Metabolismo
Os inibidores do metabolismo são compostos que interferem nas vias metabólicas, alterando a produção e utilização de energia dentro das células. Esses inibidores são usados para estudar a regulação do metabolismo, o papel das vias metabólicas em doenças como o câncer e o diabetes, e para desenvolver novas estratégias terapêuticas. Os inibidores do metabolismo podem direcionar várias enzimas e processos envolvidos na glicólise, na oxidação de ácidos graxos e em outras funções metabólicas. Na CymitQuimica, oferecemos uma ampla gama de inibidores do metabolismo de alta qualidade para apoiar sua pesquisa em bioquímica, distúrbios metabólicos e desenvolvimento de medicamentos.
Subcategorias de "Metabolismo"
- AhR(41 produtos)
- Aminopeptidase(67 produtos)
- CETP(18 produtos)
- Anidrase carbónica(178 produtos)
- Caseína quinase(130 produtos)
- DHFR(33 produtos)
- Descarboxilase(4 produtos)
- Desidrogenase(271 produtos)
- FAAH(64 produtos)
- FXR(58 produtos)
- Factor Xa(80 produtos)
- Sintase de Ácidos graxos(33 produtos)
- Ferroptose(215 produtos)
- GR(3 produtos)
- GSNOR(3 produtos)
- Glucoquinase(54 produtos)
- HIF/HIF Prolil-Hidroxilase(142 produtos)
- HMG-CoA Reductase(33 produtos)
- Hidroxilase(30 produtos)
- IDO(82 produtos)
- LDL(8 produtos)
- Lipase(98 produtos)
- Lipídio(58 produtos)
- Lipoxigenase(124 produtos)
- MAO(87 produtos)
- MPO(2 produtos)
- NAMPT(36 produtos)
- P450(6 produtos)
- PAI-1(25 produtos)
- PDE(166 produtos)
- PED(1 produtos)
- PKM(15 produtos)
- PPAR(164 produtos)
- Fosfolipase(82 produtos)
- ROR(42 produtos)
- Receptor de Retinóide(29 produtos)
- SGK(11 produtos)
- Tiorredoxina(12 produtos)
- Transferase(30 produtos)
- Tansportador(42 produtos)
- UGT(4 produtos)
- Inibidores de Xantina Oxidase (XO)(9 produtos)
Exibir 34 mais subcategorias
Foram encontrados 8626 produtos de "Metabolismo"
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CP-91149
CAS:<p>CP-91149 is a selective glycogen phosphorylase (GP) inhibitor with IC50 of 0.13 μM in the presence of glucose, 5- to 10-fold less potent in the absence of</p>Fórmula:C21H22ClN3O3Pureza:99.66% - 99.81%Cor e Forma:SolidPeso molecular:399.87Haloxyfop
CAS:<p>(±)-Haloxyfop (Haloxyfop Acid) is a herbicide.</p>Fórmula:C15H11ClF3NO4Pureza:99.94% - >99.99%Cor e Forma:SolidPeso molecular:361.7Tebuconazole
CAS:<p>Tebuconazole: azole fungicide, inhibits CYP51 with IC50s 0.9 μM (C. albicans) and 1.3 μM (human).</p>Fórmula:C16H22ClN3OPureza:99.21%Cor e Forma:SolidPeso molecular:307.82NFAT Inhibitor-2
CAS:<p>NFAT Inhibitor-2 is a compound used as a molecular building block.</p>Fórmula:C22H20F2N2O4SPureza:97.37%Cor e Forma:SolidPeso molecular:446.47Trandolapril
CAS:<p>Trandolapril is an orally administered angiotensin converting enzyme (ACE) inhibitor that is hydrolysed to the active diacid trandolaprilat.</p>Fórmula:C24H34N2O5Pureza:99.70% - 99.83%Cor e Forma:White PowderPeso molecular:430.54L-Alanine
CAS:<p>L-Alanine (L-2-Aminopropionic acid) is an Amino Acid. Alanine is involved in the metabolism of tryptophan and vitamin pyridoxine.</p>Fórmula:C3H7NO2Pureza:99.83%Cor e Forma:Orthorhombic Crystals From Water SolidPeso molecular:89.09Fosfructose
CAS:<p>D-fructose-1,6-diphosphate (D-fructose-1,6-diphosphate), also known as Fosfructose, is a cytoprotective natural sugar phosphate.</p>Fórmula:C6H14O12P2Pureza:99.84%Cor e Forma:SolidPeso molecular:340.12GW1929
CAS:<p>GW1929 is a potent PPAR-γ agonist (pKi: 8.84 for human PPAR-γ; pEC50s of 8.56 and 8.27 for human and murine PPAR-γ).</p>Fórmula:C30H29N3O4Pureza:98.1% - 98.21%Cor e Forma:SolidPeso molecular:495.57CM10
CAS:<p>CM10 is an aldehyde dehydrogenase 1A family(ALDH1A) inhibitor.</p>Fórmula:C20H23N3OPureza:99.84%Cor e Forma:SolidPeso molecular:321.42Aranidipine
CAS:<p>Aranidipine (MPC1304) (MPC1304) is a calcium channel antagonist with potent and long-lasting antihypertensive effects.</p>Fórmula:C19H20N2O7Pureza:99.15%Cor e Forma:SolidPeso molecular:388.37AZD7545
CAS:<p>AZD7545 is a potent PDHK inhibitor.</p>Fórmula:C19H18ClF3N2O5SPureza:99.12% - 99.96%Cor e Forma:SolidPeso molecular:478.87NCT-501
CAS:<p>NCT-501 is a potent and selective inhibitor of Aldehyde Dehydrogenase 1A1 (ALDH1A1) with IC50 of 40 nM.</p>Fórmula:C21H32N6O3Pureza:99.19%Cor e Forma:SolidPeso molecular:416.522,4-Diamino-6-hydroxypyrimidine
CAS:<p>2,4-Diamino-6-hydroxypyrimidine (DAHP) (DAHP) is a selective, specific inhibitor of GTP cyclohydrolase I, the rate limiting step for de novo pterin synthesis</p>Fórmula:C4H6N4OPureza:99.82%Cor e Forma:White Solid CrystalsPeso molecular:126.12Tetradecylthioacetic acid
CAS:<p>Synthetic fatty acid TTA has β-sulfur, resists β-oxidation, and activates PPARs, especially PPARα.</p>Fórmula:C16H32O2SPureza:99.93%Cor e Forma:SolidPeso molecular:288.49FOY 251
CAS:<p>FOY 251 is a proteinase inhibitor, and is an anti-proteolytic active metabolite camostate.</p>Fórmula:C17H19N3O7SPureza:97.11% - 99.33%Cor e Forma:SolidPeso molecular:409.41Rosiptor
CAS:<p>Rosiptor (AQX-1125) (AQX-1125) is an orally-active and specific phosphatase SHIP1 activator with anti-inflammatory effects.</p>Fórmula:C20H35NO2Pureza:99.53% - 99.73%Cor e Forma:SolidPeso molecular:321.5HA 155
CAS:<p>HA 155 (Autotaxin Inhibitor IV) is a boronic acid-based compound, inhibiting ATX with IC50 of 5.7 nM by selectively binding to its catalytic threonine.</p>Fórmula:C24H19BFNO5SPureza:99.88%Cor e Forma:SolidPeso molecular:463.29CAY 10465
CAS:<p>CAY 10465 is a selective and high-affinity AhR agonist, with a Ki of 0.2 nM, and shows no effect on estrogen receptor (Ki >100000 nM).</p>Fórmula:C15H9Cl2F3Pureza:98.80%Cor e Forma:SolidPeso molecular:317.13KML29
CAS:<p>KML29 is highly selective and effective monoacylglycerol lipase (MAGL) inhibitor.</p>Fórmula:C24H21F6NO7Pureza:98.65%Cor e Forma:SolidPeso molecular:549.42Minaprine dihydrochloride
CAS:<p>Minaprine dihydrochloride: reversible MAO-A inhibitor, mild on acetylcholinesterase, used for depression.</p>Fórmula:C17H24Cl2N4OPureza:99.43% - 99.99%Cor e Forma:SolidPeso molecular:371.3JNJ-42165279
CAS:<p>JNJ-42165279 selectively inactivates FAAH without notably affecting other enzymes, ion channels, receptors, or CYPs/hERG at 10 μM.</p>Fórmula:C18H17ClF2N4O3Pureza:99.67% - 99.88%Cor e Forma:SolidPeso molecular:410.8Nequinate
CAS:<p>Nequinate is an anticoccidial agent, preventing coccidiosis .</p>Fórmula:C22H23NO4Pureza:96.43%Cor e Forma:Light Yellow Odorless PowderPeso molecular:365.42CDN1163
CAS:<p>CDN1163 is a small molecule activator of sarco/endoplasmic reticulum Ca2+-ATPase (SERCA).</p>Fórmula:C20H20N2O2Pureza:99.83% - ≥95%Cor e Forma:SolidPeso molecular:320.39GSK0660
CAS:<p>GSK0660 is an antagonist and inverse agonist of PPARβ/δ.</p>Fórmula:C19H18N2O5S2Pureza:99.26% - ≥95%Cor e Forma:SolidPeso molecular:418.49Eprobemide
CAS:<p>Eprobemide (LIS 630) is a non-competitive reversible inhibitor of monoamine oxidase A (MAO-A).</p>Fórmula:C14H19ClN2O2Pureza:99.83%Cor e Forma:SolidPeso molecular:282.774-Nonylphenylboronic acid
CAS:<p>4-Nonylphenylboronic acid is a inhibitor of FAAH.</p>Fórmula:C15H25BO2Pureza:97.63%Cor e Forma:SolidPeso molecular:248.17BMS-779788
CAS:<p>BMS-779788 (XL-652) is an LXRα/β partial agonist (IC50: 68/14 nM).</p>Fórmula:C28H29ClN2O3SPureza:98.65% - 99.24%Cor e Forma:SolidPeso molecular:509.064-Amino-6-(trifluoromethyl)benzene-1,3-disulfonamide
CAS:<p>4-Amino-6-(trifluoromethyl)benzene-1,3-disulfonamide (4-Amino-6-(trifluoromethyl)benzene-1,3-d) is a carbonic anhydrase inhibitor, used as a potential anti-</p>Fórmula:C7H8F3N3O4S2Pureza:98.58%Cor e Forma:SolidPeso molecular:319.28Bepridil hydrochloride
CAS:<p>Bepridil hydrochloride (CERM 1978) is a calcium channel blocker and also inhibits Na+/Ca2+ exchange (NCX), sodium channels and cardiac sarcolemmal KATP channels</p>Fórmula:C24H35ClN2OPureza:99.45% - 99.68%Cor e Forma:SolidPeso molecular:403WIN 18446
CAS:<p>inhibitor of aldehyde dehydrogenase 1a2 (ALDH1a2)</p>Fórmula:C12H20Cl4N2O2Pureza:99.69%Cor e Forma:SolidPeso molecular:366.11Barnidipine hydrochloride
CAS:<p>Barnidipine HCl is a potent dihydropyridine Ca²⁺ blocker with 0.35 nM IC50 in pig coronary artery.</p>Fórmula:C27H30ClN3O6Pureza:99.88%Cor e Forma:SolidPeso molecular:528Milacemide
CAS:<p>Milacemide is a glycine prodrug and MAO-B inhibitor.</p>Fórmula:C7H16N2OPureza:98.04%Cor e Forma:SolidPeso molecular:144.21PF-9601N
CAS:<p>PF-9601N: potent, selective MAO-BI with neuroprotection in PD models.</p>Fórmula:C19H18N2OPureza:98.29%Cor e Forma:SolidPeso molecular:290.36Mitochondrial fusion promoter M1
CAS:<p>Mitochondrial fusion promoter M1, a modulator of mitochondrial dynamics, enhances mitochondrial function and cellular respiration, and has shown efficacy in</p>Fórmula:C14H10Cl4N2OPureza:99.54% - 99.54%Cor e Forma:SolidPeso molecular:364.05Oroxylin A
CAS:<p>Oroxylin A fights tumors, aids RAS therapy, promotes CaCo-2 cell apoptosis, blocks MCF-7 cell invasion and enhances leukemia treatment.</p>Fórmula:C16H12O5Pureza:98.72% - 99.55%Cor e Forma:SolidPeso molecular:284.26S29434
CAS:<p>S29434 (NMDPEF) is a potent, competitiveinhibitor of quinone reductase 2 (QR2;IC50:5-16nM).</p>Fórmula:C21H18N4O3Pureza:99.92%Cor e Forma:SolidPeso molecular:374.39Tryptophan, N-indol-3-ylacetyl- (6CI)
CAS:<p>Tryptophan, N-indol-3-ylacetyl- (6CI) (Indole-3-acetyl-L-tryptophan) is involved in regulatory mechanisms for the control of auxin activity during physiological</p>Fórmula:C21H19N3O3Pureza:99.55%Cor e Forma:SolidPeso molecular:361.4KY-226
CAS:<p>KY-226 is a potent inhibitor of protein tyrosine phosphatase 1B (PTP1B)(IC50: 0.25 μM,)</p>Fórmula:C27H31NO3S2Pureza:99.4%Cor e Forma:SolidPeso molecular:481.67trans-AUCB
CAS:<p>trans-AUCB (t-AUCB) is an effective and selective soluble epoxide hydrolase inhibitor (IC50s: 1.3 nM, 8 nM, 8 nM for hsEH, mouse sEH and rat sEH, respectively).</p>Fórmula:C24H32N2O4Pureza:99.27% - 99.66%Cor e Forma:SolidPeso molecular:412.52TMS
CAS:<p>TMS (2,3',4,5'-Tetramethoxystilbene) is a very selective and potent competitive inhibitor of P450 1B1 (CYP1A1).</p>Fórmula:C18H20O4Pureza:99.17% - 99.73%Cor e Forma:SolidPeso molecular:300.35Calcitriol
CAS:<p>Calcitriol (1,25-Dihydroxyvitamin D3) is a metabolite of vitamin D and a vitamin D receptor (VDR) agonist (IC50=0.4 nM).</p>Fórmula:C27H44O3Pureza:98.81% - 99.64%Cor e Forma:Colorless Crystalline Solid SolidPeso molecular:416.64(R)-GNE-140
CAS:<p>(R)-GNE-140 (GNE-140) is an effective LDHA/LDHB inhibitor (IC50s: 3/5 nM) and is 18-fold more potent than S enantiomer.</p>Fórmula:C25H23ClN2O3S2Pureza:98.25% - 98.91%Cor e Forma:SolidPeso molecular:499.04Firsocostat
CAS:<p>Firsocostat (GS-0976) is an inhibitor of acetyl-CoA carboxylase (ACC) dimerization that inhibits human ACC1 and ACC2 activity (IC50s of 2.1 and 6.1 nM).</p>Fórmula:C28H31N3O8SPureza:98% - 98.46%Cor e Forma:SolidPeso molecular:569.63AG-120 (racemic)
CAS:<p>AG-120 (racemic) is an oral IDH1 inhibitor with potential anti-cancer effects.</p>Fórmula:C28H22ClF3N6O3Pureza:99.56%Cor e Forma:SolidPeso molecular:582.961-Naphthaleneacetic acid potassium salt
CAS:<p>1-Naphthaleneacetic acid potassium salt (1-NAA Potassium Salt) is a synthetic phytogrowth hormone that promotes plant growth and a PLA2 inhibitor.</p>Fórmula:C12H9O2·KPureza:97.68%Cor e Forma:Off-White To Beige PowderPeso molecular:224.3Amifostine trihydrate
CAS:<p>Amifostine trihydrate (WR2721) is the first approved radioprotective drug, used to decrease the risk of kidney problems caused by treatment with cisplatin.</p>Fórmula:C5H15N2O3PS·3H2OPureza:99.71% - 99.80%Cor e Forma:SolidPeso molecular:268.27Cedirogant
CAS:<p>Cedirogant (ABBV-157) is an orally active retinoid-related orphan receptor-γt(RORγt) inverse agonist that is used for psoriasis study.</p>Fórmula:C24H20Cl3F3N2O3Pureza:99.20%Cor e Forma:SolidPeso molecular:547.78CAY10650
CAS:<p>CAY10650 is an effective inhibitor of cytosolic phospholipase A2α (cPLA2α, IC50: 12 nM).</p>Fórmula:C28H25NO6Pureza:97.33%Cor e Forma:SolidPeso molecular:471.5Enterostatin, human, mouse, rat acetate
<p>Enterostatin, human, mouse, rat acetate is a pentapeptide mainly formed in the intestine by the cleavage of secreted pancreatic procolipase.</p>Fórmula:C23H40N8O8Pureza:99.91%Cor e Forma:SolidPeso molecular:556.61TPPU
CAS:<p>TPPU is a potent inhibitor of both human and mouse sEH (IC50 of 3.7 and 2.8 nM, respectively)</p>Fórmula:C16H20F3N3O3Pureza:97.82%Cor e Forma:SolidPeso molecular:359.344-Chlorophenylurea
CAS:<p>4-Chlorophenylurea (NSC-12971) is a novel orally bioavailable inhibitor of factor Xa.</p>Fórmula:C7H7ClN2OPureza:98.87%Cor e Forma:White Granular / PrillPeso molecular:170.6Olesoxime
CAS:<p>Olesoxime (TRO 19622) (TRO19622), A Mitochondrial-Targeted Neuroprotective Compound,is an experimental neuroprotective drug.</p>Fórmula:C27H45NOPureza:99.86%Cor e Forma:SolidPeso molecular:399.65ZSET1446
CAS:<p>ZSET1446 (ST-101) is a T-type calcium channel activator potentially for the treatment of learning deficits in various types of Alzheimer disease (AD) models.</p>Fórmula:C15H12N2OPureza:99.32%Cor e Forma:SolidPeso molecular:236.27Vardenafil hydrochloride
CAS:<p>Vardenafil hydrochloride is a New Phosphodiesterase Type 5(PDE5) Inhibitor, in the Treatment of Erectile Dysfunction in Men With Diabetes</p>Fórmula:C23H33ClN6O4SPureza:99.76% - 99.86%Cor e Forma:White To Off-White Cyrstalline SolidPeso molecular:525.06CAY10698
CAS:<p>CAY10698 is a 12-lipoxygenase inhibitor (12-LO; IC50 of 5.1 μM).</p>Fórmula:C17H17N3O4S2Pureza:98.97%Cor e Forma:SolidPeso molecular:391.46BCI-215
CAS:<p>BCI-215 causes selective cancer cell cytotoxicity in part through non-redox-mediated activation of MAPK signaling</p>Fórmula:C22H22BrNOPureza:99.812%Cor e Forma:SolidPeso molecular:396.32GAK inhibitor 49
CAS:<p>GAK inhibitor 49 is a highly selective and ATP-competitive cyclin G associated kinase (GAK) inhibitor (IC50: 56 nM; Ki: 0.54 nM ).</p>Fórmula:C20H22N2O5Pureza:98.71%Cor e Forma:SolidPeso molecular:370.4Cinacalcet metabolite M4
CAS:<p>Cinacalcet metabolite M4 (Rarechem AL BW 1078) is a metabolite of Cinacalcet. Cinacalcet is an allosteric agonist of Ca receptor.</p>Fórmula:C10H12F3NPureza:97.13%Cor e Forma:SolidPeso molecular:203.2Gabapentin hydrochloride
CAS:<p>Gabapentin hydrochloride (Neurontin HCl) is a GABA analogue, used to treat seizures and neuropathic pain.</p>Fórmula:C9H17NO2·HClPureza:99.71%Cor e Forma:Off-White SolidPeso molecular:207.73-Amino-2-oxazolidinone
CAS:<p>3-Amino-2-oxazolidinone (AOZ) is the metabolite of Furazolidone. It is always be detected as a indicator of furazolidone residues in vivo.</p>Fórmula:C3H6N2O2Pureza:97.82%Cor e Forma:SolidPeso molecular:102.09Uridine 5′-triphosphate tris salt
CAS:<p>Uridine 5′-triphosphate tris salt (Uridine 5'-triphosphoric acid) is an agonist to the P2Y receptor and has been used to study concentrations of intracellular</p>Fórmula:C21H48N5O24P3Pureza:99.04% - 99.94%Cor e Forma:SolidPeso molecular:847.55Propiverine hydrochloride
CAS:<p>Propiverine is a widely used antimuscarinic drug with a mixed mode of action in the treatment of symptoms associated with overactive bladder (OAB).</p>Fórmula:C23H30ClNO3Pureza:99.93%Cor e Forma:White Crystalling PowerPeso molecular:403.94(Rac)-Brassinazole
CAS:<p>(Rac)-Brassinazole is a phytohormone with essential roles in plant growth and development, including the promotion of stem elongation and cell division.</p>Fórmula:C18H18ClN3OPureza:99.74% - 99.81%Cor e Forma:SolidPeso molecular:327.81Tetrindole mesylate
CAS:<p>Tetrindole mesylate is a MAO-A inhibitor.</p>Fórmula:C21H30N2O3SPureza:99.73%Cor e Forma:SolidPeso molecular:390.54TTA-A2
CAS:<p>TTA-A2: T-type calcium channel blocker; anticonvulsant targeting Cav3.1, Cav3.2; IC50 of 89/92 nM; potential for treating neurological conditions.</p>Fórmula:C20H21F3N2O2Pureza:99.5% - 99.9%Cor e Forma:SolidPeso molecular:378.39NDI-091143
CAS:<p>NDI-091143 is a potent and high-affinity human ATP-citrate lyase (ACLY) inhibitor with an IC50 of 2.1 nM (ADP-Glo assay),indirectly disrupting citrate binding</p>Fórmula:C20H14ClF2NO5SPureza:97.03% - ≥95%Cor e Forma:SolidPeso molecular:453.84Amino Tadalafil
CAS:<p>Amino tadalafil is a potent phosphodiesterase 5 (PDE5) inhibitor.</p>Fórmula:C21H18N4O4Pureza:99.85%Cor e Forma:White PowderPeso molecular:390.39Fatostatin
CAS:<p>Fatostatin inhibits SREBP-1/2 by binding to SCAP, blocking their ER-Golgi transport.</p>Fórmula:C18H18N2SPureza:99.92%Cor e Forma:SolidPeso molecular:294.41Tienilic Acid
CAS:<p>Tienilic Acid is a uricosuric diuretic with certain hepatotoxicity</p>Fórmula:C13H8Cl2O4SPureza:99.55%Cor e Forma:SolidPeso molecular:331.17Bocidelpar
CAS:<p>Bocidelpar is a modulator of PPARδ with an EC50 of 7.80 nM and improves mitochondrial biogenesis and function in Duchenne Muscular Dystrophy muscle cells.</p>Fórmula:C25H27F3N2O3Pureza:97.77%Cor e Forma:SolidPeso molecular:460.49BMS-986242
CAS:<p>BMS-986242 is an orally active, potent and selective inhibitor of indoleamine-2,3-dioxygenase 1 (IDO1), and it can be used for the research of cancer.</p>Fórmula:C24H24ClFN2OPureza:98.9%Cor e Forma:SolidPeso molecular:410.91SPI-112
CAS:<p>SPI-112, the SPI-112 methyl ester analog, can inhibit cellular Shp2 PTP activity.</p>Fórmula:C22H17FN4O5SPureza:97.51% - >99.99%Cor e Forma:SolidPeso molecular:468.46PF-3845
CAS:<p>PF-3845 is a potent, selective and irreversible FAAH inhibitor with Ki of 230 nM, showing negligible activity against FAAH2.</p>Fórmula:C24H23F3N4O2Pureza:99.54% - 99.58%Cor e Forma:SolidPeso molecular:456.46IDO-IN-7
CAS:<p>IDO-IN-7 (NLG-919 analogue) is a potent IDO (indoleamine-(2, 3)-dioxygenase) pathway inhibitor.</p>Fórmula:C18H22N2OPureza:99.32% - 99.9%Cor e Forma:SolidPeso molecular:282.38Dimethylfraxetin
CAS:<p>Dimethylfraxetin (6,7,8-Trimethoxycoumarin) is a Carbonic anhydrase inhibitor(Ki：0.0097 μM)</p>Fórmula:C12H12O5Pureza:99.96% - ≥95%Cor e Forma:SolidPeso molecular:236.22Pyributicarb
CAS:<p>Pyributicarb (TSH-888) is a potent activator of both CYP3A4 gene and human pregnane X receptor (hPXR).</p>Fórmula:C18H22N2O2SPureza:99.702% - ≥95%Cor e Forma:SolidPeso molecular:330.44IACS-13909
CAS:<p>IACS-13909 (BBP-398), a specific and potent allosteric inhibitor of SHP2, that suppresses signaling through the MAPK pathway.</p>Fórmula:C17H18Cl2N6Pureza:98.8%Cor e Forma:SolidPeso molecular:377.27K-Ras-PDEδ-IN-1
CAS:<p>K-Ras-PDEδ-IN-1 is a potent inhibitor of competitive K-Ras-PDEδ.It binds to the farnesyl binding pocket of PDEδ(Kd of 8 nM).</p>Fórmula:C25H26FN5O2Pureza:99.48%Cor e Forma:SolidPeso molecular:447.5Cilomilast
CAS:<p>Cilomilast (SB-207499) is a potent PDE4 inhibitor with IC50 of about 110 nM, has anti-inflammatory activity and low central nervous system activity. Phase 3.</p>Fórmula:C20H25NO4Pureza:97.37% - 99.52%Cor e Forma:White SolidPeso molecular:343.42(E/Z)-Elafibranor
CAS:<p>GFT505 (Elafibranor) (Elafibranor) is a PPARα/δ agonist with EC50s of 45 and 175 nM, respectively.</p>Fórmula:C22H24O4SPureza:98.36%Cor e Forma:SolidPeso molecular:384.49AGI-5198
CAS:<p>AGI-5198 (IDH-C35) is a highly effective and specific inhibitor of IDH1 R132H/R132C mutants (IC50: 0.07/0.16 μM).</p>Fórmula:C27H31FN4O2Pureza:97.37% - 99.23%Cor e Forma:SolidPeso molecular:462.56TM5441
CAS:<p>TM5441 is an orally bioavailable fibrinogen activator inhibitor-1 inhibitor that inhibits several cancer cell lines with IC50 values ranging from 13.9 to 51.1 μM.Cost-effective and quality-assured.Cost-effective and quality-assured.</p>Fórmula:C21H17ClN2O6Pureza:97.62% - 99.09%Cor e Forma:SolidPeso molecular:428.82LHW090-A7
CAS:<p>LHW090-A7 is an neutral endopeptidase (NEP) inhibitor, and an enzyme responsible for the metabolic inactivation of enkephalins.</p>Fórmula:C20H22ClNO4Pureza:98.26%Cor e Forma:SolidPeso molecular:375.85Voglibose
CAS:<p>Voglibose (Glustat), an N-substituted derivative of valiolamine, exhibits excellent inhibitory activity against α-glucosidases and action against hyperglycemia</p>Fórmula:C10H21NO7Pureza:98% - 99.90%Cor e Forma:White To Off-White Crystalline PowderPeso molecular:267.28Tipifarnib
CAS:<p>Tipifarnib (IND 58359), a quinolinone, inhibits farnesyl transferase, blocks Ras activation, arrests cell growth, and curbs angiogenesis.</p>Fórmula:C27H22Cl2N4OPureza:97.1% - 99.22%Cor e Forma:Off-White To Pale Beige SolidPeso molecular:489.4PNU-100440
CAS:<p>PNU-100440 is a biologically active compound. It is an intermediate in the synthesis of linezolid dimers, an impurity of the antibacterial agent Linezolid.</p>Fórmula:C14H17FN2O4Pureza:99.09%Cor e Forma:SolidPeso molecular:296.29ML-030
CAS:<p>ML-030 is a potent PDE4 inhibitor, selective for subtypes (A1, B1, B2, C1, D2) with IC50 ranging from 6.7 to 452 nM.</p>Fórmula:C20H20N4O4SPureza:97.93%Cor e Forma:SolidPeso molecular:412.46Sacubitril
CAS:<p>Sacubitril (AHU-377) is a potent NEP inhibitor with an IC50 of 5 nM. Sacubitril is a component of the heart failure medicine LCZ696.</p>Fórmula:C24H29NO5Pureza:97.72% - 97.91%Cor e Forma:SolidPeso molecular:411.49Olprinone
CAS:<p>Olprinone (Loprinone)(Loprinone) is a selective phosphodiesterase 3 (PDE3) inhibitor.Olprinone has been reported to improve microcirculation and attenuate</p>Fórmula:C14H10N4OPureza:99.68%Cor e Forma:SolidPeso molecular:250.26Raphin1 acetate
CAS:<p>Raphin1 acetate is a selective and orally bioavailable regulatory phosphatase PPP1R15B (R15B) inhibitor.</p>Fórmula:C10H12Cl2N4O2Pureza:99.95%Cor e Forma:SolidPeso molecular:291.13Indoximod
CAS:<p>Indoximod (NLG-8189) is a methylated tryptophan that inhibits IDO to boost T cell function by preventing tryptophan depletion.</p>Fórmula:C12H14N2O2Pureza:97.82% - 99.55%Cor e Forma:SolidPeso molecular:218.25Tebufenpyrad
CAS:<p>Tebufenpyrad (Comanche) (mitochondrial complex-1 inhibitors) is an agro-chemically important acaricide that functions like the known mitochondrial toxicant</p>Fórmula:C18H24ClN3OPureza:98.63% - 99.16%Cor e Forma:SolidPeso molecular:333.861,2-Didecanoyl-sn-glycero-3-phosphocholi
CAS:<p>1,2-Didecanoyl PC: synthetic phospholipid aiding peptide drug and insulin absorption.</p>Fórmula:C28H56NO8PPureza:98%Cor e Forma:SolidPeso molecular:565.72DASA-58
CAS:<p>DASA-58 is a specific and potent Pyruvate kinase M2 (PKM2) activator.</p>Fórmula:C19H23N3O6S2Pureza:96.96% - 99.28%Cor e Forma:SolidPeso molecular:453.53SC-57461A
CAS:<p>SC 57461A is a potent and specific leukotriene A4 hydrolase (LTA4H) inhibitor.</p>Fórmula:C20H26ClNO3Pureza:99.91%Cor e Forma:SolidPeso molecular:363.9BAY-218
CAS:<p>Bindarit (AF2838) is an aryl hydrocarbon receptor (AHR) antagonist.Cost-effective and quality-assured.</p>Fórmula:C20H17ClFN3O3Pureza:99.46% - 99.85%Cor e Forma:SolidPeso molecular:401.82Dalcetrapib
CAS:<p>Dalcetrapib (RO4607381), a rhCETP inhibitor (IC50=0.2 μM), increases the plasma HDL cholesterol.</p>Fórmula:C23H35NO2SPureza:97.98% - >99.99%Cor e Forma:SolidPeso molecular:389.59ML355
CAS:<p>ML355, a specific, effective 12-Lipoxygenase(12-LOX) inhibitors(IC50=0.34 μM), possess favorable ADME properties.</p>Fórmula:C21H19N3O4S2Pureza:98.02% - 98.2%Cor e Forma:SolidPeso molecular:441.52SR9238
CAS:<p>SR9238 is a synthetic agonist of liver X receptor inverse (IC50s: 214 nM and 43 nM for LXRα and LXRβ, respectively).</p>Fórmula:C31H33NO7S2Pureza:99.19% - 99.95%Cor e Forma:SolidPeso molecular:595.73RS-25344
CAS:<p>RS-25344: a strong PDE4 blocker, curbs eosinophil movement, boosts sperm motility in vitro.</p>Fórmula:C19H13N5O4Pureza:98.98%Cor e Forma:SolidPeso molecular:375.34
