in rats.Formula:C49H61N9O14S2Purity:99.14%Color and Shape:SoildMolecular weight:1064.19A3AR modulator 1
MRS8054 is an oral A3 adenosine receptor positive allosteric modulator, enhancing Cl-IB-MECA-induced activity.Formula:C23H25IN4Color and Shape:SolidMolecular weight:484.38BRD9 ligand-6
CAS:BRD9 ligand-6 serves as a ligand for the target protein in PROTAC applications. It is utilized in the synthesis of FHD-609.Formula:C21H21N3O4Color and Shape:SolidMolecular weight:379.41T-kinin
CAS:T-kinin (Ile-Ser-bradykinin) is a bradykinin-containing peptide utilized in inflammation research [1] [2].Formula:C59H89N17O14Molecular weight:1260.44Adatanserin hydrochloride
CAS:Adatanserin hydrochloride (WY50324 hydrochloride) is a 5-HT(1A)/5-HT(2) receptor ligand that is neuroprotective and may be used in the study of depression.Formula:C21H32ClN5OPurity:99.64%Color and Shape:SolidMolecular weight:405.96BAM (8-22) acetate
BAM (8-22) acetate, a proenkephalin A derivative, stimulates MrgprC11, hMrgprX1, and causes scratching in mice.Formula:C93H131N25O25SPurity:98.85%Color and Shape:SolidMolecular weight:2031.25Metaterol
CAS:Metaterol is a bioactive chemical.Formula:C11H17NO2Color and Shape:SolidMolecular weight:195.2582Fezolamine
CAS:Fezolamine: a new, non-tricyclic, oral antidepressant, selectively inhibits norepinephrine uptake over serotonin or dopamine.Formula:C20H23N3Purity:99.86%Color and Shape:SolidMolecular weight:305.42Israpafant
CAS:Israpafant: PAF receptor blocker, IC50 0.84nM, hinders platelet aggregation, eosinophil activation, boosts calcium transit, anti-nephrotoxic.Formula:C28H29ClN4SColor and Shape:SolidMolecular weight:489.07α-MSH acetate
α-MSH acetate is an endogenous neuromodulatory peptide derived from POMC and an agonist of MC4R (melanocortin receptor 4).Purity:99.71%Color and Shape:Odour SolidSatavaptan
CAS:Satavaptan is a vasopressin V2 receptor antagonist. Satavaptan improves the control of ascites in cirrhosis.Formula:C33H45N3O8SColor and Shape:SolidMolecular weight:643.79Protease-Activated Receptor-1, PAR-1 Agonist
CAS:Selective peptide agonist that mimics thrombin to activate PAR-1 receptor, enabling targeted receptor activation.Formula:C35H58N10O9Color and Shape:SolidMolecular weight:762.91
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