GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,023 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(194 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5986 products of "GPCR/G-Protein"
Sort by
Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
GLP-1R agonist 16
CAS:Compound 115a, a GLP-1R agonist, effectively activates the GLP-1 receptor with an EC50 of 0.15 nM [1].Formula:C50H58FN10O6PColor and Shape:SolidMolecular weight:945.03Galanin Receptor Ligand M35
CAS:M35, a galanin(1-13)-bradykinin(2-9) amide, acts as a galanin antagonist in rats and inhibits mouse pancreatic islets.Formula:C107H153N27O26Purity:98%Color and Shape:SolidMolecular weight:2233.6AC-264613
CAS:AC-264613 is an agonist of the GPCR protease-activated receptor 2 (PAR2). AC-264613 suppresses interferon regulatory factor 5.Formula:C19H18BrN3O2Purity:98%Color and Shape:SolidMolecular weight:400.28CB2R/FAAH modulator-1
CAS:CB2R/FAAH modulator-1: agonizes CB2R, inhibits FAAH (IC50=4 μM), alters cytokine production; used in inflammation research. Ki: CB2R=14.8 nM, CB1R=241.3 nM.Formula:C24H27NO2Purity:99.77%Color and Shape:SoildMolecular weight:361.48Ref: TM-T67896
1mg50.00€5mg105.00€1mL*10mM (DMSO)108.00€10mg154.00€25mg224.00€50mg314.00€100mg427.00€200mg575.00€Misoprostol acid
CAS:Misoprostol acid is an active metabolite of Misoprostol,can be used for non-steroidal anti-inflammatory drug-induced (NSAID) gastric ulcers.Formula:C21H36O5Purity:98%Color and Shape:SolidMolecular weight:368.51Betahistine mesylate
CAS:Betahistine mesylate (Extovyl), an H1 agonist and vasodilator, treats Meniere's disease and vascular headaches; risks with asthma/ulcers.Formula:C8H12N2·2(CH4O3S)Purity:98% - 99.85%Color and Shape:CoaMolecular weight:328.4Litoxetine HCl
Litoxetine HCl, an SSRI and 5-HT antagonist, treats urinary incontinence and relaxes rat oesophageal muscles without antimuscarinic effects.Formula:C16H20ClNOPurity:98.97% - 99.9%Color and Shape:SoildMolecular weight:277.79Ref: TM-T67956L
1mg92.00€1mL*10mM (DMSO)197.00€5mg207.00€10mg309.00€25mg527.00€50mg755.00€100mg1,044.00€GRK2-IN-1 hydrochloride (2055990-90-2 free base)
GRKs-IN-1 hydrochloride has remarkable potency against and selectivity for G protein-coupled receptor kinase 2 GRK2 (IC50: 130 nM) and GRK5 (IC50: 7.1 μM).Formula:C24H26ClFN4O4Purity:98%Color and Shape:SolidMolecular weight:488.94Prostaglandin D2 methyl ester
CAS:PGD2: made in mast cells during allergic reactions, causes vasodilation and inhibits blood clots. PGD2 methyl ester is a similar, fat-soluble prodrug.Formula:C21H34O5Color and Shape:SolidMolecular weight:366.498L-797,591
CAS:L-797,591 is a selective agonist of somatostatin receptor subtype 1.Formula:C38H49N5O2Color and Shape:SolidMolecular weight:607.83Seglitide acetate
CAS:Seglitide acetate (MK-678) is a selective agonist of sst2 somatostatin receptor.Formula:C46H60N8O9Purity:98.87%Color and Shape:SolidMolecular weight:869.02GV-150013X
CAS:GV-150013X ((S)-1-(1-(adamantan-1-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydro-1H-benzo[b][1,4]diazepin-3-yl)-3-phenylurea) is a potent CCKB antiagonist, pKiFormula:C33H34N4O3Purity:99.94%Color and Shape:SoildMolecular weight:534.65Ref: TM-T27503L
1mg90.00€5mg190.00€10mg259.00€1mL*10mM (DMSO)270.00€25mg394.00€50mg532.00€100mg698.00€200mg924.00€IRL-3630
CAS:IRL 3460 is an enantiomer.Formula:C31H40N4O6SPurity:98%Color and Shape:SolidMolecular weight:596.74Pal-Glu(OSu)-OH
CAS:Pal-Glu(OSu)-OH is a Liraglutide side chain, a GLP-1 agonist for type 2 diabetes study.Formula:C25H42N2O7Color and Shape:SolidMolecular weight:482.618Noladin ether
CAS:Noladin ether (2-AG ether) is a cannabinoid CB1 receptor agonist.Formula:C23H40O3Color and Shape:SolidMolecular weight:364.56BMS-193885
CAS:BMS-193885 is a selective, brain-penetrant, and competitive antagonist of the neuropeptide Y1 receptor with a Ki of 3.3 nM, and an IC50 of 5.9 nM for hY1.Formula:C33H42N4O6Purity:99.73%Color and Shape:SolidMolecular weight:590.71PG106 TFA
PG106 TFA is a potent hMC3 antagonist (IC50=210 nM), inactive at hMC4 (EC50=9900 nM) and hMC5 receptors.Formula:C53H70F3N13O11Color and Shape:SolidMolecular weight:1122.2GHRF, porcine
CAS:GHRF, porcine, a growth hormone releasing factor (GHRF) peptide (porcine), binds to the growth hormone secretagogue receptor (GHSR), thereby inducing theFormula:C219H365N73O66SColor and Shape:SolidMolecular weight:5108.76α-Helical CRF(9-41) TFA
α-Helical CRF(9-41) TFA acts as a competitive antagonist for the CRF2 receptor, possessing a binding constant (K B) of approximately 100 nM.Formula:C168H275F3N46O55S2Color and Shape:SolidMolecular weight:3940.42Corazonin
CAS:Corazonin, a neuropeptide in insects, regulates caste identity and behavior, mainly in workers/foragers.Formula:C62H83N17O19Color and Shape:SolidMolecular weight:1370.42
