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Metabolismo

Metabolismo

Os inibidores do metabolismo são compostos que interferem nas vias metabólicas, alterando a produção e utilização de energia dentro das células. Esses inibidores são usados para estudar a regulação do metabolismo, o papel das vias metabólicas em doenças como o câncer e o diabetes, e para desenvolver novas estratégias terapêuticas. Os inibidores do metabolismo podem direcionar várias enzimas e processos envolvidos na glicólise, na oxidação de ácidos graxos e em outras funções metabólicas. Na CymitQuimica, oferecemos uma ampla gama de inibidores do metabolismo de alta qualidade para apoiar sua pesquisa em bioquímica, distúrbios metabólicos e desenvolvimento de medicamentos.

Subcategorias de "Metabolismo"

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Foram encontrados 8626 produtos de "Metabolismo"

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  • L-Leucyl-L-Leucine methyl ester hydrochloride

    CAS:
    <p>L-Leucyl-L-Leucine methyl ester hydrochloride (Leu-Leu-ome hydrochloride) is a dipeptide condensation product of L-leucine methyl ester. Cost-effective and quality-assured.</p>
    Fórmula:C13H27ClN2O3
    Pureza:98.41% - 99.63%
    Cor e Forma:Solid
    Peso molecular:294.81
  • ETHYL 5-HYDROXY-2-METHYLINDOLE-3-CARBOXYLATE

    CAS:
    <p>ETHYL 5-HYDROXY-2-METHYLINDOLE-3-CARBOXYLATE is useful for preparation and study of hypoxia-selective cytotoxicity of indolequinone antitumor agents.</p>
    Fórmula:C12H13NO3
    Pureza:98.9%
    Cor e Forma:Off-White To Light Tan Crystalline Powder
    Peso molecular:219.24
  • FPH2

    CAS:
    <p>FPH2 (BRD-9424) (BRD-9424) is a small molecule promoting differentiation of iPS-derived hepatocytes.</p>
    Fórmula:C14H16ClN5O2S
    Pureza:>99.99% - >99.99%
    Cor e Forma:Solid
    Peso molecular:353.83
  • ML-211

    CAS:
    <p>ML-211 is a carbamate-based dual inhibitor of LYPLA1 (IC50 = 17 nM) and the related LYPLA2 (IC50 = 30 nM)</p>
    Fórmula:C25H30N4O2
    Pureza:97.07%
    Cor e Forma:Solid
    Peso molecular:418.53
  • RHC 80267

    CAS:
    <p>RHC 80267 (U-57908) is a selective inhibitor of DAGL (IC50 : 4 μM in canine platelets)</p>
    Fórmula:C20H34N4O4
    Pureza:99.54%
    Cor e Forma:White Solid
    Peso molecular:394.51
  • Alagebrium chloride

    CAS:
    <p>Alagebrium chloride (ALT711) inhibits AGEs, lowers systolic blood pressure, and benefits diastolic patients.</p>
    Fórmula:C13H14ClNOS
    Pureza:99.65% - 99.77%
    Cor e Forma:Solid
    Peso molecular:267.77
  • Edoxaban hydrochloride

    CAS:
    <p>Edoxaban (DU-176b) HCl: Oral, selective Factor Xa inhibitor, Ki 0.561 nM; prevents thromboembolic disease.</p>
    Fórmula:C24H31Cl2N7O4S
    Cor e Forma:Solid
    Peso molecular:584.52
  • Tebuconazole

    CAS:
    <p>Tebuconazole: azole fungicide, inhibits CYP51 with IC50s 0.9 μM (C. albicans) and 1.3 μM (human).</p>
    Fórmula:C16H22ClN3O
    Pureza:99.21%
    Cor e Forma:Solid
    Peso molecular:307.82
  • 1-phenyl-3,4-dihydroisochinoline

    CAS:
    1-phenyl-3,4-dihydroisochinoline: dopamine analog, interacts with CNS receptors, studied for Parkinson's, Alzheimer's, and Huntington's.
    Fórmula:C15H13N
    Pureza:98.01%
    Cor e Forma:Solid
    Peso molecular:207.27
  • Sacubitril

    CAS:
    <p>Sacubitril (AHU-377) is a potent NEP inhibitor with an IC50 of 5 nM. Sacubitril is a component of the heart failure medicine LCZ696.</p>
    Fórmula:C24H29NO5
    Pureza:97.72% - 97.91%
    Cor e Forma:Solid
    Peso molecular:411.49
  • MLCK inhibitor peptide 18 acetate


    <p>MLCK inhibitor peptide 18 acetate: Selective (IC50=50nM), 4000x more than CaM kinase II. Does not block PKA. Cell-permeable.</p>
    Fórmula:C62H109N23O13
    Pureza:99.57%
    Cor e Forma:Solid
    Peso molecular:1384.67
  • Amifostine trihydrate

    CAS:
    <p>Amifostine trihydrate (WR2721) is the first approved radioprotective drug, used to decrease the risk of kidney problems caused by treatment with cisplatin.</p>
    Fórmula:C5H15N2O3PS·3H2O
    Pureza:99.71% - 99.80%
    Cor e Forma:Solid
    Peso molecular:268.27
  • Nitecapone

    CAS:
    <p>Nitecapone is a reversible inhibitor of S-COMT (IC50 values of 300 nM in rat liver)</p>
    Fórmula:C12H11NO6
    Pureza:98.39%
    Cor e Forma:Solid
    Peso molecular:265.22
  • Haloxyfop

    CAS:
    <p>(±)-Haloxyfop (Haloxyfop Acid) is a herbicide.</p>
    Fórmula:C15H11ClF3NO4
    Pureza:99.94% - >99.99%
    Cor e Forma:Solid
    Peso molecular:361.7
  • Cilofexor

    CAS:
    <p>Cilofexor inhibits binding of a synthetic peptide, Cilofexor is a farnesoid X receptor (FXR) agonist.</p>
    Fórmula:C28H22Cl3N3O5
    Pureza:99.86% - ≥95%
    Cor e Forma:Solid
    Peso molecular:586.85
  • IOX4

    CAS:
    <p>IOX4 is a potent PHD2 inhibitor (IC50 = 1.6 nM)</p>
    Fórmula:C15H16N6O3
    Pureza:99.97%
    Cor e Forma:Solid
    Peso molecular:328.33
  • LXR-623

    CAS:
    <p>LXR-623 (WAY 252623) is an orally bioavailable and highly specifical synthetic modulator of LXR.</p>
    Fórmula:C21H12ClF5N2
    Pureza:97.91% - 99.24%
    Cor e Forma:Solid
    Peso molecular:422.78
  • PDE10-IN-1

    CAS:
    <p>PDE10-IN-1 (SEP-0372814) is used for treating CNS and metabolic disorders.</p>
    Fórmula:C21H19N7
    Pureza:99.65%
    Cor e Forma:Solid
    Peso molecular:369.42
  • AG-120 (racemic)

    CAS:
    <p>AG-120 (racemic) is an oral IDH1 inhibitor with potential anti-cancer effects.</p>
    Fórmula:C28H22ClF3N6O3
    Pureza:99.56%
    Cor e Forma:Solid
    Peso molecular:582.96
  • Olprinone

    CAS:
    <p>Olprinone (Loprinone)(Loprinone) is a selective phosphodiesterase 3 (PDE3) inhibitor.Olprinone has been reported to improve microcirculation and attenuate</p>
    Fórmula:C14H10N4O
    Pureza:99.68%
    Cor e Forma:Solid
    Peso molecular:250.26
  • Firsocostat

    CAS:
    <p>Firsocostat (GS-0976) is an inhibitor of acetyl-CoA carboxylase (ACC) dimerization that inhibits human ACC1 and ACC2 activity (IC50s of 2.1 and 6.1 nM).</p>
    Fórmula:C28H31N3O8S
    Pureza:98% - 98.46%
    Cor e Forma:Solid
    Peso molecular:569.63
  • Barnidipine

    CAS:
    <p>Barnidipine (YM-09730-5(Free base)) is a calcium channel blocker.</p>
    Fórmula:C27H29N3O6
    Pureza:99.98%
    Cor e Forma:Solid
    Peso molecular:491.54
  • Eliglustat

    CAS:
    <p>Eliglustat (Genz 99067) is an oral inhibitor of glucosylceramide synthase which is used in the therapy of type 1 Gaucher disease.</p>
    Fórmula:C23H36N2O4
    Pureza:99% - 99.70%
    Cor e Forma:Solid
    Peso molecular:404.54
  • Fexaramine

    CAS:
    <p>Fexaramine is a small molecule farnesoid X receptor (FXR) agonist with 100-fold increased affinity compared to natural compounds.</p>
    Fórmula:C32H36N2O3
    Pureza:98.87% - 99.61%
    Cor e Forma:Solid
    Peso molecular:496.64
  • DG172 dihydrochloride

    CAS:
    <p>DG172 dihydrochloride (DG-172 dihydrochloride) is an antagonist of PPARβ/δ(IC50 : 27 nM).</p>
    Fórmula:C20H22BrCl2N3
    Pureza:99.87%
    Cor e Forma:Solid
    Peso molecular:455.2
  • NCT-503

    CAS:
    <p>NCT-503 is a phosphoglycerate dehydrogenase (PHGDH) inhibitor with no activity against other dehydrogenases. NCT-503 has antitumor activity. Cost-effective and quality-assured.</p>
    Fórmula:C20H23F3N4S
    Pureza:98.91% - 99.84%
    Cor e Forma:Solid
    Peso molecular:408.48
  • BVT 2733

    CAS:
    <p>BVT 2733 is a new, non-steroidal, isoform-specific inhibitor of 11β-HSD1.</p>
    Fórmula:C17H21ClN4O3S2
    Pureza:98% - 99.64%
    Cor e Forma:Solid
    Peso molecular:428.96
  • NCT-501 hydrochloride

    CAS:
    <p>NCT-501 hydrochloride: potent, selective ALDH1A1 inhibitor based on theophylline; IC50 of 40 nM; highly discriminant against other ALDHs.</p>
    Fórmula:C21H33ClN6O3
    Cor e Forma:Solid
    Peso molecular:452.98
  • 3,4, 5-trimethoxyphenylacetic acid

    CAS:
    <p>3,4,5-trimethoxyphenylacetic acid: used in organic synthesis, mainly for carboxyl group conversion.</p>
    Fórmula:C11H14O5
    Pureza:99.84%
    Cor e Forma:White Crystalline Powder
    Peso molecular:226.23
  • ML348

    CAS:
    <p>ML348 (GNF-Pf-1127) is a selective and reversible lysophospholipase 1 (LYPLA1) inhibitor (IC50 = 210 nM).</p>
    Fórmula:C18H17ClF3N3O3
    Pureza:99% - 99.88%
    Cor e Forma:Solid
    Peso molecular:415.79
  • BIA 10-2474

    CAS:
    <p>BIA 10-2474 is a long-acting reversible inhibitor of FAAH that increases levels of the neurotransmitter anandamide in the nervous system.</p>
    Fórmula:C16H20N4O2
    Pureza:99.27%
    Cor e Forma:Solid
    Peso molecular:300.36
  • Nifursol

    CAS:
    <p>Nifursol is a livestock feed additive and antiobiotic used to prevent the growth of histomonas.</p>
    Fórmula:C12H7N5O9
    Pureza:97.18%
    Peso molecular:365.21
  • Enasidenib

    CAS:
    <p>Enasidenib (AG-221) is an orally available inhibitor of specific mutant forms of the mitochondrial enzyme isocitrate dehydrogenase type 2 (IDH2), with potential</p>
    Fórmula:C19H17F6N7O
    Pureza:98% - >99.99%
    Cor e Forma:Solid
    Peso molecular:473.38
  • 2,3-dihydrothieno-Thiadiazole Carboxylate

    CAS:
    <p>2,3-dihydrothieno-Thiadiazole Carboxylate is a CYP450 (CYP2E1 and CYP2B4) inhibitor.</p>
    Fórmula:C6H4N2O2S2
    Pureza:99.05%
    Cor e Forma:Solid
    Peso molecular:200.24
  • Tiplaxtinin

    CAS:
    <p>Tiplaxtinin (Tiplasinin)(PAI-039) is a selective and orally efficacious inhibitor of plasminogen activator inhibitor-1 (PAI-1) with IC50 of 2.7 uM.</p>
    Fórmula:C24H16F3NO4
    Pureza:99.16% - 99.93%
    Cor e Forma:Solid
    Peso molecular:439.38
  • BIM-46187 4HCl

    CAS:
    <p>BIM-46187 4HCl (PH-064 4HCl) is a heterotrimeric G-protein complex inhibitor.</p>
    Fórmula:C44H62Cl4N8O2S2
    Pureza:99.26% - 99.63%
    Cor e Forma:Solid
    Peso molecular:940.95
  • FEMA 4774

    CAS:
    <p>FEMA 4774 (S9632) is a positive allosteric modulator of T1R2/T1R3. FEMA4774 shows obvious enhancement of the sweetness of sucrose in sensory evaluation tests</p>
    Fórmula:C19H25N3O4
    Pureza:99.97%
    Cor e Forma:Solid
    Peso molecular:359.42
  • Perfluorooctanoic acid

    CAS:
    <p>Perfluorooctanoic acid (PFOA) (PFOA) is a persistent and widespread industry-made chemical.</p>
    Fórmula:C8HF15O2
    Pureza:99.70%
    Cor e Forma:White To Off-White Powder Othersolid
    Peso molecular:414.07
  • Nicardipine

    CAS:
    Nicardipine (Cardene), a calcium channel blockers belonging to the dihydropyridine class, is a drug used to treat angina and high blood pressure.
    Fórmula:C26H29N3O6
    Pureza:99.56%
    Cor e Forma:Solid
    Peso molecular:479.52
  • Lodenafil

    CAS:
    <p>Lodenafil (Hydroxyhomosildenafil) is a potent PDE5 inhibitor, with treatment of erectile dysfunction (ED)</p>
    Fórmula:C23H32N6O5S
    Pureza:99.92%
    Cor e Forma:Solid
    Peso molecular:504.6
  • Cedirogant

    CAS:
    <p>Cedirogant (ABBV-157) is an orally active retinoid-related orphan receptor-γt(RORγt) inverse agonist that is used for psoriasis study.</p>
    Fórmula:C24H20Cl3F3N2O3
    Pureza:99.20%
    Cor e Forma:Solid
    Peso molecular:547.78
  • BMS-303141

    CAS:
    <p>BMS-303141 is a potent ATP-citrate lyase (ACL) inhibitor (IC50: 0.13 uM, human recombinant ACL).</p>
    Fórmula:C19H15Cl2NO4S
    Pureza:98% - 99.47%
    Cor e Forma:Solid
    Peso molecular:424.3
  • 1-Naphthyl phosphate potassium salt

    CAS:
    <p>1-Naphthyl phosphate potassium salt inhibits non-specific phosphatase.</p>
    Fórmula:C10H7K2O4P
    Pureza:99%
    Cor e Forma:Solid
    Peso molecular:300.33
  • Cyclosporine

    CAS:
    <p>Cyclosporine is a calcineurin phosphatase pathway inhibitor, used as an immunosuppressant drug to prevent rejection in organ transplantation.</p>
    Fórmula:C62H111N11O12
    Pureza:99.68%
    Cor e Forma:White Powder
    Peso molecular:1202.61
  • 3PO

    CAS:
    <p>3PO inhibits PFKFB3 (IC50: 22.9 µM) and cancer cell growth (IC50: 1.4-24 µM), reducing glucose uptake and key cellular metabolites.</p>
    Fórmula:C13H10N2O
    Pureza:99.56% - 99.67%
    Cor e Forma:Solid
    Peso molecular:210.23
  • Tryptophan, N-indol-3-ylacetyl- (6CI)

    CAS:
    <p>Tryptophan, N-indol-3-ylacetyl- (6CI) (Indole-3-acetyl-L-tryptophan) is involved in regulatory mechanisms for the control of auxin activity during physiological</p>
    Fórmula:C21H19N3O3
    Pureza:99.55%
    Cor e Forma:Solid
    Peso molecular:361.4
  • TM5275 sodium

    CAS:
    <p>TM5275 sodium (TM5275 sodium salt) is an inhibitor of plasminogen activator inhibitor 1 (PAI-1).</p>
    Fórmula:C28H27ClN3NaO5
    Pureza:98.8% - 99.74%
    Cor e Forma:Solid
    Peso molecular:543.98
  • 3-Methylglutaric acid

    CAS:
    <p>Methylglutaric acid, a leucine byproduct, is linked to two metabolic disorders, detected in patient urine.</p>
    Fórmula:C6H10O4
    Pureza:98.64%
    Cor e Forma:Solid
    Peso molecular:146.14
  • CP671305

    CAS:
    <p>CP671305 is an orally active, potent and selective inhibitor of phosphodiesterase-4-D.</p>
    Fórmula:C23H19FN2O7
    Pureza:99.39%
    Cor e Forma:Solid
    Peso molecular:454.4
  • Enoximone

    CAS:
    <p>Enoximone is a selective inhibitor of phosphodiesterase III (PDE3), with treatment of congestive heart failure.</p>
    Fórmula:C12H12N2O2S
    Pureza:98.53%
    Cor e Forma:Solid
    Peso molecular:248.3
  • Isradipine

    CAS:
    <p>Isradipine (PN 200-110), a dihydropyridine, is an antihypertensive calcium channel blocker that dilates arteries and reduces resistance.</p>
    Fórmula:C19H21N3O5
    Pureza:99.84% - 99.95%
    Cor e Forma:Yellow Solid
    Peso molecular:371.39
  • Pentamidine dihydrochloride

    CAS:
    <p>Pentamidine dihydrochloride (MP-601205 dihydrochloride) is an aromatic diamidine agent with activity against a number of microorganisms including protozoa (</p>
    Fórmula:C19H26Cl2N4O2
    Pureza:99.80%
    Cor e Forma:Solid
    Peso molecular:413.34
  • THPP-1

    CAS:
    <p>THPP-1 is a potent and orally bioavailable inhibitor of PDE10A(Ki of 1 nM and 1.3 nM for human and rat PDE10A, respectively).</p>
    Fórmula:C23H21ClN6O3
    Pureza:99.46%
    Cor e Forma:Solid
    Peso molecular:464.9
  • Ethoxzolamide

    CAS:
    <p>Ethoxzolamide (L-643786) is a carbonic anhydrase inhibitor.</p>
    Fórmula:C9H10N2O3S2
    Pureza:98.27% - 99.62%
    Cor e Forma:Crystals From Ethyl Acetate + Skellysolve B Solid
    Peso molecular:258.32
  • 1-Stearoyl-2-arachidonoyl-sn-glycero-3-phosphocholine

    CAS:
    <p>1-Stearoyl-2-arachidonoyl-sn-glycero-3-phosphocholine is an endogenous metabolite that has been found in the aging mouse brain.</p>
    Fórmula:C46H84NO8P
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:810.13
  • n-acetylciprofloxacin

    CAS:
    <p>n-acetylciprofloxacin (3-Quinolinecarboxylic acid, 7-(4-acetyl-1-piperazinyl)-1-cyclopropyl-6-fluoro-1) is inhibitor of H37Rv.</p>
    Fórmula:C19H20FN3O4
    Pureza:99.83%
    Cor e Forma:Solid
    Peso molecular:373.38
  • Oroxylin A

    CAS:
    <p>Oroxylin A fights tumors, aids RAS therapy, promotes CaCo-2 cell apoptosis, blocks MCF-7 cell invasion and enhances leukemia treatment.</p>
    Fórmula:C16H12O5
    Pureza:98.72% - 99.55%
    Cor e Forma:Solid
    Peso molecular:284.26
  • YM-58483

    CAS:
    <p>YM-58483 (BTP2) is a specific and effective inhibitor of CRAC channels and subsequent Ca2+ signals.</p>
    Fórmula:C15H9F6N5OS
    Pureza:99.33% - 99.64%
    Cor e Forma:Solid
    Peso molecular:421.32
  • MAGL-IN-4

    CAS:
    <p>MAGL-IN-4 (His121 ARG57) is one of the monoacylglycerol lipase (MAGL) inhibitors in central nervous system-related diseases.</p>
    Fórmula:C18H21ClN2O4
    Pureza:99.79%
    Cor e Forma:Solid
    Peso molecular:364.82
  • Mitochondrial fusion promoter M1

    CAS:
    <p>Mitochondrial fusion promoter M1, a modulator of mitochondrial dynamics, enhances mitochondrial function and cellular respiration, and has shown efficacy in</p>
    Fórmula:C14H10Cl4N2O
    Pureza:99.54% - 99.54%
    Cor e Forma:Solid
    Peso molecular:364.05
  • Norathiol

    CAS:
    <p>Norathiol (N-methyl-N-dithiocarboxyglucamine) is a metal chelator that promotes the excretion of 109Cd and may be used in the treatment of cadmium poisoning.</p>
    Fórmula:C8H17NO5S2
    Cor e Forma:Solid
    Peso molecular:271.35
  • MCU-i4

    CAS:
    <p>MCU-i4 is a novel negative modulator of the MCU, binding MICU1 and impairing muscle cell growth.</p>
    Fórmula:C23H27N3O2
    Pureza:99.45% - 99.98%
    Cor e Forma:Solid
    Peso molecular:377.48
  • CTPI-2

    CAS:
    <p>CTPI-2 inhibits SLC25A1 (KD: 3.5 μM), glycolysis, PPARγ, GLUT4, has anti-tumor effects, and combats NASH and diet-induced obesity.</p>
    Fórmula:C13H9ClN2O6S
    Pureza:97.23%
    Cor e Forma:Solid
    Peso molecular:356.74
  • Bis(maltolato)oxovanadium(IV)

    CAS:
    <p>BMOV: oral pan-PTP inhibitor, mimics insulin, anti-diabetic, improves heart function in diabetes, IC50s: 126-201 nM.</p>
    Fórmula:C12H10O7V
    Pureza:99.65% - 99.918%
    Cor e Forma:Solid
    Peso molecular:317.15
  • Ponalrestat

    CAS:
    <p>Ponalrestat is an aldose reductase inhibitor.</p>
    Fórmula:C17H12BrFN2O3
    Pureza:97.34% - 99.86%
    Cor e Forma:Solid
    Peso molecular:391.19
  • PF-9601N

    CAS:
    <p>PF-9601N: potent, selective MAO-BI with neuroprotection in PD models.</p>
    Fórmula:C19H18N2O
    Pureza:98.29%
    Cor e Forma:Solid
    Peso molecular:290.36
  • Milacemide

    CAS:
    <p>Milacemide is a glycine prodrug and MAO-B inhibitor.</p>
    Fórmula:C7H16N2O
    Pureza:98.04%
    Cor e Forma:Solid
    Peso molecular:144.21
  • CAY10650

    CAS:
    <p>CAY10650 is an effective inhibitor of cytosolic phospholipase A2α (cPLA2α, IC50: 12 nM).</p>
    Fórmula:C28H25NO6
    Pureza:97.33%
    Cor e Forma:Solid
    Peso molecular:471.5
  • SGC-GAK-1

    CAS:
    <p>SGC-GAK-1 is a selective cyclin G-associated kinase (GAK) inhibitor (Ki: 3.1 nM).</p>
    Fórmula:C18H17BrN2O3
    Pureza:99.85%
    Cor e Forma:Solid
    Peso molecular:389.24
  • Lomerizine dihydrochloride

    CAS:
    <p>Lomerizine dihydrochloride (KB-2796) is an antagonist of L- and T-type voltage-gated calcium channels used to treat migraine.</p>
    Fórmula:C27H30F2N2O3·2HCl
    Pureza:99.26% - 99.80%
    Cor e Forma:Colourless Crystalline Solid
    Peso molecular:541.46
  • Soticlestat

    CAS:
    <p>Soticlestat (OV935) is a potent, selective and orally active cholesterol 24-hydroxylase (CYP46A1) inhibitor.</p>
    Fórmula:C23H23N3O2
    Pureza:99.79%
    Cor e Forma:Solid
    Peso molecular:373.45
  • Torcetrapib

    CAS:
    <p>Torcetrapib (CP-529414), a CETP inhibitor, curbs cholesteryl ester movement from HDL to LDL/VLDL; failed Phase III trials due to mortality increase.</p>
    Fórmula:C26H25F9N2O4
    Pureza:98% - 99.59%
    Cor e Forma:Lipid
    Peso molecular:600.47
  • N-(p-amylcinnamoyl) Anthranilic Acid

    CAS:
    <p>N-(p-amylcinnamoyl) Anthranilic Acid (ACA) is a broad spectrum Phospholipase A2 (PLA2) inhibitor and TRP channel blocker.</p>
    Fórmula:C21H23NO3
    Pureza:99.35% - 99.67%
    Cor e Forma:Solid
    Peso molecular:337.41
  • Azumolene

    CAS:
    <p>Azumolene (EU4093 free base)</p>
    Fórmula:C13H9BrN4O3
    Pureza:98.1% - 98.35%
    Cor e Forma:Solid
    Peso molecular:349.14
  • CVT-12012

    CAS:
    <p>CVT-12012 is an orally bioavailable inhibitor of stearoyl-CoA desaturase (SCD; IC50 = 6.1 nM in HepG2 cells).</p>
    Fórmula:C21H21F3N4O3
    Pureza:99.56%
    Cor e Forma:Solid
    Peso molecular:434.41
  • AKBA

    CAS:
    <p>AKBA (3-O-Acetyl-11-keto-beta-boswellic acid), a natural component from frankincense, is a novel activator of Nrf2.</p>
    Fórmula:C32H48O5
    Pureza:97.85% - 99.77%
    Cor e Forma:Solid
    Peso molecular:512.72
  • D159687

    CAS:
    <p>D159687 is a selective PDE4D inhibitor,had a procognitive profile as it improved memory in the novel object recognition test but had no antidepressant benefit.</p>
    Fórmula:C21H19ClN2O2
    Pureza:97.57%
    Cor e Forma:Solid
    Peso molecular:366.84
  • Fmoc-Ser(O-α-D-GalNAc(OAc)3)-OH

    CAS:
    <p>Fmoc-Ser(O-α-D-GalNAc(OAc)3)-OH (Fmoc-Ser(Ac3AcNH-α-Gal)-OH) is an anti-tumor drug</p>
    Fórmula:C32H36N2O13
    Pureza:98% - ≥98%
    Cor e Forma:Solid
    Peso molecular:656.63
  • DS-1001b

    CAS:
    <p>DS-1001b is an inhibitor of mutant IDH-1 (Isocitrate Dehydrogenase-1)</p>
    Fórmula:C29H29Cl3FN3O4
    Pureza:99.81%
    Cor e Forma:Solid
    Peso molecular:608.92
  • DY268

    CAS:
    <p>DY268 is a compound based on trisubstituted pyrazolamide without any FXR agonist activity and cytotoxicity and can be used as an effective FXR antagonist.</p>
    Fórmula:C30H32N4O5S
    Pureza:99.43% - 99.75%
    Cor e Forma:Solid
    Peso molecular:560.66
  • ML198

    CAS:
    <p>ML198: Activates &amp; chaperones glucocerebrosidase; a potential Gaucher disease treatment lead.</p>
    Fórmula:C17H14N4O
    Pureza:98.31%
    Cor e Forma:Solid
    Peso molecular:290.32
  • AKR1C3-IN-4

    CAS:
    <p>AKR1C3-IN-4: potent, selective AKR1C3 inhibitor, IC50 = 0.56 μM, potential for CRPC research.</p>
    Fórmula:C14H10F3NO2
    Pureza:98.59%
    Cor e Forma:Solid
    Peso molecular:281.23
  • Oxiconazole

    CAS:
    <p>Oxiconazole is a broad-spectrum imidazole antifungal, inhibiting ergosterol biosynthesi by disrupting cytochrome P450 enzymes (lanosterol 14- α demethylase).</p>
    Fórmula:C18H13Cl4N3O
    Pureza:99.99%
    Cor e Forma:Solid
    Peso molecular:429.13
  • AZD7325

    CAS:
    <p>AZD7325 (AZD-7325) is a GABA-Aα2,3 -selective receptor modulator.</p>
    Fórmula:C19H19FN4O2
    Pureza:99.83%
    Cor e Forma:Solid
    Peso molecular:354.38
  • IDO1-IN-1

    CAS:
    <p>IDO1-IN-1 (2 HzBTZ) is an indoleamine 2,3-dioxygenase 1 (IDO1) inhibitor.</p>
    Fórmula:C7H7N3S
    Pureza:99.36%
    Cor e Forma:Slightly Yellow To Beige-Green Crystalline Powder
    Peso molecular:165.22
  • EMAC10101d

    CAS:
    <p>compound EMAC10101d, bearing a 2,4-dichorophenyl substituent in position 4 of the dihydrothiazole ring, was the most potent and selective toward hCA II with an</p>
    Fórmula:C17H15Cl2N3O2S2
    Pureza:99.96%
    Cor e Forma:Solid
    Peso molecular:428.36
  • Imeglimin hydrochloride

    CAS:
    <p>Imeglimin hydrochloride (EMD 387008 hydrochloride) is an oral hypoglycemic agent. Imeglimin improves insulin sensitivity.Cost-effective and quality-assured.</p>
    Fórmula:C6H14ClN5
    Pureza:99.25% - 99.94%
    Cor e Forma:Solid
    Peso molecular:191.66
  • PHPS1

    CAS:
    <p>PHPS1 blocks Shp2, halts Shp2-E76K-induced Erk1/2 activation, and stops tumor cell growth.</p>
    Fórmula:C21H15N5O6S
    Pureza:99.08%
    Cor e Forma:Solid
    Peso molecular:465.44
  • PF-05221304

    CAS:
    <p>PF-05221304 (NSC-170984) is an orally active, liver-targeted inhibitor of acetyl-CoA carboxylase (ACC), a rate-limiting enzymes for fatty acid synthesis.</p>
    Fórmula:C28H30N4O5
    Pureza:98.82% - 99.50%
    Cor e Forma:Solid
    Peso molecular:502.56
  • Cintirorgon

    CAS:
    <p>Cintirorgon (LYC-55716) is a selective, oral agonist of RORγ. Cintirorgon modulates gene expression of RORγ expressing T lymphocyte immune cells.</p>
    Fórmula:C27H23F6NO6S
    Pureza:99.92%
    Cor e Forma:Solid
    Peso molecular:603.53
  • hnps-PLA Inhibitor

    CAS:
    <p>Hnps-PLA Inhibitor is an inhibitor of human nonpancreatic secretory Phospholipase A (hnps-PLA).</p>
    Fórmula:C21H21N3O4
    Pureza:99.68%
    Cor e Forma:Solid
    Peso molecular:379.41
  • 4-Bromo-3-hydroxybenzoic acid

    CAS:
    <p>4-bromo-3-hydroxybenzoic acid is a potent inhibitor of the enzyme histidine decarboxylase.</p>
    Fórmula:C7H5BrO3
    Pureza:98.11%
    Cor e Forma:Solid
    Peso molecular:217.02
  • WWL 154

    CAS:
    <p>WWL 154 is an serine hydrolase (SH) and fatty acid amide hydrolase FAAH-4 inhibitor.</p>
    Fórmula:C18H19N3O5
    Pureza:99.22%
    Cor e Forma:Solid
    Peso molecular:357.36
  • 1-Aminobenzotriazole

    CAS:
    <p>1-Aminobenzotriazole (ABT) (ABT) is a non-specific cytochrome P450 (CYP) inhibitor.</p>
    Fórmula:C6H6N4
    Pureza:98% - 99.54%
    Cor e Forma:Yellow To Beige Or Light Brown Crystalline Powder
    Peso molecular:134.14
  • Choline Fenofibrate

    CAS:
    <p>Choline Fenofibrate (Trilipix) is a choline formulation of fenofibrate, a synthetic phenoxy-isobutyric acid derivate and prodrug with antihyperlipidemic</p>
    Fórmula:C22H28ClNO5
    Pureza:98.82%
    Cor e Forma:Solid
    Peso molecular:421.91
  • Avasimibe

    CAS:
    <p>Avasimibe (PD-148515): Oral ACAT inhibitor, prevents arterial cholesterol buildup; IC50: 3.3 μM. Hinders CYP2C9/1A2/2C19; IC50: 2.9/13.9/26.5 μM.</p>
    Fórmula:C29H43NO4S
    Pureza:98.39% - 99.91%
    Cor e Forma:Solid
    Peso molecular:501.72
  • UK-371804

    CAS:
    <p>UK-371804: potent uPA blocker; candidate for chronic skin ulcer preclinical studies.</p>
    Fórmula:C14H16ClN5O4S
    Pureza:95.81% - 99.77%
    Cor e Forma:Solid
    Peso molecular:385.83
  • UC-1728

    CAS:
    <p>UC-1728 (t-TUCB) is an effective rabbit soluble epoxide hydrolase inhibitor (IC50: 2 nM on rabbit liver).</p>
    Fórmula:C21H21F3N2O5
    Pureza:99.88%
    Cor e Forma:Solid
    Peso molecular:438.4
  • OU749

    CAS:
    <p>OU749 is a γ-glutamyl transferase (GGT) inhibitor with an intrinsic Ki of 17.6 μM.</p>
    Fórmula:C16H15N3O3S2
    Pureza:99.50%
    Cor e Forma:Solid
    Peso molecular:361.44
  • Conduritol B epoxide

    CAS:
    <p>Conduritol B epoxide is an irreversible inhibitor of β-glucosidase (GCase).</p>
    Fórmula:C6H10O5
    Pureza:99.85% - ≥98%
    Cor e Forma:White Crystalline Solid
    Peso molecular:162.14
  • ML-​226

    CAS:
    <p>ML226 is a α/β hydrolase domain-containing protein 11 (ABHD11) inhibitor that inhibits ABHD11 in vitro and in situ.</p>
    Fórmula:C23H26N4O2
    Pureza:99.61%
    Cor e Forma:Solid
    Peso molecular:390.48
  • PF-07038124

    CAS:
    <p>PF-07038124 inhibits PDE4B2 (IC50=0.5 nM), IFNγ (IC50=1.06 nM), IL4 (IC50=4.1 nM), and IL-13 (IC50=125 nM).</p>
    Fórmula:C18H22BNO4
    Cor e Forma:Solid
    Peso molecular:327.18
  • N6022

    CAS:
    <p>N6022(IC50 of 8 nM) is an effective, reversible, and selective S-Nitrosoglutathione reductase(GSNOR) inhibitor.</p>
    Fórmula:C24H22N4O3
    Pureza:98.24% - 98.32%
    Cor e Forma:Solid
    Peso molecular:414.46
  • LJ570

    CAS:
    <p>LJ570 is the first PPARα/γ dual agonist (PPARα,PPARγ with EC50s of 1.05 and 0.12 μM, respectively[)</p>
    Fórmula:C27H22O3
    Pureza:99.64%
    Cor e Forma:Solid
    Peso molecular:394.46
  • URB602

    CAS:
    <p>URB602 is a specific monoacylglycerol lipase (MGL) inhibitor, which inhibits rat brain MGL (IC50: 28±4 μM) through a noncompetitive mechanism.</p>
    Fórmula:C19H21NO2
    Pureza:99.64% - 99.9%
    Cor e Forma:Off-White Solid
    Peso molecular:295.38
  • Fenretinide

    CAS:
    <p>Fenretinide (4-HPR) is an orally-active synthetic retinoid derivative with potential antineoplastic and chemopreventive activities.</p>
    Fórmula:C26H33NO2
    Pureza:98% - 99.68%
    Cor e Forma:Yellow Powder
    Peso molecular:391.55
  • CD437

    CAS:
    <p>CD437 (AHPN) is a specifc Retinoic Acid Receptor γ (RARγ) agonist.</p>
    Fórmula:C27H26O3
    Pureza:98.92% - 99.63%
    Cor e Forma:Solid
    Peso molecular:398.49
  • BPTES

    CAS:
    <p>BPTES(IC50 of 0.16 μM) is an effective and specific GlutamiN/Ase GLS1 (KGA) inhibitor.</p>
    Fórmula:C24H24N6O2S3
    Pureza:95.83% - 99.64%
    Cor e Forma:Solid
    Peso molecular:524.68
  • MPO-IN-28

    CAS:
    <p>MPO-IN-28 is a novel potent, irreversible Myeloperoxidase (MPO) inhibitor with IC50 of 44 nM.</p>
    Fórmula:C11H13N5O
    Pureza:98.04%
    Cor e Forma:Solid
    Peso molecular:231.25
  • HA130

    CAS:
    <p>HA130 is a selective ATX (autotaxin) inhibitor.</p>
    Fórmula:C24H19BFNO5S
    Pureza:98.26% - ≥95%
    Cor e Forma:Solid
    Peso molecular:463.29
  • EAAT2 activator 1

    CAS:
    <p>EAAT2 activator 1 (3-[(2-Chloro-6-fluorobenzyl)thio]-6-pyridin-2-ylpyridazine) is a thiopyridazine derivative that has been found to increase EAAT2 protein</p>
    Fórmula:C16H11ClFN3S
    Pureza:98.86%
    Cor e Forma:Solid
    Peso molecular:331.8
  • 1-Cyclohexyl-3-dodecyl urea

    CAS:
    <p>1-Cyclohexyl-3-dodecyl urea (NCND) is a highly selective soluble epoxide hydrolase (sEH) inhibitor.</p>
    Fórmula:C19H38N2O
    Pureza:99.59%
    Cor e Forma:Solid
    Peso molecular:310.52
  • ASP-9521

    CAS:
    <p>ASP-9521 is a selective, potent and orally active indole-based AKR1C3 inhibitor with an IC50 of 11 nM for human AKR1C3.Cost-effective and quality-assured.</p>
    Fórmula:C19H26N2O3
    Pureza:95.11% - 96.96%
    Cor e Forma:Solid
    Peso molecular:330.42
  • Pinaverium bromide

    CAS:
    <p>Pinaverium bromide is an calcium channel blocker with Antispasmodic and effectively relieves pain, diarrhea and intestinal discomfort.</p>
    Fórmula:C26H41Br2NO4
    Pureza:99.52%
    Cor e Forma:White Crystalline Powder
    Peso molecular:591.42
  • Nitrofurazone

    CAS:
    <p>Nitrofurazone (Furacilin) is a topical anti-infective agent effective against gram-negative and gram-positive bacteria.</p>
    Fórmula:C6H6N4O4
    Pureza:99.87%
    Cor e Forma:Pale Yellow Needles Solution) 6 0 - 6 5 Alkaline Solutions Are Dark Orange (Ntp 1992)
    Peso molecular:198.14
  • Linrodostat

    CAS:
    <p>Linrodostat (BMS-986205) is a selective indoleamine 2, 3-dioxygenase 1 (IDO1) inhibitor.</p>
    Fórmula:C24H24ClFN2O
    Pureza:99.54% - 99.71%
    Cor e Forma:Solid
    Peso molecular:410.91
  • PF-06282999

    CAS:
    <p>PF-06282999 is a potent and selective myeloperoxidase inhibitor which is potentially useful for the treatment of cardiovascular diseases.</p>
    Fórmula:C13H12ClN3O3S
    Pureza:98.15% - 98.28%
    Cor e Forma:Solid
    Peso molecular:325.77
  • NS-638

    CAS:
    <p>NS-638 is a Ca2+-channel blocker. It can block K+-stimulated intracellular Ca2+-elevation (IC50: 3.4 μM).</p>
    Fórmula:C15H11ClF3N3
    Pureza:98.44%
    Cor e Forma:Solid
    Peso molecular:325.72
  • Pentamidine

    CAS:
    <p>Pentamidine is an antifungal and antiprotozoal agent, interacting directly with the pathogen genome by binding to AT-rich regions of duplex DNA and the minor</p>
    Fórmula:C19H24N4O2
    Pureza:98.64% - 99.67%
    Cor e Forma:Crystallizes As Colorless Plates From Water Solid
    Peso molecular:340.42
  • 2-hydroxymethyl benzoic acid

    CAS:
    <p>2-hydroxymethyl benzoic acid is a principal metabolite of the phthalidyl moiety in man.</p>
    Fórmula:C8H8O3
    Pureza:98.36%
    Cor e Forma:Solid
    Peso molecular:152.15
  • Alrestatin

    CAS:
    <p>Alrestatin (AY-22284) is a specific inhibitor of aldose reductase and attenuates glucose-induced angiotensin II production in rat vascular smooth muscle in</p>
    Fórmula:C14H9NO4
    Pureza:99.23%
    Cor e Forma:Solid
    Peso molecular:255.2256
  • GOT1 inhibitor-1

    CAS:
    <p>GOT1 inhibitor-1 (GOT1 inhibitor 2c) is a novel, potent and non-covalent inhibitor of glutamate oxaloacetate transaminase 1 (GOT1) with an IC50 of 8.2 uM.</p>
    Fórmula:C19H19ClN4O
    Pureza:99.70%
    Cor e Forma:Solid
    Peso molecular:354.83
  • SR8278

    CAS:
    <p>SR8278 is an REV-ERBα antagonist(EC50 = 0.47 μM), blocking activation of the receptor by the synthetic agonist GSK 4112</p>
    Fórmula:C18H19NO3S2
    Pureza:99.44% - 99.73%
    Cor e Forma:Solid
    Peso molecular:361.48
  • BRL-50481

    CAS:
    <p>BRL-50481 is a novel and selective inhibitor of PDE7 with IC50s of 0.15, 12.1, 62 and 490 μM for PDE7A, PDE7B, PDE4 and PDE3, respectively.</p>
    Fórmula:C9H12N2O4S
    Pureza:99.66%
    Cor e Forma:Solid
    Peso molecular:244.27
  • Toloxatone

    CAS:
    <p>Toloxatone (MD 69276) is a reversible monoamine oxidase A (MAOA) inhibitor.</p>
    Fórmula:C11H13NO3
    Pureza:98.58%
    Cor e Forma:Solid
    Peso molecular:207.23
  • BI-187004

    CAS:
    <p>BI-187004 is an 11β-hydroxysteroid dehydrogenase 1 inhibitor.</p>
    Fórmula:C21H18N4O
    Pureza:98.63%
    Cor e Forma:Solid
    Peso molecular:342.39
  • Gonadorelin Acetate (33515-09-2 free base)

    CAS:
    <p>Gonadorelin Acetate (33515-09-2 free base) (Luteinizing Hormone Releasing Hormone (LH-RH)) is hypothalamic neuropeptide which plays a key role in the control of</p>
    Fórmula:C59H83N17O17
    Pureza:99.42% - 99.46%
    Cor e Forma:White Or Off-White Powder
    Peso molecular:1302.39
  • Pirinixic Acid

    CAS:
    <p>Pirinixic Acid (NSC 310038) is a synthetic thiacetic acid derivative used in biomedical research, a peroxisome proliferator that activates specific PPAR.</p>
    Fórmula:C14H14ClN3O2S
    Pureza:98.27% - 99.92%
    Cor e Forma:Solid
    Peso molecular:323.8
  • AUDA

    CAS:
    <p>AUDA is an inhibitor of sEH(IC50 values of 18 and 69 nM for the mouse and human enzymes, respectively)</p>
    Fórmula:C23H40N2O3
    Pureza:99.50%
    Cor e Forma:Solid
    Peso molecular:392.58
  • BW-A 78U

    CAS:
    <p>BW-A 78U is a PDE4 inhibitor (IC50: 3 μM). It is not inhibition on the lipopolysaccharide (LPS)-induced TNF-α release.</p>
    Fórmula:C13H12FN5
    Pureza:99.45%
    Cor e Forma:Solid
    Peso molecular:257.27
  • GSK805

    CAS:
    <p>GSK805 is a potent, orally bioavailable and CNS-penetrant RORγt inhibitor.Cost-effective and quality-assured.</p>
    Fórmula:C23H18Cl2F3NO4S
    Pureza:98% - ≥95%
    Cor e Forma:Solid
    Peso molecular:532.36
  • Telaglenastat

    CAS:
    <p>Telaglenastat (CB 839) (IC50 of 24 nM), an effective, specific, and oral inhibitor, which is bioavailable glutaminase, for recombinant human GAC.</p>
    Fórmula:C26H24F3N7O3S
    Pureza:97.57% - 99.89%
    Cor e Forma:Solid
    Peso molecular:571.57
  • Pargyline

    CAS:
    <p>Pargyline (Pargylamine) is a monoamine oxidase inhibitor with antihypertensive properties.</p>
    Fórmula:C11H13N
    Pureza:95.64% - 97.21%
    Cor e Forma:Solid
    Peso molecular:159.23
  • PfDHODH-IN-2

    CAS:
    <p>PfDHODH-IN-2: powerful antimalarial, blocks PfDHODH (IC50: 1.11 μM), for malaria research.</p>
    Fórmula:C13H12ClNO3S
    Pureza:98.9%
    Cor e Forma:Solid
    Peso molecular:297.76
  • Pentamidine isethionate

    CAS:
    <p>Pentamidine isethionate (Pentamidine diisethionate) is a synthetic amidine derivative, Pentamidine Isethionate is an antiprotozoal and antifungal agent.</p>
    Fórmula:C23H36N4O10S2
    Pureza:98% - 99.83%
    Cor e Forma:Slight Butyric Odor Very Bitter Taste Ph (5% Aqueous Solution) 4 5-6 5 (Ntp 1992)
    Peso molecular:592.68
  • FG-2216

    CAS:
    <p>FG-2216 (YM-311) is a HIF-prolyl hydroxylase inhibitor for the PDH2 enzyme; orally bioavailable and induced reversible and significant Epo induction in vivo.</p>
    Fórmula:C12H9ClN2O4
    Pureza:97.1% - >99.99%
    Cor e Forma:Solid
    Peso molecular:280.66
  • RGX-104

    CAS:
    <p>RGX-104 (RGX-104 free Acid) free Acid is an agonist of potent liver-X nuclear hormone receptor (LXR)</p>
    Fórmula:C34H33ClF3NO3
    Pureza:98.79% - 99.53%
    Cor e Forma:Solid
    Peso molecular:596.08
  • LOX-IN-3 dihydrochloride

    CAS:
    <p>LOX-IN-3 dihydrochloride is an inhibitor of lysyl oxidase (LOX).</p>
    Fórmula:C13H15Cl2FN2O2S
    Pureza:99.96%
    Cor e Forma:Solid
    Peso molecular:353.24
  • Cobicistat

    CAS:
    <p>Cobicistat (GS-9350): A carbamate, thiazole derivative, and CYP3A inhibitor used to boost anti-HIV drugs for treating HIV.</p>
    Fórmula:C40H53N7O5S2
    Pureza:97.36% - 99.62%
    Cor e Forma:Solid
    Peso molecular:776.02
  • Glycerol 3-phosphate biscyclohexylammonium salt

    CAS:
    <p>Glycerol 3-phosphate biscyclohexylammonium salt is an endogenous metabolite produced by cytosolic glycerol 3-phosphate dehydrogenase pathway.</p>
    Fórmula:C15H35N2O6P
    Pureza:99.94%
    Cor e Forma:Solid
    Peso molecular:370.42
  • ARM1

    CAS:
    <p>ARM1 is a potent inhibitor of aminopeptidase and epoxide hydrolase. The IC50 values are 7.61 µM for aminopeptidase and 12.4 µM for epoxide hydrolase.</p>
    Fórmula:C16H14N2S
    Pureza:99.36%
    Cor e Forma:Solid
    Peso molecular:266.36
  • (±)-Amiflamine

    CAS:
    <p>(±)-Amiflamine (2-dimethylphenethylamine) is an inhibitor of reversible MAO-A.</p>
    Fórmula:C12H20N2
    Pureza:97.24%
    Cor e Forma:Solid
    Peso molecular:192.3
  • Bempedoic acid

    CAS:
    <p>Bempedoic acid (ETC1002) is an orally available, once-daily LDL-C lowering small molecule designed to lower elevated levels of LDL-C.</p>
    Fórmula:C19H36O5
    Pureza:99.85% - 99.94%
    Cor e Forma:Solid
    Peso molecular:344.49
  • Efonidipine hydrochloride monoethanolate

    CAS:
    <p>Efonidipine HCl monoethanolate is a calcium blocker, boosts dehydroepiandrosterone sulfate in NCI-H295R cells.</p>
    Fórmula:C36H45ClN3O8P
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:714.18
  • 1-Ethynylpyrene

    CAS:
    <p>1-Ethynylpyrene is an aryl acetylenic inhibitor of CYTP450 1A1(IC50=0.18 μM), 1A2(IC50 = 0.32 μM), and 2B1(IC50 = 0.04 μM).</p>
    Fórmula:C18H10
    Pureza:98.48%
    Cor e Forma:Solid
    Peso molecular:226.27
  • Suvecaltamide

    CAS:
    <p>Suvecaltamide (MK-8998) as potent inhibitors of T-type calcium channels.</p>
    Fórmula:C20H23F3N2O2
    Pureza:99.29% - 99.70%
    Cor e Forma:Solid
    Peso molecular:380.4
  • Diflubenzuron

    CAS:
    <p>Diflubenzuron (Larvakil) is a benzoyl-urea insecticide, found to be a potent inhibitor of melanosome synthesis in mouse melanoma cells.</p>
    Fórmula:C14H9ClF2N2O2
    Pureza:99.58% - 99.96%
    Cor e Forma:Colorless Crystals Diflubenzuron Is A Colorless To Yellow Crystals Used As A Selective Insecticide
    Peso molecular:310.68
  • (Rac)-LB-100

    CAS:
    <p>LB-100, a novel Protein Phosphatase 2A (PP2A) inhibitor, sensitizes malignant meningioma cells to the therapeutic effects of radiation</p>
    Fórmula:C13H20N2O4
    Pureza:97.11% - 99.77%
    Cor e Forma:Solid
    Peso molecular:268.31
  • 2,5-Di-tert-butylhydroquinone

    CAS:
    <p>2,5-Di-tert-butylhydroquinone (BHQ) is an effective and selective endoplasmic reticulum Ca2+-ATPase inhibitor.</p>
    Fórmula:C14H22O2
    Pureza:97.11%
    Cor e Forma:Pelletslargecrystals
    Peso molecular:222.32
  • kb NB 142-70

    CAS:
    <p>kb NB 142-70 is a selective protein kinase D (PKD) inhibitor (IC50 values are 28.3, 58.7 and 53.2 nM for PKD1, 2 and 3 respectively).</p>
    Fórmula:C11H9NO2S2
    Pureza:98.15% - ≥95%
    Cor e Forma:Solid
    Peso molecular:251.32
  • AGN 193109

    CAS:
    <p>AGN 193109, a retinoid analog, is a potent and specific antagonist of RARs (Kds: 2 nM, 2 nM, and 3 nM for RARα, RARβ, and RARγ).</p>
    Fórmula:C28H24O2
    Pureza:99.87% - 99.89%
    Cor e Forma:Solid
    Peso molecular:392.49
  • D-Valine

    CAS:
    <p>D-Valine (H-D-Val-OH) is the enantiomer of L-Valine.</p>
    Fórmula:C5H11NO2
    Pureza:99.93%
    Cor e Forma:White Crystals
    Peso molecular:117.15
  • GSK2033

    CAS:
    <p>GSK2033 is an antagonist of LXR (pIC50s: 7 and 7.4 for LXRα or LXRβ, respectively).</p>
    Fórmula:C29H28F3NO5S2
    Pureza:99.70%
    Cor e Forma:Solid
    Peso molecular:591.66
  • IDO5L

    CAS:
    <p>IDO5L (INCB024360 analogue) is an effective IDO1 inhibitor(IC50=10 nM).</p>
    Fórmula:C9H7ClFN5O2
    Pureza:99.49% - 99.75%
    Cor e Forma:Solid
    Peso molecular:271.64
  • Tedizolid

    CAS:
    <p>Tedizolid (DA-7157)is a novel oxazolidinone-class antibiotic that inhibits bacterial protein synthesis by binding to the 23S ribosomal RNA of the 50S subunit of</p>
    Fórmula:C17H15FN6O3
    Pureza:96.97% - 99.89%
    Cor e Forma:Solid
    Peso molecular:370.34
  • Pimecrolimus

    CAS:
    <p>Pimecrolimus, a calcineurin inhibitor, binds FKBP-12, blocking calcium-dependent signals.</p>
    Fórmula:C43H68ClNO11
    Pureza:99.53% - 99.87%
    Cor e Forma:White Crystalline Powder
    Peso molecular:810.45
  • SI-113

    CAS:
    <p>SI-113 is a potent and selective inhibitor of SGK1, a serine/threonine protein kinase, that modulates several oncogenic signaling cascades.</p>
    Fórmula:C23H24N6O
    Pureza:98.93%
    Cor e Forma:Solid
    Peso molecular:400.48
  • IDF-11774

    CAS:
    <p>IDF-11774 is a HIF-1 inhibitor.It reduces hif-1α HRE luciferase activity (IC50 = 3.65 μM).</p>
    Fórmula:C23H32N2O2
    Pureza:98.05%
    Cor e Forma:Solid
    Peso molecular:368.51
  • Tepoxalin

    CAS:
    <p>Tepoxalin (RWJ 20485), potential asthma and osteoarthritis drug, inhibits COX-1, COX-2, and 5-LOX with low IC50 values.</p>
    Fórmula:C20H20ClN3O3
    Pureza:99.94%
    Cor e Forma:Solid
    Peso molecular:385.84
  • ZINC13466751

    CAS:
    <p>ZINC13466751 is a potent HIF-1α/von Hippel-Lindau interaction inhibitor(IC50 = 2.0 µM).</p>
    Fórmula:C20H21N5O2
    Pureza:99.8%
    Cor e Forma:Solid
    Peso molecular:363.41
  • Olumacostat Glasaretil

    CAS:
    <p>Olumacostat glasaretil is a small molecule inhibitor of acetyl coenzyme A carboxylase (ACC). It has been used in trials studying the treatment of Acne Vulgaris.</p>
    Fórmula:C26H43NO7
    Pureza:97.79% - 99.34%
    Cor e Forma:Solid
    Peso molecular:481.62
  • Ingliforib

    CAS:
    <p>Ingliforib (CP 368296) is a novel glycogen phosphorylase inhibitor,has antihyperglycemic and cardioprotective properties.</p>
    Fórmula:C23H24ClN3O5
    Pureza:99.04% - 99.30%
    Cor e Forma:Solid
    Peso molecular:457.91
  • Biotin sulfone

    CAS:
    <p>Biotin sulfone is an oxidized form of biotin.</p>
    Fórmula:C10H16N2O5S
    Pureza:95.51%
    Cor e Forma:Solid
    Peso molecular:276.31
  • G3335 Acetate


    <p>G3335 Acetate was discovered to be a novel PPARgamma antagonist.</p>
    Fórmula:C18H23N3O7
    Pureza:99.75%
    Cor e Forma:Solid
    Peso molecular:393.39
  • BCI hydrochloride

    CAS:
    <p>BCI hydrochloride ((E)-BCI hydrochloride) is a DUSP6 inhibitor that inhibits RANKL-mediated osteoclastogenesis and attenuates oophorectomy-induced bone loss.</p>
    Fórmula:C22H24ClNO
    Pureza:99.95%
    Cor e Forma:Solid
    Peso molecular:353.89
  • PKM2-IN-1

    CAS:
    <p>PKM2-IN-1 (compound 3k) displays PKM2 inhibitory activity with the IC50 value of 2.95 μM. The IC50 value for PKM1 is 4-5-fold higher than that for PKM2.</p>
    Fórmula:C18H19NO2S2
    Pureza:99.49% - 99.68%
    Cor e Forma:Solid
    Peso molecular:345.48
  • GW604714X

    CAS:
    <p>GW604714X (2,4-Thiazolidinedione, 5-[[5-[6-(4-acetyl-1-piperazinyl)-3-nitro-2-pyridinyl]-2-fluorophenyl]methylene]-) were found to be potent inhibitors of</p>
    Fórmula:C21H18FN5O5S
    Pureza:98.05%
    Cor e Forma:Solid
    Peso molecular:471.46
  • SDZ285428

    CAS:
    <p>SDZ285428 is a CYP24A1 inhibitor.</p>
    Fórmula:C24H20ClN3O
    Pureza:97.51%
    Cor e Forma:Solid
    Peso molecular:401.89
  • 1-Ethynylnaphthalene

    CAS:
    <p>1-Ethynylnaphthalene is a selective inhibitor of cytochrome P450 IB1</p>
    Fórmula:C12H8
    Pureza:99.05%
    Cor e Forma:Yellow To Brown Liquid
    Peso molecular:152.19
  • F1063-0967

    CAS:
    <p>F1063-0967 is a Dual-specificity phosphatase 26 (DUSP26) inhibitor with an IC50 of 11.62 μM.</p>
    Fórmula:C24H24N2O5S2
    Pureza:97.77%
    Cor e Forma:Solid
    Peso molecular:484.59
  • M1001

    CAS:
    <p>M1001 is a HIF-2α agonist.</p>
    Fórmula:C17H17N3O2S
    Pureza:98.83%
    Cor e Forma:Solid
    Peso molecular:327.4
  • CDC25B-IN-2

    CAS:
    <p>BIA is an inhibitor of the interaction between TMBIM6 and mTORC2, which ultimately blocks AKT activation and cancer progression.</p>
    Fórmula:C15H12N2O3
    Pureza:99.12%
    Cor e Forma:Solid
    Peso molecular:268.27
  • FPL 62064

    CAS:
    <p>FPL 62064 is a potent dual inhibitor of 5-lipoxygenase (5-LOX) and COX (IC50 of 3.5 μM and 3.1 μM for RBL-1 cytosolic 5-lipoxygenase and prostaglandin</p>
    Fórmula:C16H15N3O
    Pureza:98.79%
    Cor e Forma:Solid
    Peso molecular:265.31
  • all-trans-4-Oxoretinoic acid

    CAS:
    <p>all-trans-4-Oxoretinoic acid (all-trans 4-Keto Retinoic Acid) is an active metabolite of vitamin A.</p>
    Fórmula:C20H26O3
    Pureza:98.52%
    Cor e Forma:Solid
    Peso molecular:314.42
  • Ervogastat

    CAS:
    <p>Ervogastat (PF-06865571) is a potent and well-tolerated diacylglycerol acyltransferase 2 inhibitor.</p>
    Fórmula:C21H21N5O4
    Pureza:99.97%
    Cor e Forma:Solid
    Peso molecular:407.42
  • Galeterone

    CAS:
    <p>Galeterone (VN 124) is an oral androgen receptor modulator/CYP17 inhibitor with antiandrogen properties, targeting prostate cancer growth.</p>
    Fórmula:C26H32N2O
    Pureza:99.47% - 99.773%
    Cor e Forma:Solid
    Peso molecular:388.55
  • Heparin sodium salt

    CAS:
    <p>Heparin sodium, a sulfated glycosaminoglycan, acts as an anticoagulant and inhibits exosome-cell interactions.</p>
    Fórmula:C26H42N2NaO37S5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:1157.89
  • BMS-687453

    CAS:
    <p>BMS-687453 is a potent and selective PPAR alpha agonist, with an EC(50) of 10 nM for human PPARalpha and approximately 410-fold selectivity vs human PPARgamma</p>
    Fórmula:C22H21ClN2O6
    Pureza:99.4%
    Cor e Forma:Solid
    Peso molecular:444.86
  • RORγt inverse agonist 13

    CAS:
    <p>RORγt inverse agonist 13 (Compound 3i) is a potent, orally active and selective RORγt inverse agonist (IC50=63.8 nM), with improved drug-like properties[1].</p>
    Fórmula:C23H17Cl2F3N2O4
    Pureza:99.04%
    Cor e Forma:Solid
    Peso molecular:513.29
  • Tosedostat

    CAS:
    <p>Tosedostat (CHR-2797), an oral M1 aminopeptidase inhibitor, turns into CHR-79888, blocks tumor cell proteins, causing cell death.</p>
    Fórmula:C21H30N2O6
    Pureza:98.14% - 99.4%
    Cor e Forma:Solid
    Peso molecular:406.47
  • TCS 401

    CAS:
    <p>TCS 401 is a selective inhibitor of protein-tyrosine phosphatase 1B (PTP1B; Ki = 0.29 μM)</p>
    Fórmula:C10H11ClN2O5S
    Pureza:98.15%
    Cor e Forma:Solid
    Peso molecular:306.72
  • GEBR-7b

    CAS:
    <p>GEBR-7b (3-(Cyclopentyloxy)-4-methoxybenzaldehyde) is a phosphodiesterase-4 (PDE4) inhibitor.</p>
    Fórmula:C13H16O3
    Pureza:99.533%
    Cor e Forma:Solid
    Peso molecular:220.26
  • α-Amylase

    CAS:
    <p>α-Amylase, a hydrolase enzyme, catalyzes the hydrolysis of internal α-1,4-glycosidic linkages in starch, producing glucose and maltose.</p>
    Pureza:98%
    Cor e Forma:Solid
  • Ro 61-8048

    CAS:
    Ro 61-8048 is a potent and selective inhibitor of kynurenine hydroxylase with an IC50 value of 37 nM.
    Fórmula:C17H15N3O6S2
    Pureza:98% - >99.99%
    Cor e Forma:Solid
    Peso molecular:421.45
  • palovarotene

    CAS:
    <p>Palovarotene (Ro 3300074) is an agonist of nuclear retinoic acid receptor γ (RAR-γ).</p>
    Fórmula:C27H30N2O2
    Pureza:97.88% - 98.05%
    Cor e Forma:Solid
    Peso molecular:414.54
  • Malotilate

    CAS:
    <p>Malotilate (Kantec) is a medicine used for the therapy of liver cirrhosis.</p>
    Fórmula:C12H16O4S2
    Pureza:99.79% - 99.79%
    Cor e Forma:Solid
    Peso molecular:288.38
  • NSC 65809

    CAS:
    <p>NSC-65809 (Raphin1) is a selective inhibitor of R15B.</p>
    Fórmula:C8H8Cl2N4
    Pureza:99.37%
    Cor e Forma:Solid
    Peso molecular:231.08
  • FT113

    CAS:
    <p>FT113 is a novel potent inhibitor of fatty acid synthase (fasn, IC50 : 213 nM),and exhibits anti-cancer activity</p>
    Fórmula:C22H20FN3O4
    Pureza:97.05%
    Cor e Forma:Solid
    Peso molecular:409.41
  • Anti-Inflammatory Peptide 1 Acetate


    <p>Anti-Inflammatory Peptide 1 Acetate (C45H82N12O14S2) inhibits PLA2 to reduce inflammation and pain.</p>
    Fórmula:C47H86N12O16S2
    Pureza:98.95%
    Cor e Forma:Solid
    Peso molecular:1139.39
  • LDHA-IN-4

    CAS:
    <p>LDHA-IN-4 (AZ33) is an LDHA inhibitor. Binding affinity to 6-His-tagged human LDHA expressed in E.coli BL21 (DE3) by SPR analysis with an active value of 93 nM.</p>
    Fórmula:C25H27N3O6S
    Pureza:98.17% - 99.68%
    Cor e Forma:Solid
    Peso molecular:497.56
  • H2S Donor 5a

    CAS:
    <p>H2S Donor 5a is a H2S donor that could mimic the slow and continuous H(2)S generation process.</p>
    Fórmula:C14H11NO2S
    Pureza:99.68%
    Cor e Forma:Solid
    Peso molecular:257.31
  • Indisulam

    CAS:
    <p>Indisulam (E 7070) is a dual-action anticancer drug, blocking G1/S cell cycle transition by degrading cyclin E and activating p53/p21.</p>
    Fórmula:C14H12ClN3O4S2
    Pureza:98.68% - 99.77%
    Cor e Forma:Solid
    Peso molecular:385.85
  • (E,E)-RAMB4

    CAS:
    <p>PTP1B-IN-8 is a potent and selective inhibitor of protein tyrosine phosphatase-1B (PTP1B).</p>
    Fórmula:C19H13Cl4NO
    Pureza:96.03%
    Cor e Forma:Solid
    Peso molecular:413.12
  • Ziconotide Acetate (107452-89-1 free base)

    CAS:
    <p>Ziconotide Acetate (Prialt, 107452-89-1) is an analgesic for neuropathic pain, acting on N-type calcium channels to block pain signals.</p>
    Fórmula:C102H172N36O32S7
    Pureza:99.52% - 99.87%
    Cor e Forma:Solid
    Peso molecular:2639.2
  • PHD-1-IN-1

    CAS:
    <p>PHD-1-IN-1 is a potent inhibitor of hypoxia-inducible factor prolylhydroxylase domain-1 (PHD-1) enzyme(IC50 = 0.034 μM).</p>
    Fórmula:C13H8N4
    Pureza:99.74%
    Cor e Forma:Solid
    Peso molecular:220.23
  • Pyridaben

    CAS:
    <p>Pyridaben is a METI acaricide that inhibits mitochondrial electron transport at complex I (METI; Ki = 0.36 nmol/mg protein in rat brain mitochondria).</p>
    Fórmula:C19H25ClN2OS
    Pureza:97.11% - 99.75%
    Cor e Forma:Solid
    Peso molecular:364.93
  • Betrixaban hydrochloride(330942-05-7(free base))


    <p>Betrixaban hydrochloride(330942-05-7(free base)) (PRT054021 hydrochloride) is a potent, selective, and orally efficacious factor Xa (fXa) inhibitor (IC50: 1.5</p>
    Fórmula:C23H23Cl2N5O3
    Pureza:99.54%
    Cor e Forma:Solid
    Peso molecular:488.36
  • VY-3-135

    CAS:
    <p>VY-3-135 is an orally active, stable and specific acetyl-CoA synthetase 2 (ACSS2) inhibitor.Cost-effective and quality-assured.</p>
    Fórmula:C26H27N3O3
    Pureza:99.25% - 99.79%
    Cor e Forma:Solid
    Peso molecular:429.51
  • A939572

    CAS:
    <p>A939572 is stearoyl-CoA desaturase1 (SCD1) inhibitor with IC50 values of &lt;4 nM for mSCD1 and 37 nM for hSCD1.</p>
    Fórmula:C20H22ClN3O3
    Pureza:99.96% - ≥95%
    Cor e Forma:Solid
    Peso molecular:387.86
  • Verdiperstat

    CAS:
    <p>Verdiperstat (AZD 3241) is a selective, irreversible, orally active myeloperoxidase inhibitor for neurodegenerative brain diseases.</p>
    Fórmula:C11H15N3O2S
    Pureza:99.36%
    Cor e Forma:Solid
    Peso molecular:253.32