GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,023 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(194 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5990 products of "GPCR/G-Protein"
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β-MSH, human
CAS:beta-MSH, human is an endogenous peptide hormone and neurotransmitter by POMC, an agonist of MC4-R (melanocortin 4 receptor).Formula:C118H174N34O35SPurity:98%Color and Shape:SolidMolecular weight:2660.92RF9
CAS:RF9 is an effective and selective antagonist of the Neuropeptide FF receptor (Kis: 58±5 and 75±9 nM for hNPFF1R and hNPFF2R, respectively).Formula:C26H38N6O3Purity:98%Color and Shape:SolidMolecular weight:482.62Cetirizine methyl ester
CAS:Cetirizine methyl ester is a Cetirizine impurity, a long-acting, oral H1-antihistamine and hydroxyzine metabolite.Formula:C22H27ClN2O3Color and Shape:SolidMolecular weight:402.91GS-2278
CAS:GS-2278 is an antagonist of LPAR1 (lysophosphatidic acid receptor 1) with potential applications in the study of idiopathic pulmonary fibrosis (IPF).Formula:C22H16F5N9O3Color and Shape:SolidMolecular weight:549.41Cetirizine Impurity D
CAS:Cetirizine Impurity D, an antihistamine derivative, acts as a long-lasting H1-receptor antagonist with antiallergic effects.Formula:C30H28Cl2N2Color and Shape:SolidMolecular weight:487.4612-epi Leukotriene B4
CAS:LTB4 is made enzymatically (12(R)-specific) and non-enzymatically (6-trans-12-epi mix). 12-epi LTB4 has low receptor activity.Formula:C20H32O4Color and Shape:SolidMolecular weight:336.472O-Desethyl Dapagliflozin
CAS:O-Desethyl Dapagliflozin (Empagliflozin-4) is a SGLT2 inhibitor, IC50=33nM.Formula:C19H21ClO6Purity:98.33%Color and Shape:SolidMolecular weight:380.82Ref: TM-T67849
1mg54.00€5mg114.00€1mL*10mM (DMSO)128.00€10mg177.00€25mg304.00€50mg445.00€100mg647.00€PACAP-38 (16-38), human, mouse, rat
CAS:PACAP-38 (16-38), human, mouse, rat demonstrates potent, efficacious, and sustained stimulatory effects on sympathetic neuronal NPY and catecholamine productionFormula:C123H215N39O28SPurity:98%Color and Shape:SolidMolecular weight:2720.33NF 340
CAS:P2Y11 antagonistFormula:C37H30N4Na4O15S4Purity:98%Color and Shape:SolidMolecular weight:990.87ACTH (11-24)
CAS:ACTH (11-24) is an adrenocorticotrophin fragment, stimulates cortisol, and antagonizes ACTH (1-39)/(1-10) in adrenal cells.Formula:C77H134N24O16Purity:98%Color and Shape:SolidMolecular weight:1652.04Stressin I
Potent CRF1 agonist; Ki: 1.5 nM (CRF1), 224 nM (CRF2). Boosts ACTH, enhances stool frequency after i.p. administration.Formula:C203H337N57O56Purity:98%Color and Shape:SolidMolecular weight:4472.24Antipsychotic agent-2
Compound 11: potent antipsychotic, binds 5-HT1A/2A/2C, D2, H1 receptors; K is 56.6-1140 nM, BBB permeable.Formula:C22H26FN5OColor and Shape:SolidMolecular weight:395.47Prepro VIP (81-122), human
CAS:Prepro VIP (81-122), human is a prepro-vasoactive intestinal polypeptide (VIP) derived peptide, corresponding to residues 81-122.Formula:C202H325N53O64SPurity:98%Color and Shape:SolidMolecular weight:4552.13[Leu31,Pro34]-Neuropeptide Y(human,rat)
CAS:High affinity neuropeptide Y Y1 receptor agonist (Ki = 0.39 nM). Also shows affinity for Y4 and Y5 receptors.Formula:C189H284N54O56SPurity:98%Color and Shape:SolidMolecular weight:4241MRS 2365
CAS:Highly potent, selective P2Y1 receptor agonistFormula:C13H19N5O9P2SPurity:98%Color and Shape:SolidMolecular weight:483.33[Gly8]-GLP-1(7-37) acetate
[Gly8]-GLP-1(7-37) acetate is a derivative of GLP-1, where glycine at position 8 is replaced with alanine. [Gly8]-GLP-1(7-37) acetate is also a peptide fragment of the GLP-1 receptor (GLP-1R) agonist, Dulaglutide.Color and Shape:Odour SolidAlosetron
CAS:Alosetron, a 5-HT3 antagonist, is used for the management of severe diarrhea-predominant irritable bowel syndrome (IBS) in women only.Formula:C17H18N4OPurity:98%Color and Shape:Crystalline PowderMolecular weight:294.36LEK 8804
CAS:LEK 8804 is a 5-HT(2) receptor antagonist and 5-HT(1A) receptor agonist.Formula:C19H19N3OColor and Shape:SolidMolecular weight:305.37Hemopressin (human, mouse)
CAS:Endogenous peptide, inhibits ep24.15/24.16/ACE with Ki of 27.76/3.43/1.87 μM. Lowers blood pressure, CB1 inverse agonist, reduces pain in vivo.Formula:C50H79N13O12Purity:98%Color and Shape:SolidMolecular weight:1054.26α1A-AR Degrader 9c
CAS:α1A-AR Degrader 9c is a potent, selective, and reversible PROTAC degrader targeting the α1A adrenergic receptor (α1A-AR) with a DC50 of 2.86 μM.Formula:C38H43N11O11Purity:98%Color and Shape:SolidMolecular weight:829.82
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