GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,017 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(194 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5983 products of "GPCR/G-Protein"
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MCL0129
CAS:MCL0129, a selective and non-peptidergic melanocortin 4 (MC4) receptor antagonist, is a potential treatment for cachexia.Formula:C34H47FN4OPurity:98%Color and Shape:SolidMolecular weight:546.76Desmethyl Mirtazapine (hydrochloride)
CAS:Desmethyl mirtazapine is a metabolite of the antidepressant mirtazapine.1It is formed from mirtazapine by the cytochrome P450 (CYP) isoform CYP3A4.Formula:C16H18ClN3Color and Shape:SolidMolecular weight:287.79NK3R-IN-2
NK3R-IN-2 is an orally active NK3R inhibitor with an IC50 of 330.50 nM against human NK3R. It can penetrate the blood-brain barrier and exhibits excellent NK3R binding affinity in CHO-K1 cells (IC50= 87.31 nM). NK3R-IN-2 effectively suppresses luteinizing hormone (LH) levels and is applicable for research on hormone-related diseases.Color and Shape:Odour SolidUrocortin II, human
Human urocortin (hUcn) II is a new member of the corticotropin-releasing-factor (CRF) family. It selectively binds to the CRF2 receptor.Formula:C194H339N63O54SPurity:98%Color and Shape:SolidMolecular weight:4450.2815(R)-17-phenyl trinor Prostaglandin F2α
CAS:17-phenyl trinor Prostaglandin F2α N-ethyl amide (17-phenyl trinor PGF2α) is an F-series prostaglandin analog which has been approved for use as an ocularFormula:C23H32O5Color and Shape:SolidMolecular weight:388.5Apigenin 6,8-di-C-α-L-arabinopyranoside
CAS:Apigenin 6,8-di-C-alpha-L-arabinopyranoside is a useful organic compound for research related to life sciences.Formula:C25H26O13Color and Shape:SolidMolecular weight:534.47MLS1082
CAS:MLS1082 is a D1-like dopamine receptor (D1R) orthosteric modulatothat stimulates G-protein signaling upon dopamine activation for neurodegenerative disorders.Formula:C24H23N3O2Purity:99.53%Color and Shape:SolidMolecular weight:385.46ent-Prostaglandin E2
CAS:Enzymatic PGE2 is optically pure; radical peroxidation makes it racemic. In oxidative stress, rac-PGE2 forms via 15-E2t-isoprostane.
Formula:C20H32O5Color and Shape:SolidMolecular weight:352.4715-methoxy-α-Ethyltryptamine
CAS:5-Methoxy-alpha-ethyltryptamine is a psychoactive substance that can cause various effects. It belongs to the tryptamine chemical class and can be used for various psychoactive and stimulant effects.
Formula:C13H18N2OPurity:98.25%Color and Shape:SolidMolecular weight:218.29HAEGTFTSDVS
CAS:HAEGTFTSDVS is the first N-terminal 1-11 residues of GLP-1 peptide.Formula:C48H71N13O20Purity:98%Color and Shape:SolidMolecular weight:1150.18CB2R/FAAH modulator-3
CAS:CB2R/FAAH modulator-3 (compound 27) is a modulator targeting at CB2R and FAAH.Formula:C22H31NO2Purity:99.81%Color and Shape:SoildMolecular weight:341.49TE-8105
TE-8105 is a GLP-1 receptor agonist that demonstrates prolonged and enhanced efficacy in models of diabetes, obesity, and non-alcoholic steatohepatitis (NASH).Color and Shape:Odour SolidJmv 179
CAS:Jmv 179 is an antagonist of the cholecystokinin receptor.Formula:C51H67N7O15SColor and Shape:SolidMolecular weight:1050.19Tafluprost ethyl amide
CAS:Tafluprost ethyl amide is a prostaglandin derivative.Formula:C24H33F2NO4Color and Shape:SolidMolecular weight:437.521,2,3-Trilinoelaidoyl-rac-glycerol
CAS:1,2,3-Trilinoelaidoyl-glycerol is a TAG with linoelaidic acid; reduces rat serum thromboxane B2, PGF2, and PGE.Formula:C57H98O6Color and Shape:SolidMolecular weight:879.405Glucagon Receptor Antagonist Inactive Control
CAS:Glucagon Receptor Antagonist Inactive Control is a Glucagon receptor antagonist that can be used in related research in the field of life sciences.Formula:C21H23BrN2OSColor and Shape:SolidMolecular weight:431.394-Oxo-5-phenylpentanoic aci
CAS:4-Oxo-5-phenylpentanoic aci is a useful organic compound for research related to life sciences. The catalog number is T125056 and the CAS number is 3183-15-1.Formula:C11H12O3Color and Shape:SolidMolecular weight:192.2145(S),6(R)-11-trans DiHETE
CAS:5(S),6(R)-11-trans DiHETE, a C-11 isomer of 5(S),6(R)-DiHETE, occurs in rat kidneys, formed enzymatically; not a soybean lipoxygenase substrate.Formula:C20H32O4Color and Shape:SolidMolecular weight:336.47Olcegepant hydrochloride
CAS:Olcegepant hydrochloride (BIBN-4096 hydrochloride) is a selective calcitonin gene-related peptide 1 (CGRP1) receptor antagonist.Formula:C38H48Br2ClN9O5Purity:99.69%Color and Shape:SolidMolecular weight:906.113-hydroxy Desloratidine
CAS:3-hydroxy Desloratidine is a major metabolite of desloratadine , a tricyclic antagonist of the histamine H1 receptor.Formula:C19H19ClN2OColor and Shape:SolidMolecular weight:326.82
