GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,018 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(194 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5983 products of "GPCR/G-Protein"
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Adenosine receptor agonist 1
Compound 6m, an A3 adenosine receptor (AR) partial agonist, exhibits a K i value of 6.7 nM as an adenosine receptor agonist.Formula:C12H14ClN5O2SeColor and Shape:SolidMolecular weight:374.68Lys-Bradykinin
CAS:Endogenous bradykinin receptor agonistFormula:C56H85N17O12Purity:98%Color and Shape:SolidMolecular weight:1188.38Calcitonin (8-32), salmon
CAS:Calcitonin (8-32), salmon: selective amylin receptor antagonist, regulates calcium/phosphorus, thyroid origin, 32-aa peptide.Formula:C119H198N36O37Purity:98%Color and Shape:SolidMolecular weight:2725.06Anthramycin
CAS:Anthramycin: a PBD family antibiotic with antitumor effects and CNS cholecystokinin antagonist properties in mice.Formula:C16H17N3O4Color and Shape:SolidMolecular weight:315.32Fluphenazine free base
CAS:Flufenazine: antipsychotic for schizophrenia, blocks dopamine D2 receptors, reduces hallucinations and delusions.Formula:C22H26F3N3OSColor and Shape:SolidMolecular weight:437.52β2AR/M-receptor agonist-1
CAS:β2AR/M-receptor agonist-1 (example 131), a muscarinic antagonist and β2 adrenoceptor agonist (MABA), exhibits dual potency towards β2 adrenoceptor andFormula:C43H56BrN3O7Color and Shape:SolidMolecular weight:806.821,8-Cineole
CAS:Eucalyptol, a natural monoterpenoid and cyclic ether found in eucalyptus species, effectively controls excessive airway mucus secretion and asthma by inhibiting pro-inflammatory cytokines. It serves as an efficacious treatment for non-purulent sinusitis, reducing inflammation and pain when applied topically, and demonstrating leukemic cell-killing capabilities in vitro.Formula:C10H18OPurity:97.44% - 97.44%Color and Shape:SolidMolecular weight:154.25Secretin, porcine
CAS:Porcine secretin: 27-amino acid peptide for diagnosing pancreatic dysfunction and gastrinoma, stimulates bicarbonate fluid.Formula:C130H220N44O41·xC2H4O2Purity:98%Color and Shape:SolidMolecular weight:N/ABMS-604992 dihydrochloride
CAS:BMS-604992 dihydrochloride is a selective GHSR agonist with high affinity (Ki=2.3 nM) and potent activity (EC50=0.4 nM), stimulating rodent appetite.Formula:C24H33Cl2N7O5Color and Shape:SolidMolecular weight:570.47ELA-21 (human)
CAS:Apelin receptor agonist with high affinity for normal/PAH hearts (pKi 9.31/9.46). Blocks cAMP, promotes β-arrestin in vitro. Part of ELA-32.Formula:C112H184N40O25S3Purity:98%Color and Shape:SolidMolecular weight:2587.12Apelin-17(human, bovine)
CAS:Endogenous apelin receptor agonist. Potently inhibits forskolin-stimulated cAMP accumulation (pIC50 = 9.94).Formula:C96H156N34O20SPurity:98%Color and Shape:SolidMolecular weight:2138.56L-796,778
CAS:L-796,778 is an SST3 agonist and a selective ligand of SST3, which can increase the level of cAMP in the body.Formula:C29H40N6O7Purity:99.24%Color and Shape:SolidMolecular weight:584.66Ref: TM-T32511
1mg175.00€5mg404.00€10mg592.00€25mg888.00€50mg1,243.00€100mg1,701.00€500mg3,402.00€1mL*10mM (DMSO)522.00€PAR650097
PAR650097 is a humanized monoclonal antibody targeting PAR2, used in migraine research.Purity:96.67% (SEC-HPLC) - 98.83% (SEC-HPLC)Color and Shape:LiquidMolecular weight:144.1 kDaCYM5442 hydrochloride
CAS:CYM 5442 HCl: potent, selective S1P1 agonist (EC50 = 1.35 nM), induces MAPK activation & lymphopenia, brain-penetrant.Formula:C23H28ClN3O4Color and Shape:SolidMolecular weight:445.94P2Y14 antagonist 1
P2Y14 antagonist 1 (compound 45) is a highly selective and orally active P2Y14 receptor antagonist with an IC50 value of 0.70 nM. It demonstrates significant anti-inflammatory effects by effectively reducing pulmonary infiltration of immune cells and inflammatory responses through the inhibition of the NLRP3 signaling pathway. P2Y14 antagonist 1 is suitable for studying acute lung injury.Formula:C24H21N3O3Color and Shape:SolidMolecular weight:399.442YM 16638
CAS:YM 16638 is an LT antagonist that can be used to study antigen-induced early and late airway responses in allergic sheep.Formula:C18H22N2O5S3Purity:99.18%Color and Shape:SolidMolecular weight:442.57Sphingosine-1-phosphate (d16:1)
CAS:C16 S1P binds S1P1/EDG-1 (115%), S1P3/EDG-3 (83%), S1P2/EDG-5 (103%) receptors; elevated in glaucoma.
Formula:C16H34NO5PColor and Shape:SolidMolecular weight:351.424Dexbrompheniramine maleate
CAS:Dexbrompheniramine is an antihistamine used for hay fever and urticaria, blocking H1 receptors in the body.Formula:C20H23BrN2O4Color and Shape:SolidMolecular weight:435.318Neuropeptide S(Rat)
CAS:Potent endogenous neuropeptide S receptor (NSPR) agonist (EC50 = 3.2 nM).Formula:C95H160N34O27Purity:98%Color and Shape:SolidMolecular weight:2210.52BMS 193885
CAS:BMS 193885 is a selective and competitive neuropeptide Y(1) receptor antagonist with affinity of 3.3 nM.Formula:C36H48N4O9Purity:98%Color and Shape:SolidMolecular weight:680.79
