GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,022 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(194 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5983 products of "GPCR/G-Protein"
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ACTH (11-24)
CAS:ACTH (11-24) is an adrenocorticotrophin fragment, stimulates cortisol, and antagonizes ACTH (1-39)/(1-10) in adrenal cells.Formula:C77H134N24O16Purity:98%Color and Shape:SolidMolecular weight:1652.04AZP-531
CAS:Azp-531 is a disacylated ghrelin used to improve blood sugar control and weight loss.Formula:C40H63N15O13Purity:98%Color and Shape:SolidMolecular weight:962.02Xanthine amine congener dihydrochloride
CAS:XAC dihydrochloride is an Adenosine A1 and A2 receptor antagonist with IC50s of 1.8 nM and 114 nM, also a mouse convulsant.Formula:C21H30Cl2N6O4Color and Shape:SolidMolecular weight:501.41Triazolomethylindole-3-acetic acid
CAS:Triazolomethylindole-3-acetic acid is a metabolite of Rizatriptan, which acts as an agonist for the serotonin (5-HT) receptor subtypes 5-HT1B and 5-HT1D.Formula:C13H12N4O2Color and Shape:SolidMolecular weight:256.26(Ala13)-Apelin-13
CAS:(Ala13)-Apelin-13 is a useful organic compound for research related to life sciences. The catalog number is T35374 and the CAS number is 568565-11-7.Formula:C63H107N23O16SPurity:98%Color and Shape:SolidMolecular weight:1474.75Levocarnitine propionate hydrochloride
CAS:Levocarnitine propionate hydrochloride (ST-261) is used for the treatment of the deterioration of renal function, congestive heart failure, and other diseases.Formula:C10H20ClNO4Purity:90% - 99.77%Color and Shape:SolidMolecular weight:253.72Eledoisin Related Peptide
CAS:Eledoisin Related Peptide (Eledoisin RP) is a tachykinin receptor ligand.Formula:C34H58N8O6SPurity:98%Color and Shape:SolidMolecular weight:706.94Brexpiprazole S-oxide
CAS:Brexpiprazole S-oxide is the main metabolite of Brexpiprazole, a human 5-HT1A and dopamine receptor partial agonist (Ki: 0.12, 0.3 nM).Formula:C25H27N3O3SPurity:98%Color and Shape:SolidMolecular weight:449.57Succinate/succinate receptor antagonist 1
CAS:Potent succinate receptor antagonist with IC50 of 20 μM; blocks gingival succinate signaling, may treat periodontal disease.
Formula:C17H15N3OPurity:99.53%Color and Shape:SoildMolecular weight:277.325-HT2C agonist-4
CAS:Compound 3i, a 5-HT2C agonist-4, acts as an agonist for the 5-HT2C receptor with an EC50 of 5.7 nM. It is capable of reducing locomotor activity in zebrafish larvae.Formula:C24H25N5OColor and Shape:SolidMolecular weight:399.49HL2-m5
CAS:HL2-m5 is an inhibitor of the sonic hedgehog/patched (Shh/PTCH1) interaction, with a Kd for Shh of 170 nM. It effectively inhibits the activation of the Hedgehog signaling pathway and the transcription of Gli-controlled genes, with an IC50 of 230 nM.Formula:C70H101N15O24S3Color and Shape:SolidMolecular weight:1632.83Amisulpride hydrochloride
CAS:Amisulpride is an antagonist of 5-HT7 receptor and dopamine D2 and D3 receptors. It modulates beta 2- arresting signaling and increases neurite outgrowth.Formula:C17H28ClN3O4SColor and Shape:SolidMolecular weight:405.94Spns2-IN-2
Spns2-IN-2 (compound 3a) is an inhibitor of SPNS2.Formula:C22H30ClN3O2Color and Shape:SolidMolecular weight:403.95HDAC6-IN-49
HDAC6-IN-49 (Compound 3) is an inhibitor of HDAC, with IC50 values of 0.012 and 0.735 µM against HDAC6 and HDAC1, respectively. Additionally, it inhibits MAO-B, cholinesterase (ChE), histamine receptor (H3R), and serotonin 6 receptor (5-HT6R). HDAC6-IN-49 exhibits neuroprotective effects in SH-SY5Y cells and enhances cognitive functions and motor abilities in fruit fly models of Parkinson's disease and C. elegans models of Alzheimer's disease.Color and Shape:Odour SolidAdrenocorticotropic Hormone (ACTH) (1-39), rat
CAS:ACTH (1-39), rat: potent MC2 agonist, forms fragments in vitro, isolated by HPLC, characterized by amino acids and NH2-terminus.Formula:C210H315N57O57SPurity:98%Color and Shape:SolidMolecular weight:4582.23RF9 acetate
RF9 acetate is an effective and selective antagonist of Neuropeptide FF receptor with Ki values of 58 and 75 nM for hNPFF1R and hNPFF2R, respectively.Formula:C28H42N6O5Purity:99.77%Color and Shape:SolidMolecular weight:542.67Ref: TM-T16738L
1mg65.00€5mg125.00€1mL*10mM (DMSO)167.00€10mg182.00€25mg325.00€50mg467.00€100mg645.00€200mg868.00€β-CGRP, human
CAS:β-CGRP, human ,a 37-amino acid peptide,is the beta form of Calcitonin-gene-related peptide (β-CGRP), involved extensively in regulation of the cardiovascularFormula:C162H267N51O48S3Purity:98%Color and Shape:SolidMolecular weight:3793.4111-deoxy Prostaglandin E2
CAS:11-deoxy PGE2 is a synthetic PGE2 analog, a potent bronchoconstrictor, 5-30x stronger than PGF2α on human respiratory muscles.Formula:C20H32O4Color and Shape:SolidMolecular weight:336.47CB1R agonist 1
CB1R agonist 1 (Compound '1350) is a potent full agonist of the cannabinoid-1 receptor (CB1R) with a Ki value of 0.95 nM. It demonstrates significant pain-relieving effects in various pain models, including acute thermal pain, inflammatory pain, and neuropathic pain.Formula:C20H18F3N3O3SColor and Shape:SolidMolecular weight:437.435α-CGRP, rat
CAS:Endogenous neuropeptide, potent vasodilatorFormula:C162H262N50O52S2Purity:98%Color and Shape:SolidMolecular weight:3806.25
