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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 6011 products of "GPCR/G-Protein"

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  • 5-OMe-UDP trisodium salt

    CAS:
    Potent P2Y6 agonist
    Formula:C10H16N2O13P2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:434.19

    Ref: TM-T22525

    25mg
    To inquire
    50mg
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    100mg
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  • BAM(8-22) TFA


    BAM(8-22) TFA activates Mrgprs, induces mouse scratching, and is a proenkephalin A derivative.
    Formula:C93H128F3N25O25S
    Color and Shape:Solid
    Molecular weight:2085.22

    Ref: TM-T75862

    5mg
    To inquire
    50mg
    To inquire
  • PG106

    CAS:
    Selective hMC3 receptor antagonist (IC50 = 210 nM). Exhibits no activity at hMC4 receptors and hMC5 receptors.
    Formula:C51H69N13O9
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1008.19

    Ref: TM-TP1952

    1mg
    250.00€
  • Sar-[D-Phe8]-des-Arg9-Bradykinin

    CAS:
    Potent bradykinin B1 agonist, EC50 = 9.02 nM, enzyme resistant, induces hypotension and angiogenesis.
    Formula:C47H66N12O11
    Purity:98%
    Color and Shape:Solid
    Molecular weight:975.11

    Ref: TM-TP1917

    1mg
    207.00€
  • Hydroxybupropion

    CAS:
    Hydroxybupropion is the major active metabolite of Bupropion and an antagonist of nACh receptor. Hydroxybupropion inhibits norepinephrine uptake (IC50 = 1.7 μM).
    Formula:C13H18ClNO2
    Purity:99.73%
    Color and Shape:Off-White Solid
    Molecular weight:255.74

    Ref: TM-T11588

    1mg
    94.00€
    5mg
    193.00€
    1mL*10mM (DMSO)
    220.00€
    10mg
    314.00€
    25mg
    516.00€
    50mg
    737.00€
    100mg
    1,007.00€
  • Adrenomedullin (11-50), rat

    CAS:
    Adrenomedullin 11-50 rat is a peptide, stimulates CGRP1 receptor for vasodilation, used in bone growth research.
    Formula:C194H304N58O59S4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:4521.17

    Ref: TM-TP1625

    100mg
    To inquire
    500mg
    To inquire
  • RXFP3/4 agonist 1

    CAS:
    RXFP3/4 agonist 1 is a relaxin family peptide 3/4 receptor (RXFP3/4) agonist(EC50s of 82/2 nM, respectivley).
    Formula:C20H22ClN5O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:383.88

    Ref: TM-T12785

    25mg
    2,178.00€
    50mg
    2,862.00€
    100mg
    3,870.00€
  • WS 9326A

    CAS:
    WS 9326A is an antagonist of tachykinin receptor from Streptomyces violaceusniger.
    Formula:C54H68N8O13
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1037.181

    Ref: TM-T26333

    25mg
    1,369.00€
  • Luteinizing Hormone Releasing Hormone (LH-RH), salmon

    CAS:
    LH-RH: a hypothalamus-made pituitary hormone, key in reproductive control.
    Formula:C60H73N15O13
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1212.31

    Ref: TM-TP1112

    1mg
    79.00€
    5mg
    163.00€
    10mg
    284.00€
  • Tirzepatide hydrochloride


    Tirzepatide HCl is a dual GIP and GLP-1 receptor agonist.
    Formula:C225H349N48O68Cl
    Purity:98%
    Color and Shape:Solid
    Molecular weight:4849.91

    Ref: TM-TP1110

    1mg
    240.00€
    5mg
    628.00€
  • 13,14-dihydro-15-keto Prostaglandin F1α

    CAS:
    13,14-dihydro-15-keto Prostaglandin F1α (13,14-dihydro-15-keto PGF1α) is a metabolite of PGF1α that has been reported in the rat stomach.
    Formula:C20H36O5
    Color and Shape:Solid
    Molecular weight:356.5

    Ref: TM-T36148

    500µg
    112.00€
    1mg
    200.00€
    5mg
    828.00€
    10mg
    1,431.00€
  • Orexin B, human

    CAS:
    Orexin B, human agonizes Orexin receptors (OX1 Ki=420 nM, OX2 Ki=36 nM), promotes feeding in rats, and is a neuropeptide.
    Formula:C123H212N44O35S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:2899.34

    Ref: TM-TP1139

    500µg
    1,288.00€
  • Navafenterol

    CAS:
    AZD-8871, a potential COPD and asthma treatment, may work well with ICS.
    Formula:C38H42N6O6S2
    Color and Shape:Solid
    Molecular weight:742.91

    Ref: TM-T30264

    25mg
    To inquire
    50mg
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    100mg
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  • [D-Glp1,D-Phe2,D-Trp3,6]-LH-RH

    CAS:
    [D-Glp1,D-Phe2,D-Trp3,6]-LH-RH is a synthetic LHRH analog and a GnRH receptor antagonist.
    Formula:C67H84N16O13
    Color and Shape:Solid
    Molecular weight:1321.48

    Ref: TM-T76350

    5mg
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    50mg
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  • Spantide acetate


    Spantide acetate is a selective antagonist of NK1 receptor with Kis of 230 nM and 8150 nM for NK1 and NK2.

    Formula:C77H112N20O15
    Purity:98.9200%
    Color and Shape:Solid
    Molecular weight:1557.84

    Ref: TM-T20413L

    1mg
    129.00€
    5mg
    329.00€
    10mg
    525.00€
    25mg
    848.00€
    50mg
    1,159.00€
    100mg
    1,568.00€
    500mg
    3,117.00€
  • Adrenomedullin (AM) (22-52), human TFA


    Adrenomedullin (AM) human (22-52) is a truncated NH2 TFA-modified adrenal medullary receptor antagonist.
    Formula:C161H253N46F3O50
    Purity:98%
    Color and Shape:Solid
    Molecular weight:3690.06

    Ref: TM-TP1256

    100mg
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    500mg
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  • [His1,Nle27] GHRF (1-32), amide, human

    CAS:

    [His1,Nle27] GHRF (1-32), amide, human is a potent GHRH analog with high GHRHR affinity.

    Formula:C159H265N51O46
    Color and Shape:Solid
    Molecular weight:3627.12

    Ref: TM-T76317

    5mg
    To inquire
    50mg
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  • ANP [Des18-22] 4-23 amide rat

    CAS:
    ANP [Des18-22] 4-23 amide rat is a peptide fragment of rat atrial natriuretic peptide (ANP) that specifically binds to NPR-C.
    Formula:C64H107N25O19S2
    Color and Shape:Solid
    Molecular weight:1594.82

    Ref: TM-TP3030

    10mg
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    50mg
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  • SAR441255


    SAR441255 is a potent unimolecular peptide that acts as a GLP-1/GIP/GCG receptor triagonist, demonstrating balanced activation across all three target receptors
    Color and Shape:Odour Solid

    Ref: TM-T81214

    5mg
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    50mg
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  • LY 293284

    CAS:
    LY 293284 is a potent, selective full agonist of 5-HT1A receptor with anxiogenic effects in animal studies.
    Formula:C19H26N2O
    Color and Shape:Solid
    Molecular weight:298.42

    Ref: TM-T27914

    25mg
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    50mg
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    100mg
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