GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(251 products)
- Adrenergic Receptor(3,028 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(218 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(36 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(42 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(61 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 6012 products of "GPCR/G-Protein"
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Sarafotoxin S6c
CAS:Highly selective ETB endothelin receptor agonist (Ki values are 0.29 and 28000 nM at ETB and ETA receptors respectively).Formula:C103H147N27O37S5Purity:98%Color and Shape:SolidMolecular weight:2516Vapitadine
CAS:Vapitadine is a non-sedative antihistamine compound that relieves itching caused by atopic dermatitis.Formula:C17H20N4OPurity:99.77% - 99.86%Color and Shape:SoildMolecular weight:296.37Cannabigerorcin
CAS:Cannabigerorcin, a phytocannabinoid, serves as an analytical reference standard. It is designated for research and forensic applications.Formula:C17H24O2Color and Shape:SolidMolecular weight:260.377Glucagon (19-29), human
CAS:Glucagon, a 29-amino-acid hormone, is produced by alpha cells in the pancreas' islets of Langerhans.Formula:C61H89N15O18SPurity:98%Color and Shape:SolidMolecular weight:1352.53ELA-21 (human)
CAS:Apelin receptor agonist with high affinity for normal/PAH hearts (pKi 9.31/9.46). Blocks cAMP, promotes β-arrestin in vitro. Part of ELA-32.Formula:C112H184N40O25S3Purity:98%Color and Shape:SolidMolecular weight:2587.12allo-Yohimbine
CAS:allo-Yohimbine is a biochemical.Formula:C21H26N2O3Color and Shape:SolidMolecular weight:354.44L-803087 TFA
CAS:L-803087 TFA: potent sst4 agonist, Ki=0.7 nM, >280x selective vs other somatostatin receptors; boosts AMPA, heightens seizures.Formula:C27H30F5N5O5Color and Shape:SolidMolecular weight:599.55Flunarizine
CAS:Flunarizine is an orally administered peripheral vasodilator, a dual blocker of voltage-gated Na+/Ca2+ channels and a D2 dopamine receptor antagonist.Formula:C26H26F2N2Purity:99.9%Color and Shape:SolidMolecular weight:404.50Labradimil
CAS:Labradimil, a bradykinin B2 agonist, boosts brain drug delivery and tumor survival rates.Formula:C49H75N15O12SPurity:98%Color and Shape:SolidMolecular weight:1098.29α-Helical CRF(9-41)
CAS:Corticotropin-releasing factor receptor antagonist (Ki values are 17, 5 and 0.97 at human CRF1, rat CRF2α and mouse CRF2β receptors respectively).Formula:C166H274N46O53S2Purity:98%Color and Shape:SolidMolecular weight:3827PAF C-16 Carboxylic Acid
CAS:PAF C-16, a natural phospholipid, triggers neutrophil migration, ROS, IL-6 production, and is linked to necrotizing enterocolitis.Formula:C26H52NO9PColor and Shape:SolidMolecular weight:553.67V-0219 hydrochloride
V-0219 hydrochloride: oral GLP-1R PAM for obesity-linked diabetes study.
Formula:C20H26ClF3N4O2Purity:99.97%Color and Shape:SoildMolecular weight:446.89Etelcalcetide
CAS:Etelcalcetide (AMG 416), a synthetic peptide CaSR activator, treats secondary hyperparathyroidism in hemodialysis patients.Formula:C38H73N21O10S2Purity:98%Color and Shape:SolidMolecular weight:1048.26VIP(Guinea pig)
CAS:Neuropeptide with many biological actionsFormula:C147H239N43O42S2Purity:98%Color and Shape:SolidMolecular weight:3344.86AZP-531
CAS:Azp-531 is a disacylated ghrelin used to improve blood sugar control and weight loss.Formula:C40H63N15O13Purity:98%Color and Shape:SolidMolecular weight:962.025-HT6 inverse agonist 1
CAS:5-HT6 inverse agonist 1 (Compound 33) is an antagonist of the 5-HT6 receptor with a Ki of 23 nM and a Kb of 6.62 nM. This compound can inhibit 5-HT6R-mediated Cdk5 and mTOR signaling pathways and reduce tactile allodynia induced by spinal nerve ligation (SNL) in rat models.Formula:C22H22Cl2FN3O3SColor and Shape:SolidMolecular weight:498.4(+)-Cloprostenol
CAS:(+)-Cloprostenol is a analogue of prostaglandin F2α (PGF2α), and is selective prostaglandin receptor agonistic.Formula:C22H29ClO6Purity:98%Color and Shape:SolidMolecular weight:424.92EP4-IN-1
CAS:EP4-IN-1: Potent EP4 receptor inhibitor with anti-tumor, anti-inflammatory, and analgesic properties.Formula:C27H24N2O4Purity:99.94%Color and Shape:SoildMolecular weight:440.49Carbazochrome salicylate
CAS:Carbazochrome salicylate can be used as a coagulant.Formula:C17H18N4NaO6Color and Shape:White Crystalline PowderMolecular weight:397.343N-0500 HCl
CAS:N-0500 HCl, a potent DA receptor agonist, displaces [3H]DP_x005f_x0002_5,6-ADTN with an IC50 of 3nM.Formula:C15H22ClNO2Purity:98.85% - 99.54%Color and Shape:SolidMolecular weight:283.79
