
Metabolismo
Os inibidores do metabolismo são compostos que interferem nas vias metabólicas, alterando a produção e utilização de energia dentro das células. Esses inibidores são usados para estudar a regulação do metabolismo, o papel das vias metabólicas em doenças como o câncer e o diabetes, e para desenvolver novas estratégias terapêuticas. Os inibidores do metabolismo podem direcionar várias enzimas e processos envolvidos na glicólise, na oxidação de ácidos graxos e em outras funções metabólicas. Na CymitQuimica, oferecemos uma ampla gama de inibidores do metabolismo de alta qualidade para apoiar sua pesquisa em bioquímica, distúrbios metabólicos e desenvolvimento de medicamentos.
Subcategorias de "Metabolismo"
- AhR(41 produtos)
- Aminopeptidase(67 produtos)
- CETP(18 produtos)
- Anidrase carbónica(177 produtos)
- Caseína quinase(130 produtos)
- DHFR(32 produtos)
- Descarboxilase(4 produtos)
- Desidrogenase(267 produtos)
- FAAH(63 produtos)
- FXR(58 produtos)
- Factor Xa(80 produtos)
- Sintase de Ácidos graxos(32 produtos)
- Ferroptose(215 produtos)
- GR(3 produtos)
- GSNOR(3 produtos)
- Glucoquinase(53 produtos)
- HIF/HIF Prolil-Hidroxilase(142 produtos)
- HMG-CoA Reductase(32 produtos)
- Hidroxilase(30 produtos)
- IDO(82 produtos)
- LDL(8 produtos)
- Lipase(96 produtos)
- Lipídio(59 produtos)
- Lipoxigenase(124 produtos)
- MAO(87 produtos)
- MPO(2 produtos)
- NAMPT(36 produtos)
- P450(6 produtos)
- PAI-1(25 produtos)
- PDE(166 produtos)
- PED(1 produtos)
- PKM(15 produtos)
- PPAR(164 produtos)
- Fosfolipase(82 produtos)
- ROR(42 produtos)
- Receptor de Retinóide(29 produtos)
- SGK(11 produtos)
- Tiorredoxina(12 produtos)
- Transferase(30 produtos)
- Tansportador(42 produtos)
- UGT(4 produtos)
- Inibidores de Xantina Oxidase (XO)(9 produtos)
Exibir 34 mais subcategorias
Foram encontrados 8595 produtos de "Metabolismo"
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ZK824190 hydrochloride
CAS:<p>ZK824190 hydrochloride, an oral selective uPA inhibitor (IC50: 237 nM), also inhibits tPA (1600 nM) and Plasmin (1850 nM), used in multiple sclerosis research.</p>Fórmula:C22H21ClF2N2O4Cor e Forma:SolidPeso molecular:450.87β-Aminopropionitrile hydrochloride
CAS:<p>β-Aminopropionitrile hydrochloride is a selective, oral, irreversible inhibitor of lysyl oxidase (LOX) that reduces metastatic seeding potential.</p>Fórmula:C3H7ClN2Pureza:99.32%Cor e Forma:SolidPeso molecular:106.55PF-8380
CAS:<p>PF-8380 is an effective and orally available autotaxin inhibitor (IC50: 2.8 nM, in isolated enzyme assay; 101 nM, in the human whole blood).</p>Fórmula:C22H21Cl2N3O5Pureza:98.70% - 99.25%Cor e Forma:SolidPeso molecular:478.33MLCK inhibitor peptide 18 acetate
<p>MLCK inhibitor peptide 18 acetate: Selective (IC50=50nM), 4000x more than CaM kinase II. Does not block PKA. Cell-permeable.</p>Fórmula:C62H109N23O13Pureza:99.57%Cor e Forma:SolidPeso molecular:1384.67Nanterinone mesylate
CAS:<p>Nanterinone Mesylate is the mesylate form of Nanterinone that is a novel positive inotropic and balanced vasodilator.</p>Fórmula:C16H19N3O4SCor e Forma:SolidPeso molecular:349.421-deacetyldeflazacort
CAS:<p>21-deacetyldeflazacort is a metabolite of Deflazacort, which is a systemic corticosteroid and a derivative of prednisolone.</p>Fórmula:C23H29NO5Pureza:99.96%Cor e Forma:SolidPeso molecular:399.486-Hydroxy-4-methylcoumarin
CAS:<p>6-Hydroxy-4-methylcoumarin (6-Hydroxy-4-Methyl-2H-Chromen-2-One) is a secondary metabolite of coumarin, which has anticancer effects.</p>Fórmula:C10H8O3Pureza:98.93%Cor e Forma:SolidPeso molecular:176.17WWL229
CAS:<p>WWL229 selectively inhibits Ces3 without affecting Ces1f, ABHD6, or other serine hydrolases, mimicking WWL113 in adipocytes.</p>Fórmula:C16H22N2O5Pureza:98.14%Cor e Forma:SolidPeso molecular:322.36Linrodostat mesylate
CAS:<p>Linrodostat (BMS-986205) is an oral IDO1 inhibitor that boosts immune response and has anti-cancer properties.</p>Fórmula:C25H28ClFN2O4SPureza:98%Cor e Forma:SolidPeso molecular:507.02CP-640186
CAS:<p>CP-640186 is an isozyme-nonselective ACCase inhibitor. The IC50s of CP-640186 is 53 nM and 61 nM for rat liver ACC1 and rat skeletal muscle ACC2 respectively.</p>Fórmula:C30H35N3O3Pureza:99.87%Cor e Forma:SolidPeso molecular:485.62Mibefradil dihydrochloride
CAS:<p>Mibefradil dihydrochloride (Ro 40-5967 (dihydrochloride)) is an blocker of calcium channel with moderate selectivity for T-type Ca2+ channels (T-type and L-type</p>Fórmula:C29H40Cl2FN3O3Pureza:99.45% - 99.72%Cor e Forma:SolidPeso molecular:568.557-Ethoxy-4-Methylcoumarin
CAS:<p>7-Ethoxy-4-Methylcoumarin: fragrant, organic, enzyme inhibitor; used in drug effect studies.</p>Fórmula:C12H12O3Pureza:99.50%Cor e Forma:SolidPeso molecular:204.22MK-8245
CAS:<p>MK-8245 is a liver-targeting SCD inhibitor for human SCD1 (IC50: 1 nM) and for rat/mouse SCD1 (IC50: 3 nM), with anti-diabetic and anti-dyslipidemic function.</p>Fórmula:C17H16BrFN6O4Pureza:97.58% - 99%Cor e Forma:SolidPeso molecular:467.25Indoximod
CAS:<p>Indoximod (NLG-8189) is a methylated tryptophan that inhibits IDO to boost T cell function by preventing tryptophan depletion.</p>Fórmula:C12H14N2O2Pureza:97.82% - 99.55%Cor e Forma:SolidPeso molecular:218.256-Aminonicotinamide
CAS:<p>6-Aminonicotinamide (6-AN) is a well-established inhibitor of the NADP+-dependent enzyme.</p>Fórmula:C6H7N3OPureza:98.99% - 99.4%Cor e Forma:Physical Description White Crystalline Solid (Ntp 1992)Peso molecular:137.14ABT-639
CAS:<p>ABT-639 is a potent and selective T-type calcium channel blocker.</p>Fórmula:C20H20ClF2N3O3SPureza:99.12% - 99.77%Cor e Forma:SolidPeso molecular:455.91Edoxaban hydrochloride
CAS:<p>Edoxaban (DU-176b) HCl: Oral, selective Factor Xa inhibitor, Ki 0.561 nM; prevents thromboembolic disease.</p>Fórmula:C24H31Cl2N7O4SCor e Forma:SolidPeso molecular:584.52L-778123 Dihydrochloride
CAS:<p>L-778123 blocks FPTase/GGPTase-I, halts Ki-Ras prenylation, has acceptable toxicity with radiotherapy in advanced pancreatic cancer.</p>Fórmula:C22H22Cl3N5OCor e Forma:SolidPeso molecular:478.802Gcase activator 1
CAS:<p>Gcase activator 1 (LTI-291) is a glucocerebrosidase (Gcase) activator.</p>Fórmula:C20H30N4O2Pureza:99.25% - 99.31%Cor e Forma:SolidPeso molecular:358.48(E)-2-Decenoic acid
CAS:<p>(E)-2-Decenoic acid (trans-2-Decenoic acid) is an unsaturated fatty acid found in royal jelly produced from the mandibular gland secretions of honeybees.</p>Fórmula:C10H18O2Pureza:98%Cor e Forma:SolidPeso molecular:170.25Alkaline Phosphatase
CAS:<p>Alkaline phosphatase is a membrane-bound glycoprotein that catalyzes the hydrolysis of phosphate monoesters under alkaline conditions. High-Quality, Low-Cost!</p>Pureza:≥98%Cor e Forma:SolidPeso molecular:N/ABrinzolamide hydrochloride
<p>Brinzolamide (AL-4862) HCl selectively inhibits carbonic anhydrase II, reducing IOP for glaucoma research. IC50: 3.2 nM.</p>Cor e Forma:Solid4-methyl-2-(4-(trifluoromethyl)phenyl)thiazole-5-carboxylic acid
CAS:<p>4-methyl-2-(4-(trifluoromethyl)phenyl)thiazole-5-carboxylic acid is used as a pharmaceutical intermediate.</p>Fórmula:C12H8F3NO2SPureza:99.35%Cor e Forma:SolidPeso molecular:287.26Crisaborole
CAS:<p>Crisaborole (AN-2728) is a Phosphodiesterase 4 Inhibitor.</p>Fórmula:C14H10BNO3Pureza:99.70%Cor e Forma:SolidPeso molecular:251.052,3-dihydroxy-3-methylbutanoic acid
CAS:<p>2,3-dihydroxy-3-methylbutanoic acid, a leucine metabolite, boosts muscle growth by activating mTOR.</p>Fórmula:C5H10O4Pureza:99.03%Cor e Forma:SolidPeso molecular:134.1305AKR1C3-IN-1
CAS:<p>AKR1C3-IN-1 is a potent and selective inhibitor of AKR1C3(IC50 of 13 nM).</p>Fórmula:C16H15NO4SPureza:98.02%Cor e Forma:SolidPeso molecular:317.36sun
CAS:<p>Sun(4H-Furo[3,2-b]pyrrole-5-carboxylic acid) is an orally active and potent inhibitor of DAAO (DAO)</p>Fórmula:C7H5NO3Pureza:99.61%Cor e Forma:SolidPeso molecular:151.12Aldicarb sulfone
CAS:<p>Aldicarb sulfone is a cholinesterase inhibitor .</p>Fórmula:C7H14N2O4SPureza:99.05%Cor e Forma:Aldicarb Sulfone Is A White Crystalline Solid InsecticidePeso molecular:222.26SPI-112
CAS:<p>SPI-112, the SPI-112 methyl ester analog, can inhibit cellular Shp2 PTP activity.</p>Fórmula:C22H17FN4O5SPureza:97.51% - >99.99%Cor e Forma:SolidPeso molecular:468.46Navoximod
CAS:<p>Navoximod (GDC-0919) (NLG- 919, GDC-0919) is a potent indoleamine-(2,3)-dioxygenase (IDO) pathway inhibitor (Ki/EC50: 7 nM/75 nM).</p>Fórmula:C18H21FN2O2Pureza:99.37%Cor e Forma:SolidPeso molecular:316.37SR 16832
CAS:<p>SR 16832: Dual-site PPARγ inhibitor; outperforms GW 9662, T 0070907 in ligand binding, transcription inhibition.</p>Fórmula:C17H12ClN3O4Pureza:99.6%Cor e Forma:SolidPeso molecular:357.75Carbutamide
CAS:<p>Carbutamide is a sulfonylurea antidiabetic agent with hypoglycemic activity.</p>Fórmula:C11H17N3O3SPureza:98.77%Cor e Forma:Crystals SolidPeso molecular:271.34Fatostatin
CAS:<p>Fatostatin inhibits SREBP-1/2 by binding to SCAP, blocking their ER-Golgi transport.</p>Fórmula:C18H18N2SPureza:99.92%Cor e Forma:SolidPeso molecular:294.41Vardenafil hydrochloride trihydrate
CAS:<p>Vardenafil hydrochloride trihydrate (BAY38-9456) is a new type PDE inhibitor with IC50 of 0.7 and 180 nM for PDE5 and PDE1, respectively.</p>Fórmula:C23H32N6O4S·HCl·3H2OPureza:99.77%Cor e Forma:SolidPeso molecular:579.11NSC-226572
CAS:<p>NSC-226572, a synthetic alliin analog from cruciferous veggies, turns into thiosulfinate via alliinase.</p>Fórmula:C4H9NO3SPureza:99.48%Cor e Forma:SolidPeso molecular:151.18G6PDi-1
CAS:<p>G6PDi-1 is an effective G6PD inhibitor. It depletes NADPH and decreases inflammatory cytokine production.</p>Fórmula:C14H12N4OSPureza:98.69%Cor e Forma:SolidPeso molecular:284.34Piclamilast
CAS:<p>Piclamilast (RP 73401) is a PDE4 inhibitor.</p>Fórmula:C18H18Cl2N2O3Pureza:98.28% - 99.57%Cor e Forma:SolidPeso molecular:381.25Zolamide
CAS:<p>Zolamide (CL 5343) may be used to prevent altitude sickness and reduce the symptoms.</p>Fórmula:C2H4N4O2S2Pureza:99.75%Cor e Forma:SolidPeso molecular:180.21Zinc Phytate
CAS:<p>Zinc Phytate, present in food, plays a crucial role in human nutrient absorption.</p>Fórmula:C6H6O24P6Zn6Pureza:98%Cor e Forma:SolidPeso molecular:1040Fmoc-Gly-Thr(psi(Me,Me)pro)-OH
CAS:<p>Fmoc-Gly-Thr(psi(Me,Me)pro)-OH is a polypeptide composed of two amino acids.</p>Fórmula:C24H26N2O6Pureza:97.35%Cor e Forma:SolidPeso molecular:438.47ML-211
CAS:<p>ML-211 is a carbamate-based dual inhibitor of LYPLA1 (IC50 = 17 nM) and the related LYPLA2 (IC50 = 30 nM)</p>Fórmula:C25H30N4O2Pureza:97.07%Cor e Forma:SolidPeso molecular:418.531-phenyl-3,4-dihydroisochinoline
CAS:<p>1-phenyl-3,4-dihydroisochinoline: dopamine analog, interacts with CNS receptors, studied for Parkinson's, Alzheimer's, and Huntington's.</p>Fórmula:C15H13NPureza:98.01%Cor e Forma:SolidPeso molecular:207.27O-Succinylhomoserine
CAS:<p>O-Succinylhomoserine (O-Succinyl-L-homoserine) is an intermediate in the synthesis of cystathionine by E coli..</p>Fórmula:C8H13NO6Pureza:≥98%Cor e Forma:SolidPeso molecular:219.19L(+)-Leucinol
CAS:<p>L(+)-Leucinol is a potent inhibitor of leucine aminopeptidase.</p>Fórmula:C6H15NOPureza:98%Cor e Forma:Clear Colorless To Slightly Yellow LiquidPeso molecular:117.193-METHOXY-DL-TYROSINE
CAS:<p>3-Methoxy-DL-Tyrosine: natural, non-essential amino, precursor to dopamine, may aid in treating Parkinson's, depression, obesity.</p>Fórmula:C10H13NO4Pureza:99.90%Cor e Forma:SolidPeso molecular:211.21LXR-623
CAS:<p>LXR-623 (WAY 252623) is an orally bioavailable and highly specifical synthetic modulator of LXR.</p>Fórmula:C21H12ClF5N2Pureza:97.91% - 99.24%Cor e Forma:SolidPeso molecular:422.78BVT 2733
CAS:<p>BVT 2733 is a new, non-steroidal, isoform-specific inhibitor of 11β-HSD1.</p>Fórmula:C17H21ClN4O3S2Pureza:98% - 99.64%Cor e Forma:SolidPeso molecular:428.96Dimethyl DL-Glutamate (hydrochloride)
CAS:<p>Dimethyl DL-glutamate boosts insulin release in response to glucose.</p>Fórmula:C7H14ClNO4Pureza:≥95%Cor e Forma:SolidPeso molecular:211.64GW0742
CAS:<p>GW0742 (GW610742) is an effective and specific PPARδ agonist (EC50: 1 nM/1.1 μM/2 μM, for human PPARδ/α/γ).</p>Fórmula:C21H17F4NO3S2Pureza:99.75% - 99.85%Cor e Forma:SolidPeso molecular:471.49RGX-104 hydrochloride
CAS:<p>RGX-104 hydrochloride (SB742881) is a small molecule LXR agonist that regulates innate immunity using transcriptional activation of the ApoE gene.</p>Fórmula:C34H34Cl2F3NO3Pureza:99.49%Cor e Forma:SolidPeso molecular:632.54Mildronate
CAS:<p>Mildronate (Meldonium) is an inhibitor of biosynthesis of L-carnitine by gamma-butyrobetaine (GBB) hydroxylase and as a competitive inhibitor of renal carnitine</p>Fórmula:C6H14N2O2Pureza:99.94%Cor e Forma:White Crystalline PowderPeso molecular:146.19SU0268
CAS:<p>SU0268 is a potent and specific 8-Oxoguanine DNA glycosylase 1 (OGG1) inhibitor.</p>Fórmula:C26H25N3O4SPureza:99.97% - 99.98%Cor e Forma:SolidPeso molecular:475.56N-Valyltryptophan
CAS:<p>N-Valyltryptophan (Val-trp) is an incomplete breakdown product of protein catabolism or protein digestion.</p>Fórmula:C16H21N3O3Pureza:97.52%Cor e Forma:SolidPeso molecular:303.36Epacadostat
CAS:<p>Epacadostat (INCB 024360) is an oral, potent and selective IDO1 inhibitor with IC50 value of 71.8 nM.Cost-effective and quality-assured.</p>Fórmula:C11H13BrFN7O4SPureza:98% - >99.99%Cor e Forma:SolidPeso molecular:438.23Levofloxacin N-oxide
CAS:<p>Levofloxacin N-oxide is an impurity isolated from levofloxacin.</p>Fórmula:C18H20FN3O5Pureza:99.84%Cor e Forma:SolidPeso molecular:377.372-Hydroxycaprylic acid
CAS:<p>2-Hydroxycaprylic acid (2-hydroxyoctanoic acid) belongs to the class of organic compounds known as medium-chain fatty acids.</p>Fórmula:C8H16O3Pureza:98% - 99.84%Cor e Forma:SolidPeso molecular:160.21DMOG
CAS:<p>DMOG (Dimethyloxalylglycine), an antagonist of the α-ketoglutarate cofactor, is an inhibitor for HIF prolyl hydroxylase.</p>Fórmula:C6H9NO5Pureza:80.23% - 99.98%Cor e Forma:SolidPeso molecular:175.14ML355
CAS:<p>ML355, a specific, effective 12-Lipoxygenase(12-LOX) inhibitors(IC50=0.34 μM), possess favorable ADME properties.</p>Fórmula:C21H19N3O4S2Pureza:98.02% - 98.2%Cor e Forma:SolidPeso molecular:441.52RS-25344
CAS:<p>RS-25344: a strong PDE4 blocker, curbs eosinophil movement, boosts sperm motility in vitro.</p>Fórmula:C19H13N5O4Pureza:98.98%Cor e Forma:SolidPeso molecular:375.34L-Homocystine
CAS:<p>Homocystine briefly forms before turning into cystathionine via vitamin B6; linked to schizophrenia and neural tube defects; folic acid lowers risk.</p>Fórmula:C8H16N2O4S2Pureza:99.79%Cor e Forma:SolidPeso molecular:268.35YM976
CAS:<p>YM976 is an orally active PDE4 inhibitor (IC50:2.2 nM)</p>Fórmula:C17H16ClN3OPureza:99.84%Cor e Forma:SolidPeso molecular:313.78UK-5099
CAS:<p>UK-5099 (PF-1005023) is a potent MPC inhibitor with an IC50 of 50 nM in rat heart mitochondria.</p>Fórmula:C18H12N2O2Pureza:97.39% - >99.99%Cor e Forma:SolidPeso molecular:288.3ML351
CAS:<p>ML351 is a potent and selective inhibitor of human 15-lipoxygenase-1 (15 LOX)(IC50: 200 nM).</p>Fórmula:C15H11N3OPureza:97.67%Cor e Forma:SolidPeso molecular:249.27Osoresnontrine
CAS:<p>Osoresnontrine is a potent and selective inhibitor of PDE9A (IC50 of 52 nM),and can be used in the research of memory.</p>Fórmula:C16H17N5O2Pureza:99.93%Cor e Forma:SolidPeso molecular:311.34GW3965 hydrochloride
CAS:<p>GW3965 hydrochloride (GW3965 HCl) is an effective and specific LXR agonist for hLXRα/β (EC50: 190/30 nM).</p>Fórmula:C33H31ClF3NO3·HClPureza:98.9% - 99.51%Cor e Forma:SolidPeso molecular:618.51PDM2
CAS:<p>PDM 2 is a potent and selective aryl hydrocarbon receptor (AhR) antagonist.</p>Fórmula:C14H9Cl3Pureza:99.44%Cor e Forma:SolidPeso molecular:283.58WWL70
CAS:<p>WWL70 is a selective alpha/beta hydrolase domain 6 inhibitors (IC50: 70 nM).</p>Fórmula:C27H23N3O3Pureza:98.38% - 98.53%Cor e Forma:SolidPeso molecular:437.49Verdiperstat
CAS:<p>Verdiperstat (AZD 3241) is a selective, irreversible, orally active myeloperoxidase inhibitor for neurodegenerative brain diseases.</p>Fórmula:C11H15N3O2SPureza:99.36%Cor e Forma:SolidPeso molecular:253.32A939572
CAS:<p>A939572 is stearoyl-CoA desaturase1 (SCD1) inhibitor with IC50 values of <4 nM for mSCD1 and 37 nM for hSCD1.</p>Fórmula:C20H22ClN3O3Pureza:99.96% - ≥95%Cor e Forma:SolidPeso molecular:387.86VY-3-135
CAS:<p>VY-3-135 is an orally active, stable and specific acetyl-CoA synthetase 2 (ACSS2) inhibitor.Cost-effective and quality-assured.</p>Fórmula:C26H27N3O3Pureza:99.25% - 99.79%Cor e Forma:SolidPeso molecular:429.51Barnidipine hydrochloride
CAS:<p>Barnidipine HCl is a potent dihydropyridine Ca²⁺ blocker with 0.35 nM IC50 in pig coronary artery.</p>Fórmula:C27H30ClN3O6Pureza:99.88%Cor e Forma:SolidPeso molecular:528Betrixaban hydrochloride(330942-05-7(free base))
<p>Betrixaban hydrochloride(330942-05-7(free base)) (PRT054021 hydrochloride) is a potent, selective, and orally efficacious factor Xa (fXa) inhibitor (IC50: 1.5</p>Fórmula:C23H23Cl2N5O3Pureza:99.54%Cor e Forma:SolidPeso molecular:488.36Pyridaben
CAS:<p>Pyridaben is a METI acaricide that inhibits mitochondrial electron transport at complex I (METI; Ki = 0.36 nmol/mg protein in rat brain mitochondria).</p>Fórmula:C19H25ClN2OSPureza:97.11% - 99.75%Cor e Forma:SolidPeso molecular:364.93Tuna AI acetate
<p>Tuna AI acetate is an inhibitor of angiotensin-converting enzyme (ACE) in non-competitive manner derived from tuna muscle.</p>Fórmula:C46H68N12O14Pureza:98.49%Cor e Forma:SolidPeso molecular:1013.1Dichlorphenamide
CAS:<p>Dichlorphenamide (Diclofenamide) is a carbonic anhydrase inhibitor that is used in the treatment of glaucoma.</p>Fórmula:C6H6Cl2N2O4S2Pureza:96.87% - 97.25%Cor e Forma:Needles From Dimethylsulfoxide + Water SolidPeso molecular:305.16Ziritaxestat
CAS:<p>Ziritaxestat (GLPG1690), an autotaxin inhibitor, currently being evaluated in an exploratory phase 2 study in idiopathic pulmonary fibrosis patients.</p>Fórmula:C30H33FN8O2SPureza:97% - 99.85%Cor e Forma:SolidPeso molecular:588.7TEPP-46
CAS:<p>TEPP-46 (ML265) is an activator of pyruvate kinase M2 (PKM2), selective for PKM1, PKL and PKR. TEPP-46 has antitumor activity. Cost-effective and quality-assured.</p>Fórmula:C17H16N4O2S2Pureza:98.21% - 98.77%Cor e Forma:SolidPeso molecular:372.46Tipifarnib
CAS:<p>Tipifarnib (IND 58359), a quinolinone, inhibits farnesyl transferase, blocks Ras activation, arrests cell growth, and curbs angiogenesis.</p>Fórmula:C27H22Cl2N4OPureza:97.1% - 99.22%Cor e Forma:Off-White To Pale Beige SolidPeso molecular:489.4Fabomotizole hydrochloride
CAS:<p>Fabomotizole hydrochloride (CM346 hydrochloride) 是一种具有抗焦虑和神经保护作用的化合物。</p>Fórmula:C15H22ClN3O2SPureza:99.54% - >99.99%Cor e Forma:SolidPeso molecular:343.87PHD-1-IN-1
CAS:<p>PHD-1-IN-1 is a potent inhibitor of hypoxia-inducible factor prolylhydroxylase domain-1 (PHD-1) enzyme(IC50 = 0.034 μM).</p>Fórmula:C13H8N4Pureza:99.74%Cor e Forma:SolidPeso molecular:220.23Sacubitril hemicalcium salt
CAS:<p>Sacubitril hemicalcium salt (AHU377 calcium salt) is a potent NEP inhibitor with an IC50 of 5 nM.</p>Fórmula:C48H56CaN2O10Pureza:99.86% - 99.93%Cor e Forma:SolidPeso molecular:861.06Inosine
CAS:<p>Inosine (NSC-20262), an endogenous purine nucleoside produced by the catabolism of adenosine, is an agonist of adenosine receptors A1R and A2AR. Low-Cost!</p>Fórmula:C10H12N4O5Pureza:99.51% - 99.89%Cor e Forma:SolidPeso molecular:268.23Bay K 8644
CAS:<p>Bay K 8644 (SQ 28,873) is a potent, selective activator of L-type Ca2+ channel with IC50 of 17.3 nM.</p>Fórmula:C16H15F3N2O4Pureza:99.41%Cor e Forma:Yellow PowderPeso molecular:356.3Glyco-Obeticholic acid
CAS:<p>Glyco-Obeticholic acid is an active metabolite of Obeticholic acid. Obeticholic acid is an agonist of the farnesoid X receptor (FXR).</p>Fórmula:C28H47NO5Pureza:99.77% - 99.95%Cor e Forma:SolidPeso molecular:477.682,3-dihydro-1H-indene-5-sulfonamide
CAS:<p>2,3-dihydro-1H-indene-5-sulfonamide is Carbonic anhydrase 12 (human) inhibitor.</p>Fórmula:C9H11NO2SPureza:99.89%Cor e Forma:SolidPeso molecular:197.25YM-750
CAS:<p>YM-750 is a potent inhibitor of acyl-CoA:cholesterol acyltransferase (ACAT), with an IC50 value of 0.18 μM.</p>Fórmula:C31H36N2OPureza:99.96%Cor e Forma:SolidPeso molecular:452.63Tuftsin 3TFA
CAS:<p>Tuftsin 3TFA is a tetrapeptide. It is a macrophage/microglial activator.</p>Fórmula:C27H43F9N8O12Pureza:>99.99%Cor e Forma:SolidPeso molecular:842.664-Amino-6-(trifluoromethyl)benzene-1,3-disulfonamide
CAS:<p>4-Amino-6-(trifluoromethyl)benzene-1,3-disulfonamide (4-Amino-6-(trifluoromethyl)benzene-1,3-d) is a carbonic anhydrase inhibitor, used as a potential anti-</p>Fórmula:C7H8F3N3O4S2Pureza:98.58%Cor e Forma:SolidPeso molecular:319.28(R)-3-Hydroxy-4,4-dimethyldihydrofuran-2(3H)-one
CAS:<p>Pantolactone belongs to the class of organic compounds known as gamma-butyrolactones. gamma-Butyrolactones are compounds containing a gamma-butyrolactone moiety, which consists of an aliphatic five-member ring with four carbon atoms, one oxygen atom, and </p>Fórmula:C6H10O3Pureza:99.41%Cor e Forma:White Crystalline Powder Or CrystalsPeso molecular:130.14BMS-779788
CAS:<p>BMS-779788 (XL-652) is an LXRα/β partial agonist (IC50: 68/14 nM).</p>Fórmula:C28H29ClN2O3SPureza:98.65% - 99.24%Cor e Forma:SolidPeso molecular:509.06Ziconotide Acetate (107452-89-1 free base)
CAS:<p>Ziconotide Acetate (Prialt, 107452-89-1) is an analgesic for neuropathic pain, acting on N-type calcium channels to block pain signals.</p>Fórmula:C102H172N36O32S7Pureza:99.52% - 99.87%Cor e Forma:SolidPeso molecular:2639.2Nepicastat hydrochloride
CAS:<p>Nepicastat hydrochloride (RS-25560-197 hydrochloride) is a selective, orally active, dopamine-beta-hydroxylase inhibitor that crosses the blood-brain barrier.</p>Fórmula:C14H15F2N3S·HClPureza:98.35% - 99.74%Cor e Forma:SolidPeso molecular:331.81Nicardipine
CAS:Nicardipine (Cardene), a calcium channel blockers belonging to the dihydropyridine class, is a drug used to treat angina and high blood pressure.Fórmula:C26H29N3O6Pureza:99.56%Cor e Forma:SolidPeso molecular:479.52Enoxaparin sodium
CAS:<p>Enoxaparin, a low-weight heparin approved by FDA for STEMI, enhances antithrombin and prevents clotting by inhibiting factors XIa, IXa, Xa, IIa.</p>Fórmula:C42H59N3Na4O35S2Pureza:98%Cor e Forma:SolidPeso molecular:1322GSK256066
CAS:<p>GSK256066 is a selective PDE4B(equal affinity to isoforms A-D) inhibitor with IC50 of 3.2 pM, >380, 000-fold selectivity versus PDE1/2/3/5/6 and >2500-fold</p>Fórmula:C27H26N4O5SPureza:99.60% - 99.66%Cor e Forma:SolidPeso molecular:518.58Clinofibrate
CAS:<p>Clinofibrate lowers lipids, blocks HMGCR (IC50: 0.47 mM), and controls cholesterol/triacylglycerides.</p>Fórmula:C28H36O6Pureza:>99.99%Cor e Forma:White Crystalline PowderPeso molecular:468.58Eprobemide
CAS:<p>Eprobemide (LIS 630) is a non-competitive reversible inhibitor of monoamine oxidase A (MAO-A).</p>Fórmula:C14H19ClN2O2Pureza:99.83%Cor e Forma:SolidPeso molecular:282.77Calcineurin Autoinhibitory Peptide acetate
<p>Calcineurin Autoinhibitory Peptide acetate is a selectivecalcineurin phosphatase inhibitor(IC50 ~ 10 μM).</p>Fórmula:C252H417N78O82S4Pureza:97.24%Cor e Forma:SolidPeso molecular:5979.74SR1078
CAS:<p>SR1078 is an agonist of retinoic acid receptor-related orphan receptor (ROR)α/γ.</p>Fórmula:C17H10F9NO2Pureza:99.58%Cor e Forma:SolidPeso molecular:431.25EBPC
CAS:<p>EBPC is an inhibitor of aldose reductase.</p>Fórmula:C14H15NO4Pureza:99.55%Cor e Forma:SolidPeso molecular:261.27

