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Metabolismo

Metabolismo

Os inibidores do metabolismo são compostos que interferem nas vias metabólicas, alterando a produção e utilização de energia dentro das células. Esses inibidores são usados para estudar a regulação do metabolismo, o papel das vias metabólicas em doenças como o câncer e o diabetes, e para desenvolver novas estratégias terapêuticas. Os inibidores do metabolismo podem direcionar várias enzimas e processos envolvidos na glicólise, na oxidação de ácidos graxos e em outras funções metabólicas. Na CymitQuimica, oferecemos uma ampla gama de inibidores do metabolismo de alta qualidade para apoiar sua pesquisa em bioquímica, distúrbios metabólicos e desenvolvimento de medicamentos.

Subcategorias de "Metabolismo"

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Foram encontrados 8595 produtos de "Metabolismo"

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  • ZK824190 hydrochloride

    CAS:
    <p>ZK824190 hydrochloride, an oral selective uPA inhibitor (IC50: 237 nM), also inhibits tPA (1600 nM) and Plasmin (1850 nM), used in multiple sclerosis research.</p>
    Fórmula:C22H21ClF2N2O4
    Cor e Forma:Solid
    Peso molecular:450.87
  • β-Aminopropionitrile hydrochloride

    CAS:
    <p>β-Aminopropionitrile hydrochloride is a selective, oral, irreversible inhibitor of lysyl oxidase (LOX) that reduces metastatic seeding potential.</p>
    Fórmula:C3H7ClN2
    Pureza:99.32%
    Cor e Forma:Solid
    Peso molecular:106.55
  • PF-8380

    CAS:
    <p>PF-8380 is an effective and orally available autotaxin inhibitor (IC50: 2.8 nM, in isolated enzyme assay; 101 nM, in the human whole blood).</p>
    Fórmula:C22H21Cl2N3O5
    Pureza:98.70% - 99.25%
    Cor e Forma:Solid
    Peso molecular:478.33
  • MLCK inhibitor peptide 18 acetate


    <p>MLCK inhibitor peptide 18 acetate: Selective (IC50=50nM), 4000x more than CaM kinase II. Does not block PKA. Cell-permeable.</p>
    Fórmula:C62H109N23O13
    Pureza:99.57%
    Cor e Forma:Solid
    Peso molecular:1384.67
  • Nanterinone mesylate

    CAS:
    <p>Nanterinone Mesylate is the mesylate form of Nanterinone that is a novel positive inotropic and balanced vasodilator.</p>
    Fórmula:C16H19N3O4S
    Cor e Forma:Solid
    Peso molecular:349.4
  • 21-deacetyldeflazacort

    CAS:
    <p>21-deacetyldeflazacort is a metabolite of Deflazacort, which is a systemic corticosteroid and a derivative of prednisolone.</p>
    Fórmula:C23H29NO5
    Pureza:99.96%
    Cor e Forma:Solid
    Peso molecular:399.48
  • 6-Hydroxy-4-methylcoumarin

    CAS:
    <p>6-Hydroxy-4-methylcoumarin (6-Hydroxy-4-Methyl-2H-Chromen-2-One) is a secondary metabolite of coumarin, which has anticancer effects.</p>
    Fórmula:C10H8O3
    Pureza:98.93%
    Cor e Forma:Solid
    Peso molecular:176.17
  • WWL229

    CAS:
    <p>WWL229 selectively inhibits Ces3 without affecting Ces1f, ABHD6, or other serine hydrolases, mimicking WWL113 in adipocytes.</p>
    Fórmula:C16H22N2O5
    Pureza:98.14%
    Cor e Forma:Solid
    Peso molecular:322.36
  • Linrodostat mesylate

    CAS:
    <p>Linrodostat (BMS-986205) is an oral IDO1 inhibitor that boosts immune response and has anti-cancer properties.</p>
    Fórmula:C25H28ClFN2O4S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:507.02
  • CP-640186

    CAS:
    <p>CP-640186 is an isozyme-nonselective ACCase inhibitor. The IC50s of CP-640186 is 53 nM and 61 nM for rat liver ACC1 and rat skeletal muscle ACC2 respectively.</p>
    Fórmula:C30H35N3O3
    Pureza:99.87%
    Cor e Forma:Solid
    Peso molecular:485.62
  • Mibefradil dihydrochloride

    CAS:
    <p>Mibefradil dihydrochloride (Ro 40-5967 (dihydrochloride)) is an blocker of calcium channel with moderate selectivity for T-type Ca2+ channels (T-type and L-type</p>
    Fórmula:C29H40Cl2FN3O3
    Pureza:99.45% - 99.72%
    Cor e Forma:Solid
    Peso molecular:568.55
  • 7-Ethoxy-4-Methylcoumarin

    CAS:
    <p>7-Ethoxy-4-Methylcoumarin: fragrant, organic, enzyme inhibitor; used in drug effect studies.</p>
    Fórmula:C12H12O3
    Pureza:99.50%
    Cor e Forma:Solid
    Peso molecular:204.22
  • MK-8245

    CAS:
    <p>MK-8245 is a liver-targeting SCD inhibitor for human SCD1 (IC50: 1 nM) and for rat/mouse SCD1 (IC50: 3 nM), with anti-diabetic and anti-dyslipidemic function.</p>
    Fórmula:C17H16BrFN6O4
    Pureza:97.58% - 99%
    Cor e Forma:Solid
    Peso molecular:467.25
  • Indoximod

    CAS:
    <p>Indoximod (NLG-8189) is a methylated tryptophan that inhibits IDO to boost T cell function by preventing tryptophan depletion.</p>
    Fórmula:C12H14N2O2
    Pureza:97.82% - 99.55%
    Cor e Forma:Solid
    Peso molecular:218.25
  • 6-Aminonicotinamide

    CAS:
    <p>6-Aminonicotinamide (6-AN) is a well-established inhibitor of the NADP+-dependent enzyme.</p>
    Fórmula:C6H7N3O
    Pureza:98.99% - 99.4%
    Cor e Forma:Physical Description White Crystalline Solid (Ntp 1992)
    Peso molecular:137.14
  • ABT-639

    CAS:
    <p>ABT-639 is a potent and selective T-type calcium channel blocker.</p>
    Fórmula:C20H20ClF2N3O3S
    Pureza:99.12% - 99.77%
    Cor e Forma:Solid
    Peso molecular:455.91
  • Edoxaban hydrochloride

    CAS:
    <p>Edoxaban (DU-176b) HCl: Oral, selective Factor Xa inhibitor, Ki 0.561 nM; prevents thromboembolic disease.</p>
    Fórmula:C24H31Cl2N7O4S
    Cor e Forma:Solid
    Peso molecular:584.52
  • L-778123 Dihydrochloride

    CAS:
    <p>L-778123 blocks FPTase/GGPTase-I, halts Ki-Ras prenylation, has acceptable toxicity with radiotherapy in advanced pancreatic cancer.</p>
    Fórmula:C22H22Cl3N5O
    Cor e Forma:Solid
    Peso molecular:478.802
  • Gcase activator 1

    CAS:
    <p>Gcase activator 1 (LTI-291) is a glucocerebrosidase (Gcase) activator.</p>
    Fórmula:C20H30N4O2
    Pureza:99.25% - 99.31%
    Cor e Forma:Solid
    Peso molecular:358.48
  • (E)-2-Decenoic acid

    CAS:
    <p>(E)-2-Decenoic acid (trans-2-Decenoic acid) is an unsaturated fatty acid found in royal jelly produced from the mandibular gland secretions of honeybees.</p>
    Fórmula:C10H18O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:170.25
  • Alkaline Phosphatase

    CAS:
    <p>Alkaline phosphatase is a membrane-bound glycoprotein that catalyzes the hydrolysis of phosphate monoesters under alkaline conditions. High-Quality, Low-Cost!</p>
    Pureza:≥98%
    Cor e Forma:Solid
    Peso molecular:N/A
  • Brinzolamide hydrochloride


    <p>Brinzolamide (AL-4862) HCl selectively inhibits carbonic anhydrase II, reducing IOP for glaucoma research. IC50: 3.2 nM.</p>
    Cor e Forma:Solid
  • 4-methyl-2-(4-(trifluoromethyl)phenyl)thiazole-5-carboxylic acid

    CAS:
    <p>4-methyl-2-(4-(trifluoromethyl)phenyl)thiazole-5-carboxylic acid is used as a pharmaceutical intermediate.</p>
    Fórmula:C12H8F3NO2S
    Pureza:99.35%
    Cor e Forma:Solid
    Peso molecular:287.26
  • Crisaborole

    CAS:
    <p>Crisaborole (AN-2728) is a Phosphodiesterase 4 Inhibitor.</p>
    Fórmula:C14H10BNO3
    Pureza:99.70%
    Cor e Forma:Solid
    Peso molecular:251.05
  • 2,3-dihydroxy-3-methylbutanoic acid

    CAS:
    <p>2,3-dihydroxy-3-methylbutanoic acid, a leucine metabolite, boosts muscle growth by activating mTOR.</p>
    Fórmula:C5H10O4
    Pureza:99.03%
    Cor e Forma:Solid
    Peso molecular:134.1305
  • AKR1C3-IN-1

    CAS:
    <p>AKR1C3-IN-1 is a potent and selective inhibitor of AKR1C3(IC50 of 13 nM).</p>
    Fórmula:C16H15NO4S
    Pureza:98.02%
    Cor e Forma:Solid
    Peso molecular:317.36
  • sun

    CAS:
    <p>Sun(4H-Furo[3,2-b]pyrrole-5-carboxylic acid) is an orally active and potent inhibitor of DAAO (DAO)</p>
    Fórmula:C7H5NO3
    Pureza:99.61%
    Cor e Forma:Solid
    Peso molecular:151.12
  • Aldicarb sulfone

    CAS:
    <p>Aldicarb sulfone is a cholinesterase inhibitor .</p>
    Fórmula:C7H14N2O4S
    Pureza:99.05%
    Cor e Forma:Aldicarb Sulfone Is A White Crystalline Solid Insecticide
    Peso molecular:222.26
  • SPI-112

    CAS:
    <p>SPI-112, the SPI-112 methyl ester analog, can inhibit cellular Shp2 PTP activity.</p>
    Fórmula:C22H17FN4O5S
    Pureza:97.51% - >99.99%
    Cor e Forma:Solid
    Peso molecular:468.46
  • Navoximod

    CAS:
    <p>Navoximod (GDC-0919) (NLG- 919, GDC-0919) is a potent indoleamine-(2,3)-dioxygenase (IDO) pathway inhibitor (Ki/EC50: 7 nM/75 nM).</p>
    Fórmula:C18H21FN2O2
    Pureza:99.37%
    Cor e Forma:Solid
    Peso molecular:316.37
  • SR 16832

    CAS:
    <p>SR 16832: Dual-site PPARγ inhibitor; outperforms GW 9662, T 0070907 in ligand binding, transcription inhibition.</p>
    Fórmula:C17H12ClN3O4
    Pureza:99.6%
    Cor e Forma:Solid
    Peso molecular:357.75
  • Carbutamide

    CAS:
    <p>Carbutamide is a sulfonylurea antidiabetic agent with hypoglycemic activity.</p>
    Fórmula:C11H17N3O3S
    Pureza:98.77%
    Cor e Forma:Crystals Solid
    Peso molecular:271.34
  • Fatostatin

    CAS:
    <p>Fatostatin inhibits SREBP-1/2 by binding to SCAP, blocking their ER-Golgi transport.</p>
    Fórmula:C18H18N2S
    Pureza:99.92%
    Cor e Forma:Solid
    Peso molecular:294.41
  • Vardenafil hydrochloride trihydrate

    CAS:
    <p>Vardenafil hydrochloride trihydrate (BAY38-9456) is a new type PDE inhibitor with IC50 of 0.7 and 180 nM for PDE5 and PDE1, respectively.</p>
    Fórmula:C23H32N6O4S·HCl·3H2O
    Pureza:99.77%
    Cor e Forma:Solid
    Peso molecular:579.11
  • NSC-226572

    CAS:
    <p>NSC-226572, a synthetic alliin analog from cruciferous veggies, turns into thiosulfinate via alliinase.</p>
    Fórmula:C4H9NO3S
    Pureza:99.48%
    Cor e Forma:Solid
    Peso molecular:151.18
  • G6PDi-1

    CAS:
    <p>G6PDi-1 is an effective G6PD inhibitor. It depletes NADPH and decreases inflammatory cytokine production.</p>
    Fórmula:C14H12N4OS
    Pureza:98.69%
    Cor e Forma:Solid
    Peso molecular:284.34
  • Piclamilast

    CAS:
    <p>Piclamilast (RP 73401) is a PDE4 inhibitor.</p>
    Fórmula:C18H18Cl2N2O3
    Pureza:98.28% - 99.57%
    Cor e Forma:Solid
    Peso molecular:381.25
  • Zolamide

    CAS:
    <p>Zolamide (CL 5343) may be used to prevent altitude sickness and reduce the symptoms.</p>
    Fórmula:C2H4N4O2S2
    Pureza:99.75%
    Cor e Forma:Solid
    Peso molecular:180.21
  • Zinc Phytate

    CAS:
    <p>Zinc Phytate, present in food, plays a crucial role in human nutrient absorption.</p>
    Fórmula:C6H6O24P6Zn6
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:1040
  • Fmoc-Gly-Thr(psi(Me,Me)pro)-OH

    CAS:
    <p>Fmoc-Gly-Thr(psi(Me,Me)pro)-OH is a polypeptide composed of two amino acids.</p>
    Fórmula:C24H26N2O6
    Pureza:97.35%
    Cor e Forma:Solid
    Peso molecular:438.47
  • ML-211

    CAS:
    <p>ML-211 is a carbamate-based dual inhibitor of LYPLA1 (IC50 = 17 nM) and the related LYPLA2 (IC50 = 30 nM)</p>
    Fórmula:C25H30N4O2
    Pureza:97.07%
    Cor e Forma:Solid
    Peso molecular:418.53
  • 1-phenyl-3,4-dihydroisochinoline

    CAS:
    <p>1-phenyl-3,4-dihydroisochinoline: dopamine analog, interacts with CNS receptors, studied for Parkinson's, Alzheimer's, and Huntington's.</p>
    Fórmula:C15H13N
    Pureza:98.01%
    Cor e Forma:Solid
    Peso molecular:207.27
  • O-Succinylhomoserine

    CAS:
    <p>O-Succinylhomoserine (O-Succinyl-L-homoserine) is an intermediate in the synthesis of cystathionine by E coli..</p>
    Fórmula:C8H13NO6
    Pureza:≥98%
    Cor e Forma:Solid
    Peso molecular:219.19
  • L(+)-Leucinol

    CAS:
    <p>L(+)-Leucinol is a potent inhibitor of leucine aminopeptidase.</p>
    Fórmula:C6H15NO
    Pureza:98%
    Cor e Forma:Clear Colorless To Slightly Yellow Liquid
    Peso molecular:117.19
  • 3-METHOXY-DL-TYROSINE

    CAS:
    <p>3-Methoxy-DL-Tyrosine: natural, non-essential amino, precursor to dopamine, may aid in treating Parkinson's, depression, obesity.</p>
    Fórmula:C10H13NO4
    Pureza:99.90%
    Cor e Forma:Solid
    Peso molecular:211.21
  • LXR-623

    CAS:
    <p>LXR-623 (WAY 252623) is an orally bioavailable and highly specifical synthetic modulator of LXR.</p>
    Fórmula:C21H12ClF5N2
    Pureza:97.91% - 99.24%
    Cor e Forma:Solid
    Peso molecular:422.78
  • BVT 2733

    CAS:
    <p>BVT 2733 is a new, non-steroidal, isoform-specific inhibitor of 11β-HSD1.</p>
    Fórmula:C17H21ClN4O3S2
    Pureza:98% - 99.64%
    Cor e Forma:Solid
    Peso molecular:428.96
  • Dimethyl DL-Glutamate (hydrochloride)

    CAS:
    <p>Dimethyl DL-glutamate boosts insulin release in response to glucose.</p>
    Fórmula:C7H14ClNO4
    Pureza:≥95%
    Cor e Forma:Solid
    Peso molecular:211.64
  • GW0742

    CAS:
    <p>GW0742 (GW610742) is an effective and specific PPARδ agonist (EC50: 1 nM/1.1 μM/2 μM, for human PPARδ/α/γ).</p>
    Fórmula:C21H17F4NO3S2
    Pureza:99.75% - 99.85%
    Cor e Forma:Solid
    Peso molecular:471.49
  • RGX-104 hydrochloride

    CAS:
    <p>RGX-104 hydrochloride (SB742881) is a small molecule LXR agonist that regulates innate immunity using transcriptional activation of the ApoE gene.</p>
    Fórmula:C34H34Cl2F3NO3
    Pureza:99.49%
    Cor e Forma:Solid
    Peso molecular:632.54
  • Mildronate

    CAS:
    <p>Mildronate (Meldonium) is an inhibitor of biosynthesis of L-carnitine by gamma-butyrobetaine (GBB) hydroxylase and as a competitive inhibitor of renal carnitine</p>
    Fórmula:C6H14N2O2
    Pureza:99.94%
    Cor e Forma:White Crystalline Powder
    Peso molecular:146.19
  • SU0268

    CAS:
    <p>SU0268 is a potent and specific 8-Oxoguanine DNA glycosylase 1 (OGG1) inhibitor.</p>
    Fórmula:C26H25N3O4S
    Pureza:99.97% - 99.98%
    Cor e Forma:Solid
    Peso molecular:475.56
  • N-Valyltryptophan

    CAS:
    <p>N-Valyltryptophan (Val-trp) is an incomplete breakdown product of protein catabolism or protein digestion.</p>
    Fórmula:C16H21N3O3
    Pureza:97.52%
    Cor e Forma:Solid
    Peso molecular:303.36
  • Epacadostat

    CAS:
    <p>Epacadostat (INCB 024360) is an oral, potent and selective IDO1 inhibitor with IC50 value of 71.8 nM.Cost-effective and quality-assured.</p>
    Fórmula:C11H13BrFN7O4S
    Pureza:98% - >99.99%
    Cor e Forma:Solid
    Peso molecular:438.23
  • Levofloxacin N-oxide

    CAS:
    <p>Levofloxacin N-oxide is an impurity isolated from levofloxacin.</p>
    Fórmula:C18H20FN3O5
    Pureza:99.84%
    Cor e Forma:Solid
    Peso molecular:377.37
  • 2-Hydroxycaprylic acid

    CAS:
    <p>2-Hydroxycaprylic acid (2-hydroxyoctanoic acid) belongs to the class of organic compounds known as medium-chain fatty acids.</p>
    Fórmula:C8H16O3
    Pureza:98% - 99.84%
    Cor e Forma:Solid
    Peso molecular:160.21
  • DMOG

    CAS:
    <p>DMOG (Dimethyloxalylglycine), an antagonist of the α-ketoglutarate cofactor, is an inhibitor for HIF prolyl hydroxylase.</p>
    Fórmula:C6H9NO5
    Pureza:80.23% - 99.98%
    Cor e Forma:Solid
    Peso molecular:175.14
  • ML355

    CAS:
    <p>ML355, a specific, effective 12-Lipoxygenase(12-LOX) inhibitors(IC50=0.34 μM), possess favorable ADME properties.</p>
    Fórmula:C21H19N3O4S2
    Pureza:98.02% - 98.2%
    Cor e Forma:Solid
    Peso molecular:441.52
  • RS-25344

    CAS:
    <p>RS-25344: a strong PDE4 blocker, curbs eosinophil movement, boosts sperm motility in vitro.</p>
    Fórmula:C19H13N5O4
    Pureza:98.98%
    Cor e Forma:Solid
    Peso molecular:375.34
  • L-Homocystine

    CAS:
    <p>Homocystine briefly forms before turning into cystathionine via vitamin B6; linked to schizophrenia and neural tube defects; folic acid lowers risk.</p>
    Fórmula:C8H16N2O4S2
    Pureza:99.79%
    Cor e Forma:Solid
    Peso molecular:268.35
  • YM976

    CAS:
    <p>YM976 is an orally active PDE4 inhibitor (IC50:2.2 nM)</p>
    Fórmula:C17H16ClN3O
    Pureza:99.84%
    Cor e Forma:Solid
    Peso molecular:313.78
  • UK-5099

    CAS:
    <p>UK-5099 (PF-1005023) is a potent MPC inhibitor with an IC50 of 50 nM in rat heart mitochondria.</p>
    Fórmula:C18H12N2O2
    Pureza:97.39% - >99.99%
    Cor e Forma:Solid
    Peso molecular:288.3
  • ML351

    CAS:
    <p>ML351 is a potent and selective inhibitor of human 15-lipoxygenase-1 (15 LOX)(IC50: 200 nM).</p>
    Fórmula:C15H11N3O
    Pureza:97.67%
    Cor e Forma:Solid
    Peso molecular:249.27
  • Osoresnontrine

    CAS:
    <p>Osoresnontrine is a potent and selective inhibitor of PDE9A (IC50 of 52 nM),and can be used in the research of memory.</p>
    Fórmula:C16H17N5O2
    Pureza:99.93%
    Cor e Forma:Solid
    Peso molecular:311.34
  • GW3965 hydrochloride

    CAS:
    <p>GW3965 hydrochloride (GW3965 HCl) is an effective and specific LXR agonist for hLXRα/β (EC50: 190/30 nM).</p>
    Fórmula:C33H31ClF3NO3·HCl
    Pureza:98.9% - 99.51%
    Cor e Forma:Solid
    Peso molecular:618.51
  • PDM2

    CAS:
    <p>PDM 2 is a potent and selective aryl hydrocarbon receptor (AhR) antagonist.</p>
    Fórmula:C14H9Cl3
    Pureza:99.44%
    Cor e Forma:Solid
    Peso molecular:283.58
  • WWL70

    CAS:
    <p>WWL70 is a selective alpha/beta hydrolase domain 6 inhibitors (IC50: 70 nM).</p>
    Fórmula:C27H23N3O3
    Pureza:98.38% - 98.53%
    Cor e Forma:Solid
    Peso molecular:437.49
  • Verdiperstat

    CAS:
    <p>Verdiperstat (AZD 3241) is a selective, irreversible, orally active myeloperoxidase inhibitor for neurodegenerative brain diseases.</p>
    Fórmula:C11H15N3O2S
    Pureza:99.36%
    Cor e Forma:Solid
    Peso molecular:253.32
  • A939572

    CAS:
    <p>A939572 is stearoyl-CoA desaturase1 (SCD1) inhibitor with IC50 values of &lt;4 nM for mSCD1 and 37 nM for hSCD1.</p>
    Fórmula:C20H22ClN3O3
    Pureza:99.96% - ≥95%
    Cor e Forma:Solid
    Peso molecular:387.86
  • VY-3-135

    CAS:
    <p>VY-3-135 is an orally active, stable and specific acetyl-CoA synthetase 2 (ACSS2) inhibitor.Cost-effective and quality-assured.</p>
    Fórmula:C26H27N3O3
    Pureza:99.25% - 99.79%
    Cor e Forma:Solid
    Peso molecular:429.51
  • Barnidipine hydrochloride

    CAS:
    <p>Barnidipine HCl is a potent dihydropyridine Ca²⁺ blocker with 0.35 nM IC50 in pig coronary artery.</p>
    Fórmula:C27H30ClN3O6
    Pureza:99.88%
    Cor e Forma:Solid
    Peso molecular:528
  • Betrixaban hydrochloride(330942-05-7(free base))


    <p>Betrixaban hydrochloride(330942-05-7(free base)) (PRT054021 hydrochloride) is a potent, selective, and orally efficacious factor Xa (fXa) inhibitor (IC50: 1.5</p>
    Fórmula:C23H23Cl2N5O3
    Pureza:99.54%
    Cor e Forma:Solid
    Peso molecular:488.36
  • Pyridaben

    CAS:
    <p>Pyridaben is a METI acaricide that inhibits mitochondrial electron transport at complex I (METI; Ki = 0.36 nmol/mg protein in rat brain mitochondria).</p>
    Fórmula:C19H25ClN2OS
    Pureza:97.11% - 99.75%
    Cor e Forma:Solid
    Peso molecular:364.93
  • Tuna AI acetate


    <p>Tuna AI acetate is an inhibitor of angiotensin-converting enzyme (ACE) in non-competitive manner derived from tuna muscle.</p>
    Fórmula:C46H68N12O14
    Pureza:98.49%
    Cor e Forma:Solid
    Peso molecular:1013.1
  • Dichlorphenamide

    CAS:
    <p>Dichlorphenamide (Diclofenamide) is a carbonic anhydrase inhibitor that is used in the treatment of glaucoma.</p>
    Fórmula:C6H6Cl2N2O4S2
    Pureza:96.87% - 97.25%
    Cor e Forma:Needles From Dimethylsulfoxide + Water Solid
    Peso molecular:305.16
  • Ziritaxestat

    CAS:
    <p>Ziritaxestat (GLPG1690), an autotaxin inhibitor, currently being evaluated in an exploratory phase 2 study in idiopathic pulmonary fibrosis patients.</p>
    Fórmula:C30H33FN8O2S
    Pureza:97% - 99.85%
    Cor e Forma:Solid
    Peso molecular:588.7
  • TEPP-46

    CAS:
    <p>TEPP-46 (ML265) is an activator of pyruvate kinase M2 (PKM2), selective for PKM1, PKL and PKR. TEPP-46 has antitumor activity. Cost-effective and quality-assured.</p>
    Fórmula:C17H16N4O2S2
    Pureza:98.21% - 98.77%
    Cor e Forma:Solid
    Peso molecular:372.46
  • Tipifarnib

    CAS:
    <p>Tipifarnib (IND 58359), a quinolinone, inhibits farnesyl transferase, blocks Ras activation, arrests cell growth, and curbs angiogenesis.</p>
    Fórmula:C27H22Cl2N4O
    Pureza:97.1% - 99.22%
    Cor e Forma:Off-White To Pale Beige Solid
    Peso molecular:489.4
  • Fabomotizole hydrochloride

    CAS:
    <p>Fabomotizole hydrochloride (CM346 hydrochloride) 是一种具有抗焦虑和神经保护作用的化合物。</p>
    Fórmula:C15H22ClN3O2S
    Pureza:99.54% - >99.99%
    Cor e Forma:Solid
    Peso molecular:343.87
  • PHD-1-IN-1

    CAS:
    <p>PHD-1-IN-1 is a potent inhibitor of hypoxia-inducible factor prolylhydroxylase domain-1 (PHD-1) enzyme(IC50 = 0.034 μM).</p>
    Fórmula:C13H8N4
    Pureza:99.74%
    Cor e Forma:Solid
    Peso molecular:220.23
  • Sacubitril hemicalcium salt

    CAS:
    <p>Sacubitril hemicalcium salt (AHU377 calcium salt) is a potent NEP inhibitor with an IC50 of 5 nM.</p>
    Fórmula:C48H56CaN2O10
    Pureza:99.86% - 99.93%
    Cor e Forma:Solid
    Peso molecular:861.06
  • Inosine

    CAS:
    <p>Inosine (NSC-20262), an endogenous purine nucleoside produced by the catabolism of adenosine, is an agonist of adenosine receptors A1R and A2AR. Low-Cost!</p>
    Fórmula:C10H12N4O5
    Pureza:99.51% - 99.89%
    Cor e Forma:Solid
    Peso molecular:268.23
  • Bay K 8644

    CAS:
    <p>Bay K 8644 (SQ 28,873) is a potent, selective activator of L-type Ca2+ channel with IC50 of 17.3 nM.</p>
    Fórmula:C16H15F3N2O4
    Pureza:99.41%
    Cor e Forma:Yellow Powder
    Peso molecular:356.3
  • Glyco-Obeticholic acid

    CAS:
    <p>Glyco-Obeticholic acid is an active metabolite of Obeticholic acid. Obeticholic acid is an agonist of the farnesoid X receptor (FXR).</p>
    Fórmula:C28H47NO5
    Pureza:99.77% - 99.95%
    Cor e Forma:Solid
    Peso molecular:477.68
  • 2,3-dihydro-1H-indene-5-sulfonamide

    CAS:
    <p>2,3-dihydro-1H-indene-5-sulfonamide is Carbonic anhydrase 12 (human) inhibitor.</p>
    Fórmula:C9H11NO2S
    Pureza:99.89%
    Cor e Forma:Solid
    Peso molecular:197.25
  • YM-750

    CAS:
    <p>YM-750 is a potent inhibitor of acyl-CoA:cholesterol acyltransferase (ACAT), with an IC50 value of 0.18 μM.</p>
    Fórmula:C31H36N2O
    Pureza:99.96%
    Cor e Forma:Solid
    Peso molecular:452.63
  • Tuftsin 3TFA

    CAS:
    <p>Tuftsin 3TFA is a tetrapeptide. It is a macrophage/microglial activator.</p>
    Fórmula:C27H43F9N8O12
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:842.66
  • 4-Amino-6-(trifluoromethyl)benzene-1,3-disulfonamide

    CAS:
    <p>4-Amino-6-(trifluoromethyl)benzene-1,3-disulfonamide (4-Amino-6-(trifluoromethyl)benzene-1,3-d) is a carbonic anhydrase inhibitor, used as a potential anti-</p>
    Fórmula:C7H8F3N3O4S2
    Pureza:98.58%
    Cor e Forma:Solid
    Peso molecular:319.28
  • (R)-3-Hydroxy-4,4-dimethyldihydrofuran-2(3H)-one

    CAS:
    <p>Pantolactone belongs to the class of organic compounds known as gamma-butyrolactones. gamma-Butyrolactones are compounds containing a gamma-butyrolactone moiety, which consists of an aliphatic five-member ring with four carbon atoms, one oxygen atom, and </p>
    Fórmula:C6H10O3
    Pureza:99.41%
    Cor e Forma:White Crystalline Powder Or Crystals
    Peso molecular:130.14
  • BMS-779788

    CAS:
    <p>BMS-779788 (XL-652) is an LXRα/β partial agonist (IC50: 68/14 nM).</p>
    Fórmula:C28H29ClN2O3S
    Pureza:98.65% - 99.24%
    Cor e Forma:Solid
    Peso molecular:509.06
  • Ziconotide Acetate (107452-89-1 free base)

    CAS:
    <p>Ziconotide Acetate (Prialt, 107452-89-1) is an analgesic for neuropathic pain, acting on N-type calcium channels to block pain signals.</p>
    Fórmula:C102H172N36O32S7
    Pureza:99.52% - 99.87%
    Cor e Forma:Solid
    Peso molecular:2639.2
  • Nepicastat hydrochloride

    CAS:
    <p>Nepicastat hydrochloride (RS-25560-197 hydrochloride) is a selective, orally active, dopamine-beta-hydroxylase inhibitor that crosses the blood-brain barrier.</p>
    Fórmula:C14H15F2N3S·HCl
    Pureza:98.35% - 99.74%
    Cor e Forma:Solid
    Peso molecular:331.81
  • Nicardipine

    CAS:
    Nicardipine (Cardene), a calcium channel blockers belonging to the dihydropyridine class, is a drug used to treat angina and high blood pressure.
    Fórmula:C26H29N3O6
    Pureza:99.56%
    Cor e Forma:Solid
    Peso molecular:479.52
  • Enoxaparin sodium

    CAS:
    <p>Enoxaparin, a low-weight heparin approved by FDA for STEMI, enhances antithrombin and prevents clotting by inhibiting factors XIa, IXa, Xa, IIa.</p>
    Fórmula:C42H59N3Na4O35S2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:1322
  • GSK256066

    CAS:
    <p>GSK256066 is a selective PDE4B(equal affinity to isoforms A-D) inhibitor with IC50 of 3.2 pM, &gt;380, 000-fold selectivity versus PDE1/2/3/5/6 and &gt;2500-fold</p>
    Fórmula:C27H26N4O5S
    Pureza:99.60% - 99.66%
    Cor e Forma:Solid
    Peso molecular:518.58
  • Clinofibrate

    CAS:
    <p>Clinofibrate lowers lipids, blocks HMGCR (IC50: 0.47 mM), and controls cholesterol/triacylglycerides.</p>
    Fórmula:C28H36O6
    Pureza:>99.99%
    Cor e Forma:White Crystalline Powder
    Peso molecular:468.58
  • Eprobemide

    CAS:
    <p>Eprobemide (LIS 630) is a non-competitive reversible inhibitor of monoamine oxidase A (MAO-A).</p>
    Fórmula:C14H19ClN2O2
    Pureza:99.83%
    Cor e Forma:Solid
    Peso molecular:282.77
  • Calcineurin Autoinhibitory Peptide acetate


    <p>Calcineurin Autoinhibitory Peptide acetate is a selectivecalcineurin phosphatase inhibitor(IC50 ~ 10 μM).</p>
    Fórmula:C252H417N78O82S4
    Pureza:97.24%
    Cor e Forma:Solid
    Peso molecular:5979.74
  • SR1078

    CAS:
    <p>SR1078 is an agonist of retinoic acid receptor-related orphan receptor (ROR)α/γ.</p>
    Fórmula:C17H10F9NO2
    Pureza:99.58%
    Cor e Forma:Solid
    Peso molecular:431.25
  • EBPC

    CAS:
    <p>EBPC is an inhibitor of aldose reductase.</p>
    Fórmula:C14H15NO4
    Pureza:99.55%
    Cor e Forma:Solid
    Peso molecular:261.27