GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,030 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(159 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(196 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(42 products)
- Opioid Receptor(325 products)
- PAFR(14 products)
- PKA(58 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5982 products of "GPCR/G-Protein"
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Pasireotide
CAS:Pasireotide (SOM 230) is a cyclohexapeptide, mimicking somatostatin with high affinity for sst1/2/3/4/5 receptors (pKi=8.2/9.0/9.1/<7.0/9.9).Formula:C58H66N10O9Purity:98%Color and Shape:SolidMolecular weight:1047.21MAO-B-IN-3
MAO-B-IN-3 is a reversible, selective inhibitor of monoamine oxidase B (MAO-B) with an IC50 of 96 nM and demonstrates affinity for the 5-HT6 receptor with a Ki
Formula:C24H25N3O2Purity:98%Color and Shape:SolidMolecular weight:387.47Orexin B, rat, mouse TFA
Orexin B, rat/mouse TFA, activates OX1-R & OX2-R receptors, influencing food intake, energy, and sleep regulation.Formula:C128H216F3N45O36SColor and Shape:SolidMolecular weight:3050.42(±)5-iPF2α-VI
CAS:Isoprostanes are prostaglandin (PG)-like products of free-radical induced lipid peroxidation.Formula:C20H34O5Color and Shape:SolidMolecular weight:354.487[D-Phe12]-Bombesin
CAS:Bombesin receptor antagonist
Formula:C74H112N22O18SPurity:98%Color and Shape:SolidMolecular weight:1629.88GLP-1 receptor agonist 9 citrate
GLP-1 receptor agonist 9 citrate is an agonist of GLP-1.
Formula:C38H39ClFN3O12Purity:98.76%Color and Shape:SolidMolecular weight:784.18Xanthine amine congener dihydrochloride
CAS:XAC dihydrochloride is an Adenosine A1 and A2 receptor antagonist with IC50s of 1.8 nM and 114 nM, also a mouse convulsant.Formula:C21H30Cl2N6O4Color and Shape:SolidMolecular weight:501.41α-CGRP(human)
CAS:Endogenous calcitonin gene-related peptide receptor (CGRP) agonist.Formula:C163H267N51O49S2Purity:98%Color and Shape:SolidMolecular weight:3789.33SGLT1/2-IN-2
CAS:SGLT1/2-IN-2 is a chemical compound with robust dual inhibitory properties, exhibiting potent activities against SGLT1 (IC50 = 96 nM) and SGLT2 (IC50 = 1.3 nM).Formula:C23H26F2O7Color and Shape:SolidMolecular weight:452.451α-Helical CRF(9-41)
CAS:Corticotropin-releasing factor receptor antagonist (Ki values are 17, 5 and 0.97 at human CRF1, rat CRF2α and mouse CRF2β receptors respectively).Formula:C166H274N46O53S2Purity:98%Color and Shape:SolidMolecular weight:3827Adrenomedullin (16-31), human TFA
Human adrenomedullin (16-31) TFA, fragment 16-31, binds CGRP1 receptor, raises rat blood pressure, not cats’.Formula:C84H130F3N25O23S2Color and Shape:SolidMolecular weight:1979.21Angiopeptin TFA
CAS:Angiopeptin TFA: somatostatin analogue, sst2/sst5 partial agonist (IC50: 0.26/6.92 nM), suppresses GH & IGF-1, for atherosclerosis research.Formula:C58H73F6N11O14S2Color and Shape:SolidMolecular weight:1326.39CH 275
CAS:Potent sst1 agonist with 30.9 nM IC50; selective over sst2-5; inhibits somatostatin in rat nucleus accumbens.Formula:C74H96N14O15S2Purity:98%Color and Shape:SolidMolecular weight:1485.8HAEGTFTSDVS
CAS:HAEGTFTSDVS is the first N-terminal 1-11 residues of GLP-1 peptide.Formula:C48H71N13O20Purity:98%Color and Shape:SolidMolecular weight:1150.18Amylin (8-37), human
CAS:Human-derived Amylin (8-37) is a vasodilator in rat arteries and forms aggregates linked to type II diabetes.Formula:C138H216N42O45Color and Shape:SolidMolecular weight:3183.495Spns2-IN-2
Spns2-IN-2 (compound 3a) is an inhibitor of SPNS2.Formula:C22H30ClN3O2Color and Shape:SolidMolecular weight:403.95Pancreatic polypeptide TFA
Pancreatic polypeptide TFA acts as a neuropeptide Y (NPY) Y4/Y5 receptor agonist.Color and Shape:Odour SolidNeuropeptide Y (13-36), amide, human
CAS:Neuropeptide Y (13-36), amide, human is a neuropeptide Y receptor agonist.Formula:C134H207N41O36SPurity:98%Color and Shape:SolidMolecular weight:3000.4Lys-[Hyp3]-Bradykinin
CAS:Lys-[Hyp3]-Bradykinin, a human urine-derived kinin and bradykinin agonist, is used for inflammation research.Formula:C56H85N17O13Color and Shape:SolidMolecular weight:1204.38AM-0466
CAS:AM-0466 has a wide range of applications in life science related research.Formula:C27H19F3N4O4SColor and Shape:SolidMolecular weight:552.52Human growth hormone-releasing factor
CAS:GHRH from the hypothalamus prompts the pituitary to produce/release GH by attaching to the GHRHR.Formula:C215H358N72O66SPurity:98%Color and Shape:SolidMolecular weight:5039.65Icatibant
CAS:Icatibant is a selective and specific antagonist of the bradykinin B2 receptor (IC50 and Ki: 1.07 nM and 0.798 nM respectively).Formula:C59H89N19O13SPurity:98%Color and Shape:White SolidMolecular weight:1304.52Dulaglutide
CAS:Dulaglutide (LY2189265) is a GLP-1 receptor agonist for studying type 2 diabetes mellitus (T2DM).Color and Shape:SolidRF9 acetate
RF9 acetate is an effective and selective antagonist of Neuropeptide FF receptor with Ki values of 58 and 75 nM for hNPFF1R and hNPFF2R, respectively.Formula:C28H42N6O5Purity:99.77%Color and Shape:SolidMolecular weight:542.67Ref: TM-T16738L
1mg65.00€5mg125.00€10mg182.00€25mg325.00€50mg467.00€100mg645.00€200mg868.00€1mL*10mM (DMSO)167.00€P2Y6R antagonist 1
P2Y6R antagonist 1 (compound 5ab) is a selective, orally active antagonist of P2Y6R, featuring an IC50 value of 19.6 nM. This compound also exhibits anti-inflammatory properties.Color and Shape:Odour Solid15(S)-15-methyl Prostaglandin D2
CAS:15(S)-15-methyl PGD2 is a stable PGD2 analog that induces vasoconstriction, raises blood pressure, and shows strong antifertility effects.Formula:C21H34O5Color and Shape:SolidMolecular weight:366.49Amylin (IAPP), feline TFA
Amylin (IAPP), feline TFA: 37-amino acid peptide; inhibits insulin/glucagon; secreted by pancreatic β-cells.
Formula:C167H271F3N52O56S2Color and Shape:SolidMolecular weight:4024.47(Pro34)-Peptide YY (human)
CAS:(Pro34)-Peptide YY (human) is a highly Y 1 -selective full agonist of Peptide YY /neuropeptide Y receptors [1] .Formula:C194H294N54O56Color and Shape:SolidMolecular weight:4278.73HDAC6-IN-49
HDAC6-IN-49 (Compound 3) is an inhibitor of HDAC, with IC50 values of 0.012 and 0.735 µM against HDAC6 and HDAC1, respectively. Additionally, it inhibits MAO-B, cholinesterase (ChE), histamine receptor (H3R), and serotonin 6 receptor (5-HT6R). HDAC6-IN-49 exhibits neuroprotective effects in SH-SY5Y cells and enhances cognitive functions and motor abilities in fruit fly models of Parkinson's disease and C. elegans models of Alzheimer's disease.Color and Shape:Odour SolidCortistatin 14, human, rat
CAS:Cortistatin 14: a neuropeptide similar to somatostatin; induces sleep, depresses neuronal activity; found in cortex, hippocampus.Formula:C81H113N19O19S2Purity:98%Color and Shape:SolidMolecular weight:1721.01Antisauvagine-30
CAS:CRF2 receptor antagonist; Kd 1.4 nM (mCRF2β), 153.6 nM (rCRF1). Blocks sauvagine-induced cAMP in cells & stress-related responses in mice.
Formula:C161H274N48O46SPurity:98%Color and Shape:SolidMolecular weight:3650.29BAY-747
CAS:BAY-747: oral, brain-penetrant sGC stimulator; improves rat memory, cognition, lowers blood pressure, aids Duchenne muscular dystrophy.Formula:C22H26F2N4O2Color and Shape:SolidMolecular weight:416.46Adrenocorticotropic Hormone (ACTH) (1-39), rat
CAS:ACTH (1-39), rat: potent MC2 agonist, forms fragments in vitro, isolated by HPLC, characterized by amino acids and NH2-terminus.Formula:C210H315N57O57SPurity:98%Color and Shape:SolidMolecular weight:4582.23PACAP (1-27), human, ovine, rat
CAS:PACAP (1-27) (the N-terminal fragment of PACAP-38) is a novel neuropeptides originally isolated from bovine hypothalamus, also found in humans and rats.Formula:C142H224N40O39SPurity:98%Color and Shape:SolidMolecular weight:3147.66d[Cha4]-AVP TFA
d[Cha4]-AVP TFA: potent, selective V1b agonist, K i 1.2 nM, favors V1b over V1a, V2, oxytocin receptors.Formula:C52H72F3N13O13S2Color and Shape:SolidMolecular weight:1208.33des-Gln14-Ghrelin TFA
Des-Gln14-Ghrelin TFA, a ligand for GHSR, boosts [Ca2+]i with an EC50 of 2.4 nM in CHO-GHSR62 cells.Formula:C144H238F3N43O42Color and Shape:SolidMolecular weight:3300.69Syk Inhibitor II hydrochloride
CAS:Syk signaling is key in lupus. Syk inhibitors reduce inflammation and sepsis severity in FcgRIIb-/- mice, lowering cytokines and organ damage.
Formula:C14H16ClF3N6OPurity:99.05%Color and Shape:SolidMolecular weight:376.778-iso-15-keto Prostaglandin F2α
CAS:8-iso-15-keto Prostaglandin F2α (8-iso-15-keto PGF2α) is a metabolite of the isoprostane 8-iso PGF2α in rabbits, monkeys, and humans.Formula:C20H32O5Color and Shape:SolidMolecular weight:352.471Cinnamtannin A2
CAS:Cinnamtannin A2, a tetrameric procyanidin, boosts GLP-1, insulin, CRH expression, and has antioxidant, anti-diabetic, nephroprotective properties.
Formula:C60H50O24Color and Shape:SolidMolecular weight:1155.02CB1R agonist 1
CB1R agonist 1 (Compound '1350) is a potent full agonist of the cannabinoid-1 receptor (CB1R) with a Ki value of 0.95 nM. It demonstrates significant pain-relieving effects in various pain models, including acute thermal pain, inflammatory pain, and neuropathic pain.
Formula:C20H18F3N3O3SColor and Shape:SolidMolecular weight:437.435Cortistatin 14, human, rat acetate
Cortistatin 14, human, rat acetate is a neuropeptide having structural similarity to somatostatin-14 and shows anticonvulsive, neuroprotective effects andFormula:C80H112N18O19S2Purity:97.86%Color and Shape:SolidMolecular weight:1693.98GI-560192
CAS:GI-560192 (RL-0070933), a potent smo modulator, EC50: 0.02µM; affects smoothened in cilia via hedgehog signaling.Formula:C20H16N2O2Purity:99.53%Color and Shape:SoildMolecular weight:316.35Ref: TM-T64351
1mg85.00€5mg170.00€10mg250.00€25mg371.00€50mg522.00€100mg712.00€200mg954.00€1mL*10mM (DMSO)170.00€β2AR/M-receptor agonist-1
CAS:β2AR/M-receptor agonist-1 (example 131), a muscarinic antagonist and β2 adrenoceptor agonist (MABA), exhibits dual potency towards β2 adrenoceptor andFormula:C43H56BrN3O7Color and Shape:SolidMolecular weight:806.82Cortistatin-29 (rat) (trifluoroacetate salt)
CAS:Cortistatin-29, similar to somatostatin-28, derives from preprocortistatin and binds to SST receptors 1-5 with varying IC50 values.Formula:C161H240N46O41S2Color and Shape:SolidMolecular weight:3540.09Apelin-36(human)
CAS:Endogenous APJ agonist, EC50=20nM, regulates cardiovascular function, fluid balance, and feeding; blocks certain HIV strains.Formula:C184H297N69O43SPurity:98%Color and Shape:SolidMolecular weight:4195.87Antipsychotic agent-2
Compound 11: potent antipsychotic, binds 5-HT1A/2A/2C, D2, H1 receptors; K is 56.6-1140 nM, BBB permeable.Formula:C22H26FN5OColor and Shape:SolidMolecular weight:395.47Dipentylone hydrochloride
CAS:Dipentylone hydrochloride (Bk-dmbdp HCl) is a psychoactive synthetic cathinone and sympathomimetic stimulant. Its inhibitory activity towards the dopamine transporter (IC50=0.233µM) is tenfold higher than that towards NET and SERT, inhibiting dopamine uptake and stimulating locomotor activity in mice.Formula:C14H20ClNO3Purity:99.94%Color and Shape:SolidMolecular weight:285.77DSP-1053
CAS:Dsp-1053 is a powerful SERT (Ki=1.02 nM) inhibitor with partial 5-HT1A receptor (Ki=5.05 nM) agonizing activity.Formula:C26H32BrNO4Purity:98%Color and Shape:SolidMolecular weight:502.44Albenatide
CAS:Albenatide is a modified analog of exendin 4 conjugated to recombinant human albumin.
Formula:C26H47N7O9SPurity:98%Color and Shape:SolidMolecular weight:633.76[Nle11]-Substance P
CAS:'[Nle11]-Substance P is a gut and brain peptide, resisting methionine oxidation and causing excitatory neural effects.'
Formula:C64H100N18O13Purity:98%Color and Shape:SolidMolecular weight:1329.59Endothelin 1 (swine, human), Alexa Fluor 488-labeled
Synthetic human/swine Endothelin 1 peptide, tagged with Alexa Fluor 488, acts as a strong vasoconstrictor via ET A/B receptors.Color and Shape:SolidMolecular weight:2848.4Ethoxyquin Dimer
CAS:Ethoxyquin dimer is an antioxidant, metabolite of ethoxyquin, that protects fish meal/oil fats but can cause liver damage in mice.Formula:C28H36N2O2Color and Shape:SolidMolecular weight:432.608VIP36
VIP36 is an agonist of the cannabinoid type 1 receptor (CB1) with analgesic properties. It reduces the recruitment of inhibitory proteins, thereby exerting its pain-relieving effects, and is applicable in research related to chronic pain.Formula:C27H35FN6O4Color and Shape:SolidMolecular weight:526.603Relaxin H3 (human) TFA
Relaxin H3 (human) (TFA) is a relaxin peptide that exerts antifibrotic effects through the RXFP1 receptor.Formula:C237H374N70O69S6·xC2HF3O2SU 4029 dihydrochloride
CAS:SU 4029 dihydrochloride is a bioactive chemical.Formula:C9H21Cl2N3OColor and Shape:SolidMolecular weight:258.19(3R,5R,6S)-Atogepant
(3R,5R,6S)-Atogepant (MK-8031) is a CGRP antagonist enantiomer used in migraine research.Formula:C29H23F6N5O3Color and Shape:SolidMolecular weight:603.52S 16474
CAS:S 16474 is an antagonist of Neurokinin-1 Receptor.Formula:C44H48N6NaO8Purity:98%Color and Shape:SolidMolecular weight:811.892GRL018-21
GRL018-21 is a potent, highly selective inhibitor of G protein-coupled receptor kinase 5 (GRK5), exhibiting an IC50 of 10 nM [1].Color and Shape:Odour SolidPF-9184
CAS:PF-9184 inhibits human mPGES-1 selectively, with an IC50 of 16.5 nM, and reduces IL-1β-stimulated PGE2 production in vitro.Formula:C21H14Cl2N2O4SPurity:97.43%Color and Shape:SolidMolecular weight:461.32[D-Glp1,D-Phe2,D-Trp3,6]-LH-RH
CAS:[D-Glp1,D-Phe2,D-Trp3,6]-LH-RH is a synthetic LHRH analog and a GnRH receptor antagonist.Formula:C67H84N16O13Color and Shape:SolidMolecular weight:1321.48INCB 3284 dimesylate
CAS:INCB 3284 dimesylate: oral CCR2 antagonist, blocks MCP-1/hCCR2 binding (IC50: 3.7 nM), potential in acute liver failure research.Formula:C28H39F3N4O10S2Purity:98%Color and Shape:SolidMolecular weight:712.76AZP-531
CAS:Azp-531 is a disacylated ghrelin used to improve blood sugar control and weight loss.Formula:C40H63N15O13Purity:98%Color and Shape:SolidMolecular weight:962.02Imelciment
CAS:Imelciment (REGN-9035) is a humanised monoclonal antibody targeting NPR1, which can be used for research into heart failure.Purity:95%Color and Shape:SoildProtease-Activated Receptor-1 antagonist 2
CAS:Orally active PAR-1 antagonist with 7 nM IC50; potential for CVD research.Formula:C24H23F2N3O2Color and Shape:SolidMolecular weight:423.46Heterobivalent ligand-1
Heterobivalent ligand-1 targets A2A-D2 receptor heteromer with affinity: Kd for A2A=2.1 nM, D2=0.13 nM.Formula:C86H115FN16O21Color and Shape:SolidMolecular weight:1727.93Adrenomedullin (16-31), human
CAS:Adrenomedullin (16-31), human is amino acid residues 16-31 fragment of human adrenomedullin (hADM).Formula:C82H129N25O21S2Purity:98%Color and Shape:SolidMolecular weight:1865.19Cenderitide
CAS:Cenderitide fuses CNP with DNP, stimulates pGC-A/B, ups cGMP, curbs aldosterone, and aids GFR, not affecting BP—used in heart failure studies.Formula:C158H263N49O50S3Color and Shape:SolidMolecular weight:3745.27Cannabidiolic acid methyl ester
CAS:Cannabidiolic acid methyl ester (HU-580) is an orally active analogue of cannabidiolic acid. It enhances the activation of 5-HT1A receptors and increases the expression of c-Fos and NeuN in specific hypothalamic nuclei in rats. Cannabidiolic acid methyl ester exhibits anti-nausea, anxiolytic, and anti-nociceptive effects.Formula:C23H32O4Color and Shape:SolidMolecular weight:372.5CB2R probe 1
CAS:CB2R Probe 1, a cannabinoid 2 receptor (CB2R) fluorescent probe, exhibits both safety and environmental friendliness, boasting a dissociation constant (K i) of
Formula:C36H42N4O4Color and Shape:SolidMolecular weight:594.74Prostaglandin F1α
CAS:Prostaglandin F1α (PGF1α) is a lipid mediator and an endogenous metabolite of prostacyclin, regulate smooth muscle contraction.Formula:C20H36O5Color and Shape:SolidMolecular weight:356.5L-threo Lysosphingomyelin (d18:1)
CAS:L-threo Lysosphingomyelin, a natural S1P receptor agonist, has EC50s: 19.3 nM (hS1P1), 131.8 nM (hS1P3), 313.3 nM (hS1P2).Formula:C23H49N2O5PColor and Shape:SolidMolecular weight:464.6212(S)-HpEPE
CAS:12(S)-HpEPE, a fatty acid created by 12-lipoxygenase on EPA, has unclear biological activities but may resemble 12(S)-HpETE.
Formula:C20H30O4Color and Shape:SolidMolecular weight:334.456Poly-D-lysine hydrobromide (MW 1000-5000)
Poly-D-lysine hydrobromide (PDLHB) (MW 1000-5000) is a synthetically produced polymeric substrate widely used in neural cell culture. Additionally, Poly-D-lysine hydrobromide acts as a CaSR agonist peptide.Color and Shape:Odour SolidCyclosomatostatin TFA
Cyclosomatostatin TFA blocks SST receptor, reduces CRC cell growth, ALDH+ size, and sphere-formation.Formula:C46H58F3N7O8Color and Shape:SolidMolecular weight:893.99(Trp7,β-Ala8)-Neurokinin A (4-10)
CAS:(Trp7,β-Ala8)-Neurokinin A (4-10) is a potent neurokinin-3 (NK3) antagonist [1] .Formula:C41H57N9O10SColor and Shape:SolidMolecular weight:868.01Sauvagine TFA
Sauvagine TFA: frog-derived, 40-amino-acid CRF agonist; stimulates ACTH release, affects diuresis, cardiovascular system, endocrine glands.Formula:C204H347F3N56O65S1Color and Shape:SolidMolecular weight:4713.33D5R agonist 1
D5R Agonist 1 (Compound 5j) is a selective, orally active partial agonist of the D5 receptor that can penetrate the blood-brain barrier (EC50: 269.7 nM). It has been demonstrated to enhance cognitive abilities in a scopolamine-induced amnesia model.Color and Shape:Odour SolidHaloperidol D4
CAS:Haloperidol D4 is deuterium-labeled haloperidol.Formula:C21H23ClFNO2Purity:98%Color and Shape:SolidMolecular weight:379.89Neurokinin A(4-10) TFA
Neurokinin A (4-10) TFA is a tachykinin NK 2 receptor agonist [1] .Formula:C36H55F3N8O12SColor and Shape:SolidMolecular weight:880.93Efranarelaxin alfa
CAS:Efranarelaxin alfa is an agonist of the relaxin receptor. It shows potential for research in cardiovascular diseases and tissue repair.Color and Shape:LiquidBrexpiprazole S-oxide D8
CAS:Brexpiprazole S-oxide D8 (DM-3411 D8) is a deuterium-labeled metabolite of Brexpiprazole, a partial agonist at 5-HT1A and dopamine receptors.Formula:C25H19D8N3O3SPurity:98%Color and Shape:SolidMolecular weight:457.61BAY-6672 hydrochloride
CAS:BAY-6672 hydrochloride is a potent, selective antagonist of the human Prostaglandin F (FP) receptor, exhibiting an IC50 value of 11 nM.Formula:C26H28BrCl2N3O3Color and Shape:SolidMolecular weight:581.33Poly-D-lysine hydrobromide (MW 150000-300000)
Poly-D-lysine hydrobromide (MW 150000-300000) enhances neural cell adhesion in culture and acts as a calcium-sensing receptor agonist peptide in research.Color and Shape:Odour SolidGlucagon-like peptide 1 (1-37), human
CAS:Human GLP-1 (1-37) is a potent GLP-1 receptor agonist without impact on rat food intake or insulin secretion.Formula:C186H275N51O59Purity:98%Color and Shape:SolidMolecular weight:4169.48FR 113680
CAS:FR 113680 is a tripeptide substance P antagonist with NK1 receptor selectivity.Formula:C35H39N5O6Purity:98%Color and Shape:SolidMolecular weight:625.726Leukotriene B4 Ethanolamide
CAS:LTB4 binds to BLT1 (high affinity) and BLT2. LTB4-EA, a metabolite, is a stronger BLT1 antagonist, suggesting anti-inflammatory properties.Formula:C22H37NO4Color and Shape:SolidMolecular weight:379.541Prepro-ANF (56-92), human
CAS:Human prepro-ANF (56-92) activates renal guanylate cyclase and boosts its activity.Formula:C173H270N44O57Color and Shape:SolidMolecular weight:3878.26RWJ 676070
CAS:RWJ 676070 is an antagonist of vasopressin V1A/V2 receptor.Formula:C30H26ClFN2O5Color and Shape:SolidMolecular weight:548.99(S)-V-0219 hydrochloride
(S)-V-0219 hydrochloride, a GLP-1R PAM, triggers calcium in hGLP-1R HEK cells, lowers glucose in mice, and reduces fasting hunger.Formula:C20H26ClF3N4O2Color and Shape:SolidMolecular weight:446.89GLI1-IN-3
GLI1-IN-3 (Compound 11a) is a triterpenoid-like compound that inhibits Hedgehog signaling in cancer cells with GLI1 overexpression. It suppresses the proliferation of non-small cell lung cancer and prostate cancer cell lines with excessive Hh signaling activation. Additionally, GLI1-IN-3 reduces the expression of GLI1 protein and its target genes associated with tumor progression and proliferation in A549 and DU-145 cancer cells.Color and Shape:Odour SolidZoliprofen
CAS:Zoliprofen: potent, oral NSAID with anti-inflammatory, antipyretic, analgesic effects. Exceeds ibuprofen's efficacy in rats and rabbits.Formula:C12H11NO3SPurity:99.62%Color and Shape:SolidMolecular weight:249.29Ref: TM-T68025
1mg85.00€5mg170.00€10mg256.00€25mg480.00€50mg655.00€100mg933.00€500mg1,872.00€1mL*10mM (DMSO)168.00€Besipirdine hydrochloride
CAS:Besipirdine hydrochloride is a non-receptor-dependent cholinomimetic compound with cardiovascular activity that inhibits the uptake of biogenic amines.
Formula:C16H18ClN3Purity:98.45%Color and Shape:SoildMolecular weight:287.79GS-2278
CAS:GS-2278 is an antagonist of LPAR1 (lysophosphatidic acid receptor 1) with potential applications in the study of idiopathic pulmonary fibrosis (IPF).Formula:C22H16F5N9O3Color and Shape:SolidMolecular weight:549.41Lys-[Des-Arg9]Bradykinin
CAS:Selective bradykinin B1 agonist with Ki 0.12 nM; inactive at B2 (>30,000 nM). Lowers blood pressure, more potent than Des-Arg9-Bradykinin.Formula:C50H73N13O11Purity:98%Color and Shape:SolidMolecular weight:1032.21Protease-Activated Receptor-1, PAR-1 Agonist TFA
PAR-1 Agonist TFA: Selective peptide, mimics thrombin, activates PAR-1 receptor.Color and Shape:LiquidChemerin-9, Mouse
CAS:Chemokine-like receptor 1 (CMKLR1) agonist (EC50 = 42 nM). Corresponds to C-terminal of full length mouse Chemerin, amino acids 148 - 156.Formula:C51H68N10O12Color and Shape:SolidMolecular weight:1013.163Exendin-3/4 (59-86)
Exendin-3/4 (59-86) is a Exendin-4 peptide derivative.Formula:NAPurity:98%Color and Shape:SolidMolecular weight:3055.49Pentagastrin meglumine
CAS:Pentagastrin meglumine is a synthetic pentapeptide that has effects like gastrin when given parenterally.Formula:C44H66N8O14SColor and Shape:SolidMolecular weight:963.11Human follicular gonadotropin releasing peptide
CAS:Human Follicular Gonadotropin Releasing Peptide (hF-GRP) is a hormonal peptide that, in vitro, can induce the secretion of pituitary luteinizing hormone (LH)Formula:C68H94N22O27Color and Shape:SolidMolecular weight:1651.615-OMe-UDP trisodium salt
CAS:Potent P2Y6 agonistFormula:C10H16N2O13P2Purity:98%Color and Shape:SolidMolecular weight:434.19
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