GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(251 products)
- Adrenergic Receptor(3,029 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(218 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(36 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(42 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(61 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 6012 products of "GPCR/G-Protein"
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Tirzepatide hydrochloride
Tirzepatide HCl is a dual GIP and GLP-1 receptor agonist.Formula:C225H349N48O68ClPurity:98%Color and Shape:SolidMolecular weight:4849.91Lisuride maleate
CAS:Lisuride maleate is a non-selective dopamine agonist and G-protein-biased 5-HT2A receptor agonist capable of blocking prolactin release.Formula:C24H30N4O5Purity:99.85%Color and Shape:SolidMolecular weight:454.52Ref: TM-T8775
1mg204.00€5mg627.00€1mL*10mM (DMSO)627.00€10mg898.00€25mg1,346.00€50mg1,745.00€100mg2,382.00€7-Hydroxy-PIPAT maleate
CAS:7-Hydroxy-PIPAT maleate is a D3R agonist.Formula:C16H22INOColor and Shape:SolidMolecular weight:371.262Apelin-36(human)
CAS:Endogenous APJ agonist, EC50=20nM, regulates cardiovascular function, fluid balance, and feeding; blocks certain HIV strains.Formula:C184H297N69O43SPurity:98%Color and Shape:SolidMolecular weight:4195.87IRAK inhibitor 4 trans
IRAK inhibitor 4 targets and blocks IRAK4 activity; refers to its trans molecular configuration.Formula:C33H35F3N6O3Purity:98%Color and Shape:SolidMolecular weight:620.66Urocortin, rat
CAS:Endogenous CRF agonist. Ki values are 13, 1.5 and 0.97 nM for hCRF1, rCRF2α and mCRF2β respectively.Formula:C206H338N62O64Purity:98%Color and Shape:SolidMolecular weight:4707.26VIP(Guinea pig)
CAS:Neuropeptide with many biological actionsFormula:C147H239N43O42S2Purity:98%Color and Shape:SolidMolecular weight:3344.86SR 142948 TFA
SR 142948 TFA is an orally active, selective non-peptide neurotensin receptor (NT) antagonist, displaying IC50 values of 1.19 nM in h-NTR1-CHO cells, 0.32 nM in HT-29 cells, and 3.96 nM in adult rat brain. In HT-29 cells, it counteracts NT-induced inositol monophosphate formation with an IC50 of 3.9 nM. It blocks NT-induced hypothermia, analgesia, and turning behavior in vivo and can cross the blood-brain barrier, making it useful for research in psychiatric disorders.Color and Shape:Odour SolidMisoprostol acid
CAS:Misoprostol acid is an active metabolite of Misoprostol,can be used for non-steroidal anti-inflammatory drug-induced (NSAID) gastric ulcers.Formula:C21H36O5Purity:98%Color and Shape:SolidMolecular weight:368.51Add 4743
CAS:Add 4743 is an analog of sitoglitazone, which is also a fat-forming agent.Formula:C18H23NO4SColor and Shape:SolidMolecular weight:349.44Δ9-THCH
CAS:Δ9-THCH, a phytocannabinoid analytical reference standard, is present in a Cannabis variety cultivated for medicinal use. In the United States, it is classified as a Schedule I compound. This product is designated for research and forensic applications.Formula:C22H32O2Color and Shape:SolidMolecular weight:328.49sGnRH-A
CAS:sGnRH-A, a salmon GnRH analog, boosts growth hormone and induces ovulation for artificial insemination.Formula:C64H83N17O12Color and Shape:SolidMolecular weight:1282.45CKLF1-C27 TFA
CKLF1-C27 peptide activates ERK1/2 via CCR4, competes with CKLF1, promotes HUVEC growth, and has psoriasis research potential.Formula:C153H244F3N39O39Color and Shape:SolidMolecular weight:3310.8IRL-3630
CAS:IRL 3460 is an enantiomer.Formula:C31H40N4O6SPurity:98%Color and Shape:SolidMolecular weight:596.74CB1-IN-3
CB1-IN-3 (Compound 6i) is a potent inhibitor of the cannabinoid receptor type 1 (CB1). It holds potential for research in obesity, inflammation, and neurological disorders.Color and Shape:Odour SolidColulintide
CAS:Colulintide is an analog of amylin, utilized in obesity research.Color and Shape:SolidEletriptan
CAS:Eletriptan, second-generation triptans used to treat migraines, is used as an abortion drug.Formula:C22H26N2O2SColor and Shape:SolidMolecular weight:382.522,3-dinor Thromboxane B1
CAS:TXB2 released from platelets becomes 11-dehydro and 2,3-dinor TXB2. Rats excrete 2,3-dinor TXB1, a reliable thromboxane biosynthesis marker.Formula:C18H32O6Color and Shape:SolidMolecular weight:344.448ELA-21 (human)
CAS:Apelin receptor agonist with high affinity for normal/PAH hearts (pKi 9.31/9.46). Blocks cAMP, promotes β-arrestin in vitro. Part of ELA-32.Formula:C112H184N40O25S3Purity:98%Color and Shape:SolidMolecular weight:2587.12S(-)-Bisoprolol fumarate
CAS:S(-)-Bisoprolol fumarate is a selective β1-blocker for hypertension and heart research.Formula:C18H31NO4·xC4H4O4Color and Shape:SolidMolecular weight:441.521
