GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,004 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(155 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(192 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(326 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5970 products of "GPCR/G-Protein"
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Canine KP-10
Canine KP-10 is a potent kisspeptin that induces a significant gonadotropin and estradiol response in female dogs during estrus.Color and Shape:Odour SolidSLB1122168 formic
SLB1122168 is a potent inhibitor of Spns2-mediated sphingosine-1-phosphate (S1P) release, exhibiting an IC50 value of 94 nM [1].Formula:C23H37N3O3Purity:98%Color and Shape:SolidMolecular weight:403.56N6-Benzyl-5'-ethylcarboxamido adenosine
CAS:N6-Benzyl-5'-ethylcarboxamido adenosine is a selective A3 adenosine receptor agonist.Formula:C19H22N6O4Color and Shape:SolidMolecular weight:398.42L-692429 HCl
CAS:L-692,429 is a novel non-peptide growth hormone secretagin.Formula:C29H32ClN7O2Color and Shape:SolidMolecular weight:546.06S1R agonist 2 hydrochloride
Compound 8b hydrochloride, a selective S1R agonist, exhibits affinity with K i s of 1.1 nM for S1R and 88 nM for S2R.Formula:C21H28ClNOPurity:98%Color and Shape:SolidMolecular weight:345.91Neuromedin S (human)
CAS:Neuromedin S (human) is a 33-amino acid neuropeptide identified as an endogenous ligand for the orphan G-protein coupled receptor (GPCR) FM-4/TGR-1, acting onColor and Shape:SolidGM-60186
GM-60186, a potent inhibitor of the 5-HT receptor 2B (HTR2B) with an IC50 of 257 nM, effectively suppresses the proliferation and migration of colorectal cancer cells.Formula:C30H33FN2O4Color and Shape:SolidMolecular weight:504.59Alkyne-βAG-TOCA
Alkyne-βAG-TOCA is an octreotide derivative that targets somatostatin receptor subtype 2 (SST2). It is utilized in the synthesis and research of radioconjugates (RDC).Formula:C48H65N11O15S2Color and Shape:SolidMolecular weight:1100.22γ3-MSH
CAS:γ3-MSH, originating from the N-terminal segment of pro-opiomelanocortin (POMC), induces aldosterone secretion in cultured human adrenal tumor cells [1].Formula:C126H188N44O37SColor and Shape:SolidMolecular weight:2943.18RFRP-1(human)
CAS:Endogenous NPFF agonist with EC50 of 0.0011 nM (NPFF2) and 29 nM (NPFF1); reduces cardiac function and raises prolactin in rats. GnIH homolog.Formula:C67H101N19O14SPurity:98%Color and Shape:SolidMolecular weight:1428.72Maridebart
CAS:Maridebart is a humanized IgG1-kappa monoclonal antibody that targets the GIPR (gastric inhibitory polypeptide receptor) [1].Color and Shape:LiquidK1-70
K1-70 is a humanized antibody targeting TSHR, used in the study of autoimmune diseases and endocrine disorders.Color and Shape:LiquidMolecular weight:143.54 kDaGFB-024
GFB-024 is a humanized antibody targeting CB1, which can be used to study obesity.Color and Shape:LiquidMolecular weight:146.12 kDa[Ala11,D-Leu15]-Orexin B acetate
[Ala11,D-Leu15]-Orexin B acetate is a selective agonist of orexin-2 receptor (OX2) with an EC50 of 0.13 nM, showing 400-fold selectivity over OX1 (52 nM).Formula:C122H210N44O37SPurity:98.18%Color and Shape:SolidMolecular weight:2917.31(±)14(15)-EpETE
CAS:(±)14(15)-EpETE is an intestinal microbial lipid metabolite that attenuates cisplatin chemotherapy-induced nausea in rats by inhibiting Substance P release.Formula:C20H30O3Color and Shape:SolidMolecular weight:318.45Triamterene
CAS:Triamterene is a barosensitive epithelial sodium channel (ENaC) blocker with a diuretic effect. It can also act as an inhibitor of the TGR5 receptor, reducing GLP-1 secretion and cAMP level increases induced by TGR5 activation in a dose-dependent manner.Formula:C12H11N7Purity:99.77%Color and Shape:Yellow Yellow SolidMolecular weight:253.26Minaprine
CAS:Minaprine is a reversible inhibitor of MAO-A, used in the treatment of various depressive states.Formula:C17H22N4OPurity:98%Color and Shape:SolidMolecular weight:298.38Galanin-Like Peptide (porcine)
CAS:Galanin-Like Peptide (porcine) is a 60 amino acid neuropeptide originally isolated from the porcine hypothalamus.Formula:C281H443N81O78Purity:98%Color and Shape:SolidMolecular weight:6204.02CCR6 antagonist 1
CAS:CCR6 antagonist 1 blocks CCL20/CCR6, aiding autoimmune and IBD research.
Formula:C17H12F3NO2Purity:99.83%Color and Shape:SoildMolecular weight:319.28CUR61414 hydrochloride
CUR61414 hydrochloride: potent cell-permeable Hedgehog pathway inhibitor, IC50=100-200 nM, selectively targets Smo (Ki=44 nM), induces cancer cell apoptosis.Formula:C31H43ClN4O5Purity:94.05%Color and Shape:SolidMolecular weight:587.15
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