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Metabolismo

Metabolismo

Os inibidores do metabolismo são compostos que interferem nas vias metabólicas, alterando a produção e utilização de energia dentro das células. Esses inibidores são usados para estudar a regulação do metabolismo, o papel das vias metabólicas em doenças como o câncer e o diabetes, e para desenvolver novas estratégias terapêuticas. Os inibidores do metabolismo podem direcionar várias enzimas e processos envolvidos na glicólise, na oxidação de ácidos graxos e em outras funções metabólicas. Na CymitQuimica, oferecemos uma ampla gama de inibidores do metabolismo de alta qualidade para apoiar sua pesquisa em bioquímica, distúrbios metabólicos e desenvolvimento de medicamentos.

Subcategorias de "Metabolismo"

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Foram encontrados 8626 produtos de "Metabolismo"

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  • Lodenafil

    CAS:
    <p>Lodenafil (Hydroxyhomosildenafil) is a potent PDE5 inhibitor, with treatment of erectile dysfunction (ED)</p>
    Fórmula:C23H32N6O5S
    Pureza:99.92%
    Cor e Forma:Solid
    Peso molecular:504.6
  • Aranidipine

    CAS:
    <p>Aranidipine (MPC1304) (MPC1304) is a calcium channel antagonist with potent and long-lasting antihypertensive effects.</p>
    Fórmula:C19H20N2O7
    Pureza:99.15%
    Cor e Forma:Solid
    Peso molecular:388.37
  • Tebufenpyrad

    CAS:
    <p>Tebufenpyrad (Comanche) (mitochondrial complex-1 inhibitors) is an agro-chemically important acaricide that functions like the known mitochondrial toxicant</p>
    Fórmula:C18H24ClN3O
    Pureza:98.63% - 99.16%
    Cor e Forma:Solid
    Peso molecular:333.86
  • Fluorometholone Acetate

    CAS:
    <p>Fluorometholone Acetate (Oxylone acetate) is a synthetic corticosteroid, used in the treatment of steroid responsive inflammatory conditions of the eye.</p>
    Fórmula:C24H31FO5
    Pureza:99.76%
    Cor e Forma:Solid
    Peso molecular:418.50
  • 3-(2-Naphthalenyl)-1-(3-pyridinyl)-2-propen-1-one

    CAS:
    <p>DMU2105 is a specific CYP1B1 inhibitor(CYP1B1 and CYP1A1 with IC50 of 10 nM and 742 nM, respectively)</p>
    Fórmula:C18H13NO
    Pureza:99.37%
    Cor e Forma:Solid
    Peso molecular:259.3
  • Lofemizole

    CAS:
    <p>Lofemizole is an antagonist of CYP1A2.</p>
    Fórmula:C10H9ClN2
    Pureza:97.11%
    Cor e Forma:Solid
    Peso molecular:192.64
  • Fondaparinux sodium

    CAS:
    <p>Fondaparinux sodium (SR-90107A) is an antithrombin-dependent factor Xa inhibitor with antithrombotic activity.</p>
    Fórmula:C31H43N3Na10O49S8
    Pureza:98% - >99.99%
    Cor e Forma:Solid
    Peso molecular:1728.08
  • G6PDi-1

    CAS:
    <p>G6PDi-1 is an effective G6PD inhibitor. It depletes NADPH and decreases inflammatory cytokine production.</p>
    Fórmula:C14H12N4OS
    Pureza:98.69%
    Cor e Forma:Solid
    Peso molecular:284.34
  • UNC6934

    CAS:
    <p>UNC6934 is a chemical probe targeting the N-terminal PWWP (PWWP1) domain of NSD2.</p>
    Fórmula:C24H21N5O4
    Pureza:98.67%
    Cor e Forma:Solid
    Peso molecular:443.45
  • Izilendustat hydrochloride

    CAS:
    <p>Izilendustat hydrochloride inhibits prolyl hydroxylase, stabilizing HIF-1α/HIF-2, with potential to treat various HIF-1α diseases.</p>
    Fórmula:C22H29Cl2N3O4
    Cor e Forma:Solid
    Peso molecular:470.39
  • PRL-3 Inhibitor I

    CAS:
    <p>PRL-3 Inhibitor I (BR-1) is a phosphatase of regenerating liver 3 (PRL-3) inhibitor which blocks the migration and invasion of metastatic cancer cells.</p>
    Fórmula:C17H11Br2NO2S2
    Pureza:98.11%
    Cor e Forma:Solid
    Peso molecular:485.21
  • Edoxaban Tosylate Monohydrate

    CAS:
    <p>Edoxaban(DU-176) is an oral factor Xa (FXa) inhibitor in clinical development for stroke prevention.</p>
    Fórmula:C31H40ClN7O8S2
    Pureza:99.86% - 99.91%
    Cor e Forma:Solid
    Peso molecular:738.27
  • ISX-9

    CAS:
    <p>ISX-9 (Isoxazole 9) is necessary to activate neuron-specific genes as neurogenesis inducer.</p>
    Fórmula:C11H10N2O2S
    Pureza:97.81% - ≥95%
    Cor e Forma:Solid
    Peso molecular:234.27
  • Tetradecylthioacetic acid

    CAS:
    <p>Synthetic fatty acid TTA has β-sulfur, resists β-oxidation, and activates PPARs, especially PPARα.</p>
    Fórmula:C16H32O2S
    Pureza:99.93%
    Cor e Forma:Solid
    Peso molecular:288.49
  • Elafibranor

    CAS:
    <p>Elafibranor (GFT505) is an agonist of the peroxisome proliferator-activated receptor-α (PPAR-α) and peroxisome proliferator-activated receptor-δ (PPAR-δ) with</p>
    Fórmula:C22H24O4S
    Pureza:98.42% - 98.78%
    Cor e Forma:Solid
    Peso molecular:384.49
  • BMS-986242

    CAS:
    <p>BMS-986242 is an orally active, potent and selective inhibitor of indoleamine-2,3-dioxygenase 1 (IDO1), and it can be used for the research of cancer.</p>
    Fórmula:C24H24ClFN2O
    Pureza:98.9%
    Cor e Forma:Solid
    Peso molecular:410.91
  • SGC-GAK-1

    CAS:
    <p>SGC-GAK-1 is a selective cyclin G-associated kinase (GAK) inhibitor (Ki: 3.1 nM).</p>
    Fórmula:C18H17BrN2O3
    Pureza:99.85%
    Cor e Forma:Solid
    Peso molecular:389.24
  • Lomerizine dihydrochloride

    CAS:
    <p>Lomerizine dihydrochloride (KB-2796) is an antagonist of L- and T-type voltage-gated calcium channels used to treat migraine.</p>
    Fórmula:C27H30F2N2O3·2HCl
    Pureza:99.26% - 99.80%
    Cor e Forma:Colourless Crystalline Solid
    Peso molecular:541.46
  • Soticlestat

    CAS:
    <p>Soticlestat (OV935) is a potent, selective and orally active cholesterol 24-hydroxylase (CYP46A1) inhibitor.</p>
    Fórmula:C23H23N3O2
    Pureza:99.79%
    Cor e Forma:Solid
    Peso molecular:373.45
  • Torcetrapib

    CAS:
    <p>Torcetrapib (CP-529414), a CETP inhibitor, curbs cholesteryl ester movement from HDL to LDL/VLDL; failed Phase III trials due to mortality increase.</p>
    Fórmula:C26H25F9N2O4
    Pureza:98% - 99.59%
    Cor e Forma:Lipid
    Peso molecular:600.47
  • N-(p-amylcinnamoyl) Anthranilic Acid

    CAS:
    <p>N-(p-amylcinnamoyl) Anthranilic Acid (ACA) is a broad spectrum Phospholipase A2 (PLA2) inhibitor and TRP channel blocker.</p>
    Fórmula:C21H23NO3
    Pureza:99.35% - 99.67%
    Cor e Forma:Solid
    Peso molecular:337.41
  • Azumolene

    CAS:
    <p>Azumolene (EU4093 free base)</p>
    Fórmula:C13H9BrN4O3
    Pureza:98.1% - 98.35%
    Cor e Forma:Solid
    Peso molecular:349.14
  • CVT-12012

    CAS:
    <p>CVT-12012 is an orally bioavailable inhibitor of stearoyl-CoA desaturase (SCD; IC50 = 6.1 nM in HepG2 cells).</p>
    Fórmula:C21H21F3N4O3
    Pureza:99.56%
    Cor e Forma:Solid
    Peso molecular:434.41
  • AKBA

    CAS:
    <p>AKBA (3-O-Acetyl-11-keto-beta-boswellic acid), a natural component from frankincense, is a novel activator of Nrf2.</p>
    Fórmula:C32H48O5
    Pureza:97.85% - 99.77%
    Cor e Forma:Solid
    Peso molecular:512.72
  • D159687

    CAS:
    <p>D159687 is a selective PDE4D inhibitor,had a procognitive profile as it improved memory in the novel object recognition test but had no antidepressant benefit.</p>
    Fórmula:C21H19ClN2O2
    Pureza:97.57%
    Cor e Forma:Solid
    Peso molecular:366.84
  • Fmoc-Ser(O-α-D-GalNAc(OAc)3)-OH

    CAS:
    <p>Fmoc-Ser(O-α-D-GalNAc(OAc)3)-OH (Fmoc-Ser(Ac3AcNH-α-Gal)-OH) is an anti-tumor drug</p>
    Fórmula:C32H36N2O13
    Pureza:98% - ≥98%
    Cor e Forma:Solid
    Peso molecular:656.63
  • DS-1001b

    CAS:
    <p>DS-1001b is an inhibitor of mutant IDH-1 (Isocitrate Dehydrogenase-1)</p>
    Fórmula:C29H29Cl3FN3O4
    Pureza:99.81%
    Cor e Forma:Solid
    Peso molecular:608.92
  • DY268

    CAS:
    <p>DY268 is a compound based on trisubstituted pyrazolamide without any FXR agonist activity and cytotoxicity and can be used as an effective FXR antagonist.</p>
    Fórmula:C30H32N4O5S
    Pureza:99.43% - 99.75%
    Cor e Forma:Solid
    Peso molecular:560.66
  • ML198

    CAS:
    <p>ML198: Activates &amp; chaperones glucocerebrosidase; a potential Gaucher disease treatment lead.</p>
    Fórmula:C17H14N4O
    Pureza:98.31%
    Cor e Forma:Solid
    Peso molecular:290.32
  • AKR1C3-IN-4

    CAS:
    <p>AKR1C3-IN-4: potent, selective AKR1C3 inhibitor, IC50 = 0.56 μM, potential for CRPC research.</p>
    Fórmula:C14H10F3NO2
    Pureza:98.59%
    Cor e Forma:Solid
    Peso molecular:281.23
  • Oxiconazole

    CAS:
    <p>Oxiconazole is a broad-spectrum imidazole antifungal, inhibiting ergosterol biosynthesi by disrupting cytochrome P450 enzymes (lanosterol 14- α demethylase).</p>
    Fórmula:C18H13Cl4N3O
    Pureza:99.99%
    Cor e Forma:Solid
    Peso molecular:429.13
  • AZD7325

    CAS:
    <p>AZD7325 (AZD-7325) is a GABA-Aα2,3 -selective receptor modulator.</p>
    Fórmula:C19H19FN4O2
    Pureza:99.83%
    Cor e Forma:Solid
    Peso molecular:354.38
  • IDO1-IN-1

    CAS:
    <p>IDO1-IN-1 (2 HzBTZ) is an indoleamine 2,3-dioxygenase 1 (IDO1) inhibitor.</p>
    Fórmula:C7H7N3S
    Pureza:99.36%
    Cor e Forma:Slightly Yellow To Beige-Green Crystalline Powder
    Peso molecular:165.22
  • EMAC10101d

    CAS:
    <p>compound EMAC10101d, bearing a 2,4-dichorophenyl substituent in position 4 of the dihydrothiazole ring, was the most potent and selective toward hCA II with an</p>
    Fórmula:C17H15Cl2N3O2S2
    Pureza:99.96%
    Cor e Forma:Solid
    Peso molecular:428.36
  • Imeglimin hydrochloride

    CAS:
    <p>Imeglimin hydrochloride (EMD 387008 hydrochloride) is an oral hypoglycemic agent. Imeglimin improves insulin sensitivity.Cost-effective and quality-assured.</p>
    Fórmula:C6H14ClN5
    Pureza:99.25% - 99.94%
    Cor e Forma:Solid
    Peso molecular:191.66
  • PHPS1

    CAS:
    <p>PHPS1 blocks Shp2, halts Shp2-E76K-induced Erk1/2 activation, and stops tumor cell growth.</p>
    Fórmula:C21H15N5O6S
    Pureza:99.08%
    Cor e Forma:Solid
    Peso molecular:465.44
  • PF-05221304

    CAS:
    <p>PF-05221304 (NSC-170984) is an orally active, liver-targeted inhibitor of acetyl-CoA carboxylase (ACC), a rate-limiting enzymes for fatty acid synthesis.</p>
    Fórmula:C28H30N4O5
    Pureza:98.82% - 99.50%
    Cor e Forma:Solid
    Peso molecular:502.56
  • Cintirorgon

    CAS:
    <p>Cintirorgon (LYC-55716) is a selective, oral agonist of RORγ. Cintirorgon modulates gene expression of RORγ expressing T lymphocyte immune cells.</p>
    Fórmula:C27H23F6NO6S
    Pureza:99.92%
    Cor e Forma:Solid
    Peso molecular:603.53
  • hnps-PLA Inhibitor

    CAS:
    <p>Hnps-PLA Inhibitor is an inhibitor of human nonpancreatic secretory Phospholipase A (hnps-PLA).</p>
    Fórmula:C21H21N3O4
    Pureza:99.68%
    Cor e Forma:Solid
    Peso molecular:379.41
  • 4-Bromo-3-hydroxybenzoic acid

    CAS:
    <p>4-bromo-3-hydroxybenzoic acid is a potent inhibitor of the enzyme histidine decarboxylase.</p>
    Fórmula:C7H5BrO3
    Pureza:98.11%
    Cor e Forma:Solid
    Peso molecular:217.02
  • WWL 154

    CAS:
    <p>WWL 154 is an serine hydrolase (SH) and fatty acid amide hydrolase FAAH-4 inhibitor.</p>
    Fórmula:C18H19N3O5
    Pureza:99.22%
    Cor e Forma:Solid
    Peso molecular:357.36
  • 1-Aminobenzotriazole

    CAS:
    <p>1-Aminobenzotriazole (ABT) (ABT) is a non-specific cytochrome P450 (CYP) inhibitor.</p>
    Fórmula:C6H6N4
    Pureza:98% - 99.54%
    Cor e Forma:Yellow To Beige Or Light Brown Crystalline Powder
    Peso molecular:134.14
  • Choline Fenofibrate

    CAS:
    <p>Choline Fenofibrate (Trilipix) is a choline formulation of fenofibrate, a synthetic phenoxy-isobutyric acid derivate and prodrug with antihyperlipidemic</p>
    Fórmula:C22H28ClNO5
    Pureza:98.82%
    Cor e Forma:Solid
    Peso molecular:421.91
  • Avasimibe

    CAS:
    <p>Avasimibe (PD-148515): Oral ACAT inhibitor, prevents arterial cholesterol buildup; IC50: 3.3 μM. Hinders CYP2C9/1A2/2C19; IC50: 2.9/13.9/26.5 μM.</p>
    Fórmula:C29H43NO4S
    Pureza:98.39% - 99.91%
    Cor e Forma:Solid
    Peso molecular:501.72
  • UK-371804

    CAS:
    <p>UK-371804: potent uPA blocker; candidate for chronic skin ulcer preclinical studies.</p>
    Fórmula:C14H16ClN5O4S
    Pureza:95.81% - 99.77%
    Cor e Forma:Solid
    Peso molecular:385.83
  • UC-1728

    CAS:
    <p>UC-1728 (t-TUCB) is an effective rabbit soluble epoxide hydrolase inhibitor (IC50: 2 nM on rabbit liver).</p>
    Fórmula:C21H21F3N2O5
    Pureza:99.88%
    Cor e Forma:Solid
    Peso molecular:438.4
  • OU749

    CAS:
    <p>OU749 is a γ-glutamyl transferase (GGT) inhibitor with an intrinsic Ki of 17.6 μM.</p>
    Fórmula:C16H15N3O3S2
    Pureza:99.50%
    Cor e Forma:Solid
    Peso molecular:361.44
  • Conduritol B epoxide

    CAS:
    <p>Conduritol B epoxide is an irreversible inhibitor of β-glucosidase (GCase).</p>
    Fórmula:C6H10O5
    Pureza:99.85% - ≥98%
    Cor e Forma:White Crystalline Solid
    Peso molecular:162.14
  • ML-​226

    CAS:
    <p>ML226 is a α/β hydrolase domain-containing protein 11 (ABHD11) inhibitor that inhibits ABHD11 in vitro and in situ.</p>
    Fórmula:C23H26N4O2
    Pureza:99.61%
    Cor e Forma:Solid
    Peso molecular:390.48
  • PF-07038124

    CAS:
    <p>PF-07038124 inhibits PDE4B2 (IC50=0.5 nM), IFNγ (IC50=1.06 nM), IL4 (IC50=4.1 nM), and IL-13 (IC50=125 nM).</p>
    Fórmula:C18H22BNO4
    Cor e Forma:Solid
    Peso molecular:327.18
  • N6022

    CAS:
    <p>N6022(IC50 of 8 nM) is an effective, reversible, and selective S-Nitrosoglutathione reductase(GSNOR) inhibitor.</p>
    Fórmula:C24H22N4O3
    Pureza:98.24% - 98.32%
    Cor e Forma:Solid
    Peso molecular:414.46
  • LJ570

    CAS:
    <p>LJ570 is the first PPARα/γ dual agonist (PPARα,PPARγ with EC50s of 1.05 and 0.12 μM, respectively[)</p>
    Fórmula:C27H22O3
    Pureza:99.64%
    Cor e Forma:Solid
    Peso molecular:394.46
  • URB602

    CAS:
    <p>URB602 is a specific monoacylglycerol lipase (MGL) inhibitor, which inhibits rat brain MGL (IC50: 28±4 μM) through a noncompetitive mechanism.</p>
    Fórmula:C19H21NO2
    Pureza:99.64% - 99.9%
    Cor e Forma:Off-White Solid
    Peso molecular:295.38
  • Fenretinide

    CAS:
    <p>Fenretinide (4-HPR) is an orally-active synthetic retinoid derivative with potential antineoplastic and chemopreventive activities.</p>
    Fórmula:C26H33NO2
    Pureza:98% - 99.68%
    Cor e Forma:Yellow Powder
    Peso molecular:391.55
  • CD437

    CAS:
    <p>CD437 (AHPN) is a specifc Retinoic Acid Receptor γ (RARγ) agonist.</p>
    Fórmula:C27H26O3
    Pureza:98.92% - 99.63%
    Cor e Forma:Solid
    Peso molecular:398.49
  • BPTES

    CAS:
    <p>BPTES(IC50 of 0.16 μM) is an effective and specific GlutamiN/Ase GLS1 (KGA) inhibitor.</p>
    Fórmula:C24H24N6O2S3
    Pureza:95.83% - 99.64%
    Cor e Forma:Solid
    Peso molecular:524.68
  • MPO-IN-28

    CAS:
    <p>MPO-IN-28 is a novel potent, irreversible Myeloperoxidase (MPO) inhibitor with IC50 of 44 nM.</p>
    Fórmula:C11H13N5O
    Pureza:98.04%
    Cor e Forma:Solid
    Peso molecular:231.25
  • HA130

    CAS:
    <p>HA130 is a selective ATX (autotaxin) inhibitor.</p>
    Fórmula:C24H19BFNO5S
    Pureza:98.26% - ≥95%
    Cor e Forma:Solid
    Peso molecular:463.29
  • EAAT2 activator 1

    CAS:
    <p>EAAT2 activator 1 (3-[(2-Chloro-6-fluorobenzyl)thio]-6-pyridin-2-ylpyridazine) is a thiopyridazine derivative that has been found to increase EAAT2 protein</p>
    Fórmula:C16H11ClFN3S
    Pureza:98.86%
    Cor e Forma:Solid
    Peso molecular:331.8
  • 1-Cyclohexyl-3-dodecyl urea

    CAS:
    <p>1-Cyclohexyl-3-dodecyl urea (NCND) is a highly selective soluble epoxide hydrolase (sEH) inhibitor.</p>
    Fórmula:C19H38N2O
    Pureza:99.59%
    Cor e Forma:Solid
    Peso molecular:310.52
  • ASP-9521

    CAS:
    <p>ASP-9521 is a selective, potent and orally active indole-based AKR1C3 inhibitor with an IC50 of 11 nM for human AKR1C3.Cost-effective and quality-assured.</p>
    Fórmula:C19H26N2O3
    Pureza:95.11% - 96.96%
    Cor e Forma:Solid
    Peso molecular:330.42
  • Pinaverium bromide

    CAS:
    <p>Pinaverium bromide is an calcium channel blocker with Antispasmodic and effectively relieves pain, diarrhea and intestinal discomfort.</p>
    Fórmula:C26H41Br2NO4
    Pureza:99.52%
    Cor e Forma:White Crystalline Powder
    Peso molecular:591.42
  • Nitrofurazone

    CAS:
    <p>Nitrofurazone (Furacilin) is a topical anti-infective agent effective against gram-negative and gram-positive bacteria.</p>
    Fórmula:C6H6N4O4
    Pureza:99.87%
    Cor e Forma:Pale Yellow Needles Solution) 6 0 - 6 5 Alkaline Solutions Are Dark Orange (Ntp 1992)
    Peso molecular:198.14
  • Linrodostat

    CAS:
    <p>Linrodostat (BMS-986205) is a selective indoleamine 2, 3-dioxygenase 1 (IDO1) inhibitor.</p>
    Fórmula:C24H24ClFN2O
    Pureza:99.54% - 99.71%
    Cor e Forma:Solid
    Peso molecular:410.91
  • PF-06282999

    CAS:
    <p>PF-06282999 is a potent and selective myeloperoxidase inhibitor which is potentially useful for the treatment of cardiovascular diseases.</p>
    Fórmula:C13H12ClN3O3S
    Pureza:98.15% - 98.28%
    Cor e Forma:Solid
    Peso molecular:325.77
  • NS-638

    CAS:
    <p>NS-638 is a Ca2+-channel blocker. It can block K+-stimulated intracellular Ca2+-elevation (IC50: 3.4 μM).</p>
    Fórmula:C15H11ClF3N3
    Pureza:98.44%
    Cor e Forma:Solid
    Peso molecular:325.72
  • Pentamidine

    CAS:
    <p>Pentamidine is an antifungal and antiprotozoal agent, interacting directly with the pathogen genome by binding to AT-rich regions of duplex DNA and the minor</p>
    Fórmula:C19H24N4O2
    Pureza:98.64% - 99.67%
    Cor e Forma:Crystallizes As Colorless Plates From Water Solid
    Peso molecular:340.42
  • 2-hydroxymethyl benzoic acid

    CAS:
    <p>2-hydroxymethyl benzoic acid is a principal metabolite of the phthalidyl moiety in man.</p>
    Fórmula:C8H8O3
    Pureza:98.36%
    Cor e Forma:Solid
    Peso molecular:152.15
  • Alrestatin

    CAS:
    <p>Alrestatin (AY-22284) is a specific inhibitor of aldose reductase and attenuates glucose-induced angiotensin II production in rat vascular smooth muscle in</p>
    Fórmula:C14H9NO4
    Pureza:99.23%
    Cor e Forma:Solid
    Peso molecular:255.2256
  • GOT1 inhibitor-1

    CAS:
    <p>GOT1 inhibitor-1 (GOT1 inhibitor 2c) is a novel, potent and non-covalent inhibitor of glutamate oxaloacetate transaminase 1 (GOT1) with an IC50 of 8.2 uM.</p>
    Fórmula:C19H19ClN4O
    Pureza:99.70%
    Cor e Forma:Solid
    Peso molecular:354.83
  • SR3335

    CAS:
    <p>SR3335 (ML 176) is a selective inverse agonist of RORα, competitively inhibiting the binding of 25-hydroxycholesterol to the ligand binding domain (Ki: 220 nM).</p>
    Fórmula:C13H9F6NO3S2
    Pureza:99.77%
    Cor e Forma:Solid
    Peso molecular:405.34
  • AZ876

    CAS:
    <p>AZ876 is a potent, highly selective LXR agonist with Ki/EC50 of 7/6 nM and 11/73 nM for hLXRα and hLXRβ respectively.</p>
    Fórmula:C24H29N3O3S
    Pureza:99.86%
    Cor e Forma:Solid
    Peso molecular:439.57
  • SR8278

    CAS:
    <p>SR8278 is an REV-ERBα antagonist(EC50 = 0.47 μM), blocking activation of the receptor by the synthetic agonist GSK 4112</p>
    Fórmula:C18H19NO3S2
    Pureza:99.44% - 99.73%
    Cor e Forma:Solid
    Peso molecular:361.48
  • BRL-50481

    CAS:
    <p>BRL-50481 is a novel and selective inhibitor of PDE7 with IC50s of 0.15, 12.1, 62 and 490 μM for PDE7A, PDE7B, PDE4 and PDE3, respectively.</p>
    Fórmula:C9H12N2O4S
    Pureza:99.66%
    Cor e Forma:Solid
    Peso molecular:244.27
  • Toloxatone

    CAS:
    <p>Toloxatone (MD 69276) is a reversible monoamine oxidase A (MAOA) inhibitor.</p>
    Fórmula:C11H13NO3
    Pureza:98.58%
    Cor e Forma:Solid
    Peso molecular:207.23
  • Obafistat

    CAS:
    <p>Obafistat is a potent inhibitor of aldo-keto reductase AKR1C3 with an IC50 of 1.2 nM for human AKR1C3.</p>
    Fórmula:C15H16FN5O3S
    Pureza:99.71%
    Cor e Forma:Solid
    Peso molecular:365.38
  • BI-187004

    CAS:
    <p>BI-187004 is an 11β-hydroxysteroid dehydrogenase 1 inhibitor.</p>
    Fórmula:C21H18N4O
    Pureza:98.63%
    Cor e Forma:Solid
    Peso molecular:342.39
  • U-104

    CAS:
    <p>U-104 (NSC-213841) is an effective carbonic anhydrase (CA) inhibitor for CA IX( Ki=45.1 nM) and CA XII(Ki=4.5 nM).</p>
    Fórmula:C13H12FN3O3S
    Pureza:98.76% - 99.88%
    Cor e Forma:Solid
    Peso molecular:309.32
  • Gonadorelin Acetate (33515-09-2 free base)

    CAS:
    <p>Gonadorelin Acetate (33515-09-2 free base) (Luteinizing Hormone Releasing Hormone (LH-RH)) is hypothalamic neuropeptide which plays a key role in the control of</p>
    Fórmula:C59H83N17O17
    Pureza:99.42% - 99.46%
    Cor e Forma:White Or Off-White Powder
    Peso molecular:1302.39
  • Pirinixic Acid

    CAS:
    <p>Pirinixic Acid (NSC 310038) is a synthetic thiacetic acid derivative used in biomedical research, a peroxisome proliferator that activates specific PPAR.</p>
    Fórmula:C14H14ClN3O2S
    Pureza:98.27% - 99.92%
    Cor e Forma:Solid
    Peso molecular:323.8
  • AUDA

    CAS:
    <p>AUDA is an inhibitor of sEH(IC50 values of 18 and 69 nM for the mouse and human enzymes, respectively)</p>
    Fórmula:C23H40N2O3
    Pureza:99.50%
    Cor e Forma:Solid
    Peso molecular:392.58
  • p-Fluoro-L-phenylalanine

    CAS:
    <p>p-Fluoro-L-phenylalanine: TH substrate, studies enzyme regulation, binds E. coli L-leucine receptor, KD 0.26μM.</p>
    Fórmula:C9H10FNO2
    Pureza:99.63%
    Cor e Forma:White To Off-White Powder
    Peso molecular:183.18
  • BW-A 78U

    CAS:
    <p>BW-A 78U is a PDE4 inhibitor (IC50: 3 μM). It is not inhibition on the lipopolysaccharide (LPS)-induced TNF-α release.</p>
    Fórmula:C13H12FN5
    Pureza:99.45%
    Cor e Forma:Solid
    Peso molecular:257.27
  • GSK805

    CAS:
    <p>GSK805 is a potent, orally bioavailable and CNS-penetrant RORγt inhibitor.Cost-effective and quality-assured.</p>
    Fórmula:C23H18Cl2F3NO4S
    Pureza:98% - ≥95%
    Cor e Forma:Solid
    Peso molecular:532.36
  • 2-Bromo-4'-hydroxyacetophenone

    CAS:
    <p>2-Bromo-4'-hydroxyacetophenone(PTP Inhibitor I) is a cell-permeable, PTP inhibitor that covalently blocks the catalytic domain of the SHP-1(ΔSH2).</p>
    Fórmula:C8H7BrO2
    Pureza:98.64%
    Cor e Forma:Clear Colorless To Light Yellow Liquid
    Peso molecular:215.04
  • Telaglenastat

    CAS:
    <p>Telaglenastat (CB 839) (IC50 of 24 nM), an effective, specific, and oral inhibitor, which is bioavailable glutaminase, for recombinant human GAC.</p>
    Fórmula:C26H24F3N7O3S
    Pureza:97.57% - 99.89%
    Cor e Forma:Solid
    Peso molecular:571.57
  • Pargyline

    CAS:
    <p>Pargyline (Pargylamine) is a monoamine oxidase inhibitor with antihypertensive properties.</p>
    Fórmula:C11H13N
    Pureza:95.64% - 97.21%
    Cor e Forma:Solid
    Peso molecular:159.23
  • PfDHODH-IN-2

    CAS:
    <p>PfDHODH-IN-2: powerful antimalarial, blocks PfDHODH (IC50: 1.11 μM), for malaria research.</p>
    Fórmula:C13H12ClNO3S
    Pureza:98.9%
    Cor e Forma:Solid
    Peso molecular:297.76
  • Pentamidine isethionate

    CAS:
    <p>Pentamidine isethionate (Pentamidine diisethionate) is a synthetic amidine derivative, Pentamidine Isethionate is an antiprotozoal and antifungal agent.</p>
    Fórmula:C23H36N4O10S2
    Pureza:98% - 99.83%
    Cor e Forma:Slight Butyric Odor Very Bitter Taste Ph (5% Aqueous Solution) 4 5-6 5 (Ntp 1992)
    Peso molecular:592.68
  • FG-2216

    CAS:
    <p>FG-2216 (YM-311) is a HIF-prolyl hydroxylase inhibitor for the PDH2 enzyme; orally bioavailable and induced reversible and significant Epo induction in vivo.</p>
    Fórmula:C12H9ClN2O4
    Pureza:97.1% - >99.99%
    Cor e Forma:Solid
    Peso molecular:280.66
  • JZL 184

    CAS:
    <p>JZL 184 is a potent and selective inhibitor of MAGL with IC50 of 8 nM and 4 μM for inhibition of MAGL and FAAH in mouse brain membranes respectively.</p>
    Fórmula:C27H24N2O9
    Pureza:97.56% - 99.31%
    Cor e Forma:Solid
    Peso molecular:520.49
  • RGX-104

    CAS:
    <p>RGX-104 (RGX-104 free Acid) free Acid is an agonist of potent liver-X nuclear hormone receptor (LXR)</p>
    Fórmula:C34H33ClF3NO3
    Pureza:98.79% - 99.53%
    Cor e Forma:Solid
    Peso molecular:596.08
  • KPT9274

    CAS:
    <p>KPT9274 (PAK4-IN-1) is a non-competitive dual inhibitor of PAK4 and NAMPT(IC50= ~120 nM). It is an orally bioavailable small molecule.</p>
    Fórmula:C35H29F3N4O3
    Pureza:99.75% - 99.93%
    Cor e Forma:Solid
    Peso molecular:610.62
  • LOX-IN-3 dihydrochloride

    CAS:
    <p>LOX-IN-3 dihydrochloride is an inhibitor of lysyl oxidase (LOX).</p>
    Fórmula:C13H15Cl2FN2O2S
    Pureza:99.96%
    Cor e Forma:Solid
    Peso molecular:353.24
  • Cobicistat

    CAS:
    <p>Cobicistat (GS-9350): A carbamate, thiazole derivative, and CYP3A inhibitor used to boost anti-HIV drugs for treating HIV.</p>
    Fórmula:C40H53N7O5S2
    Pureza:97.36% - 99.62%
    Cor e Forma:Solid
    Peso molecular:776.02
  • Glycerol 3-phosphate biscyclohexylammonium salt

    CAS:
    <p>Glycerol 3-phosphate biscyclohexylammonium salt is an endogenous metabolite produced by cytosolic glycerol 3-phosphate dehydrogenase pathway.</p>
    Fórmula:C15H35N2O6P
    Pureza:99.94%
    Cor e Forma:Solid
    Peso molecular:370.42
  • ARM1

    CAS:
    <p>ARM1 is a potent inhibitor of aminopeptidase and epoxide hydrolase. The IC50 values are 7.61 µM for aminopeptidase and 12.4 µM for epoxide hydrolase.</p>
    Fórmula:C16H14N2S
    Pureza:99.36%
    Cor e Forma:Solid
    Peso molecular:266.36
  • (±)-Amiflamine

    CAS:
    <p>(±)-Amiflamine (2-dimethylphenethylamine) is an inhibitor of reversible MAO-A.</p>
    Fórmula:C12H20N2
    Pureza:97.24%
    Cor e Forma:Solid
    Peso molecular:192.3
  • Cecropin P1, porcine acetate


    <p>Cecropin P1, porcine acetate is an antibacterial peptide found in Hyalophora cecropia and pig intestine.</p>
    Fórmula:C149H257N45O45
    Pureza:95.4% - 98%
    Cor e Forma:Solid
    Peso molecular:3398.91
  • Bempedoic acid

    CAS:
    <p>Bempedoic acid (ETC1002) is an orally available, once-daily LDL-C lowering small molecule designed to lower elevated levels of LDL-C.</p>
    Fórmula:C19H36O5
    Pureza:99.85% - 99.94%
    Cor e Forma:Solid
    Peso molecular:344.49