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G-protein Coupled Receptors and 7-TM Receptors

G-protein Coupled Receptors and 7-TM Receptors

G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.

Found 5800 products of "G-protein Coupled Receptors and 7-TM Receptors"

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  • Doxylamine succinate

    CAS:
    <p>Doxylamine Succinate is a pyridine derivate histamine H1 antagonist with pronounced sedative properties.</p>
    Formula:C21H28N2O5
    Purity:99.61%
    Color and Shape:5 1 (Ntp 1992)
    Molecular weight:388.46
  • Retatrutide sodium salt


    Retatrutide sodium salt is a glucagon receptor and glucagon-like peptide-1 receptor agonist for the study of type 2 diabetes mellitus.
    Purity:99.97%
    Color and Shape:Soild
  • Vibozilimod

    CAS:
    Vibozilimod (SCD-044) is S1P receptor-1 (S1PR1) agonist .
    Formula:C29H36ClN3O5
    Purity:99.97%
    Color and Shape:Solid
    Molecular weight:542.07
  • Tabernanthalog fumarate

    CAS:
    <p>Tabernanthalog fumarate is a 5-HT2A agonist that promotes neuronal growth and reduces alcohol consumption in mice, producing antidepressant-like effects.</p>
    Formula:C18H22N2O5
    Purity:99.83%
    Color and Shape:Soild
    Molecular weight:346.38
  • Ranitidine Hydrochloride

    CAS:
    Ranitidine Hydrochloride (AH19065) is a competitive and reversible inhibitor of histamine H2-receptor antagonists with antacid activity.
    Formula:C13H23ClN4O3S
    Purity:99.30% - 99.49%
    Color and Shape:Solid
    Molecular weight:350.86
  • Ramelteon

    CAS:
    <p>Ramelteon (TAK-375) is a Melatonin Receptor Agonist. The mechanism of action of ramelteon is as a Melatonin Receptor Agonist.</p>
    Formula:C16H21NO2
    Purity:97.21% - 99.92%
    Color and Shape:Crystalline Solid
    Molecular weight:259.34
  • Cimetidine

    CAS:
    <p>Cimetidine (SKF-92334) is a histamine congener, it competitively inhibits HISTAMINE binding to HISTAMINE H2 RECEPTORS.</p>
    Formula:C10H16N6S
    Purity:99.82%
    Color and Shape:Crystals Physical Description White Crystals With A Slight Sulfur-Mercaptan Odor (Ntp 1992)
    Molecular weight:252.34
  • Cetirizine dihydrochloride

    CAS:
    Cetirizine dihydrochloride is a potent non-drowsy antihistamine for allergies and asthma.
    Formula:C21H27Cl3N2O3
    Purity:99.4% - 99.97%
    Color and Shape:Solid
    Molecular weight:461.81
  • Domperidone

    CAS:
    <p>Domperidone (R33812)(Motilium) is a dopamine blocker and an antidopaminergic reagent.</p>
    Formula:C22H24ClN5O2
    Purity:98% - 99.82%
    Color and Shape:Solid
    Molecular weight:425.91
  • Evatanepag

    CAS:
    <p>Evatanepag (CP-533536) is a selective EP2 agonist for bone formation with 0.3 nM EC50, promoting fracture healing in rats.</p>
    Formula:C25H28N2O5S
    Purity:97.09%
    Color and Shape:Solid
    Molecular weight:468.57
  • Mirabegron

    CAS:
    <p>Mirabegron (YM178) is a beta-3 adrenergic agonist that is used for treatment of overactive bladder syndrome.</p>
    Formula:C21H24N4O2S
    Purity:99.64%
    Color and Shape:Light Yellow To Yellow Solid
    Molecular weight:396.51
  • Naftidrofuryl oxalate

    CAS:
    <p>Naftidrofuryl oxalate treats peripheral/cerebral vascular issues, boosts cell oxidation, is spasmolytic, and may block 5HT-2 serotonin receptors.</p>
    Formula:C26H35NO7
    Purity:97.12% - 98.38%
    Color and Shape:Solid
    Molecular weight:473.56
  • Tetrabenazine

    CAS:
    Tetrabenazine (Ro 1-9569) is a drug formerly used as an antipsychotic and treatment of various movement disorders.
    Formula:C19H27NO3
    Purity:98% - 99.91%
    Color and Shape:White To Off-White White To Off-White Solid
    Molecular weight:317.42
  • GANT 58

    CAS:
    <p>GANT 58 (NSC-75503) is a potent antagonist of Gli. Which inhibits GLI1-induced transcription (IC50: 5 μM).</p>
    Formula:C24H16N4S
    Purity:99.53%
    Color and Shape:Solid
    Molecular weight:392.48
  • Terazosin hydrochloride

    CAS:
    <p>Terazosin HCl (Hytrin) treats BPH and hypertension by blocking alpha1, affecting bladder and vessel muscles.</p>
    Formula:C19H26ClN5O4
    Purity:99.69% - 99.91%
    Color and Shape:Solid
    Molecular weight:423.89
  • Vapreotide acetate

    CAS:
    Vapreotide acetate (BMY-41606 acetate) is an antagonist of the neurokinin-1 (NK1) receptor (IC50: 330 nM).
    Formula:C59H74N12O11S2
    Purity:99.89%
    Color and Shape:Solid
    Molecular weight:1191.42
  • BIBO3304 TFA

    CAS:
    BIBO3304 TFA: Oral, selective NPY Y1 receptor blocker; IC50: 0.38 nM (human), 0.72 nM (rat).
    Formula:C31H36F3N7O5
    Purity:99.5%
    Color and Shape:Solid
    Molecular weight:643.66
  • Tolamolol

    CAS:
    Tolamolol is a selective β-adrenergic blocker that significantly reduces the degree of exercise-induced inhibition of the S-T segment and can be used in the
    Formula:C19H24N2O4
    Purity:98.59%
    Color and Shape:Solid
    Molecular weight:344.4
  • Terbutaline

    CAS:
    Terbutaline is a short-acting agonist of β2-adrenergic receptor (β2-AR) . It is an active metabolite of bambuterol
    Formula:C12H19NO3
    Purity:99.12%
    Color and Shape:Solid
    Molecular weight:225.3
  • Relamorelin

    CAS:
    Relamorelin(BIM28131, RM131) is a selective and potent ghrelin/growth hormone secretagogue receptor (GHSR) agonist.Cost-effective and quality-assured.
    Formula:C43H50N8O5S
    Purity:99.26% - >99.99%
    Color and Shape:Solid
    Molecular weight:790.97
  • Aripiprazole Lauroxil

    CAS:
    <p>Aripiprazole lauroxil, the N-acyloxymethyl prodrug form of aripiprazole, a long-acting injectable (LAI) antipsychotic.</p>
    Formula:C36H51Cl2N3O4
    Purity:99.64%
    Color and Shape:Solid
    Molecular weight:660.71
  • Alfuzosin hydrochloride

    CAS:
    <p>Alfuzosin hydrochloride (Alfuzosin HCl) is an α1 adrenergic receptor antagonist. It applies to treat benign prostatic hyperplasia (BPH).</p>
    Formula:C19H27N5O4·HCl
    Purity:99.78%
    Color and Shape:White To Off-White Solid
    Molecular weight:425.91
  • ALLO-2

    CAS:
    ALLO-2 is a Inhibitor of Drug-Resistant Smo Mutant.It inhibits Smo agonist Hh-Ag1.5-induced luciferase expression in TM3-Gli-Luc cells with IC50 of 6 nM.
    Formula:C18H12F3N5O
    Purity:99.19%
    Color and Shape:Solid
    Molecular weight:371.32
  • Traxanox

    CAS:
    Traxanox: oral diuretic, boosts phagocytosis in mice/rats, reverses antibody production inhibition in BALB/c mice.
    Formula:C13H6ClN5O2
    Purity:98.37%
    Color and Shape:Solid
    Molecular weight:299.67
  • Brompheniramine maleate

    CAS:
    Brompheniramine maleate (Dimotane) is an antagonist against histamine H1 receptors.
    Formula:C16H19BrN2·C4H4O4
    Purity:99.80%
    Color and Shape:Crystal Powder
    Molecular weight:435.31
  • Benztropine mesylate

    CAS:
    <p>Benztropine mesylate (Benztropine methanesulfonate) is a centrally active muscarinic antagonist that has been used in the symptomatic treatment of PARKINSON</p>
    Formula:C21H25NO·CH4SO3
    Purity:98.41% - 99.96%
    Color and Shape:White Crystalline Powder; Odourless Or Almost Odourless
    Molecular weight:403.53
  • CCR2-RA-[R]

    CAS:
    <p>CCR2-RA-[R] is a C-C chemokine receptor type 2 (CCR2) allosteric antagonist (IC50: 103 nM).</p>
    Formula:C18H19ClFNO3
    Purity:99.7%
    Color and Shape:Solid
    Molecular weight:351.8
  • Clozapine

    CAS:
    <p>Clozapine (HF 1854) is a tricylic dibenzodiazepine, classified as an atypical antipsychotic agent.</p>
    Formula:C18H19ClN4
    Purity:99.91% - 99.93%
    Color and Shape:Yellow Crystals From Acetone-Petroleum Ether Solid
    Molecular weight:326.82
  • Risperidone

    CAS:
    Risperidone (R 64 766) is a selective blocker of dopamine D2 receptors and serotonin 5-HT2 receptors that act as an atypical antipsychotic agent.
    Formula:C23H27FN4O2
    Purity:99.73%
    Color and Shape:Crystalline Solid
    Molecular weight:410.48
  • Isoprenaline hydrochloride

    CAS:
    Isoprenaline hydrochloride (NCI-c55630) is a potent beta-adrenergic agonist with the peripheral vasodilator, bronchodilator, and cardiac stimulating properties.
    Formula:C11H18ClNO3
    Purity:98% - 99.65%
    Color and Shape:Turn Brownish-Pink Upon Prolonged Exposure To Air (Ntp 1992)
    Molecular weight:247.719
  • INCB-9471

    CAS:
    INCB-9471 is a CCR5 antagonist with anti-HIV activity and inhibits the interaction between HIV-1 gp120.
    Formula:C30H40F3N5O2
    Purity:98.80%
    Color and Shape:Solid
    Molecular weight:559.666
  • PF429242 dihydrochloride

    CAS:
    <p>PF429242 dihydrochloride can reversibly inhibit S1P (IC50 of 175 nM).</p>
    Formula:C25H37Cl2N3O2
    Purity:99.68%
    Color and Shape:Solid
    Molecular weight:482.49
  • Sumatriptan succinate

    CAS:
    Sumatriptan succinate (GR 43175), a serotonin1 (5-HT1) receptor agonist, is used in the acute treatment of a migraine headache.
    Formula:C18H27N3O6S
    Purity:97.53% - 99.51%
    Color and Shape:White Powder
    Molecular weight:413.49
  • Salbutamol

    CAS:
    Salbutamol (Albuterol) stimulates beta2-adrenergic receptors in the lungs, thereby activating the enzyme adenylate cyclase that catalyzes the conversion of ATP to cyclic-3', 5'-adenosine monophosphate (cAMP).
    Formula:C13H21NO3
    Purity:91.59% - 99.9%
    Color and Shape:White To Off-White Crystalline Solid Solid
    Molecular weight:239.31
  • Droperidol

    CAS:
    <p>Droperidol (Dehydrobenzperidol) is a Dopamine-2 Receptor Antagonist. The mechanism of action of droperidol is as a Dopamine D2 Antagonist.</p>
    Formula:C22H22FN3O2
    Purity:97.16% - 98%
    Color and Shape:Solid
    Molecular weight:379.43
  • Alprenolol

    CAS:
    <p>Alprenolol (Alpheprol) is a non-selective β-adrenergic receptor (β-AR) antagonist that is also an antagonist of the serotonin (5-HT) receptor subtypes 5-HT1A</p>
    Formula:C15H23NO2
    Purity:99.72% - 99.78%
    Color and Shape:Solid
    Molecular weight:249.35
  • Nardeterol HCl


    <p>Nardeterol HCl is a β-adrenergic receptor partial agonist used in the study of the central nervous system.CAS 번호13460-73-83-4</p>
    Formula:C20H25ClFN3O2
    Purity:97.72% - 98.65%
    Color and Shape:Soild
    Molecular weight:393.88
  • Ezlopitant

    CAS:
    <p>Ezlopitant (CJ-11974) is a small molecule neurokinin-1-receptor (NK1) antagonist used to treat nausea, vomiting and pain.</p>
    Formula:C31H38N2O
    Purity:97.49%
    Color and Shape:Solid
    Molecular weight:454.65
  • Fenoterol

    CAS:
    Fenoterol is an agonist of β2-adrenergic receptor It is classed as sympathomimetic beta agonist and asthma medication.
    Formula:C17H21NO4
    Purity:98.29%
    Color and Shape:Solid
    Molecular weight:303.35
  • Amylin, amide, human

    CAS:
    Amylin, amide, human(DAP Amide) is a 37-amino acid peptide hormone co-secreted with insulin to regulate postprandial glucose levels.
    Formula:C165H261N51O55S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:3903.28
  • Tropisetron hydrochloride

    CAS:
    <p>Tropisetron hydrochloride (Tropisetron HCl) is a selective, competitive serotonin 5-HT3 receptor antagonist, with antinauseant and antiemetic activities.</p>
    Formula:C17H21ClN2O2
    Purity:99.72% - 99.83%
    Color and Shape:Solid
    Molecular weight:320.82
  • Gevotroline

    CAS:
    Gevotroline, a chemical in palm wine that can be used to treat psychosis, is a 5-HT2 receptor antagonist that can be used to study behavioral disorders.
    Formula:C19H20FN3
    Purity:99.45%
    Color and Shape:Solid
    Molecular weight:309.38
  • Chlorpheniramine maleate

    CAS:
    <p>Chlorpheniramine maleate (NCI-C55265) is a histamine H1 antagonist used in allergic reactions, hay fever, rhinitis, urticaria, and asthma.</p>
    Formula:C20H23ClN2O4
    Purity:99.64% - 99.98%
    Color and Shape:Odorless White Crystalline Solid Or White Powder With A Bitter Taste
    Molecular weight:390.87
  • Anatibant 2HCl

    CAS:
    <p>Anatibant 2HCl is a small molecule bradykinin B2 receptor antagonist for the treatment of neurological disorders and may be used in the study of brain injury.</p>
    Formula:C34H36Cl2N6O5S·2ClH
    Purity:99.17% - 99.58%
    Color and Shape:Soild
    Molecular weight:784.58
  • (Rac)-MGV354

    CAS:
    <p>(Rac)-MGV354: a racemic sGC activator; EC50s &lt;0.5 nM (CHO cells), 5 nM (GTM-3 E cells).</p>
    Formula:C35H37N5O3
    Purity:99.26%
    Color and Shape:Solid
    Molecular weight:575.7
  • Strontium ranelate

    CAS:
    <p>Strontium ranelate (S12911), a strontium (II) salt of the ranelic acid, is a medication for osteoporosis and can slow the course of osteoarthritis of the knee.</p>
    Formula:C12H6N2O8S·2Sr
    Purity:98.97%
    Color and Shape:Crystalline Solid
    Molecular weight:513.49
  • Volagidemab

    CAS:
    <p>Anti-CD34 Antibody is a CHO-expressed humanized monoclonal antibody targeting CD34, which can be used for the study of neurological and cardiovascular diseases.</p>
    Purity:97.8% (SDS-PAGE); 98% (SEC-HPLC) - 97.8% (SDS-PAGE); 98% (SEC-HPLC)
    Color and Shape:Liquid
  • p-MPPI hydrochloride

    CAS:
    <p>p-MPPI hydrochloride is a selective antagonist of 5-HT1A receptor, and has antidepressant and anxiolytic-like effects.</p>
    Formula:C25H28ClIN4O2
    Purity:99.95%
    Color and Shape:Solid
    Molecular weight:578.87
  • Vilazodone

    CAS:
    <p>Vilazodone (SB659746A): an SSRI and 5-HT-1A agonist, boosts serotonin to treat depression and anxiety.</p>
    Formula:C26H27N5O2
    Purity:99.61%
    Color and Shape:Light Yellow Solid
    Molecular weight:441.52
  • (1R,5S,6r)-N-(2-methyl-1-((3-methylpyridin-2-yl)oxy)propan-2-yl)-3-azabicyclo[3.1.0]hexane-6-carboxamide L(+)-Tartaric acid

    CAS:
    (1R,5S,6r)-N-(2-methyl-1-((3-methylpyridin-2-yl)oxy)propan-2-yl)-3-azabicyclo[3.1.0]hexane-6-carboxamide L(+)-Tartaric acid is a potential SSTR4 agonist.
    Formula:C20H29N3O8
    Purity:99.72%
    Color and Shape:Soild
    Molecular weight:439.46
  • Ifenprodil Tartrate

    CAS:
    <p>Ifenprodil is a selective NMDA receptor (glutamate) antagonist.</p>
    Formula:C21H27NO2C4H6O6
    Purity:99.02% - 99.55%
    Color and Shape:Solid
    Molecular weight:400.49
  • JNJ-39758979

    CAS:
    <p>JNJ-39758979: selective H4 receptor antagonist, Kis 12.5/5.3/25 nM (human/mouse/monkey), blocks histamine cAMP inhibition (pA2 7.9).</p>
    Formula:C11H19N5
    Purity:98.33% - 99.62%
    Color and Shape:Solid
    Molecular weight:221.3
  • 2-Bromo-6-methoxynaphthalene

    CAS:
    2-Bromo-6-methoxynaphthalene was used in the synthesis of nabumetone [4-(6-methoxy-2-naphthalenyl)-2-butanone] by Heck reaction.
    Formula:C11H9BrO
    Purity:98.51%
    Color and Shape:White To Off-White Powder
    Molecular weight:237.09
  • Ziprasidone hydrochloride monohydrate

    CAS:
    Ziprasidone hydrochloride monohydrate (CP 88059) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of the antipsychotic
    Formula:C21H21ClN4OS·HCl·H2O
    Purity:98% - 99.83%
    Color and Shape:Off-White Powder
    Molecular weight:467.12
  • Imidazolidinyl urea

    CAS:
    <p>Imidazolidinyl urea (Imidurea) is an antimicrobial preservative used in cosmetics.</p>
    Formula:C11H16N8O8
    Purity:98.6%
    Color and Shape:White Fluid Powder With Slight Characteristic Odor
    Molecular weight:388.29
  • AM095 free acid

    CAS:
    AM095 (free acid) is a potent LPA1 receptor antagonist (IC50s: 0.98 and 0.73 μM for recombinant human or mouse LPA1).
    Formula:C27H24N2O5
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:456.49
  • DREADD agonist 21

    CAS:
    <p>DREADD agonist 21 is a potent agonist of human muscarinic acetylcholine M3 receptors (EC50=1.7 nM).</p>
    Formula:C17H18N4
    Purity:99.94%
    Color and Shape:Solid
    Molecular weight:278.35
  • (R)-Elagolix

    CAS:
    (R)-Elagolix (NBI-56418) is an orally active, highly selective, short-term potent antagonist of the non-peptide gonadotropin-releasing hormone receptor.
    Formula:C32H30F5N3O5
    Purity:99.08%
    Color and Shape:Solid
    Molecular weight:631.59
  • Lafutidine

    CAS:
    <p>Lafutidine (FRG-8813) is a newly developed histamine H(2)-receptor antagonist, which can inhibit gastric acid secretion.</p>
    Formula:C22H29N3O4S
    Purity:98.55%
    Color and Shape:Yellowish White Crystalline Powder
    Molecular weight:431.55
  • Alarelin Acetate

    CAS:
    Alarelin Acetate is a synthetic GnRH agonist which can directly inhibit proliferation and DNA synthesis of rat GSMC through GnRH receptors.
    Formula:C56H78N16O12
    Purity:99.81% - >99.99%
    Color and Shape:White Powder
    Molecular weight:1167.34
  • Erenumab

    CAS:
    <p>Erenumab: human antibody blocking CGRP receptors to prevent migraines.</p>
    Purity:99.43% (SEC-HPLC) - > 95%
    Color and Shape:Liquid
    Molecular weight:146.2 kDa
  • Ciproquazone

    CAS:
    Ciproquazone has analgesic activity and is used to treat spondylitis.
    Formula:C19H18N2O2
    Purity:99.66%
    Color and Shape:Solid
    Molecular weight:306.36
  • Anamorelin

    CAS:
    <p>Anamorelin (ONO-7643) is a novel ghrelin receptor agonist (EC50: 0.74 nM in the FLIPR assay).</p>
    Formula:C31H42N6O3
    Purity:99.35% - 99.94%
    Color and Shape:Solid
    Molecular weight:546.7
  • Centanafadine hydrochloride

    CAS:
    Centanafadine HCl is a NE/DA reuptake inhibitor, also affects serotonin (IC50: NE 6 nM, DA 38 nM, serotonin 83 nM).
    Formula:C15H16ClN
    Purity:99.65%
    Color and Shape:Solid
    Molecular weight:245.75
  • Mizolastine

    CAS:
    Mizolastine (SL 850324), an antihistamine with IC50 of 47 nM, treats allergies like hay fever and hives.
    Formula:C24H25FN6O
    Purity:98% - 99.75%
    Color and Shape:Solid
    Molecular weight:432.49
  • 2',5'-Dideoxyadenosine

    CAS:
    2',5'-Dideoxyadenosine is a potent and non-competitive adenylyl cyclase inhibitor via binding the P-site (IC50: 3 μM).
    Formula:C10H13N5O2
    Purity:99.55%
    Color and Shape:White Solid
    Molecular weight:235.24
  • JP1302 dihydrochloride

    CAS:
    JP1302 dihydrochloride: selective α2C-adrenoceptor antagonist; Ki=28 nM, Kb=16 nM.
    Formula:C24H26Cl2N4
    Purity:99.61%
    Color and Shape:Solid
    Molecular weight:441.4
  • Sulpiride

    CAS:
    Sulpiride (Aiglonyl) is a dopamine D2-receptor antagonist, used therapeutically as an antidepressant, antipsychotic, and as a digestive aid.
    Formula:C15H23N3O4S
    Purity:99.94%
    Color and Shape:White Crystalline Powder
    Molecular weight:341.43
  • (±) Clopidogrel hydrogen sulfate

    CAS:
    (±) Clopidogrel hydrogen sulfate (Iscover) , an antiplatelet agent pharmacologically and structurally analogous to ticlopidine, is used to inhibit blood clots
    Formula:C16H16ClNO2S·H2SO4
    Purity:98.67% - 99.04%
    Color and Shape:Colorless To Light Yellow Liquid
    Molecular weight:419.9
  • Molindone hydrochloride

    CAS:
    <p>Molindone hydrochloride (EN-1733A) is an indole derivative effective in schizophrenia and other psychoses by blocking the effects of dopamine in the brain.</p>
    Formula:C16H24N2O2·HCl
    Purity:99% - 99.99%
    Color and Shape:Solid
    Molecular weight:312.84
  • CB1 antagonist 2

    CAS:
    CB1 antagonist 2 (AM4113) is caimabinoid 1 (CB1) antagonist which inhibits CB1 in vivo with an IC50 of 25.5 nM.
    Formula:C17H12Cl3N3O
    Purity:99.75%
    Color and Shape:Solid
    Molecular weight:380.66
  • Granisetron hydrochloride

    CAS:
    <p>Granisetron hydrochloride (Granisetron HCl) is a serotonin receptor (5HT-3 selective) antagonist that has been used as an antiemetic for cancer chemotherapy</p>
    Formula:C18H25ClN4O
    Purity:99.88% - 99.93%
    Color and Shape:White To Off-White Crystalline Solid
    Molecular weight:348.87
  • Desipramine hydrochloride

    CAS:
    Desipramine hydrochloride (Norimipramine) ,a secondary amine tricyclic antidepressant (TCA), is the hydrochloride salt form of desipramine.
    Formula:C18H23ClN2
    Purity:99.58% - 99.94%
    Color and Shape:White To Off-White Powder
    Molecular weight:302.842
  • CD80-IN-3

    CAS:
    CD80-IN-3 is a potent CD80 inhibitor and inhibits CD80/CD28 interaction (Kd: 125 nM; EC50: 630 nM).
    Formula:C17H10FN3O3
    Purity:98.08%
    Color and Shape:Solid
    Molecular weight:323.28
  • (S)-(-)-Atenolol

    CAS:
    (S)-(-)-Atenolol has beta-adrenergic blocking effects.
    Formula:C14H22N2O3
    Purity:99.31% - 99.81%
    Color and Shape:Solid
    Molecular weight:266.34
  • Bisoprolol hemifumarate

    CAS:
    Bisoprolol, a selective beta-1 adrenergic receptor antagonist, selectively and competitively binds to and blocks beta-1 adrenergic receptors in the heart,
    Formula:C20H33NO6
    Purity:98.69% - 99.84%
    Color and Shape:White To Offf-White Powder
    Molecular weight:383.49
  • Olodaterol

    CAS:
    Olodaterol is a novel, long-acting beta2-adrenergic agonist (LABA) that exerts its pharmacological effect by binding and activating beta2-adrenergic receptors
    Formula:C21H26N2O5
    Purity:98.9%
    Color and Shape:Solid
    Molecular weight:386.45
  • Tolazoline hydrochloride

    CAS:
    Tolazoline hydrochloride (NSC35110 (hydrochloride)) is a non-selective competitive α-adrenergic receptor antagonist used in treatment of persistent pulmonary
    Formula:C10H13ClN2
    Purity:99.67%
    Color and Shape:Pale Yellow Crystalline Solid
    Molecular weight:196.68
  • Lofepramine

    CAS:
    <p>Lofepramine (Leo 640) is a potent tricyclic antidepressant that is extensively metabolized to desipramine.</p>
    Formula:C26H27ClN2O
    Purity:98.38%
    Color and Shape:Crystals From Methanol Or Acetone Solid
    Molecular weight:418.96
  • Dexchlorpheniramine Maleate

    CAS:
    <p>Dexchlorpheniramine Maleate, an antihistamine with anticholinergic effects, treats allergies like hay fever. It's the active isomer of chlorpheniramine.</p>
    Formula:C20H23ClN2O4
    Purity:99.58%
    Color and Shape:White Or Almost White Crystalline Powder
    Molecular weight:390.86
  • Isoxsuprine hydrochloride

    CAS:
    Isoxsuprine hydrochloride (Isolait) is a beta-adrenergic agonist that causes direct relaxation of uterine and vascular smooth muscle.
    Formula:C18H24ClNO3
    Purity:99.38%
    Color and Shape:Crystals From Water Solid
    Molecular weight:337.84
  • PF-04995274

    CAS:
    PF-04995274: potent, selective partial 5-HT4R agonist; EC50 0.26-0.47 nM; brain penetrant; may treat Alzheimer's cognitive issues.
    Formula:C23H32N2O6
    Purity:99.52%
    Color and Shape:Solid
    Molecular weight:432.51
  • AZ084

    CAS:
    AZ084 is a potent, selective, allosteric, and oral active CCR8 antagonist (Ki: 0.9 nM). It has the potential to treat asthma.
    Formula:C26H34N4O2
    Purity:97.12%
    Color and Shape:Solid
    Molecular weight:434.57
  • Ondansetron hydrochloride dihydrate

    CAS:
    Ondansetron hydrochloride dihydrate (GR 38032) is a competitive serotonin type 3 receptor antagonist,which has reported anxiolytic and neuroleptic properties.
    Formula:C18H19N3O·HCl·2H2O
    Purity:99.92%
    Color and Shape:White Crystal Powder
    Molecular weight:365.86
  • Sergliflozin A

    CAS:
    Sergliflozin A is a selective SGLT2 inhibitor that induces diabetes in a dose-dependent manner. It reduces hyperglycemia.
    Formula:C20H24O7
    Purity:99.71%
    Color and Shape:Solid
    Molecular weight:376.4
  • Prostaglandin E1

    CAS:
    Alprostadil (PGE1) is a natural vasodilator that also inhibits platelets and induces bronchodilation, used in erectile dysfunction treatment.
    Formula:C20H34O5
    Purity:99.78% - >99.99%
    Color and Shape:Solid
    Molecular weight:354.48
  • Hydroxyzine Pamoate

    CAS:
    Hydroxyzine Pamoate (Bobsule) is a histamine H1 receptor antagonist that is effective in the treatment of chronic urticaria and histamine-mediated pruritus.
    Formula:C44H43ClN2O8
    Purity:99.49%
    Color and Shape:Solid
    Molecular weight:763.27
  • Cinnarizine

    CAS:
    <p>Cinnarizine is a piperazine, blocks H1-receptor &amp; Ca-channels, has vasodilating &amp; antiemetic effects, may cause Parkinson-like symptoms.</p>
    Formula:C26H28N2
    Purity:99.94%
    Color and Shape:Solid
    Molecular weight:368.51
  • REV 5901A

    CAS:
    <p>REV 5901A (REV 5901 HCl) is a leukotriene receptor antagonist and 5-LOX inhibitor with antimicrobial activity that attenuates the growth of colon cancer in mice</p>
    Formula:C22H26ClNO2
    Purity:98.04%
    Color and Shape:Soild
    Molecular weight:371.90
  • PF-5190457

    CAS:
    PF-5190457 is an effective and selective ghrelin receptor inverse agonist (pKi: 8.36).
    Formula:C29H32N6OS
    Purity:99.34%
    Color and Shape:Solid
    Molecular weight:512.67
  • Atomoxetine hydrochloride

    CAS:
    <p>Atomoxetine HCl (LY 139603) is a selective non-stimulant ADHD drug that blocks norepinephrine reuptake, enhancing focus and reducing impulsivity.</p>
    Formula:C17H22ClNO
    Purity:99.86%
    Color and Shape:White Solid
    Molecular weight:291.82
  • [Leu15]-Gastrin I, human

    CAS:
    [Leu15]-Gastrin I, human is a variant of Gastrin I, modulating the binding of cholecystokinin to mucosal membranes.
    Formula:C98H126N20O31
    Purity:98.02% - 98.84%
    Color and Shape:Solid
    Molecular weight:2080.16
  • Sertraline hydrochloride

    CAS:
    <p>Sertraline hydrochloride (Sertraline HCl) is a selective serotonin uptake inhibitor that is used in the treatment of depression.</p>
    Formula:C17H18Cl3N
    Purity:99.12% - 99.89%
    Color and Shape:Solid Powder
    Molecular weight:342.691
  • Iobenguane sulfate

    CAS:
    Iobenguane sulfate is used in radioiodinated form to diagnose and treat adrenergic tumors.
    Formula:C8H10IN3H2O4S
    Purity:99.04%
    Color and Shape:Solid
    Molecular weight:324.12
  • Bromperidol

    CAS:
    Bromperidol (R-11333) is a butyrophenone derivative and it is a potent and long-acting neuroleptic.
    Formula:C21H23BrFNO2
    Purity:99.89%
    Color and Shape:Tan Solid
    Molecular weight:420.32
  • Doxofylline

    CAS:
    Doxofylline (Doxophylline) is a methylxanthine derivative with the presence of a dioxolane group in position 7.
    Formula:C11H14N4O4
    Purity:99.958% - >99.99%
    Color and Shape:Solid
    Molecular weight:266.25
  • (-)-GSK598809 hydrochloride

    CAS:
    <p>(-)-GSK598809 hydrochloride, a DRD3 selective antagonist, may correct reward deficits in substance dependence.</p>
    Formula:C22H24ClF4N5OS
    Purity:98.36%
    Color and Shape:Soild
    Molecular weight:517.97
  • Bromopride

    CAS:
    Bromopride (Valopride), a metoclopramide-like dopamine antagonist and prokinetic, is an antiemetic not sold in the US or UK.
    Formula:C14H22BrN3O2
    Purity:99.95%
    Color and Shape:Solid
    Molecular weight:344.25
  • Carvedilol EP IMpurity E

    CAS:
    <p>Carvedilol EP IMpurity E (Carvedilol USP E) is used as a pharmaceutical intermediate.</p>
    Formula:C9H14ClNO2
    Purity:99.53%
    Color and Shape:White To Almost White Solid Crystalline
    Molecular weight:203.666
  • Indusatumab

    CAS:
    <p>Indusatumab (5F9 Monoclonal antibody) is an anti-human GUCY2C (Guanylate cyclase 2C) monoclonal antibody that can be used to synthesize antibody-drug conjugate.</p>
    Purity:> 95% - > 95%
    Color and Shape:Liquid
    Molecular weight:145.18 kDa