GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,023 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(194 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5986 products of "GPCR/G-Protein"
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Zoliprofen
CAS:Zoliprofen: potent, oral NSAID with anti-inflammatory, antipyretic, analgesic effects. Exceeds ibuprofen's efficacy in rats and rabbits.Formula:C12H11NO3SPurity:99.62%Color and Shape:SolidMolecular weight:249.29Ref: TM-T68025
1mg80.00€1mL*10mM (DMSO)159.00€5mg167.00€10mg244.00€25mg455.00€50mg622.00€100mg883.00€500mg1,773.00€Tiflucarbine
CAS:Tiflucarbine is a potential non-selective 5-HT agonist with antidepressant activity.Tiflucarbine dose-dependently increased the specific activity of solubleFormula:C16H17FN2SPurity:97.71%Color and Shape:SolidMolecular weight:288.38MAO-B-IN-3
MAO-B-IN-3 is a reversible, selective inhibitor of monoamine oxidase B (MAO-B) with an IC50 of 96 nM and demonstrates affinity for the 5-HT6 receptor with a KiFormula:C24H25N3O2Purity:98%Color and Shape:SolidMolecular weight:387.47[D-Trp34]-Neuropeptide Y
CAS:Potent NPY Y5 receptor agonist (pEC50 = 7.82); highly selective; induces hyperphagia, body weight gain; orally active.Formula:C196H289N55O56Purity:98%Color and Shape:SolidMolecular weight:4311.77Pasireotide (diaspartate)
CAS:Pasireotide diaspartate (SOM230) has high agonist activity at sst1/2/3/5, less at sst4; it's antiproliferative and proapoptotic.Formula:C66H80N12O17Color and Shape:SolidMolecular weight:1313.41Jmv 167
CAS:Jmv 167 is an antagonist of the Cholecystokinin receptor.Formula:C51H68N8O14SPurity:98%Color and Shape:SolidMolecular weight:1049.21O-2172
CAS:O-2172 is a carbocyclic analogue serving as an inhibitor of dopamine transporter (DAT), exhibiting IC50 values of 47 nM for DAT and 7000 nM for the serotonin transporter (SERT).Formula:C14H16Cl2O2Color and Shape:SolidMolecular weight:287.18APJ receptor agonist 10
CAS:APJ receptor agonist 10 (Compound I choline salt) modulates the activity of the APJ receptor, making it useful for pulmonary hypertension research. Compared to its free form, this compound exhibits improved bioavailability.Formula:C26H36N7O6SColor and Shape:SolidMolecular weight:574.67HTR2A antagonist 1
HTR2A antagonist 1 (Compound 15f) is an HTR2A antagonist with an IC50 of 42.79 nM. It induces sub-G1 cell cycle arrest and apoptosis in colorectal cancer cells by activating the p53/p21/caspase 3 signaling pathway. HTR2A antagonist 1 exhibits good liver microsomal stability and is useful for colorectal cancer research.Formula:C35H43Cl2F2N5O4Color and Shape:SolidMolecular weight:706.65Vapitadine
CAS:Vapitadine is a non-sedative antihistamine compound that relieves itching caused by atopic dermatitis.Formula:C17H20N4OPurity:99.77% - 99.86%Color and Shape:SoildMolecular weight:296.37CAY10606
CAS:CAY10606 has a wide range of applications in life science related research.
Formula:C22H18ClNO3Color and Shape:SolidMolecular weight:379.84Adrenomedullin (AM) (22-52), human TFA
Adrenomedullin (AM) human (22-52) is a truncated NH2 TFA-modified adrenal medullary receptor antagonist.Formula:C161H253N46F3O50Purity:98%Color and Shape:SolidMolecular weight:3690.06D-Epinephrine
CAS:D-Epinephrine: a hormone and drug, boosts heart rate, muscle blood flow, pupil size, and sugar levels in stress responses.
Formula:C9H13NO3Color and Shape:SolidMolecular weight:183.2S1PR1 modulator 1
CAS:S1PR1 modulator 1 is a selective inhibitor of S1PR1 with a pIC50 of 7.6.Formula:C23H24N2O3SPurity:99.69%Color and Shape:SolidMolecular weight:408.51P2Y14 antagonist 1
P2Y14 antagonist 1 (compound 45) is a highly selective and orally active P2Y14 receptor antagonist with an IC50 value of 0.70 nM. It demonstrates significant anti-inflammatory effects by effectively reducing pulmonary infiltration of immune cells and inflammatory responses through the inhibition of the NLRP3 signaling pathway. P2Y14 antagonist 1 is suitable for studying acute lung injury.Formula:C24H21N3O3Color and Shape:SolidMolecular weight:399.442Vapreotide
CAS:Vapreotide is an antagonist of the neurokinin-1 (NK1) receptor (IC50: 330 nM).Formula:C57H70N12O9S2Purity:98%Color and Shape:SolidMolecular weight:1131.38Olcegepant hydrochloride
CAS:Olcegepant hydrochloride (BIBN-4096 hydrochloride) is a selective calcitonin gene-related peptide 1 (CGRP1) receptor antagonist.Formula:C38H48Br2ClN9O5Purity:99.69%Color and Shape:SolidMolecular weight:906.11ACTH (4-11)
CAS:ACTH (4-11) is a peptide fragment of adrenocorticotropic hormone, a peptide hormone found in the brain that is involved in the biological stress response.Formula:C50H71N15O11SPurity:98%Color and Shape:SolidMolecular weight:1090.26Protease-Activated Receptor-1 antagonist 2
CAS:Orally active PAR-1 antagonist with 7 nM IC50; potential for CVD research.Formula:C24H23F2N3O2Color and Shape:SolidMolecular weight:423.46Cholecystokinin Octapeptide, desulfated TFA
CAS:Cholecystokinin Octapeptide, desulfated TFA, is a synthetic octapeptide derived from Cholecystokinin (CCK) that has undergone desulfation.Formula:C51H63F3N10O15S2Color and Shape:SolidMolecular weight:1177.24
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