GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,024 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(194 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5990 products of "GPCR/G-Protein"
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(D-Ser4,D-Ser(tBu)6,Azagly10)-LHRH
CAS:Analog of LHRH, stimulates LH and FSH release, controls reproduction.Formula:C59H84N18O14Color and Shape:SolidMolecular weight:1269.41CYM5442 hydrochloride
CAS:CYM 5442 HCl: potent, selective S1P1 agonist (EC50 = 1.35 nM), induces MAPK activation & lymphopenia, brain-penetrant.Formula:C23H28ClN3O4Color and Shape:SolidMolecular weight:445.94AY 254
CAS:AY 254: Potent PAR2 agonist, ERK1/2 activation (EC50=2 nM), limits caspase 3/8, aids HT29 cell healing, boosts IL-8.
Formula:C30H49N9O6Color and Shape:SolidMolecular weight:631.779Senktide TFA
Senktide TFA is a potent and selective neurokinin 3 (NK3) receptor agonist with an EC50 of 0.5-3 nM, while showing significantly weaker activity on NK1 receptors (EC50=35 µM). It is a promising candidate for research in neurological disorders.Color and Shape:Odour Solid2-Furoyl-LIGRLO-amide
CAS:2-Furoyl-LIGRLO-amide TFA is a peptide that acts as a proteinase-activated receptor-2 (PAR2) agonist, and contains a furoyl group addition at its N-terminal.Formula:C36H63N11O8Purity:98%Color and Shape:SolidMolecular weight:777.95Cetirizine Impurity C
CAS:Cetirizine Impurity C - a metabolite of hydroxyzine, is a long-acting, oral H1-antihistamine.Formula:C21H25ClN2O3Color and Shape:SolidMolecular weight:388.8919(R)-hydroxy Prostaglandin E1
CAS:19(R)-hydroxy Prostaglandin E1 is an agonist of EP1 and EP3 receptor subtypes and exhibits contractile activity on smooth muscle and is the major prostaglandinFormula:C20H34O6Color and Shape:SolidMolecular weight:370.486Neuropeptide Y(29-64)
CAS:Neuropeptide Y(29-64) is a 36 amino acid peptide, a fragment of Neuropeptide Y.Formula:C189H284N54O58SPurity:98%Color and Shape:SolidMolecular weight:4272.7Adrenocorticotropic Hormone (ACTH) (1-39), rat TFA
Adrenocorticotropic Hormone (ACTH) (1-39), rat (TFA) is a potent melanocortin 2 receptor (MC2) agonist.Formula:C212H316F3N57O59SPurity:98%Color and Shape:SolidMolecular weight:4696.18Sibenadet hydrochloride
CAS:Sibenadet, a D2/beta2-agonist, is potential useful for the treatment of symptoms of chronic obstructive pulmonary disease.Formula:C22H29ClN2O5S2Color and Shape:SolidMolecular weight:501.06Litoxetine HCl
Litoxetine HCl, an SSRI and 5-HT antagonist, treats urinary incontinence and relaxes rat oesophageal muscles without antimuscarinic effects.Formula:C16H20ClNOPurity:98.97% - 99.9%Color and Shape:SoildMolecular weight:277.79Ref: TM-T67956L
1mg92.00€1mL*10mM (DMSO)197.00€5mg207.00€10mg309.00€25mg527.00€50mg755.00€100mg1,044.00€(+)-OSU 6162
CAS:(+)-OSU 6162 (Piperidine, 3-[3-(methylsulfonyl)phenyl]-1-propyl-, (3R)-) is an agonist of 5-HT Receptor with anti-Alzheimer and antidepressant activities.Formula:C15H23NO2SPurity:98.19%Color and Shape:SoildMolecular weight:281.41Ref: TM-T60027
1mg73.00€5mg146.00€1mL*10mM (DMSO)155.00€10mg208.00€25mg319.00€50mg447.00€100mg600.00€200mg808.00€GI-560192
CAS:GI-560192 (RL-0070933), a potent smo modulator, EC50: 0.02µM; affects smoothened in cilia via hedgehog signaling.Formula:C20H16N2O2Purity:99.53%Color and Shape:SoildMolecular weight:316.35Ref: TM-T64351
1mg85.00€5mg170.00€1mL*10mM (DMSO)170.00€10mg250.00€25mg371.00€50mg522.00€100mg712.00€200mg954.00€Ilatreotide
CAS:Ilatreotide is a Amadori compound of octreotide.Formula:C61H86N10O20S2Purity:98%Color and Shape:SolidMolecular weight:1343.53d[Leu4,Lys8]-VP acetate
d[Leu4,Lys8]-VP acetate: Vasopressin V1b agonist. Ki: rat 0.16 nM, human 0.52 nM, mouse 1.38 nM. Low antidiuretic/vasopressor effects.Formula:C49H71N11O13S2Purity:98.86%Color and Shape:SolidMolecular weight:1086.28D[LEU4,LYS8]-VP TFA
D[LEU4,LYS8]-VP TFA: V1b receptor agonist; K_i: 0.16 nM (rat), 0.52 nM (human), 1.38 nM (mouse); weak antidiuretic/vasopressor/oxytocic.Formula:C49H68F3N11O13S2Color and Shape:SolidMolecular weight:1140.25Detomidine carboxylic acid
CAS:Detomidine carboxylic acid, a urine metabolite of detomidine, is a synthetic α2-agonist, animal analgesic, with cardiac, respiratory, and diuretic effects.Formula:C12H12N2O2Purity:98%Color and Shape:SolidMolecular weight:216.24MRS 2957 triethylammonium salt
CAS:MRS 2957 triethylammonium salt is a P2Y6 agonist.Formula:C19H28N5O20P3Purity:98%Color and Shape:SolidMolecular weight:739.37γ-Glu-Abu TFA
Gamma-Glu-AbuTFA is the TFA salt form of Gamma-Glu-Abu. This compound acts as an agonist for the calcium sensing receptor (CaSR), activating CaSR in HEK-293 cells with an EC50 of 0.21 μM.Formula:C11H17F3N2O7Color and Shape:SolidMolecular weight:346.26(Phe2,Orn8)-Oxytocin acetate
(Phe2,Orn8)-Oxytocin acetate: V1 agonist with EC50 of 280 nM for rabbit epididymis contractility.Formula:C44H69N13O13S2Color and Shape:SolidMolecular weight:1052.23
![d[Leu4,Lys8]-VP acetate](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FTP1927L1.webp&w=3840&q=75)
