GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,023 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(194 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5988 products of "GPCR/G-Protein"
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Cagrilintide
CAS:Cagrilintide is a long-acting amylin analogue acting as a dual agonist of the amylin receptor and calcitonin receptor, reducing body weight and food intake.Formula:C194H312N54O59S2Color and Shape:SolidMolecular weight:4409.01(D-Phe7)-α-MSH
CAS:(D-Phe7)-α-MSH is an α-MSH analogue [1] .Formula:C77H109N21O19SColor and Shape:SolidMolecular weight:1664.88[Sar4] Substance P (4-11)
'[Sar4] Substance P (4-11) is a C-terminus fragment and agonist of Substance P.'Formula:C44H65N11O10SColor and Shape:SolidMolecular weight:940.12Satoreotide
CAS:Satoreotide (JR11) is an SSTR2 antagonist, typically conjugated with radiolabeled chelators for use in neuroendocrine tumor imaging [1].Formula:C58H72ClN15O14S2Color and Shape:SolidMolecular weight:1302.87FSLLRY-NH2
CAS:PAR2 antagonist; counters taxol effects, PKC in mice; inhibits ERK, collagen in fibroblasts; lessens dermatophyte itch in mice.Formula:C39H60N10O8Purity:98%Color and Shape:SolidMolecular weight:796.97Vanicoside E
CAS:Vanicoside E is an antioxidant and antitumor agent. Vanicoside E inhibits L-Tyrosine and L-DOPA with IC 50 s of 45.23 μM and 189.96 μM, respectively [1] [2] .Formula:C53H52O22Color and Shape:SolidMolecular weight:1040.97Neuropeptide S(Mouse) TFA
Neuropeptide S(Mouse) TFA: Endogenous NPSR agonist, EC50 3 nM, boosts Ca2+, activity, wakefulness, and lowers mouse anxiety.
Formula:C92H157F3N34O29Color and Shape:SolidMolecular weight:2296.49GHRF, bovine
CAS:bGRF(1-44)-NH2 is a bovine GH-releasing factor that stimulates GH release and synergizes with Hydrocortisone.Formula:C220H366N72O66SColor and Shape:SolidMolecular weight:5104.72BMS 193885
CAS:BMS 193885 is a selective and competitive neuropeptide Y(1) receptor antagonist with affinity of 3.3 nM.Formula:C36H48N4O9Purity:98%Color and Shape:SolidMolecular weight:680.7912-epi Leukotriene B4
CAS:LTB4 is made enzymatically (12(R)-specific) and non-enzymatically (6-trans-12-epi mix). 12-epi LTB4 has low receptor activity.Formula:C20H32O4Color and Shape:SolidMolecular weight:336.4722-Methyl-N,N-dimethyltryptamine
CAS:2-Methyl-N,N-dimethyltryptamine (2,N,N-TMT, compound 15) exhibits binding affinity for the serotonin (5-HT) receptor, with a pA2 value of 6.04. It plays a significant role in neurological disease research.Formula:C13H18N2Color and Shape:SolidMolecular weight:202.3Ki16198
CAS:Ki16198, a methyl ester derivative of Ki16425, blocks LPA1/3, weak on LPA2; inactive on LPA4/5/6. Ki values: 0.34 μM (LPA1), 0.93 μM (LPA3).Formula:C24H25ClN2O5SPurity:98.09%Color and Shape:SolidMolecular weight:488.98Adrenotensin (human)
CAS:Adrenotensin: human 153-185 fragment of Adrenomedullin precursor, a 52-amino acid peptide in CGRP hormone family.Formula:C143H224N42O43Color and Shape:SolidMolecular weight:3219.56PAMP-12 (unmodified)
CAS:PAMP-12 (unmodified), an endogenous peptide and potent MRGPRX2 (MrgX2) agonist (EC50=20-50 nM), induces hypotension by inhibiting catecholamine release fromFormula:C77H118N24O15Color and Shape:SolidMolecular weight:1619.91K41498
CAS:Potent CRF2α/β antagonist; Ki: 0.66/0.62 nM, weak for CRF1 (425 nM). Blocks sauvagine in hCRF2 cells and urocortin hypotension in rats.Formula:C162H276N48O46Purity:98%Color and Shape:SolidMolecular weight:3632.26a-Helical Corticotropin Releasing Factor (12-41)
CAS:α-Helical CRF (12-41), a 30-aa analog, curbs CRF's ACTH-stimulating effect.Formula:C152H251N43O47S2Color and Shape:SolidMolecular weight:3497.01LCKLSL acetate
LCKLSL acetate is a potent AnxA2 inhibitor, blocking tPA binding and plasmin production, with anti-angiogenic effects.Formula:C32H61N7O10SPurity:99.9%Color and Shape:SolidMolecular weight:735.93Mesoridazine Besylate
CAS:Mesoridazine Besylate (Serentil), a piperidine antipsychotic and phenothiazine, treats schizophrenia; it's a thioridazine metabolite.Formula:C27H32N2O4S3Purity:98.87%Color and Shape:SolidMolecular weight:544.75MK-7246 S enantiomer
MK-7246 S enantiomer is a potent and selective CRTH2 antagonist.Formula:C21H21FN2O4SPurity:98%Color and Shape:SolidMolecular weight:416.47Guanylin(human) TFA
Guanylin (human) TFA, a 15-amino acid peptide, activates intestinal guanylate cyclase, regulating electrolyte and water transport via cGMP.Color and Shape:Liquid
