GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,024 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(194 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5990 products of "GPCR/G-Protein"
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GR 94800
CAS:Potent and selective tachykinin NK2 receptor antagonistFormula:C49H61N9O8Purity:98%Color and Shape:SolidMolecular weight:904.0824-Hydroxy MET
CAS:4-Hydroxy MET (4-HO-MET) is a tryptamine-based new psychoactive substance (NPS), structurally similar to the endogenous neurotransmitter serotonin. It has hallucinogenic properties that affect mood, movement, and cognitive functions.Formula:C13H18N2OColor and Shape:SolidMolecular weight:218.3Navafenterol saccharinate
CAS:AZD-8871 saccharinate is a dual-acting bronchodilator which may be useful in the treatment of Chronic Obstructive Pulmonary Disease (COPD).Formula:C45H47N7O9S3Color and Shape:SolidMolecular weight:926.09des-Gln14-Ghrelin
CAS:Endogenous rat ghrelin gene variant binds GHS-R1a; strong Ca2+ release (EC50=2.4 nM); boosts GH secretion in vivo.Formula:C142H237N43O40Purity:98%Color and Shape:SolidMolecular weight:3186.7GRK-IN-1
CAS:4-Amino-5-(bromomethyl)-2-methylpyrimidine used in vitamin B1 analogs and esters synthesis.
Formula:C6H10Br3N3Color and Shape:SolidMolecular weight:363.87919(S)-HETE
CAS:19-HETE, a CYP450 arachidonic acid metabolite from kidneys, consists of 70% (S) and 30% (R) isomers and dilates renal vessels.Formula:C20H32O3Color and Shape:SolidMolecular weight:320.473Eloralintide sodium
Eloralintide sodium (LY-3841136 sodium) is an AMYR (amylin receptor) agonist applicable for studying type 2 diabetes and obesity.Formula:C201H319N49O65S2·xNaPurity:98.66%Color and Shape:SolidMolecular weight:4526.1 (free base)Tienoxolol FA
Tienoxolol FA, a beta-blocker for treating heart disease, hypertension, and ischemia.Formula:C22H30N2O7SPurity:97.05% - 98.53%Color and Shape:SoildMolecular weight:466.55JNJ-5207787
CAS:JNJ-5207787, a blood-brain barrier-crossing Y2 receptor antagonist, is >100x selective against Y1/Y4/Y5 and inhibits human/rat Y2 with pIC50s of 7.0/7.1.Formula:C32H38N4O2Purity:98%Color and Shape:SolidMolecular weight:510.67CCR6 antagonist 2
CCR6 antagonist2 (Compound 20c) acts as a CCR6 antagonist with a Ki of 1.1 nM. It inhibits CCL20-induced calcium influx with an IC50 of 4.9 nM and suppresses the chemotactic migration of CCR6+ T cells with an IC50 of 190 nM.Formula:C19H24N4O4Color and Shape:SolidMolecular weight:372.42GLP-2(1-33)(human)
CAS:GLP-2(1-33) (human) is an enteroendocrine hormone which stimulates the growth of the intestinal epithelium.Formula:C165H254N44O55SPurity:98%Color and Shape:SolidMolecular weight:3766.19Urocortin, rat
CAS:Endogenous CRF agonist. Ki values are 13, 1.5 and 0.97 nM for hCRF1, rCRF2α and mCRF2β respectively.Formula:C206H338N62O64Purity:98%Color and Shape:SolidMolecular weight:4707.26Amylin (1-37), human acetate
Amylin (1-37), human acetate, a peptide hormone containing 37 amino acids secreted by the pancreas in conjunction with insulin, inhibits glucagon secretion.Purity:96.21%Color and Shape:Odour SolidIloperidone metabolite P95
CAS:Iloperidone metabolite P95, a non-brain penetrating compound, binds 5-HT2A, α1-, α2B-, α2C-receptors with Ki of 7.08-83.18 nM.Formula:C23H25FN2O5Color and Shape:SolidMolecular weight:428.46Beraprost
CAS:Beraprost is a stable prostacyclin analog.Formula:C24H30O5Color and Shape:SolidMolecular weight:398.4920-Carboxy-Leukotriene B4
CAS:20-COOH LTB4, a metabolite of LTB4, binds BLT1 receptor and inhibits LTB4-induced neutrophil responses.Formula:C20H30O6Color and Shape:SolidMolecular weight:366.45TAK-615
CAS:TAK-615 is commonly used to study pulmonary fibrosis and is a negative allosteric modulator of LPA1 receptors.Formula:C25H22FNO4Purity:99.73%Color and Shape:SolidMolecular weight:419.44Ref: TM-T9699
1mg72.00€5mg160.00€1mL*10mM (DMSO)172.00€10mg245.00€25mg405.00€50mg572.00€100mg772.00€500mg1,539.00€11-deoxy Prostaglandin F1α
CAS:11-deoxy PGF1α is a synthetic analog of PGF1α.Formula:C20H36O4Color and Shape:SolidMolecular weight:340.5048-iso Prostaglandin E1
CAS:8-iso Prostaglandin E1 causes spasm in the pulmonary veins of dogs and also acts as a vasodilator.
Formula:C20H34O5Color and Shape:Light Yellow Crystalline SolidMolecular weight:354.48GR 64349
CAS:Potent NK2 agonist, EC50=3.7 nM in rat colon; >1000x selectivity over NK1, >300x over NK3; effective in vivo.Formula:C42H68N10O11SPurity:98%Color and Shape:SolidMolecular weight:921.12
