GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,004 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(155 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(192 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(326 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5971 products of "GPCR/G-Protein"
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(R)-Citalopram oxalate
CAS:(R)-Citalopram oxalate is a weak selective serotonin reuptake inhibitor (SSRI) that antagonises its S-isomer (escitalopram), anticonvulsant and antidepressant
Formula:C22H23FN2O5Purity:99.76%Color and Shape:White SolidMolecular weight:414.43PT-129
PT-129 is a PROTAC degrader targeting the NTF2 domain of G3BP1/2, degrading stress granules in stressed cells, suppressing proliferation.Formula:C46H48N8O12SColor and Shape:SolidMolecular weight:936.98Tafluprost acid
CAS:Tafluprost acid is a selective agonist at the prostaglandin F receptor.Formula:C22H28F2O5Color and Shape:SolidMolecular weight:410.46Nebokitug
Nebokitug is a humanized IgG1κ antibody targeting CCL24, with HumanIgG1kappa, Isotype Control serving as its corresponding isotype control.Color and Shape:Odour LiquidU 67827E
CAS:U 67827E is a long-lasting cholecystokinin agonist. It acts by decreases food intake.Formula:C53H68N10O17SPurity:98%Color and Shape:SolidMolecular weight:1149.24AA 497 HCl
CAS:AA 497, a beta-2 agonist, suppresses Ca spikes.Formula:C14H22ClNO3Color and Shape:SolidMolecular weight:287.78Anticancer agent 258
CAS:Anticanceragent 258 is an imidazo[1,2-B][1,2,4]triazole derivative that modulates nuclear receptor activity. It exhibits an EC50 of 63 nM for Nurr in N2A cells and an IC50 of 0.1 pM for Nur77 in HEK293 cells. Anticanceragent 258 is applicable in studies related to cancer, metabolic disorders, and neurological diseases.Formula:C17H12F2N4Color and Shape:SolidMolecular weight:310.3RS 18286
CAS:RS 18286 is a LHRH antagonist.Formula:C74H101Cl2N17O14Color and Shape:SolidMolecular weight:1523.6Abediterol napadisylate
CAS:Abediterol napadisylate is a novel long-acting β2-agonist in persistent asthma that is efficacy, safe, and tolerable.Formula:C60H68F4N4O14S2Purity:98%Color and Shape:SolidMolecular weight:1209.32Vapiprost
CAS:Vapiprost is an antagonist of the thromboxane receptor and a prostaglandin receptor.Formula:C30H39NO4Purity:98%Color and Shape:SolidMolecular weight:477.64Ala5-Galanin (2-11)
CAS:Ala5-Galanin (2-11) is a specific agonist for the galanin receptor 2 (GAL2R) with an affinity constant (Ki) of 258 nM [1].Formula:C54H81N13O13Purity:98%Color and Shape:SolidMolecular weight:1120.3(±)-PPCC
CAS:(±)-PPCC (oxalate) is a sigma-1 agonist that interacts with sigma-1 receptors (Ki=1.5 nM).Formula:C24H29NO3Color and Shape:SolidMolecular weight:379.49Val9-Oxytocin
CAS:Val9-Oxytocin, an Oxytocin analog where Gly9 is substituted with Val9 [1], functions as a complete antagonist of the vasopressin (V1a) receptor.Formula:C46H72N12O12S2Purity:98%Color and Shape:SolidMolecular weight:1049.27A-286501
CAS:A-286501: Oral adenosine kinase inhibitor, IC50=0.47 nM, reduces pain via non-opioid, non-NSAID ADO receptors.Formula:C11H14BrN5O2Purity:98%Color and Shape:SolidMolecular weight:328.17Ritobegron HCl
CAS:Ritobegron (KUC-7483), a β3-adrenergic agonist, targets human β-AR effectively and is highly selective for rat bladder.Formula:C23H32ClNO5Color and Shape:SolidMolecular weight:437.96Survodutide TFA
Survodutide TFA (BI 456906 TFA) is a GCGR/GLP-1R dual agonist, a peptide compound used in obesity research.Formula:C192H289N47O61·xC2HF3OC2Purity:99.29% - 99.96%Color and Shape:SolidMolecular weight:4231.62 (free base)PSB-22269
PSB-22269 is identified as a GPR17 antagonist with a Ki value of 8.91 nM. It exhibits significant inhibitory effects in cAMP and G protein activation assays. Molecular docking studies indicate that the binding site of PSB-22269 includes positively charged arginine residues and a hydrophobic pocket. PSB-22269 promotes myelin regeneration strategies, offering potential for multiple sclerosis research.Formula:C26H21NO6Color and Shape:SolidMolecular weight:443.45MRS 2957 triethylammonium salt
CAS:MRS 2957 triethylammonium salt is a P2Y6 agonist.Formula:C19H28N5O20P3Purity:98%Color and Shape:SolidMolecular weight:739.37Stressin I TFA
Stressin I (Cyclo(31-34)[DPhe12, Nle21, 38, Glu31, Lys34]Ac-hCRF(4-41)) TFA, with a K i of 1.7 nM, is a potent and selective agonist of the CRF1 receptor.Purity:98%Color and Shape:Odour Solid(S)-Azelastine hydrochloride
CAS:(S)-Azelastine HCl, an antihistamine, reduces H1R, M1R, M3R levels and inhibits HNEpC growth.Formula:C22H25Cl2N3OPurity:98%Color and Shape:SolidMolecular weight:418.36
