GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,017 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(194 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5983 products of "GPCR/G-Protein"
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α-CGRP (mouse, rat) TFA
α-CGRP (mouse, rat) TFA, a neuropeptide belonging to the calcitonin gene-related peptide (CGRP) family, is predominantly located at neuromuscular junctions andFormula:C162H262N50O52S2·C2HF3O2Purity:98%Color and Shape:Solid[Ala11,D-Leu15]-Orexin B(human)
CAS:OX2 receptor agonist with 400x selectivity vs OX1. EC50: 0.13 nM (OX2), 52 nM (OX1).Formula:C120H206N44O35SPurity:98%Color and Shape:SolidMolecular weight:2857.28Emoghrelin
CAS:Emoghrelin, extracted from Heshouwu (Polygonum multiflorum), promotes the secretion of growth hormone by activating the ghrelin receptor [1].Formula:C24H22O13Purity:98%Color and Shape:SolidMolecular weight:518.42FFN246
CAS:FFN246, a fluorescent probe, concurrently targets the serotonin transporter (SERT) and vesicular monoamine transporter 2 (VMAT2), exhibiting excitation andFormula:C15H13FN2OPurity:98%Color and Shape:SolidMolecular weight:256.27Arotinolol hydrochloride
CAS:Arotinolol HCl is a non-selective α/β-blocker, anti-hypertensive, anti-obesity, and improves aortic stiffness.Formula:C15H22ClN3O2S3Purity:99.82%Color and Shape:SolidMolecular weight:408Prolactin Releasing Peptide (1-31), human
CAS:Human Prolactin Releasing Peptide (1-31) is a potent GPR10 agonist; Ki values are 1.03 nM (human) and 0.33 nM (rat).Formula:C160H252N56O42SPurity:98%Color and Shape:SolidMolecular weight:3664.15LY 293284
CAS:LY 293284 is a potent, selective full agonist of 5-HT1A receptor with anxiogenic effects in animal studies.Formula:C19H26N2OColor and Shape:SolidMolecular weight:298.42Zicronapine fumarate
CAS:Zicronapine fumarate, an antipsychotic, targets D1/D2 & 5-HT2A receptors; may treat neuropsychiatric conditions.Formula:C26H31ClN2O4Color and Shape:SolidMolecular weight:470.99Ghrelin receptor full agonist-2
CAS:Ghrelin receptor full agonist-2 is a highly potent Ghrelin receptor full agonist.Formula:C26H28ClN5O5SColor and Shape:SolidMolecular weight:558.05Org 13011
CAS:Org 13011 has CNS activity and induces conditioned taste aversion by mediating 5-HT 1A receptors.Formula:C18H25F3N4OPurity:98.02%Color and Shape:SoildMolecular weight:370.41Ref: TM-T28258L
1mg109.00€5mg261.00€10mg374.00€25mg583.00€50mg803.00€100mg1,063.00€200mg1,431.00€1mL*10mM (DMSO)266.00€Pafenolol
CAS:Pafenolol is a P-glycoprotein modulator with a Ki value of 5.5 µM. pafenolol is an orally available and selective beta-adrenergic receptor antagonist.Formula:C18H31N3O3Purity:98.33%Color and Shape:SolidMolecular weight:337.46Lanepitant 2HCl
CAS:Lanepitant 2HCl is a non-peptide neurokinin-1 receptor antagonist that can be used to study painful neuropathy-like disorders such as migraine.Formula:C33H47Cl2N5O3Purity:98.67%Color and Shape:SolidMolecular weight:632.66S1R agonist 2
CAS:S1R agonist 2 is a selective S1R agonist with a Ki of 88 nM for S2R and 1.1 nM for S1R and is protective against ROS and NMDA-induced neurotoxicity.Formula:C21H27NOPurity:99.66%Color and Shape:SolidMolecular weight:309.45LTD4 antagonist 2
CAS:LTD4 antagonist 2 (compound 6) functions as a leukotriene D4 (LTD4) antagonist with an IC50 of 2.8 μM for the cysteinyl leukotriene 1 receptor (CysLT1R). Additionally, it acts as an agonist for the G protein-coupled bile acid receptor 1 (GPBAR1), making it applicable for research into colitis, metabolic syndrome, and other GPBAR1- and CysLT1R-related diseases.Formula:C17H13NO3Color and Shape:SolidMolecular weight:279.29Eloralintide
CAS:Eloralintide (LY 3841136) is an AMYR agonist, anticipated for research in type 2 diabetes and obesity.Formula:C201H319N49O65S2Color and Shape:SolidMolecular weight:4526.1BAY-6672 hydrochloride
CAS:BAY-6672 hydrochloride is a potent, selective antagonist of the human Prostaglandin F (FP) receptor, exhibiting an IC50 value of 11 nM.Formula:C26H28BrCl2N3O3Color and Shape:SolidMolecular weight:581.3317-TFM-PGF1α
CAS:17-TFM-PGF1α (Compound 8) is a saturated prostaglandin analog. It exhibits a high affinity and receptor selectivity for the human prostaglandin F receptor (hFP receptor), with an EC50 of 85 nM.Formula:C24H35F3O5Color and Shape:SolidMolecular weight:460.536-Fluoro-N,N-diethyltryptamine
CAS:6-Fluoro-N,N-diethyltryptamine (6-F-DET) exhibits affinity for the 5-HT2A receptor.Formula:C14H19FN2Color and Shape:SolidMolecular weight:234.31Casopitant
CAS:Casopitant (GW679769) is an orally active neurokinin-1 (NK1) receptor antagonist, researched for its potential use in managing chemotherapy-induced nausea and vomiting (CINV) and postoperative nausea and vomiting (PONV).Formula:C30H35F7N4O2Color and Shape:SolidMolecular weight:616.61PF-4363467
CAS:PF-4363467 is a dopamine D3/D2 receptor antagonist that reduces opioid-seeking behavior without the side effects associated with D2 receptors. It has a Ki value of 3.1 nM for D3R and 692 nM for D2R.Formula:C22H30N2O3SColor and Shape:SolidMolecular weight:402.55
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