GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(251 products)
- Adrenergic Receptor(3,025 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(218 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(36 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 6011 products of "GPCR/G-Protein"
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A71378
CAS:A71378 is a high potency, selectivity CCK-A receptors agonist.Formula:C48H62N8O13SPurity:98%Color and Shape:SolidMolecular weight:991.12(R)-CJ 11974
CAS:(R)-CJ 11974: non-peptide NK1 receptor antagonist, may relieve pain and prevent chemo-induced vomiting.Formula:C31H38N2OPurity:97.15%Color and Shape:SoildMolecular weight:454.65CTP-amiodarone
CTP-amiodarone, a cellular-penetrating conjugate of myocardial cell-targeting peptide and Amiodarone, exhibits anti-arrhythmic activity by blocking Na+, K+, and Ca2+ channels as well as β-adrenergic receptors.Formula:C97H131F3I2N20O25S2Color and Shape:SolidMolecular weight:2352.13Chemerin-9 (149-157) TFA
Chemerin-9 (149-157) TFA is a peptide located at positions 149-157 of chemerin-9, acting as a ChemR23/CMKLR1 agonist.Formula:C56H67F3N10O15Purity:99.77%Color and Shape:SolidMolecular weight:1177.18Clomipramine D3
CAS:Clomipramine D3 is deuterium-labeled Clomipramine, blocking serotonin, norepinephrine, dopamine transporters (Ki: 0.14, 54, 3 nM).Formula:C19H23ClN2Purity:98%Color and Shape:SolidMolecular weight:317.87Glucagon (19-29), human
CAS:Glucagon, a 29-amino-acid hormone, is produced by alpha cells in the pancreas' islets of Langerhans.Formula:C61H89N15O18SPurity:98%Color and Shape:SolidMolecular weight:1352.534-P-PDOT
CAS:4-P-PDOT (4-phenyl-2- propionamidotetralin) is a potent, selective and affinity Melatonin receptor (MT2) antagonist.Formula:C19H21NOPurity:99.91%Color and Shape:SolidMolecular weight:279.38GRK2i
CAS:GRK2 inhibitory polypeptide that specifically inhibits Gβγ activation of GRK2. Corresponds to the Gβγ-binding domain and acts as a cellular Gβγ antagonist.Formula:C153H256N50O41SPurity:98%Color and Shape:SolidMolecular weight:3484.08Neuropeptide Y (22-36)
CAS:Neuropeptide Y (22-36) is a 15-amino acid fragment of NPY, which is abundant in the mammalian brain and involved in multiple physiological functions.Formula:C85H139N29O21Purity:98%Color and Shape:SolidMolecular weight:1903.19NF157
CAS:NF157, a selective P2Y11 antagonist with pKi 7.35, lowers MMP-3/MMP-13, aiding OA treatment; IC50s: P2Y11 463 nM, P2Y1 1811 μM, P2Y2 170 μM.Formula:C49H28F2N6Na6O23S6Purity:98%Color and Shape:SolidMolecular weight:1437.1AL 34662
CAS:AL 34662 is a selective and potent 5-HT2A receptor agonist with IC50s of 0.77 nM and 1.5 nM for rat and human 5-HT2 receptors, respectively.AL 34662 is also aFormula:C10H13N3OPurity:99.97%Color and Shape:SolidMolecular weight:191.23L 152804
CAS:L 152804: Y5 receptor antagonist, reduces food intake/boosts energy, leads to weight loss in obese mice.Formula:C23H26O4Purity:99.82%Color and Shape:SolidMolecular weight:366.45Ref: TM-T15679
5mg48.00€1mL*10mM (DMSO)49.00€10mg75.00€25mg111.00€50mg170.00€100mg245.00€200mg349.00€Xanthine amine congener trihydrochloride
CAS:Xanthine amine congener trihydrochloride: potent adenosine antagonist, reverses effects of N6-cyclohexyladenosine on urine, sodium excretion, heart rate.Formula:C21H29ClN6O4Purity:98.81%Color and Shape:SolidMolecular weight:464.95YM 16638
CAS:YM 16638 is an LT antagonist that can be used to study antigen-induced early and late airway responses in allergic sheep.Formula:C18H22N2O5S3Purity:99.18%Color and Shape:SolidMolecular weight:442.57P2Y12R ligand-1
P2Y12R ligand-1 (Compound 41) is a high-affinity P2Y12 receptor ligand with a Ki of 17.1 nM. The [18F]-labeled version of P2Y12R ligand-1 is suitable for research involving brain PET imaging.Color and Shape:Odour Solid(Iso)-Landipirdine
CAS:(Iso)-Landipirdine((Iso)-RO5025181) is a selective and potent 5-HT6R antagonist.Formula:C18H19FN2O3SPurity:98.94%Color and Shape:SoildMolecular weight:362.42Tiflucarbine
CAS:Tiflucarbine is a potential non-selective 5-HT agonist with antidepressant activity.Tiflucarbine dose-dependently increased the specific activity of solubleFormula:C16H17FN2SPurity:97.71%Color and Shape:SolidMolecular weight:288.38Tocrifluor T1117
CAS:Fluorescent form of AM 251, CB1 receptor antagonistFormula:C56H53Cl2N7O5Purity:98%Color and Shape:SolidMolecular weight:974.97ELA-11(human)
CAS:Apelin receptor agonist with high affinity (Ki = 14 nM). Blocks cAMP production and promotes β-arrestin activation; derived from ELA-32.Formula:C58H90N16O13S2Purity:98%Color and Shape:SolidMolecular weight:1283.57Kadsurenin B
CAS:Kadsurenin B, a platelet-activating factor (PAF) antagonist, exhibits neuroprotective properties and has a broad spectrum of pharmacological researchFormula:C20H22O5Color and Shape:SolidMolecular weight:342.39
