GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,023 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(194 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5990 products of "GPCR/G-Protein"
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Histamine & Melatonin Receptor-Targeted Compound Library
A unique collection of xnum compounds targeting histaminergic receptor and melatonin receptor for high throughput screening (HTS) and high content screening (HCS
Color and Shape:Odour SolidANXA3 degrader 1
ANXA3 degrader 1 (Compound 18a5) is a highly selective ANXA3 degrader with activity against cancer cells. It demonstrates significant inhibitory effects in a triple-negative breast cancer (TNBC) tumor xenograft model, with a tumor growth inhibition (TGI) rate of 96%.Formula:C30H32N6O2S2Color and Shape:SolidMolecular weight:572.74BMS-753426
CAS:BMS-753426 is a potent and orally bioavailable antagonist of CCR2 .
Formula:C25H33F3N6O2Color and Shape:SolidMolecular weight:506.574(Iso)-RJW100
CAS:Potent LRH-1/NR5A2 and SF-1/NR5A1 agonist; pEC50: 6.4 (LRH-1), 7.2 (SF-1).Formula:C28H34OPurity:99.79%Color and Shape:SoildMolecular weight:386.57Ref: TM-T64363
1mg109.00€5mg241.00€1mL*10mM (DMSO)259.00€10mg354.00€25mg532.00€50mg745.00€100mg1,018.00€500mg2,035.00€CYN 154806
CAS:CYN 154806: potent sst2 antagonist; pIC50: 8.58 (sst2), 5.41 (sst1), 6.07 (sst3), 5.76 (sst4), 6.48 (sst5).Formula:C56H68N12O14S2Purity:98%Color and Shape:SolidMolecular weight:1197.34Pexopiprant
CAS:Pexopiprant, a potent oral antagonist of the prostaglandin D2 receptor 2 (DP2) with a K i value less than 100nM, is a valuable compound for asthma research.Formula:C21H17Cl2F2NO4Color and Shape:SolidMolecular weight:456.27Cianopramine hydrochloride
CAS:Cianopramine hydrochloride is a bio-active chemical.Formula:C20H24ClN3Color and Shape:SolidMolecular weight:341.88Zalospirone
CAS:Zalospirone is a 5-HT1A receptor agonist that can be used to study anxiety disorders and major depressive disorder.Formula:C24H29N5O2Purity:98.24% - 99.82%Color and Shape:SolidMolecular weight:419.52Neurokinin B
CAS:NKB, a tachykinin peptide, impacts human functions like gonadotropin-releasing hormone secretion.Formula:C55H79N13O14S2Purity:98%Color and Shape:SolidMolecular weight:1210.42HS024 TFA
HS024, a selective MC4 receptor antagonist, exhibits affinity with Ki values of 0.29, 3.29, 5.45, and 18.6 nM for MC4, MC5, MC3, and MC1 receptors, respectivelyFormula:C60H80F3N19O12S2Color and Shape:SolidMolecular weight:1380.52Tetrahydro-β-carboline
CAS:Compound Fr12161, with CAS No. 16502-01-5, is a fragment molecule that serves as an important scaffold for molecular linking, expansion, and modification. Compound Fr12161 provides a structural basis and research tool for the design and screening of novel drug candidates, and is commonly used in drug discovery, drug synthesis, and related research.Formula:C11H12N2Purity:96.31%Color and Shape:Tan SolidMolecular weight:172.2264Guanylin(human)
CAS:Peptide that activates gut guanylyl cyclase, secreted by GI mucosa, regulates water and electrolytes in gut and kidneys.Formula:C58H87N15O21S4Purity:98%Color and Shape:SolidMolecular weight:1458.65HAEGTFTSD
CAS:HAEGTFTSD is GLP-1's initial segment; GLP-1 (7-36) amide, tied to food intake, stems from preproglucagon in L-cells.Formula:C40H57N11O17Purity:98%Color and Shape:SolidMolecular weight:963.94Prostaglandin H1
CAS:Prostaglandin H1 is the cyclooxygenase metabolite of DGLA, a CRTh2 agonist and a precursor of a family of 1 anti-inflammatory prostaglandins.Formula:C20H34O5Color and Shape:SolidMolecular weight:354.487Imnopitant dihydrochloride
CAS:Imnopitant dihydrochloride is a neurokinin NK1 receptor antagonist [1] .Formula:C28H30Cl2F6N4OColor and Shape:SolidMolecular weight:623.46[D-Phe12]-Bombesin
CAS:Bombesin receptor antagonist
Formula:C74H112N22O18SPurity:98%Color and Shape:SolidMolecular weight:1629.88Dehydro Aripiprazole (hydrochloride)
CAS:Dehydro aripiprazole, an active atypical antipsychotic metabolite of aripiprazole, is formed by CYP3A4 and CYP2D6.Formula:C23H26Cl3N3O2Color and Shape:SolidMolecular weight:482.83M40
CAS:Potent, non-selective galanin receptor antagonist (Ki values are 1.82 and 5.1 nM at GAL1 and GAL2 respectively) that inhibits galanin (1-29) binding in ratFormula:C94H145N23O24Purity:98%Color and Shape:SolidMolecular weight:1981.33Neuropeptide Y (human)
CAS:Neuropeptide Y (29-64), amide, human is a biologically active 36-amino acid peptide.Formula:C189H285N55O57SPurity:98%Color and Shape:SolidMolecular weight:4271.68PACAP (6-38), human, ovine, rat
CAS:PACAP (6-38) in humans, sheep, rats: a strong inhibitor of PACAP 38, outperforms PACAP (6-27) in blocking PACAP-27-induced adenylate cyclase.Formula:C182H300N56O45SPurity:98%Color and Shape:SolidMolecular weight:4024.74
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