Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,781 products)
- Apoptosis(6,260 products)
- Cell Cycle/Checkpoint(4,792 products)
- Chromatin/Epigenetics(2,440 products)
- Cytoskeletal Signaling(1,527 products)
- DNA Damage/DNA Repair(2,968 products)
- Endocrinology/Hormones(3,706 products)
- Enzyme(3,667 products)
- GPCR/G-Protein(9,005 products)
- Immunology and Inflammation(3,874 products)
- Influenza Virus(301 products)
- JAK/STAT signaling(414 products)
- MAPK Signaling(1,248 products)
- Membrane Transporter/Ion Channel(3,033 products)
- Metabolism(10,207 products)
- Microbiology/Virology(7,591 products)
- Neuroscience(10,382 products)
- Other Inhibitors(36,042 products)
- Oxidation-Reduction(42 products)
- PI3K/Akt/mTOR Signaling(1,444 products)
- Proteases/Proteasome(1,724 products)
- Stem Cell and Derivatives(825 products)
- Tyrosine Kinase/Adaptors(2,035 products)
- Ubiquitination(1,717 products)
Show 16 more subcategories
Found 66686 products of "Inhibitors"
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ICMT-IN-25
CAS:ICMT-IN-25 (compound 37) serves as a potent inhibitor of isoprenylcysteine carboxyl methyltransferase (ICMT), exhibiting an IC50 value of 0.025 μM [1].Formula:C21H26ClNOColor and Shape:SolidMolecular weight:343.89Cap-dependent endonuclease-IN-13
CAS:Cap-dependent endonuclease-IN-13 is a potent inhibitor of cap-dependent endonuclease (CEN) and shows research potential against influenza virus infection (Formula:C25H20F2N4O4SColor and Shape:SolidMolecular weight:510.51L-689502
CAS:L-689502 is a potent HIV-l protease inhibitor (IC50: 1 nM).Formula:C39H51N3O7Purity:98%Color and Shape:SolidMolecular weight:673.84TNF-α-IN-8
CAS:TNF-α-IN-8 (compound I-42) is an isoindole-imide-based inhibitor of tumor necrosis factor-alpha (TNF-α) with applications in researching various diseasesFormula:C15H12N6O5Color and Shape:SolidMolecular weight:356.29HIV-1 protease-IN-11
CAS:HIV-1 protease-IN-11 (compound 34a), an HIV-1 protease inhibitor, demonstrates potent inhibition with an IC50 of 0.41 nM and maintains substantial efficacyFormula:C26H37N3O5SPurity:98%Color and Shape:SolidMolecular weight:503.65CD33 splicing modulator 1 hydrochloride
CAS:CD33 Splicing Modulator 1 Hydrochloride (Compound 1) is a myeloid lineage cell surface receptor CD33/Siglec 3 modulator involved in regulating microgliaFormula:C25H26ClFN6OColor and Shape:SolidMolecular weight:480.97Iganidipine
CAS:Iganidipine（NKY 722） is a new water-soluble Ca2+ antagonist with antihypertensive activity for research and neurological related diseases.Formula:C28H38N4O6Purity:96.3%Color and Shape:SolidMolecular weight:526.62Deoxynybomycin
CAS:Deoxynybomycin, a selective anti-tumor agent, inhibits topoisomerase I and induces apoptosis.Formula:C16H14N2O3Purity:98%Color and Shape:SolidMolecular weight:282.29Dicentrine, (-)-
CAS:Dicentrine (NSC-251699), an aporphinic alkaloid from plants, has strong pain relief effects in mice.Formula:C20H21NO4Purity:99.86%Color and Shape:SolidMolecular weight:339.39Ilepatril
CAS:Ilepatril, also known as AVE-7688, is a vasopeptidase inhibitor for the treatment of hypertension.Formula:C22H28N2O5SColor and Shape:SolidMolecular weight:432.53HA-29
CAS:HA-29 is an inhibitor of thromboxane A2 and prostaglandin endoperoxide receptors.Formula:C16H16N2O3Color and Shape:SolidMolecular weight:284.31Nirogacestat dihydrobromide
CAS:Potent γ-secretase inhibitor; IC50: 1.2 nM (cell), 6.2 nM (cell-free); lowers Aβ in mice/guinea pigs' brain, CSF, plasma.Formula:C27H43Br2F2N5OColor and Shape:SolidMolecular weight:651.48XDM-CBP
CAS:XDM-CBP is an effective and selective CBP/p300 bromodomain inhibitor.Formula:C21H22N2O4Purity:98%Color and Shape:SolidMolecular weight:366.41Pumaprazole
CAS:Pumaprazole (BY-841) is an antagonist of a reversible proton pump.Formula:C19H22N4O2Purity:99.91%Color and Shape:SolidMolecular weight:338.4Ref: TM-T16682
1mg92.00€5mg188.00€10mg311.00€25mg635.00€50mg1,017.00€100mg1,644.00€200mg2,213.00€1mL*10mM (DMSO)215.00€AGN-201904Z
CAS:AGN-201904Z is a slow-release, acid-resistant pro-PPI that turns into omeprazole, offering extended acid suppression.Formula:C25H25N3NaO8S2Purity:98%Color and Shape:SolidMolecular weight:582.6BF738735
CAS:<p>BF738735 is a selective inhibitor of phosphatidylinositol 4-kinase III beta (PI4KIIIβ, IC50 = 5.7 nM) showing higher activity over α(IC50 = 1.7 μM).</p>Formula:C21H19FN4O3SPurity:90%Color and Shape:SolidMolecular weight:426.46IR415
CAS:IR415 selectively interacts with Hepatitis B virus X protein (HBx, Kd = 2 nM) and blocks HBV-mediated RNAi suppression, reverses the inhibitory effect of HBxFormula:C13H14F2N4SPurity:99.85%Color and Shape:SolidMolecular weight:296.34Ref: TM-T11669
5mg46.00€10mg74.00€25mg135.00€50mg226.00€100mg335.00€200mg469.00€1mL*10mM (DMSO)49.00€USP7-IN-3
CAS:USP7-IN-3 is a potent and selective allosteric inhibitor of ubiquitin-specific protease 7 (USP7).Formula:C29H31F3N6O3Purity:98%Color and Shape:SolidMolecular weight:568.593-Oxo-5β-cholanoic acid
CAS:3-Oxo-5β-cholanoic acid (Dehydrolithocholic acid) (Dehydrolithocholic acid) is a bile acid metabolite and inhibits the differentiation of TH17 cells by directlyFormula:C24H38O3Purity:98.01% - 99.86%Color and Shape:SolidMolecular weight:374.56ICMT-IN-30
CAS:ICMT-IN-30 (compound 67) is an ICMT inhibitor with an IC50 value of 0.27 μM [1].Formula:C19H25NOSColor and Shape:SolidMolecular weight:315.47Pentiapine
CAS:Pentiapine (CGS 10746) is a novel inhibitor of dopamine release.Formula:C15H17N5SPurity:99.35%Color and Shape:SolidMolecular weight:299.39Ref: TM-T12405
1mg487.00€5mg753.00€10mg1,216.00€25mg1,691.00€50mg2,262.00€100mg3,068.00€1mL*10mM (DMSO)938.00€MF498
CAS:MF498 is a novel and selective E prostanoid receptor 4 (EP4 receptor) antagonist, displayed a strong binding affinity for the EP4 receptor (Ki: 0.7 nM).Formula:C32H33N3O7SPurity:98%Color and Shape:SolidMolecular weight:603.69Antiproliferative agent-33
CAS:Antiproliferative Agent-33 (Compound 2g) serves as an anti-proliferative, antifungal, and antibacterial agent, effectively inhibiting the proliferation of MDA-Formula:C21H26N2OColor and Shape:SolidMolecular weight:322.44UCB7362
CAS:UCB7362 (GLXC-26743) is an orally available and potent plasmepsin X (PMX) inhibitor with anti-malarial activity.UCB7362 inhibits parasite reproduction.Formula:C25H26ClN5O3Purity:97.67%Color and Shape:SolidMolecular weight:479.96Vonifimod
CAS:Vonifimod is an immunomodulator .Formula:C17H34N4O2Color and Shape:SolidMolecular weight:326.481,2-Diheptadecanoyl-sn-glycero-3-phosphorylcholine
CAS:1,2-Diheptadecanoyl-sn-glycero-3-phosphorylcholine (DHPC) is a derivative of phosphatidylcholine (PC) that exhibits biological activity, functioning as aFormula:C42H84NO8PColor and Shape:SolidMolecular weight:762.09ROCK2-IN-7
CAS:<p>ROCK2 inhibitor is a chemical compound associated with the therapeutic management of psoriasis.</p>Formula:C26H28FN5OPurity:98%Color and Shape:SolidMolecular weight:445.53Azt-pmap
CAS:AZT-PMPA, an aryl phosphate derivative of AZT and a nucleoside analogue, demonstrates anti-HIV activity[1].Formula:C20H25N6O8PPurity:98%Color and Shape:SolidMolecular weight:508.42AGN-195183
CAS:AGN 195183: RARα agonist, Kd=3 nM, selective, no RARβ/γ effect, inhibits breast cancer cells, in Phase I/II clinical trials, non-irritant.Formula:C22H22ClF2NO4Color and Shape:SolidMolecular weight:437.86KRAS G12D mutation regulator 4
CAS:KRAS G12D mutation regulator 4 can be used in studies about Ras.Formula:C33H33FN6O2Color and Shape:SolidMolecular weight:564.65Epigenetic factor-IN-1
CAS:<p>Epigenetic factor-IN-1 (40569Z) is an epigenetic factor inhibitor that exhibits potent binding affinity for SIRT7.</p>Formula:C32H34FN5O6S2Purity:98%Color and Shape:SolidMolecular weight:667.77Solitomab
CAS:Solitomab (AMG 110) is a bispecific antibody targeting CD3 and EpCAM, used in uterine/ovarian carcinosarcoma research.Purity:95%Color and Shape:Liquid(2R,4R)-APDC
CAS:(2R,4R)-APDC is a selective group II metabotropic glutamate receptors (mGluRs) agonist. It has anticonvulsant and neuroprotective effects.Formula:C6H10N2O4Purity:98%Color and Shape:SolidMolecular weight:174.15ALP/Carbonic anhydrase-IN-1
CAS:<p>Compound 1e, also known as ALP/Carbonic anhydrase-IN-1, is a dual inhibitor targeting both carbonic anhydrase (CA) isozymes II, IX, and XII, as well as alkaline</p>Formula:C15H16N2Purity:98%Color and Shape:SolidMolecular weight:224.3IR-Crizotinib
CAS:IR-Crizotinib is a conjugate of the near-infrared dye IR-786 and Crizotinib, an NF-κB-inducing kinase (NIK) inhibitor, with an IC50 of 3.381 μM for intracranialFormula:C53H57Cl2FIN7OPurity:98%Color and Shape:SolidMolecular weight:1024.88Topoisomerase I inhibitor 9
CAS:Topoisomerase I Inhibitor 9 (compound 3d), a specific inhibitor of leishmanial topoisomerase IB, exhibits antileishmanial activity, demonstrating an IC50 valueFormula:C23H15Br2FN2Purity:98%Color and Shape:SolidMolecular weight:498.19YM281
CAS:<p>YM281 is a potent EZH2 inhibitor, causes apoptosis and G0/G1 arrest, has antitumor activity in vivo, and may be researched for lymphoma.</p>Formula:C56H71N7O9SColor and Shape:SolidMolecular weight:1018.27Org 6582
CAS:Org 6582 inhibits 3-hydroxytryptamine reuptake.Formula:C13H15Cl2NColor and Shape:SolidMolecular weight:256.17PPARδ agonist 9
CAS:PPARδ agonist 9 (compound 21), with an EC50 of 3.6 nM, is effective in vivo, decreasing serum MCP-1 concentrations in mice and markedly reducing atheroscleroticFormula:C26H28ClF3N4O3SPurity:98%Color and Shape:SolidMolecular weight:569.04BIO-7662
CAS:BIO-7662 is an effective and highly selective antagonist of α4β1 integrin.Formula:C38H48N6O8SPurity:98%Color and Shape:SolidMolecular weight:748.89KUNG94
KUNG94 selectively inhibits Grp94 at 8 nM IC50, a 90 kDa Hsp90 variant in the endoplasmic reticulum.Formula:C22H18FNO3Purity:98%Color and Shape:SolidMolecular weight:363.39Bivamelagon
CAS:MC-4R Agonist 2 (Example 1), a melanocortin 4 receptor (MC4R) agonist, is employed in the research of conditions such as obesity, diabetes, inflammation, andFormula:C35H53ClN4O4Purity:100%Color and Shape:SolidMolecular weight:629.27Estrogen receptor modulator 7
CAS:Estrogen Receptor Modulator 7 is a potent modulator of estrogen receptors, utilized in cancer research [1].Formula:C30H31BCl2FNO3Purity:98%Color and Shape:SolidMolecular weight:554.29Indacrinone
CAS:Indacrinone is an investigational diuretic.Formula:C18H14Cl2O4Purity:98%Color and Shape:SolidMolecular weight:365.21Adam-20-S
CAS:Adam-20-S is a potent inhibitor of glucosinolate sulfatase, exhibiting an IC50 of 9.04 μg/mL.Formula:C17H21FN2O4SColor and Shape:SolidMolecular weight:368.42WAY-660222
CAS:WAY-660222 is an active molecule.Formula:C19H13FOColor and Shape:SolidMolecular weight:276.3Balapiravir hydrochloride
CAS:Balapiravir HCl, an NS5B inhibitor, is used potentially for the treatment of HCV infection.Formula:C21H31ClN6O8Color and Shape:SolidMolecular weight:530.96Nepaprazole
CAS:Nepaprazole (TY-11345) is a potent proton pump inhibitor; IC50: 5.8µM at pH 6.0, 9.9µM at pH 7.4. Better inhibition in weak acid.Formula:C18H19N3O2SPurity:98%Color and Shape:SolidMolecular weight:341.43AZ-TAK1
CAS:"AZ-Tak1 inhibits TAK1 kinase (IC50=0.009mM), reduces p38/ERK levels, and induces apoptosis in Mino, SP53, Jeko cells with increasing efficacy at 0.1-0.5mM."Formula:C25H28FN7O2Color and Shape:SolidMolecular weight:477.53MS934
CAS:<p>MS934, a novel VHL-recruiting MEK 1/2 degrader, exhibits potent anti-proliferative effects on HT-29 cell growth, achieving a GI50 of 0.023 μM.</p>Formula:C52H69F3IN7O6SPurity:98%Color and Shape:SolidMolecular weight:1104.11Propiolactone
CAS:<p>Propiolactone (β-propiolactone; 2-Oxetanone), a chemosterilant, effectively inactivates viruses, rendering them non-infectious.</p>Formula:C3H4O2Purity:98%Color and Shape:SolidMolecular weight:72.06MTI-31
CAS:MTI-31 (LXI-15029) is a potent oral mTORC1/2 inhibitor with a Kd of 0.20 nM, >5,000-fold selectivity, and an IC50 of 39 nM.Formula:C26H30N6O3Purity:99.97%Color and Shape:SolidMolecular weight:474.55THRβ receptor agonist-1
CAS:THRβ receptor agonist-1 is an agonist for the THRβ receptor [1].Formula:C18H12Cl2N6O4Color and Shape:SolidMolecular weight:447.23Anti-inflammatory agent 44
CAS:Compound 1 (Anti-inflammatory agent 44) is a 6-methoxyflavonol glycoside exhibiting anti-inflammatory properties, and it can be extracted from the aerial partsFormula:C43H48O25Color and Shape:SolidMolecular weight:964.83ω-3 Arachidonic acid ethyl ester
CAS:Omega-3 Arachidonic Acid ethyl ester, a rare polyunsaturated fatty acid with limited presence in dietary sources, is crucial for infant growth and developmentFormula:C22H36O2Color and Shape:SolidMolecular weight:332.52Fecosterol
CAS:Fecosterol, a metabolite derived from Saccharomyces cerevisiae, is utilized in phytosterolemia research.Formula:C28H46OColor and Shape:SolidMolecular weight:398.66Siremadlin (R Enantiomer)
CAS:Siremadlin R Enantiomer is the R enantiomer of Siremadlin. Siremadlin is a potent and highly specific inhibitor of MDM-2/p53.Formula:C26H24Cl2N6O4Purity:98%Color and Shape:SolidMolecular weight:555.41PK68
CAS:PK68 selectively inhibits RIPK1 (IC50=90nM), potentially useful in inflammation and cancer metastasis studies.Formula:C22H24N4O3SPurity:98.09% - 99.64%Color and Shape:SolidMolecular weight:424.52Ref: TM-T12493
1mg81.00€5mg170.00€10mg274.00€25mg518.00€50mg747.00€100mg938.00€1mL*10mM (DMSO)188.00€MALT1-IN-6
CAS:MALT1-IN-6 is a MALT1 protease inhibitor (Ki: 9 nM) that exhibits anticancer activity.Formula:C18H12Cl2F3N9OColor and Shape:SolidMolecular weight:498.25CGP 20376
CAS:<p>CGP 20376: Benzothiazole anthelmintic, modulates eosinophil burst, antifibrillatory, dose-dependent effects.</p>Formula:C16H20N2O3S3Purity:95.11%Color and Shape:SolidMolecular weight:384.54Stobadine
CAS:Stobadine, a potent antioxidant, safeguards endoplasmic reticulum (ER) membrane fluidity against free radical-induced changes.Formula:C13H18N2Purity:98%Color and Shape:SolidMolecular weight:202.3(-)-IHCH7041
CAS:(–)-IHCH7041 is a optical rotation negative isomer of IHCH7041.Formula:C24H35N5OColor and Shape:SolidMolecular weight:409.57Antibacterial agent 135
CAS:Antibacterial Agent 135 (example 7) effectively inhibits various bacteria, including P.Formula:C11H15N5O6SColor and Shape:SolidMolecular weight:345.33Gestonorone Capronate
CAS:Gestonorone Capronate is a progesterone used in benign prostatic hyperplasia and endometrial cancer studies.Formula:C26H38O4Purity:99.19%Color and Shape:SolidMolecular weight:414.58Ref: TM-T13703
1mg145.00€5mg319.00€10mg472.00€25mg753.00€50mg1,074.00€100mg1,444.00€1mL*10mM (DMSO)361.00€L 670548
CAS:L 670548 is an agonist of muscarinic receptor.Formula:C9H13N3OPurity:98%Color and Shape:SolidMolecular weight:179.22Vitamin CK3
CAS:Vitamin CK3 is the combination of Vitamin C and vitamin K3 and has been shown to inhibit tumor growth and lung metastasis.Formula:C17H18Na2O11SPurity:98%Color and Shape:SolidMolecular weight:476.36FK706
CAS:FK706, a human neutrophil elastase inhibitor (IC50: 83 nM, Ki: 4.2 nM), also blocks mouse and porcine elastases. Anti-inflammatory.Formula:C26H33F3N4NaO7Color and Shape:SolidMolecular weight:593.556PTAC oxalate
CAS:muscarinic receptor ligandFormula:C14H21N3O4S2Purity:98%Color and Shape:SolidMolecular weight:359.46(Iso)-MS4322
CAS:(Iso)-MS4322 ((Iso)-YS43-22) is a protein arginine methyltransferase 5 (PRMT5 ) degrader with potential anticancer activity.Formula:C55H76N10O12SPurity:99.05% - 99.79%Color and Shape:SolidMolecular weight:1101.32O-2050
CAS:O-2050: strong CB1 antagonist (Ki 2.5 nM), CB2 inhibitor (Ki 0.2 nM); reduces mouse food intake, increases activity.Formula:C23H31NO4SPurity:98%Color and Shape:SolidMolecular weight:417.56DNA gyrase B-IN-3
CAS:DNA gyrase B-IN-3 (Compound A), with an IC50 of less than 10 nM, acts as an inhibitor of bacterial DNA gyrase B and exhibits antibacterial activity against GramFormula:C14H9Cl2N3O4SPurity:98%Color and Shape:SolidMolecular weight:386.21TAM558
CAS:TAM558 is a payload molecule utilized in the synthesis of OMTX705, which is a humanized anti-fibroblast-activating protein (FAP) antibody conjugated to theFormula:C79H122N14O19SColor and Shape:SolidMolecular weight:1603.96Gusperimus trihydrochloride
CAS:Gusperimus trihydrochloride is a derivative of the antitumor antibiotic spergualin with immunosuppressant activity.Formula:C17H40Cl3N7O3Purity:98%Color and Shape:SolidMolecular weight:496.9Potassium Channel Activator 1
CAS:Potassium Channel Activator 1 aids treatment of ADHD, schizophrenia, and mood disorders by targeting the dopaminergic system.Formula:C19H23N3O3Purity:99.86%Color and Shape:SolidMolecular weight:341.4Dendrogenin A
CAS:Dendrogenin A (DDA) is a compound acting as a selective liver X receptor (LXR) modulator, cholesterol epoxide hydrolase inhibitor (Ki = 120 nM), and a metabolicFormula:C32H55N3O2Color and Shape:SolidMolecular weight:513.80Enpp-1-IN-4
CAS:Enpp-1-IN-4: potent enpp-1 inhibitor with potential in cancer research. See patent WO2019177971A1, compound 1.Formula:C19H19N5O5SColor and Shape:SolidMolecular weight:429.45Bisegliptin
CAS:Bisegliptin(KRP-104) is a small molecule compound with anti-diabetic activity.Formula:C18H26FN3O3Purity:98%Color and Shape:SolidMolecular weight:351.42AP-C6
CAS:AP-C6 is a potent inhibitor of guanosine 3',5'-cyclic monophosphate (cGMP)-dependent protein kinase II (cGKII), exhibiting a pIC50 of 6.5.Formula:C15H15N5OColor and Shape:SolidMolecular weight:281.31PAT-505
CAS:PAT-505 is an autologous epidermal growth factor inhibitor.Formula:C23H18ClF2N3O2SPurity:98.84%Color and Shape:SolidMolecular weight:473.92AMPK-IN-1
CAS:AMPK-IN-1 is an activator of the AMP-activated protein kinase (AMPK) enzyme, specifically targeting the α2β2γ1 isoform with an EC50 of 551 nM.Formula:C24H18ClN3O3Color and Shape:SolidMolecular weight:431.87PARP-1-IN-3
CAS:PARP-1-IN-3 is a potent PARP-1 inhibitor that inhibits PARP-1 and PARP-2 with IC50 values of 0.25 nM and 2.34 nM, respectively.PARP-1-IN-3 has potential anti-Formula:C21H17BrN2O3Purity:99.86%Color and Shape:SolidMolecular weight:425.28IMD-vanillin
CAS:IMD-vanillin is a novel compound characterized as an imidazoquinolinone-derived dimer with NF-κB immunomodulatory properties.Formula:C37H45N7O4Purity:98%Color and Shape:SolidMolecular weight:651.8CLP257
CAS:<p>CLP257 is a selective K+-Cl− cotransporter KCC2 activator (EC50: 616 nM) and it is inactive against NKCC1, GABAA receptors, KCC1, KCC3 or KCC4.</p>Formula:C14H14FN3O2SPurity:99.5%Color and Shape:SolidMolecular weight:307.34VU 0255035
CAS:<p>VU 0255035 is a highly selective, competitive and brain penetrant muscarinic M1 receptor antagonist with an IC50 of 130 nM.</p>Formula:C18H20N6O3S2Purity:98.09% - 98.1%Color and Shape:SolidMolecular weight:432.52LCB-2853
CAS:LCB-2853 is a potent thromboxane A2/prostaglandin H2 (TXA2/PGH2) receptor antagonist with antiplatelet aggregation, antivasospasm, and antithrombotic effects.Formula:C21H24ClNO4SPurity:97.15%Color and Shape:SolidMolecular weight:421.94BAY-204
CAS:BAY-204 is a CSNK1α/δ inhibitor that can be used in the treatment of proliferative diseases.Formula:C29H26F3N5O2Color and Shape:SolidMolecular weight:533.54RORγt inverse agonist 26
CAS:RORγt inverse agonist 26, a potent reverse agonist of RORγt, effectively modulates Th17 cell differentiation and suppresses IL-17 production.Formula:C27H21F7N2O5SColor and Shape:SolidMolecular weight:618.52L-Moses
CAS:L-45 is the first potent and cell-active bromodomain (Brd) inhibitor of p300/CBP-associated factor (PCAF) (Kd: 126±15 nM).Formula:C21H24N6Purity:98%Color and Shape:SolidMolecular weight:360.46Fosnetupitant chloride monohydrochloride
CAS:Fosnetupitant chloride monohydrochloride (Pro-netupitant chloride monohydrochloride) is a selective NK1 antagonist exhibiting high affinity for the human NK1Formula:C31H37Cl2F6N4O5PPurity:98%Color and Shape:SolidMolecular weight:761.52Gliamilide
CAS:Gliamilide is a high-potency sulfamylurea hypoglycemic agent.Formula:C23H33N5O5SColor and Shape:SolidMolecular weight:491.6Niceritrol
CAS:Niceritrol (Cardiolipol) is a niacin ester that reduces cholesterol and triglycerides in total plasma and in the VLD and LD lipoprotein fractions.Formula:C29H24N4O8Purity:97.02%Color and Shape:SolidMolecular weight:556.52Ref: TM-T19861
1mg60.00€2mg85.00€5mg109.00€10mg156.00€25mg269.00€50mg404.00€100mg597.00€1mL*10mM (DMSO)150.00€H3 receptor antagonist 1
CAS:H3 receptor antagonist 1 is used in the study of neurological diseases, histamine H3 receptor antagonist.Formula:C20H28F2N2OPurity:98%Color and Shape:SolidMolecular weight:350.45UBP316
CAS:GluR5-containing kainate receptor antagonistFormula:C20H19N3O6SPurity:98%Color and Shape:SolidMolecular weight:429.45NCT-10b
CAS:NCT-10b is a selective inhibitor of HDAC6.Formula:C21H38N2O4SPurity:98%Color and Shape:SolidMolecular weight:414.6Tyk2-IN-9
CAS:Tyk2-IN-9: selective Tyk-2 inhibitor, IC50 of 0.076 nM (TYK2-JH2), 1.8 nM (JAK1-JH2), for inflammation/autoimmune research.Formula:C20H17N9Purity:98%Color and Shape:SolidMolecular weight:383.41T 98475
CAS:gonadotropin-releasing hormone (GnRH, LHRH) receptor antagonist,orally activeFormula:C37H37F2N3O4SPurity:98%Color and Shape:SolidMolecular weight:657.77Ro 23-0364
CAS:Ro 23-0364 an imidazobenzodiazepine with mixed benzodiazepine agonist/antagonist properties.Formula:C18H13ClN4OColor and Shape:SolidMolecular weight:336.78Alclofenac
CAS:Alclofenac (W-7320) aids chronic rheumatism by affecting acute phase proteins and L-tryptophan binding.Formula:C11H11ClO3Purity:99.89%Color and Shape:SolidMolecular weight:226.66PQM130
CAS:PQM130 is a Feruloyl-Donepezil Hybrid compound against the neurotoxicity induced by Aβ1-42 oligomer (AβO) and shows anti-inflammatory activity.Formula:C23H27NO4Purity:98.73%Color and Shape:SolidMolecular weight:381.46NS5A-IN-3
CAS:NS5A-IN-3 is a potent NS5A inhibitor with high efficacy against HCV 1b, good activity on 3a, and strong metabolic stability; superior to daclatasvir.Formula:C44H44N6O8Purity:98%Color and Shape:SolidMolecular weight:784.86Cgp 6809
CAS:CGP 6809: a methylnitrosoureido-sugar derivative active against various mice/rat tumors; promising for bowel/lung cancer trials.Formula:C12H23N3O7Color and Shape:SolidMolecular weight:321.33Fenquinotrione
CAS:Fenquinotrione, a 4-hydroxyphenylpyruvate dioxygenase (HPPD) inhibitor, exhibits IC50 values of 27.2 and 44.7 nM against HPPD from rice and Arabidopsis thalianaFormula:C22H17ClN2O5Color and Shape:SolidMolecular weight:424.83Nur77 modulator 2
CAS:Nur77 modulator 2: Kd of 0.35 μM, oral anti-inflammatory, affects Nur77/mitochondria localization.Formula:C26H25NO5Color and Shape:SolidMolecular weight:431.48Anticancer agent 128
CAS:Anticancer agent 128 (compound 1) is an IAP inhibitor that covalently binds to the BIR3 domains of XIAP, cIAP1, and cIAP2, exhibiting IC50 values of 24.9 nM, 19Formula:C26H38N4O4Purity:98%Color and Shape:SolidMolecular weight:470.6Inz-5
CAS:Inz-5 is a fungal-selective inhibitor of mitochondrial cytochrome bc1. Inz-5 impairs fungal virulence. It also prevents the evolution of drug resistance.Formula:C18H14F4N6Color and Shape:SolidMolecular weight:390.34Chroman 1
CAS:Chroman 1 is a potent inhibitor of ROCK1 (IC50 = 52 pM) and ROCK2 (IC50 = 1 pM).Formula:C24H28N4O4Purity:99.67% - 99.84%Color and Shape:SolidMolecular weight:436.5Ref: TM-T14960
1mg77.00€5mg169.00€10mg264.00€25mg454.00€50mg682.00€100mg938.00€1mL*10mM (DMSO)183.00€CDKI-83
CAS:CDKI-83, a potent CDK9 inhibitor, inhibits tumor growth with GI50 <1μM and triggers apoptosis in A2780 cells, showing promise as an anti-cancer agent.Formula:C21H23N7O3S2Color and Shape:SolidMolecular weight:485.585-Iodo-indirubin-3'-monoxime
CAS:5-Iodo-indirubin-3'-monoxime is a potent GSK-3β, CDK5/P25 and CDK1/cyclin B inhibitor, competing with ATP for binding to the catalytic site of the kinase (IC50sFormula:C16H10IN3O2Color and Shape:SolidMolecular weight:403.17TC-5115
CAS:TC-5115 inhibits MLL1 enzyme at 16 nM, promising for treating MLL leukemia.Formula:C23H32N8O5SColor and Shape:SolidMolecular weight:532.62Spr 210
CAS:Spr 210 is an aldose reductase (AR) inhibitor with potential uses as a therapeutic agent for preventing and improving some diabetic complications.Formula:C18H11F3N2O3S2Color and Shape:SolidMolecular weight:424.42GLUT4 activator 1
CAS:GLUT4 activator 1 is a potent glucose transporter type 4 (GLUT4) translocation activator (EC50: 0.14 μM).Formula:C23H21FN4O3SPurity:98%Color and Shape:SolidMolecular weight:452.5TH-Z827
CAS:<p>TH-Z827 is a mutant-selective inhibitor targeting KRAS(G12D) with an IC50 of 2.4 μM, demonstrating specificity by not binding to KRAS(WT) or KRAS(G12C).</p>Formula:C30H38N6OPurity:98%Color and Shape:SolidMolecular weight:498.66Mioflazine hydrochloride
CAS:Mioflazine hydrochloride is a nucleoside transport inhibitor that acts on adenosine to improve sleep.Formula:C29H34Cl4F2N4O3Color and Shape:SolidMolecular weight:666.41ML-099
CAS:ML-099 is a pan Ras-related GTPases activator that activates Rac1, Ras, GTP-binding protein (Rab7), Rab2A and cell division cycle 42.Formula:C14H13NO2SPurity:99.73%Color and Shape:SolidMolecular weight:259.32Ref: TM-T22991
1mg48.00€2mg64.00€5mg96.00€10mg153.00€25mg305.00€50mg487.00€100mg710.00€1mL*10mM (DMSO)94.00€ERX-41
CAS:ERX-41 is an orally active, stereospecific small molecule that targets lysosomal acid lipase A (LIPA).Formula:C38H48N4O9Purity:98%Color and Shape:SolidMolecular weight:704.81CYT296
CAS:CYT296 is a chromatin de-condensation agent that enhances the efficiency of induced pluripotent stem cell (iPSC) generation mediated by defined factors (OSKM)Formula:C18H16O2SPurity:98%Color and Shape:SolidMolecular weight:296.38FGTI-2734
CAS:FGTI-2734, a dual FT/GGT-1 inhibitor (IC50: 250/520 nM), blocks KRAS membrane binding and curbs KRAS-driven pancreatic cancer.Formula:C26H31FN6O2SPurity:99.69%Color and Shape:SolidMolecular weight:510.63Ref: TM-T11282
1mg51.00€5mg119.00€10mg188.00€25mg393.00€50mg587.00€100mg835.00€1mL*10mM (DMSO)136.00€MK-386
CAS:MK-386 is a potent and selective inhibitor of human type-1 5alpha-reductase.Formula:C28H49NOColor and Shape:SolidMolecular weight:415.69ALK/EGFR-IN-1
CAS:ALK/EGFR-IN-1 (Compound 8l) is a dual inhibitor targeting both ALK and EGFR, effectively blocking their phosphorylation.Formula:C27H34ClN7O3SPurity:98%Color and Shape:SolidMolecular weight:572.12KUNG38
CAS:KUNG38 is a purine-based inhibitor of Grp94.Formula:C18H16Cl2N2O5Purity:98%Color and Shape:SolidMolecular weight:411.24SHP2/CDK4-IN-1
CAS:SHP2/CDK4-IN-1: dual inhibitor, oral, potent (IC50: SHP2 4.3 nM, CDK4 18.2 nM), hinders TNBC growth, strong antitumor effects in mice.Formula:C33H35ClF2N10OSColor and Shape:SolidMolecular weight:693.21Nurr1 agonist 8
CAS:Nurr1 agonist 8 is a low-affinity Nurr1 agonist that can be used to study neurological diseases such as Parkinson's.Formula:C14H10Cl2O3Purity:99.79%Color and Shape:SolidMolecular weight:297.13E-5324
CAS:E-5324 is potent cholesterol acyltransferase (ACAT) inhibitor (IC50s: 44 to 190 nM).Formula:C26H34N4O2Purity:98%Color and Shape:SolidMolecular weight:434.57ITK inhibitor
CAS:ITK, a kinase in T/NKT cells & mast cells, regulates TCR pathways. ITK inhibitors treat immune disorders; one is a BMS-509744 analogue.Formula:C31H39N5O4S2Color and Shape:SolidMolecular weight:609.8KRAS G12C inhibitor 28
CAS:KRAS G12C Inhibitor 28 is a compound that effectively inhibits the KRAS G12C mutation, exhibiting potent antitumor effects with an inhibitory concentration (Formula:C33H36F2N5O4PColor and Shape:SolidMolecular weight:635.64T-00127_HEV1
CAS:T-00127_HEV1 is an inhibitor of phosphatidylinositol 4-kinase III beta(PI4KIIIβ, IC50 = 60 nM).Formula:C22H29N5O3Purity:99.89%Color and Shape:SolidMolecular weight:411.5Ref: TM-T16967
1mg56.00€5mg119.00€10mg187.00€25mg375.00€50mg560.00€100mg800.00€500mg1,644.00€1mL*10mM (DMSO)246.00€YM543 free base
CAS:"YM543 is an effective, oral SGLT2 inhibitor that lowers blood glucose, useful for diabetes research."Formula:C23H24O6Color and Shape:SolidMolecular weight:396.43ARTD3/PARP3-IN-1
CAS:ARTD3/PARP3-IN-1 is a non-selective inhibitor targeting diphtheria toxin-like ADP-ribosyltransferase 3 (ARTD3)/PARP3 [1].Formula:C17H16N4O2Color and Shape:SolidMolecular weight:308.33NaPi2b Inhibitor 15
CAS:NaPi2b, key in phosphate balance, is in intestines, lungs, testes. Blocking it may treat hyperphosphatemia by lowering serum phosphate.Formula:C44H58ClF3N4O11SColor and Shape:SolidMolecular weight:943.46DCLK1-IN-2
CAS:DCLK1-IN-2 (Compound I-5) is a potent inhibitor of DCLK1, exhibiting an IC50 of 171.3 nM, and demonstrates significant antiproliferative effects on SW1990 cellFormula:C26H32N8O3SColor and Shape:SolidMolecular weight:536.65Moxestrol
CAS:Moxestrol, a synthetic estrogen, treats menopause and menstrual issues in Europe.Formula:C21H26O3Purity:98%Color and Shape:SolidMolecular weight:326.43SAR-7226 Hydrate
CAS:SAR-7226 Hydrate, a SGLT1/2 inhibitor, is used potentially for the treatment of type 2 diabetes.Formula:C18H22F4N2O7Purity:98%Color and Shape:SolidMolecular weight:454.37Carbidine dihydrochloride
CAS:Carbidine, a gamma-carboline derivative, is an atypical antipsychotic that modulates dopamine release and tyrosine hydroxylase activity.Formula:C13H20Cl2N2Purity:98.59%Color and Shape:SolidMolecular weight:275.217JTT 130
CAS:JTT 130 is an agent of hypolipidemic. It inhibits microsomal triglyceride transfer protein.Formula:C39H37F3N2O8Color and Shape:SolidMolecular weight:718.71Ogremorphin
CAS:Ogremorphin (GPR68-IN-1) is a potent inhibitor of GPR68, exhibiting an EC50 of 170 nM.it is utilized in the study of autoimmune chronic inflammatory diseases [1Formula:C21H17N3OSPurity:99.65% - 99.65%Color and Shape:SolidMolecular weight:359.44Ponicidin
CAS:Ponicidin, a diterpenoid from Rabdosia rubescens, has immunoregulatory, anti-inflammatory, anti-viral, and anti-cancer properties.Formula:C20H26O6Purity:98.98% - 99.92%Color and Shape:SolidMolecular weight:362.42β-Lactamase-IN-8
CAS:β-Lactamase-IN-8 (compound 20) is a potent and oral bioavailable broad-spectrum cyclic boronate β-lactamase inhibitor that can be used for researchingFormula:C10H14BNO4SColor and Shape:SolidMolecular weight:255.1Difluorocyclooctyne-CH2-COOH
CAS:Difluorocyclooctyne-CH2-COOH is a DIFO analogue for live-cell glycan imaging, reacting swiftly with azides sans copper catalysts.Formula:C10H12F2O2Color and Shape:SolidMolecular weight:202.2μ opioid receptor agonist 1
CAS:μ opioid receptor agonist 1 (Compound H-1a) is an optically pure oxyheterocyclic substituted pyrroloxypyrazole derivative and an MOR receptor agonist that canFormula:C26H38N4OColor and Shape:SolidMolecular weight:422.61Duocarmycin DM free base
CAS:Duocarmycin: DNA-binding, alkylating anticancer agent with a curved indole structure, used in ADCs.Formula:C26H26ClN3O3Purity:98%Color and Shape:SolidMolecular weight:463.96CBP/p300-IN-17
CAS:CBP/p300-IN-17 (compound 7) is a potent inhibitor of EP300/CBP HAT, acting on HAT EP300 (IC50: 0.18 μM) and LK2 H3K27 (IC50: 0.69 μM).Formula:C25H28N4O3Color and Shape:SolidMolecular weight:432.51Capeserod HCl
CAS:Capeserod HCl, a 5-hydroxytriptamine 4 (5-HT4) receptor agonist, is used potentially for the treatment of Alzheimer's disease.Formula:C23H26Cl2N4O4Purity:98%Color and Shape:SolidMolecular weight:493.38Tradipitant
CAS:Tradipitant (VLY-686) is an antagonist of neurokinin-1.Formula:C28H16ClF6N5OPurity:99.42%Color and Shape:SolidMolecular weight:587.9Ref: TM-T17156
1mg60.00€2mg85.00€5mg119.00€10mg187.00€25mg329.00€50mg490.00€100mg700.00€1mL*10mM (DMSO)157.00€ST1074
CAS:ST1074, a dual inhibitor of CerS2 and CerS4, promotes apoptosis and is applicable in cancer research [1].Formula:C20H36ClNO3Purity:98%Color and Shape:SolidMolecular weight:373.96WAY-649123
CAS:WAY-649123 is an active molecule that exhibits (in vitro) antagonistic properties against (alpha-1A adrenergic receptors), with a (pKi) of 8.9.Formula:C16H13F2NO3Color and Shape:SolidMolecular weight:305.286-Chloro-7-deazapurine-β-D-riboside
CAS:6-Chloro-7-deazapurine-β-D-riboside shows antifungal activity.Formula:C11H12ClN3O4Purity:98.26%Color and Shape:SolidMolecular weight:285.68Arbemnifosbuvir
CAS:Arbemnifosbuvir, a drug interfering with the nidovirus DdRp-associated nucleotidyltransferase (NiRAN) domain of non-structural protein 12 (nsp12), is utilizedFormula:C24H33FN7O7PPurity:98%Color and Shape:SolidMolecular weight:581.535-HT3-In-1
CAS:5-HT3-In-1 (compound example 8) exhabits with 5-HT3 inhibition activity.Formula:C16H21ClN4O3Purity:98%Color and Shape:SolidMolecular weight:352.82Urease Inhibitor 07
CAS:Urease Inhibitor 07 is an isosubstituted metalloproteinase inhibitor with potential activity against Mycobacterium tuberculosis strain H37Rv.Formula:C7H5N3OSPurity:99.65%Color and Shape:SolidMolecular weight:179.2DHODH-IN-22
CAS:DHODH-IN-22: potent, selective DHODH inhibitor, orally active, IC50: 0.3 nM, for AML research.Formula:C21H21ClF4N6O5Color and Shape:SolidMolecular weight:548.88EPZ011989 HCl(1598383-40-4 Free base)
CAS:EPZ011989 is a highly potent and selective oral EZH2 inhibitor with Ki value <3 nM.Formula:C35H51N5O4·HClColor and Shape:SolidMolecular weight:642.27ATR-IN-13
CAS:ATR-IN-13 is a potent inhibitor of ATR kinases (IC50: 2 nM) and can be used to study ATR kinase-mediated diseases (e.g. proliferative diseases, cancer).Formula:C24H24FN9OColor and Shape:SolidMolecular weight:473.51CJ-42794
CAS:CJ-42794 (CJ-042794) is a selective antagonist of prostaglandin E receptor subtype 4 (EP4).Formula:C22H17ClFNO4Purity:99.92%Color and Shape:SolidMolecular weight:413.83KD-3010
CAS:KD-3010 (Kalypsys) is an orally active potent and selective PPARδ agonist for the study of liver injury.Formula:C30H33F3N2O8S2Purity:99.61%Color and Shape:SolidMolecular weight:670.72VULM 1457
CAS:VULM 1457 is a potent ACAT inhibitor.Formula:C25H27N3O3SPurity:99.73%Color and Shape:SolidMolecular weight:449.57ALS-8112
CAS:ALS-8112 is a inhibitor of respiratory syncytial virus (RSV) polymerase. The 5'-triphosphate form of ALS-8112 inhibits RSV polymerase (IC50: 0.02 μM).Formula:C10H13ClFN3O4Purity:98.90%Color and Shape:SolidMolecular weight:293.68Bromochloromethotrexate
CAS:Bromochloromethotrexate is a bioactive chemical.Formula:C20H20BrClN8O5Color and Shape:SolidMolecular weight:567.78GLX481304
CAS:GLX481304 is a selective Nox-2 and Nox-4 inhibitor, exhibiting IC50 values of 1.25 μM.Formula:C23H29N7OColor and Shape:SolidMolecular weight:419.52Androgen receptor degrader-3
CAS:Androgen Receptor Degrader-3 (ARD-3) is a compound that inhibits androgen receptor signaling and promotes the degradation of the receptor, with potentialFormula:C45H51ClN8O5Purity:98%Color and Shape:SolidMolecular weight:819.39FR-217840
CAS:FR-217840: Potential anti-rheumatic drug; inhibits matrix metalloproteinases, halts joint damage.Formula:C16H18FN3O6S3Color and Shape:SolidMolecular weight:463.52T521
CAS:T521 is a selective inhibitor of the PBD of Plk1 and shows no inhibitory effect on Plk2 and Plk3.Formula:C17H14FNO5S2Purity:99.71%Color and Shape:SolidMolecular weight:395.43JG-2016
CAS:JG-2016, as a histone acetyltransferase 1 inhibitor, inhibits growth of human cancer cell lines and inhibits enzymatic activity in cellulose.Formula:C18H21ClN4O3Purity:99.00% - 99.37%Color and Shape:SolidMolecular weight:376.84Ref: TM-T82008
1mg116.00€5mg283.00€10mg455.00€25mg905.00€50mg1,454.00€100mg1,882.00€1mL*10mM (DMSO)310.00€CCT-271850
CAS:CCT-271850 is an inhibitor of the spindle checkpoint function of Monospindle 1.Formula:C24H29N7OPurity:98%Color and Shape:SolidMolecular weight:431.53Arginase inhibitor 1
CAS:Arginase inhibitor 1 is a potent inhibitor of human arginases I and II (IC50s: 223 and 509 nM).Formula:C13H27BN2O4Color and Shape:SolidMolecular weight:286.18meplazumab
CAS:<p>meplazumab is a humanized anti-CD147 antibody, as add-on therapy in patients with COVID-19 pneumonia.</p>Purity:98%Color and Shape:LiquidMolecular weight:N/APBR28
CAS:PBR28, a TSPO modulator, holds potential for preventative research in Pulmonary Arterial Hypertension (PAH) and is instrumental in brain positron emissionFormula:C21H20N2O3Purity:98%Color and Shape:SolidMolecular weight:348.4Calmidazolium chloride
CAS:Calmidazolium chloride blocks calmodulin, hinders phosphodiesterase (IC50=0.15µM), Ca2+-ATPase (IC50=0.35µM), and can induce cancer cell apoptosis.Formula:C31H23Cl7N2OPurity:98.53%Color and Shape:SolidMolecular weight:687.7Ref: TM-T10667
5mg63.00€10mg87.00€25mg145.00€50mg215.00€100mg320.00€200mg467.00€1mL*10mM (DMSO)95.00€Ianthelliformisamine B TFA
CAS:Ianthelliformisamine B TFA, an antibiotic enhancer, is used to against resistant Gram-negative bacteria.Formula:C21H27Br2F6N3O6Purity:98%Color and Shape:SolidMolecular weight:691.25(3β,20E)-24-Norchola-5,20(22)-diene-3,23-diol
CAS:(3β,20E)-24-Norchola-5,20(22)-diene-3,23-diol is a steroid-based allylic alcohol.Formula:C23H36O2Purity:98%Color and Shape:SolidMolecular weight:344.53LY52
CAS:LY52 is a matrix metalloproteinase-2 inhibitor. It acts by suppressing tumor invasion and metastasis.Formula:C22H24N4O6Purity:98%Color and Shape:SolidMolecular weight:440.45L 670630
CAS:L 670630 is a potent and orally active 5-lipoxygenase inhibitor.Formula:C25H26O3Purity:98%Color and Shape:SolidMolecular weight:374.47cis-9,10-Epoxystearic acid
CAS:cis-9,10-Epoxystearic acid (cis-9,10-Epoxyoctadecanoic acid) is an endogenous component in human urine and blood and can be produced from oleic acid by enzymicFormula:C18H34O3Purity:99.93%Color and Shape:SolidMolecular weight:298.46Unguisin A
CAS:Unguisin A is a cyclic peptide isolated from the marine-derived fungus Emericella unguis [1].Formula:C40H54N8O7Color and Shape:SolidMolecular weight:758.91HDAC-IN-53
CAS:HDAC-IN-53 inhibits HDAC1-3 with IC50s: 47, 125, 450 nM. Inactive on class II HDACs; triggers apoptosis; reduces tumor growth in mice.Formula:C23H20ClN7O2Purity:98%Color and Shape:SolidMolecular weight:461.9Gly-β-MCA
CAS:Gly-β-MCA is an orally bioactive, entero inhibitor of the farnesoid X receptor (FXR), a bile acid, used in the study of obesity and diabetes.Formula:C26H43NO6Purity:≥98.0%Color and Shape:SolidMolecular weight:465.62ELND007
CAS:ELND007 is a Gamma secretase inhibitor.Formula:C19H14F4N4O2SColor and Shape:SolidMolecular weight:438.46,9,12,15-Hexadecatetraenoic acid-ethyl ester
CAS:6,9,12,15-Hexadecatetraenoic acid-ethyl ester, an n-1PUFA, demonstrates oral activity and has been shown to lower plasma triglyceride levels in mice whenFormula:C18H28O2Color and Shape:SolidMolecular weight:276.41STING-IN-7
CAS:<p>STING-IN-7 (compound 21) serves as a potent inhibitor of the stimulator of interferon genes (STING) pathway, demonstrating an inhibitory concentration (IC50) of</p>Formula:C16H14ClN3OPurity:98%Color and Shape:SolidMolecular weight:299.76LEQ-506 HCl (1204975-42-7 free base)
LEQ506 is an orally bioavailable small-molecule Smoothened antagonist. It also has a potential antineoplastic activity.Formula:C27H31Cl2N5OPurity:98%Color and Shape:SolidMolecular weight:512.48ERK Inhibitor II (Negative control)
CAS:ERK Inhibitor II, a control, blocks ERK and insulin receptor activation, aiding diabetes research.Formula:C18H12N6OColor and Shape:SolidMolecular weight:328.33UniPR505
CAS:<p>UniPR505 is a potent EphA2 antagonist (IC50: 0.95 µM), a novel 3α-carbamoyloxy derivative with antiangiogenic properties.</p>Formula:C39H57N3O5Purity:98.23%Color and Shape:SolidMolecular weight:647.89Antiviral agent 35
CAS:<p>Antiviral agent 35 (compound 4d) serves as a potent orally active inhibitor of the influenza virus, targeting early stages of viral replication.</p>Formula:C23H18N2O4SPurity:98%Color and Shape:SolidMolecular weight:418.47Antimalarial agent 10
CAS:Compound 17b, an amino alcohol-quinoline, targets Pf3D7 (IC50: 14.9 nM) and PfW2 (IC50: 11 nM) with selectivity index >770.Formula:C23H22F6N2O2Color and Shape:SolidMolecular weight:472.42dBRD4-BD1
CAS:dBRD4-BD1 selectively inhibits and degrades BRD4 (DC50=280nM), upregulates BRD2/3, and aids in creating BRD4-specific probes.Formula:C50H53F3N8O9Color and Shape:SolidMolecular weight:967KDM2A/7A-IN-1
CAS:KDM2A/7A-IN-1 is a KDM2A/7A inhibitor with potential anti-tumour activity for the study of duodenal adenomas and ossifying fibromucoid tumours.Formula:C33H38N4OPurity:99.59%Color and Shape:SolidMolecular weight:506.68SG3-179
CAS:SG3-179 is a BET inhibitor.Formula:C28H35ClFN7O3SColor and Shape:SolidMolecular weight:604.145'-ODMT cEt N-Bzm5 C Phosphoramidite (Amidite)
CAS:5'-ODMT cEt N-Bzm5 C Phosphoramidite is a strong modified nucleic acid analog for antisense oligos.Formula:C49H56N5O9PColor and Shape:SolidMolecular weight:889.972-Methoxyestrone
CAS:2-Methoxyestrone is a methoxylated catechol estrogen and the principal metabolite of 2-hydroxyestrone, a nonuterotropic metabolite of estradiol.Formula:C19H24O3Purity:97.07% - 99.18%Color and Shape:SolidMolecular weight:300.39Ref: TM-T13481
1mg49.00€5mg97.00€10mg160.00€25mg283.00€50mg418.00€100mg615.00€200mg879.00€1mL*10mM (DMSO)106.00€Taragarestrant
CAS:Taragarestrant (D-0502), an oral estrogen receptor degrader, combats ER+ breast cancer in research.Formula:C25H25Cl2FN2O2Color and Shape:SolidMolecular weight:475.38MP7
CAS:MP7 (PDK1 inhibitor) is a inhibitor of phosphoinositide-dependent kinase-1 (PDK1).Formula:C28H22F2N4O4Purity:99.89%Color and Shape:SolidMolecular weight:516.5RSV L-protein-IN-5
CAS:RSV L-protein-IN-5 (Compound E) serves as a potent inhibitor of the Respiratory Syncytial Virus (RSV), with an EC50 value of 0.1 μM.Formula:C31H36N6O4Purity:98%Color and Shape:SolidMolecular weight:556.66USP7-IN-12
CAS:USP7-IN-12 (compound 1) is a potent, orally active inhibitor of Usp7, exhibiting an IC50 of 3.67 nM and demonstrating antiproliferative activity [1].Formula:C29H28ClFN4O2SColor and Shape:SolidMolecular weight:551.07Esterbut-6
CAS:Esterbut-6 is a potent tumor cell proliferation inhibitor in vivo by stabilizes butyric acid.Formula:C13H22O7Purity:98%Color and Shape:SolidMolecular weight:290.31Quizalofop
CAS:Quizalofop (Xylafop) is a reagent of biochemical.Formula:C17H13ClN2O4Purity:97.14%Color and Shape:SolidMolecular weight:344.75Ref: TM-T19959
5mg55.00€10mg77.00€25mg111.00€50mg164.00€100mg235.00€500mg588.00€1mL*10mM (DMSO)69.00€Dibutepinephrine
CAS:Dibutylephrine is a sympathomimetic agent.Formula:C17H25NO5Color and Shape:SolidMolecular weight:323.38ONO-0740556
CAS:ONO-0740556 is a potent agonist of the Gi-coupled human lysophosphatidic acid receptor 1 (LPA1), exhibiting an EC50 value of 0.26 nM.Formula:C20H34NO6PColor and Shape:SolidMolecular weight:415.46(+)-Apogossypol
CAS:(+)-Apogossypol is an antagonist of pan-BCL-2. (+)-Apogossypol binds to Mcl-1(Bcl-2 and Bcl-xL with EC50s of 2.6, 2.8 and 3.69 μM, respectively).Formula:C28H30O6Purity:98%Color and Shape:SolidMolecular weight:462.53Abiraterone sulfate N-oxide
CAS:Abiraterone sulfate N-oxide, a carboxylic acid and major metabolite of Abiraterone, is utilized in prostate cancer research [1] [2].Formula:C24H31NO5SColor and Shape:SolidMolecular weight:445.57AMPA receptor modulator-2
CAS:<p>AMPA receptor modulator-2 is a modulator of AMPA receptor. The pIC50 value for TARPγ2 dependent AMPA receptor is 10.1.</p>Formula:C15H6F6N4OSPurity:99.8%Color and Shape:SolidMolecular weight:404.29Antitumor agent-49
CAS:Antitumor agent-49 (Compound 10), a harmine derivative-furoxan hybrid featuring nitric oxide (NO) donating properties, exhibits cytotoxic effects against HepG2Formula:C42H41BrN4O8SColor and Shape:SolidMolecular weight:841.77
