CymitQuimica logo
Metabolismo

Metabolismo

Os inibidores do metabolismo são compostos que interferem nas vias metabólicas, alterando a produção e utilização de energia dentro das células. Esses inibidores são usados para estudar a regulação do metabolismo, o papel das vias metabólicas em doenças como o câncer e o diabetes, e para desenvolver novas estratégias terapêuticas. Os inibidores do metabolismo podem direcionar várias enzimas e processos envolvidos na glicólise, na oxidação de ácidos graxos e em outras funções metabólicas. Na CymitQuimica, oferecemos uma ampla gama de inibidores do metabolismo de alta qualidade para apoiar sua pesquisa em bioquímica, distúrbios metabólicos e desenvolvimento de medicamentos.

Subcategorias de "Metabolismo"

Exibir 34 mais subcategorias

Foram encontrados 8595 produtos de "Metabolismo"

Ordenar por

Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
produtos por página.
  • SR9238

    CAS:
    <p>SR9238 is a synthetic agonist of liver X receptor inverse (IC50s: 214 nM and 43 nM for LXRα and LXRβ, respectively).</p>
    Fórmula:C31H33NO7S2
    Pureza:99.19% - 99.95%
    Cor e Forma:Solid
    Peso molecular:595.73
  • Tiplaxtinin

    CAS:
    <p>Tiplaxtinin (Tiplasinin)(PAI-039) is a selective and orally efficacious inhibitor of plasminogen activator inhibitor-1 (PAI-1) with IC50 of 2.7 uM.</p>
    Fórmula:C24H16F3NO4
    Pureza:99.16% - 99.93%
    Cor e Forma:Solid
    Peso molecular:439.38
  • Seladelpar

    CAS:
    <p>Seladelpar (MBX 8025) has been used in trials studying the treatment of Hyperlipidemia.</p>
    Fórmula:C21H23F3O5S
    Pureza:99.18% - 99.41%
    Cor e Forma:Solid
    Peso molecular:444.46
  • XEN445

    CAS:
    <p>XEN445, a potent and selective endothelial lipase(EL) inhibitor (IC50=0.237 uM), exhibitis good ADME and PK properties.</p>
    Fórmula:C18H17F3N2O3
    Pureza:99.47% - 99.6%
    Cor e Forma:Solid
    Peso molecular:366.33
  • CP-609754

    CAS:
    <p>CP-609754 shows selective inhibition of farnesyltransferase.</p>
    Fórmula:C29H22ClN3O2
    Pureza:99.04% - 99.86%
    Cor e Forma:Solid
    Peso molecular:479.96
  • Olprinone

    CAS:
    <p>Olprinone (Loprinone)(Loprinone) is a selective phosphodiesterase 3 (PDE3) inhibitor.Olprinone has been reported to improve microcirculation and attenuate</p>
    Fórmula:C14H10N4O
    Pureza:99.68%
    Cor e Forma:Solid
    Peso molecular:250.26
  • Sacubitril

    CAS:
    <p>Sacubitril (AHU-377) is a potent NEP inhibitor with an IC50 of 5 nM. Sacubitril is a component of the heart failure medicine LCZ696.</p>
    Fórmula:C24H29NO5
    Pureza:97.72% - 97.91%
    Cor e Forma:Solid
    Peso molecular:411.49
  • StemRegenin 1

    CAS:
    <p>StemRegenin 1 (SR1) is an aryl hydrocarbon receptor (AhR) inhibitor.</p>
    Fórmula:C24H23N5OS
    Pureza:98% - 99.89%
    Cor e Forma:Solid
    Peso molecular:429.54
  • TM5441

    CAS:
    <p>TM5441 is an orally bioavailable fibrinogen activator inhibitor-1 inhibitor that inhibits several cancer cell lines with IC50 values ranging from 13.9 to 51.1 μM.Cost-effective and quality-assured.Cost-effective and quality-assured.</p>
    Fórmula:C21H17ClN2O6
    Pureza:97.62% - 99.09%
    Cor e Forma:Solid
    Peso molecular:428.82
  • γ-Glu-Phe TFA(7432-24-8 free base)


    <p>γ-Glu-Phe TFA(7432-24-8 free base) is a dipeptide composed of gamma-glutamate and phenylalanine and is a proteolytic breakdown product of larger proteins.</p>
    Fórmula:C16H19F3N2O7
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:408.33
  • Pyributicarb

    CAS:
    <p>Pyributicarb (TSH-888) is a potent activator of both CYP3A4 gene and human pregnane X receptor (hPXR).</p>
    Fórmula:C18H22N2O2S
    Pureza:99.702% - ≥95%
    Cor e Forma:Solid
    Peso molecular:330.44
  • U-73343

    CAS:
    <p>U-73343 is an inactive analog of U-73122 and can be used as a negative control. U-73122 dose-dependently inhibits acid secretion irrespective of the stimulant.</p>
    Fórmula:C29H42N2O3
    Pureza:99.06%
    Cor e Forma:Solid
    Peso molecular:466.66
  • Tazarotene

    CAS:
    <p>Tazarotene (Zorac), a synthetic topical retinoid, treats psoriasis by normalizing keratinocytes and reducing growth.</p>
    Fórmula:C21H21NO2S
    Pureza:97.01% - 99.14%
    Cor e Forma:White Solid
    Peso molecular:351.46
  • Cycloguanil hydrochloride

    CAS:
    <p>Cycloguanil hydrochloride, proguanil's metabolite, inhibits Plasmodium/human dihydrofolate reductase (Ki: 0.3/1.5 nM).</p>
    Fórmula:C11H14ClN5·ClH
    Pureza:98.72%
    Cor e Forma:Solid
    Peso molecular:288.18
  • PSB-1491

    CAS:
    <p>PSB-1491 is a selective and competitive monoamine oxidase B inhibitor with IC50 of 0.386 nM, &gt;25000-fold selective versus MAO-A.</p>
    Fórmula:C15H11Cl2N3O
    Pureza:98.41% - 99.68%
    Cor e Forma:Solid
    Peso molecular:320.17
  • Udenafil

    CAS:
    <p>Udenafil is an inhibitor of PDE5 .</p>
    Fórmula:C25H36N6O4S
    Pureza:99.90%
    Cor e Forma:Off-White Solid
    Peso molecular:516.66
  • Icerguastat

    CAS:
    <p>Icerguastat (IFB-088) is a selective inhibitor of holophosphatase. Icerguastat selectively inhibited a regulatory subunit of protein phosphatase 1 in vivo.</p>
    Fórmula:C8H9ClN4
    Pureza:97.95%
    Cor e Forma:Solid
    Peso molecular:196.64
  • Mardepodect

    CAS:
    <p>Mardepodect (PF-2545920) is a phosphodiesterase inhibitor selective for the PDE10A subtype with an IC50 of 0.37 nM, &gt;1000-fold selectivity over PDE.</p>
    Fórmula:C25H20N4O
    Pureza:99.81% - 99.94%
    Cor e Forma:Solid
    Peso molecular:392.45
  • Spinacine

    CAS:
    <p>Spinacine is a condensation product of formaldehyde and histidine and an endogenous metabolite.</p>
    Fórmula:C7H9N3O2
    Pureza:99.89% - 99.98%
    Cor e Forma:Solid
    Peso molecular:167.17
  • Mutant IDH1-IN-1

    CAS:
    <p>Mutant IDH1-IN-1 is a potent mutant IDH1 R132 h inhibitor with IC50 &lt; 0.1 uM.</p>
    Fórmula:C30H31FN4O2
    Pureza:99.49% - >99.99%
    Cor e Forma:Solid
    Peso molecular:498.59
  • 16α-Hydroxyprednisolone


    <p>16α-Hydroxyprednisolone is a stereoselective metabolite of the 22(R) epimer of the glucocorticoid budesonide</p>
    Fórmula:C21H28O6
    Pureza:99.75%
    Cor e Forma:White Solid
    Peso molecular:376.44
  • TP0463518

    CAS:
    <p>TP-0463518 is a highly potent HIF prolyl hydroxylase (PHD) inhibitor (IC50s: 13 nM and 18 nM for human and rat PHD2, respectively).</p>
    Fórmula:C20H18ClN3O6
    Pureza:99.52%
    Cor e Forma:Solid
    Peso molecular:431.83
  • JNJ-1661010

    CAS:
    <p>JNJ-1661010 (Takeda-25) is an effective and specific FAAH inhibitor (IC50: 10/ 12 nM for rat/human), shows &gt;100-fold selectivity for FAAH-1 than FAAH-2.</p>
    Fórmula:C19H19N5OS
    Pureza:99.79% - 99.97%
    Cor e Forma:Solid
    Peso molecular:365.45
  • CP-91149

    CAS:
    <p>CP-91149 is a selective glycogen phosphorylase (GP) inhibitor with IC50 of 0.13 μM in the presence of glucose, 5- to 10-fold less potent in the absence of</p>
    Fórmula:C21H22ClN3O3
    Pureza:99.66% - 99.81%
    Cor e Forma:Solid
    Peso molecular:399.87
  • Potassium 2-hydroxy-2-methylsuccinate

    CAS:
    <p>Potassium 2-hydroxy-2-methylsuccinate ((±)-2-Hydroxy-2-methylsuccinic acid dipotassium salt) is a type of endogenous metabolite.</p>
    Fórmula:C5H6K2O5
    Pureza:99.96% - ≥98%
    Cor e Forma:Solid
    Peso molecular:224.29
  • β-Aminopropionitrile

    CAS:
    <p>β-Aminopropionitrile (3-Aminopropionitrile) is a selective inhibitor of lysyl oxidase.</p>
    Fórmula:C3H6N2
    Pureza:98.29%
    Cor e Forma:Light Yellow Liquid
    Peso molecular:70.09
  • 1,2-Dipalmitoyl-sn-glycero-3-phosphoethanolamine

    CAS:
    <p>DPPE, a phospholipid, thickens membranes with Ca2+ and cholesterol.</p>
    Fórmula:C37H74NO8P
    Pureza:99.59% - 99.71%
    Cor e Forma:Solid
    Peso molecular:691.96
  • Globalagliatin

    CAS:
    <p>Globalagliatin (LY2608204) has been used in trials studying the treatment of Diabetes Mellitus, Type 2.</p>
    Fórmula:C28H37N3O3S3
    Pureza:98% - 99.49%
    Cor e Forma:Solid
    Peso molecular:559.81
  • Tebuconazole

    CAS:
    <p>Tebuconazole: azole fungicide, inhibits CYP51 with IC50s 0.9 μM (C. albicans) and 1.3 μM (human).</p>
    Fórmula:C16H22ClN3O
    Pureza:99.21%
    Cor e Forma:Solid
    Peso molecular:307.82
  • Gabapentin hydrochloride

    CAS:
    <p>Gabapentin hydrochloride (Neurontin HCl) is a GABA analogue, used to treat seizures and neuropathic pain.</p>
    Fórmula:C9H17NO2·HCl
    Pureza:99.71%
    Cor e Forma:Off-White Solid
    Peso molecular:207.7
  • RPI-1

    CAS:
    <p>RPI-1 is a competitive, potent ATP-dependent Ret kinase inhibitor.</p>
    Fórmula:C17H15NO4
    Pureza:98.91% - ≥95%
    Cor e Forma:Solid
    Peso molecular:297.31
  • Alagebrium chloride

    CAS:
    <p>Alagebrium chloride (ALT711) inhibits AGEs, lowers systolic blood pressure, and benefits diastolic patients.</p>
    Fórmula:C13H14ClNOS
    Pureza:99.65% - 99.77%
    Cor e Forma:Solid
    Peso molecular:267.77
  • Uridine 5′-triphosphate tris salt

    CAS:
    <p>Uridine 5′-triphosphate tris salt (Uridine 5'-triphosphoric acid) is an agonist to the P2Y receptor and has been used to study concentrations of intracellular</p>
    Fórmula:C21H48N5O24P3
    Pureza:99.04% - 99.94%
    Cor e Forma:Solid
    Peso molecular:847.55
  • L-Leucyl-L-Leucine methyl ester hydrochloride

    CAS:
    <p>L-Leucyl-L-Leucine methyl ester hydrochloride (Leu-Leu-ome hydrochloride) is a dipeptide condensation product of L-leucine methyl ester. Cost-effective and quality-assured.</p>
    Fórmula:C13H27ClN2O3
    Pureza:98.41% - 99.63%
    Cor e Forma:Solid
    Peso molecular:294.81
  • Liquiritin

    CAS:
    <p>Liquiritin (Liquiritigenin-4'-O-glucoside) (LIQ) is a main component among the licorice flavonoids, and possesses anti-inflammatory and anti-cancer abilities.</p>
    Fórmula:C21H22O9
    Pureza:98.16% - 98.66%
    Cor e Forma:Solid
    Peso molecular:418.39
  • TOFA

    CAS:
    <p>TOFA (MDL14514) is an allosteric inhibitor of acetyl-CoA carboxylase-α (ACCA).</p>
    Fórmula:C19H32O4
    Pureza:97.52% - 98.98%
    Cor e Forma:Solid
    Peso molecular:324.45
  • Telotristat

    CAS:
    <p>Telotristat, active metabolite of LX1606, is an oral tryptophan hydroxylase inhibitor with potential antiserotonergic effects.</p>
    Fórmula:C25H22ClF3N6O3
    Pureza:99.70%
    Cor e Forma:Solid
    Peso molecular:546.93
  • AGI-6780

    CAS:
    <p>AGI-6780 is a potent and selective inhibitor of IDH2 R140Q mutant.</p>
    Fórmula:C21H18F3N3O3S2
    Pureza:98.19% - 99.7%
    Cor e Forma:Solid
    Peso molecular:481.51
  • PF-04457845

    CAS:
    <p>PF-04457845 is a greatly and effctive FAAH inhibitor, and for hFAAH(IC50=7.2±0.63 nM) and rFAAH(IC50=7.4±0.62 nM).</p>
    Fórmula:C23H20F3N5O2
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:455.43
  • 2,4-Diamino-6-hydroxypyrimidine

    CAS:
    <p>2,4-Diamino-6-hydroxypyrimidine (DAHP) (DAHP) is a selective, specific inhibitor of GTP cyclohydrolase I, the rate limiting step for de novo pterin synthesis</p>
    Fórmula:C4H6N4O
    Pureza:99.82%
    Cor e Forma:White Solid Crystals
    Peso molecular:126.12
  • Tienilic Acid

    CAS:
    <p>Tienilic Acid is a uricosuric diuretic with certain hepatotoxicity</p>
    Fórmula:C13H8Cl2O4S
    Pureza:99.55%
    Cor e Forma:Solid
    Peso molecular:331.17
  • PFK-015

    CAS:
    <p>PFK-015 (PFK15) is an effective inhibitor of PFKFB3 (IC50: 110 nM) and inhibits PFKFB3 activity in Y cells (IC50: 20 nM).</p>
    Fórmula:C17H12N2O
    Pureza:99.7% - 99.85%
    Cor e Forma:Solid
    Peso molecular:260.29
  • IDO-IN-7

    CAS:
    <p>IDO-IN-7 (NLG-919 analogue) is a potent IDO (indoleamine-(2, 3)-dioxygenase) pathway inhibitor.</p>
    Fórmula:C18H22N2O
    Pureza:99.32% - 99.9%
    Cor e Forma:Solid
    Peso molecular:282.38
  • CP-640186 hydrochloride

    CAS:
    <p>CP-640186 hydrochloride (CP 640186 HCl) is an isozyme-nonselective acetyl-CoA carboxylase (ACC) inhibitor, including rat liver ACC1 (IC50: 53 nM) and rat</p>
    Fórmula:C30H36ClN3O3
    Pureza:98.86%
    Cor e Forma:Solid
    Peso molecular:522.08
  • Edoxaban Tosylate Monohydrate

    CAS:
    <p>Edoxaban(DU-176) is an oral factor Xa (FXa) inhibitor in clinical development for stroke prevention.</p>
    Fórmula:C31H40ClN7O8S2
    Pureza:99.86% - 99.91%
    Cor e Forma:Solid
    Peso molecular:738.27
  • Pradefovir mesylate

    CAS:
    <p>Pradefovir mesylate (Hepavir B) is converted to 9-(2-phosphonylmethoxyethyl)adenine (PMEA) in human liver microsomes with Km of 60 μM.</p>
    Fórmula:C18H23ClN5O7PS
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:519.9
  • GSK 650394

    CAS:
    <p>GSK 650394 is an inhibitor of serum- and glucocorticoid-regulated kinases (SGK). GSK 650394 has antitumor activity. Cost-effective and quality-assured.</p>
    Fórmula:C25H22N2O2
    Pureza:97.46% - >99.99%
    Cor e Forma:Solid
    Peso molecular:382.45
  • Dimethylfraxetin

    CAS:
    <p>Dimethylfraxetin (6,7,8-Trimethoxycoumarin) is a Carbonic anhydrase inhibitor(Ki:0.0097 μM)</p>
    Fórmula:C12H12O5
    Pureza:99.96% - ≥95%
    Cor e Forma:Solid
    Peso molecular:236.22
  • EMD638683

    CAS:
    <p>EMD638683,a novel SGK inhibitor with antihypertensive potency(with an IC50 of 3 μM).</p>
    Fórmula:C18H18F2N2O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:364.34
  • IACS-13909

    CAS:
    <p>IACS-13909 (BBP-398), a specific and potent allosteric inhibitor of SHP2, that suppresses signaling through the MAPK pathway.</p>
    Fórmula:C17H18Cl2N6
    Pureza:98.8%
    Cor e Forma:Solid
    Peso molecular:377.27
  • Melilotic acid

    CAS:
    <p>3-(2-Hydroxyphenyl)propanoic acid, aka melilotic acid, found in cytoplasm, in foods like herbs, beetroot, cinnamon.</p>
    Fórmula:C9H10O3
    Pureza:99.65% - 99.83%
    Cor e Forma:Solid
    Peso molecular:166.17
  • CALP3 acetate(261969-05-5 free base)


    <p>CALP3 acetate blocks Ca2+ channels, mimics elevated [Ca2+]i, activates EF hands, and regulates CaM, channels, and pumps.</p>
    Fórmula:C46H72N10O11
    Pureza:96.49%
    Cor e Forma:Solid
    Peso molecular:941.12
  • PKD-IN-1

    CAS:
    <p>CRT0066101 is an inhibitor of PKD.</p>
    Fórmula:C18H19ClN4O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:342.82
  • K-Ras-PDEδ-IN-1

    CAS:
    <p>K-Ras-PDEδ-IN-1 is a potent inhibitor of competitive K-Ras-PDEδ.It binds to the farnesyl binding pocket of PDEδ(Kd of 8 nM).</p>
    Fórmula:C25H26FN5O2
    Pureza:99.48%
    Cor e Forma:Solid
    Peso molecular:447.5
  • Cilomilast

    CAS:
    <p>Cilomilast (SB-207499) is a potent PDE4 inhibitor with IC50 of about 110 nM, has anti-inflammatory activity and low central nervous system activity. Phase 3.</p>
    Fórmula:C20H25NO4
    Pureza:97.37% - 99.52%
    Cor e Forma:White Solid
    Peso molecular:343.42
  • Minaprine dihydrochloride

    CAS:
    <p>Minaprine dihydrochloride: reversible MAO-A inhibitor, mild on acetylcholinesterase, used for depression.</p>
    Fórmula:C17H24Cl2N4O
    Pureza:99.43% - 99.99%
    Cor e Forma:Solid
    Peso molecular:371.3
  • AGI-5198

    CAS:
    <p>AGI-5198 (IDH-C35) is a highly effective and specific inhibitor of IDH1 R132H/R132C mutants (IC50: 0.07/0.16 μM).</p>
    Fórmula:C27H31FN4O2
    Pureza:97.37% - 99.23%
    Cor e Forma:Solid
    Peso molecular:462.56
  • Ethyl 3,4-dihydroxybenzoate

    CAS:
    <p>Ethyl 3,4-dihydroxybenzoate (EDHB): a prolyl hydroxylase inhibitor attenuates acute hypobaric hypoxia mediated vascular leakage in brain.</p>
    Fórmula:C9H10O4
    Pureza:99.88%
    Cor e Forma:White Crystal Or Powder
    Peso molecular:182.17
  • JNJ-42165279

    CAS:
    <p>JNJ-42165279 selectively inactivates FAAH without notably affecting other enzymes, ion channels, receptors, or CYPs/hERG at 10 μM.</p>
    Fórmula:C18H17ClF2N4O3
    Pureza:99.67% - 99.88%
    Cor e Forma:Solid
    Peso molecular:410.8
  • amflutizole

    CAS:
    <p>Amflutizole used for the treatment of gout, and is a Xanthine oxidase inhibitor</p>
    Fórmula:C11H7F3N2O2S
    Pureza:98.83%
    Cor e Forma:Solid
    Peso molecular:288.246
  • GSK0660

    CAS:
    <p>GSK0660 is an antagonist and inverse agonist of PPARβ/δ.</p>
    Fórmula:C19H18N2O5S2
    Pureza:99.26% - ≥95%
    Cor e Forma:Solid
    Peso molecular:418.49
  • Tempol

    CAS:
    <p>Tempol (Tanol) is a superoxide scavenger. It has anti-inflammatory, neuroprotective and analgesic effects.</p>
    Fórmula:C9H18NO2
    Pureza:97% - 99.74%
    Cor e Forma:4-Hydroxy-Tempo Appears As Orange Flakes Solid Flakes
    Peso molecular:172.25
  • Fraxinellone

    CAS:
    <p>1.</p>
    Fórmula:C14H16O3
    Pureza:99.35% - 99.92%
    Cor e Forma:Solid
    Peso molecular:232.27
  • SEP-0372814

    CAS:
    <p>SEP-0372814 is a potent inhibitor of PDE10.</p>
    Fórmula:C21H19N7
    Pureza:99.29%
    Cor e Forma:Solid
    Peso molecular:369.42
  • Tebufenpyrad

    CAS:
    <p>Tebufenpyrad (Comanche) (mitochondrial complex-1 inhibitors) is an agro-chemically important acaricide that functions like the known mitochondrial toxicant</p>
    Fórmula:C18H24ClN3O
    Pureza:98.63% - 99.16%
    Cor e Forma:Solid
    Peso molecular:333.86
  • 8-Azaadenosine

    CAS:
    <p>8-Azaadenosine inhibits ADAR1, blocks RNA editing, and reduces thyroid cancer cell proliferation and spread.</p>
    Fórmula:C9H12N6O4
    Pureza:99.39%
    Cor e Forma:Solid
    Peso molecular:268.23
  • SC-57461A

    CAS:
    <p>SC 57461A is a potent and specific leukotriene A4 hydrolase (LTA4H) inhibitor.</p>
    Fórmula:C20H26ClNO3
    Pureza:99.91%
    Cor e Forma:Solid
    Peso molecular:363.9
  • BMS-779788

    CAS:
    <p>BMS-779788 (XL-652) is an LXRα/β partial agonist (IC50: 68/14 nM).</p>
    Fórmula:C28H29ClN2O3S
    Pureza:98.65% - 99.24%
    Cor e Forma:Solid
    Peso molecular:509.06
  • 4-Amino-6-(trifluoromethyl)benzene-1,3-disulfonamide

    CAS:
    <p>4-Amino-6-(trifluoromethyl)benzene-1,3-disulfonamide (4-Amino-6-(trifluoromethyl)benzene-1,3-d) is a carbonic anhydrase inhibitor, used as a potential anti-</p>
    Fórmula:C7H8F3N3O4S2
    Pureza:98.58%
    Cor e Forma:Solid
    Peso molecular:319.28
  • Tuftsin 3TFA

    CAS:
    <p>Tuftsin 3TFA is a tetrapeptide. It is a macrophage/microglial activator.</p>
    Fórmula:C27H43F9N8O12
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:842.66
  • WIN 18446

    CAS:
    <p>inhibitor of aldehyde dehydrogenase 1a2 (ALDH1a2)</p>
    Fórmula:C12H20Cl4N2O2
    Pureza:99.69%
    Cor e Forma:Solid
    Peso molecular:366.11
  • Inosine

    CAS:
    <p>Inosine (NSC-20262), an endogenous purine nucleoside produced by the catabolism of adenosine, is an agonist of adenosine receptors A1R and A2AR. Low-Cost!</p>
    Fórmula:C10H12N4O5
    Pureza:99.51% - 99.89%
    Cor e Forma:Solid
    Peso molecular:268.23
  • Fomepizole

    CAS:
    <p>Fomepizole (4-Methylpyrazole), a competitive inhibitor of alcohol dehydrogenase, is used as an antidote in methanol or ethylene glycol poisoning.</p>
    Fórmula:C4H6N2
    Pureza:98.1% - 99.94%
    Cor e Forma:Yellow <13°C Solid >13°C Liquid
    Peso molecular:82.1
  • Barnidipine hydrochloride

    CAS:
    <p>Barnidipine HCl is a potent dihydropyridine Ca²⁺ blocker with 0.35 nM IC50 in pig coronary artery.</p>
    Fórmula:C27H30ClN3O6
    Pureza:99.88%
    Cor e Forma:Solid
    Peso molecular:528
  • PDM2

    CAS:
    <p>PDM 2 is a potent and selective aryl hydrocarbon receptor (AhR) antagonist.</p>
    Fórmula:C14H9Cl3
    Pureza:99.44%
    Cor e Forma:Solid
    Peso molecular:283.58
  • ABX-1431

    CAS:
    <p>ABX-1431 (Elcubragistat) is a selective and orally available CNS-penetrant monoacylglycerol lipase (MAGL/MGLL) inhibitor (IC50: 14 nM).</p>
    Fórmula:C20H22F9N3O2
    Pureza:99.8% - 99.96%
    Cor e Forma:Solid
    Peso molecular:507.39
  • ISX-9

    CAS:
    <p>ISX-9 (Isoxazole 9) is necessary to activate neuron-specific genes as neurogenesis inducer.</p>
    Fórmula:C11H10N2O2S
    Pureza:97.81% - ≥95%
    Cor e Forma:Solid
    Peso molecular:234.27
  • trifarotene

    CAS:
    <p>Trifarotene (CD5789) is a RARγ agonist, 65x more selective than RARα and 16x than RARβ, with EC50 of 7.7 nM.</p>
    Fórmula:C29H33NO4
    Pureza:99.51%
    Cor e Forma:Solid
    Peso molecular:459.58
  • Furafylline

    CAS:
    <p>Furafylline is a selective inhibitor of human cytochrome P450 (CYP)1A2 (IC50 : 0.07 μM),</p>
    Fórmula:C12H12N4O3
    Pureza:99.61%
    Cor e Forma:Solid
    Peso molecular:260.25
  • ML351

    CAS:
    <p>ML351 is a potent and selective inhibitor of human 15-lipoxygenase-1 (15 LOX)(IC50: 200 nM).</p>
    Fórmula:C15H11N3O
    Pureza:97.67%
    Cor e Forma:Solid
    Peso molecular:249.27
  • Osoresnontrine

    CAS:
    <p>Osoresnontrine is a potent and selective inhibitor of PDE9A (IC50 of 52 nM),and can be used in the research of memory.</p>
    Fórmula:C16H17N5O2
    Pureza:99.93%
    Cor e Forma:Solid
    Peso molecular:311.34
  • VAS2870

    CAS:
    <p>VAS2870 is an inhibitor of NADPH oxidase (NOX).</p>
    Fórmula:C18H12N6OS
    Pureza:99.74%
    Cor e Forma:Solid
    Peso molecular:360.39
  • Oroxylin A

    CAS:
    <p>Oroxylin A fights tumors, aids RAS therapy, promotes CaCo-2 cell apoptosis, blocks MCF-7 cell invasion and enhances leukemia treatment.</p>
    Fórmula:C16H12O5
    Pureza:98.72% - 99.55%
    Cor e Forma:Solid
    Peso molecular:284.26
  • Isradipine

    CAS:
    <p>Isradipine (PN 200-110), a dihydropyridine, is an antihypertensive calcium channel blocker that dilates arteries and reduces resistance.</p>
    Fórmula:C19H21N3O5
    Pureza:99.84% - 99.95%
    Cor e Forma:Yellow Solid
    Peso molecular:371.39
  • CP671305

    CAS:
    <p>CP671305 is an orally active, potent and selective inhibitor of phosphodiesterase-4-D.</p>
    Fórmula:C23H19FN2O7
    Pureza:99.39%
    Cor e Forma:Solid
    Peso molecular:454.4
  • Dichlorphenamide

    CAS:
    <p>Dichlorphenamide (Diclofenamide) is a carbonic anhydrase inhibitor that is used in the treatment of glaucoma.</p>
    Fórmula:C6H6Cl2N2O4S2
    Pureza:96.87% - 97.25%
    Cor e Forma:Needles From Dimethylsulfoxide + Water Solid
    Peso molecular:305.16
  • Ziritaxestat

    CAS:
    <p>Ziritaxestat (GLPG1690), an autotaxin inhibitor, currently being evaluated in an exploratory phase 2 study in idiopathic pulmonary fibrosis patients.</p>
    Fórmula:C30H33FN8O2S
    Pureza:97% - 99.85%
    Cor e Forma:Solid
    Peso molecular:588.7
  • Tryptophan, N-indol-3-ylacetyl- (6CI)

    CAS:
    <p>Tryptophan, N-indol-3-ylacetyl- (6CI) (Indole-3-acetyl-L-tryptophan) is involved in regulatory mechanisms for the control of auxin activity during physiological</p>
    Fórmula:C21H19N3O3
    Pureza:99.55%
    Cor e Forma:Solid
    Peso molecular:361.4
  • 2,3-dihydro-1H-indene-5-sulfonamide

    CAS:
    <p>2,3-dihydro-1H-indene-5-sulfonamide is Carbonic anhydrase 12 (human) inhibitor.</p>
    Fórmula:C9H11NO2S
    Pureza:99.89%
    Cor e Forma:Solid
    Peso molecular:197.25
  • Hydroxy Dimetridazole

    CAS:
    <p>Hydroxy Dimetridazole is a hydroxy metabolite of Dimetridazole which combats protozoan infections.</p>
    Fórmula:C5H7N3O3
    Pureza:99.83% - 99.85%
    Cor e Forma:Solid
    Peso molecular:157.13
  • trans-AUCB

    CAS:
    <p>trans-AUCB (t-AUCB) is an effective and selective soluble epoxide hydrolase inhibitor (IC50s: 1.3 nM, 8 nM, 8 nM for hsEH, mouse sEH and rat sEH, respectively).</p>
    Fórmula:C24H32N2O4
    Pureza:99.27% - 99.66%
    Cor e Forma:Solid
    Peso molecular:412.52
  • 3,4, 5-trimethoxyphenylacetic acid

    CAS:
    <p>3,4,5-trimethoxyphenylacetic acid: used in organic synthesis, mainly for carboxyl group conversion.</p>
    Fórmula:C11H14O5
    Pureza:99.84%
    Cor e Forma:White Crystalline Powder
    Peso molecular:226.23
  • PT-2385

    CAS:
    <p>PT-2385 is a selective HIF-2α inhibitor (Kd&lt;50 nM).</p>
    Fórmula:C17H12F3NO4S
    Pureza:98.91% - 99.55%
    Cor e Forma:Solid
    Peso molecular:383.34
  • Z944

    CAS:
    <p>Z944 is a T-type calcium channel blocker.</p>
    Fórmula:C19H27ClFN3O2
    Pureza:99.8%
    Cor e Forma:Solid
    Peso molecular:383.89
  • Barnidipine

    CAS:
    <p>Barnidipine (YM-09730-5(Free base)) is a calcium channel blocker.</p>
    Fórmula:C27H29N3O6
    Pureza:99.98%
    Cor e Forma:Solid
    Peso molecular:491.54
  • SF1670

    CAS:
    <p>SF1670 (PTPase CD45 Inhibitor) is a specific PTEN inhibitor with IC50 of 2 μM.</p>
    Fórmula:C19H17NO3
    Pureza:98.25% - 98.54%
    Cor e Forma:Solid
    Peso molecular:307.34
  • Benzolamide

    CAS:
    <p>Benzolamide (CL 11366) inhibits carbonic anhydrase effectively and low-threshold calcium currents in hippocampal pyramidal neurons.</p>
    Fórmula:C8H8N4O4S3
    Pureza:99.31%
    Cor e Forma:Solid
    Peso molecular:320.37
  • L-165041

    CAS:
    <p>L-165041 is a potent and selective agonist of the nuclear receptor PPARβ and PPARδ(Ki = 9 nM, EC50 = ~500 nM ,respectively)</p>
    Fórmula:C22H26O7
    Pureza:97.97%
    Cor e Forma:Solid
    Peso molecular:402.44
  • Lofemizole

    CAS:
    <p>Lofemizole is an antagonist of CYP1A2.</p>
    Fórmula:C10H9ClN2
    Pureza:97.11%
    Cor e Forma:Solid
    Peso molecular:192.64
  • 1-Naphthaleneacetic acid potassium salt

    CAS:
    <p>1-Naphthaleneacetic acid potassium salt (1-NAA Potassium Salt) is a synthetic phytogrowth hormone that promotes plant growth and a PLA2 inhibitor.</p>
    Fórmula:C12H9O2·K
    Pureza:97.68%
    Cor e Forma:Off-White To Beige Powder
    Peso molecular:224.3